EPA-540/1-86-026
oEPA
                      environmeniai riuieiuun
                      Agency
Office of Emergency and
Remedial Response
Washington DC 20460
                      Superfund
Off'ce of Research and Development
Office of Health and Environmental
Assessment
Environmental Criteria and
Assessment Office
Cincinnati OH 45268
                       HEALTH  EFFECTS ASSESSMENT
                       FOR  DDT

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                                           EPA/540/1-86-026
                                           September 1984
       HEALTH EFFECTS  ASSESSMENT
                  FOR DDT
    U.S. Environmental Protection  Agency
     Office of Research and Development
Office  of Health  and  Environmental Assessment
Environmental Criteria and Assessment  Office
            Cincinnati,  OH  45268
    U.S. Environmental Protection  Agency
  Office of  Emergency  and Remedial Response
Office of Solid Waste and  Emergency  Response
            Washington,  DC  20460

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                                  DISCLAIMER

    This  report  has  been funded  wholly  or  In  part by  the  United  States
Environmental  Protection  Agency under  Contract  No.  68-03-3112  to  Syracuse
Research Corporation.  It has been  subject  to  the Agency's peer and adminis-
trative review, and  1t has been  approved  for  publication as an EPA document.
Mention of  trade  names or commercial  products  does  not  constitute  endorse-
ment or recommendation for use.
                                      11

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                                    PREFACE
    This  report  summarizes and evaluates  Information  relevant  to a prelimi-
nary  Interim  assessment  of adverse health effects  associated  with DDT.   All
estimates  of  acceptable  Intakes  and  carcinogenic  potency  presented  1n  this
document  should  be considered  as preliminary and  reflect  limited resources
allocated  to  this  project.   Pertinent  toxlcologlc  and environmental  data
were  located  through  on-line literature  searches  of  the Chemical Abstracts,
TOXLINE,  CANCERLINE and  the CHEMFATE/DATALOG data  bases.   The basic  litera-
ture  searched supporting  this  document  Is  current  up  to  September,  1984.
Secondary  sources  of  Information  have also been  relied  upon 1n the prepara-
tion  of  this  report and  represent large-scale health  assessment efforts  that
entail extensive peer and  Agency  review.   The following  Office of Health and
Environmental Assessment (OHEA) sources have been extensively utilized:


    U.S.  EPA.   1980a.    Hazard   Assessment  Report  on  DDT,  ODD,  DDE.
    Environmental  Criteria  and   Assessment   Office,  Cincinnati,  OH.
    Internal report.

    U.S.   EPA.    1980b.    Ambient  Water  Quality  Criteria  for  DDT.
    Environmental  Criteria  and  Assessment Office,  Cincinnati,  OH.  EPA
    440/5-80-038.  NTIS PB 81-117491.

    U.S.  EPA.   1985.   The  Carcinogen Assessment  Group's  Evaluation  of
    the  Cardnogenlcity  of Dicofol (Kelthane), DDT,  DDE  and DDD  (TOE).
    Prepared  by  the Carcinogen Assessment Group,  OHEA,  Washington,  DC
    for  the Hazard Evaluation  Division  Office  of Pesticide  Programs.
    EPA 600/6-85-002X.  Internal Review Draft.
    The Intent in these assessments  is  to  suggest  acceptable exposure levels
whenever sufficient data  were  available.   Values were  not  derived  or larger
uncertainty  factors  were  employed  when the  variable  data  were limited  In
scope tending  to  generate conservative  (I.e.,  protective) estimates.  Never-
theless, the  interim  values  presented reflect the  relative  degree  of hazard
associated with exposure or risk to the chemical(s) addressed.

    Whenever possible, two categories of values  have  been estimated for sys-
temic toxicants (toxicants for which  cancer  is  not  the endpoint of  concern).
The  first,  the AIS  or acceptable  intake  subchronic,  is  an estimate  of  an
exposure  level  that  would not  be  expected  to cause  adverse  effects  when
exposure occurs during a  limited time  interval  (I.e.,  for  an  Interval that
does not  constitute  a  significant  portion of  the Hfespan).   This  type  of
exposure estimate  has not been  extensively used  or  rigorously  defined,  as
previous  risk  assessment  efforts   have  been  primarily  directed  towards
exposures from toxicants  in  ambient air or water where lifetime exposure  is
assumed.  Animal  data  used  for  AIS estimates  generally  include  exposures
with durations of  30-90 days.  Subchronic  human data  are  rarely available.
Reported exposures are usually  from chronic  occupational exposure situations
or from reports of acute accidental  exposure.
                                      111

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    The  AIC,  acceptable  Intake  chronic,  is  similar  In  concept  to  the  ADI
(acceptable  dally  Intake).   It   Is  an  estimate  of an  exposure level  that
would  not  be expected  to cause  adverse effects  when  exposure occurs  for  a
significant portion  of  the llfespan  [see  U.S.  EPA  (1980c)  for  a discussion
of  this  concept].   The  AIC  Is  route specific  and  estimates  acceptable
exposure  for  a  given  route with  the  Implicit  assumption that  exposure  by
other routes 1s Insignificant.

    Composite  scores  (CSs)  for  noncardnogens  have  also  been  calculated
where data  permitted.   These  values  are used for  ranking reportable quanti-
ties; the methodology for their development is explained  in U.S.  EPA (1983).

    For  compounds for which there  Is  sufficient  evidence  of  carcinogenlcity,
AIS  and AIC values  are  not derived.   For a  discussion  of risk assessment
methodology  for  carcinogens  refer to  U.S. EPA  (1980c).   Since  cancer  is  a
process  that  Is  not  characterized by  a threshold,  any exposure  contributes
an  Increment of  risk.   Consequently,  derivation of  AIS and  AIC  values  would
be  Inappropriate.   For  carcinogens,   q-|*s  have been computed  based  on  oral
and Inhalation data if available.
                                      iv

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                                   ABSTRACT
    In  order  to  place the  risk assessment  evaluation  1n  proper  context,
refer  to  the preface  of  this  document.   The  preface outlines  limitations
applicable to all documents of  this  series as  well  as  the appropriate Inter-
pretation and use of the quantitative estimates presented.
    U.S.  EPA  (1985)  estimated
orally administered DDT based on
separate studies.
a  human  q-|*
the geometric
 of  0.34
average of
(mg/kg/day) 1  for
potencies from six
    Data are  not  available for  the  evaluation  of the  potential  cardnogen-
1dty of DDT following Inhalation exposure.

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                               ACKNOWLEDGEMENTS
    The  Initial  draft  of  this  report  was  prepared  by Syracuse  Research
Corporation under  Contract No.  68-03-3112  for EPA's  Environmental  Criteria
and  Assessment  Office,  Cincinnati,  OH.   Or.  Christopher  DeRosa and  Karen
Blackburn were the Technical Project Monitors  and  Helen Ball  was',the Project
Officer.  The final documents  In  this  series  were  prepared for the Office of
Emergency and Remedial Response, Washington, DC.

    Scientists from  the  following U.S. EPA offices  provided  review comments
for this document series:

         Environmental Criteria and Assessment Office, Cincinnati, OH
         Carcinogen Assessment Group
         Office of A1r Quality Planning and Standards
         Office of Solid Waste
         Office of Toxic Substances
         Office of Drinking Water

Editorial review for the document series was provided by:

    Judith Olsen and Erma Durden
    Environmental Criteria and Assessment Office
    Cincinnati, OH

Technical support services for the document series  was provided by:

    Bette Zwayer, Pat Daunt, Karen Mann and Jacky Bohanon
    Environmental Criteria and Assessment Office
    Cincinnati, OH
                                      v1

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                          TABLE  OF  CONTENTS

1.
2.


3.








ENVIRONMENTAL CHEMISTRY AND FATE 	
ABSORPTION FACTORS IN HUMANS AND EXPERIMENTAL ANIMALS . . .
2.1.
2.2.
ORAL 	
INHALATION 	
TOXICITY IN HUMANS AND EXPERIMENTAL ANIMALS 	
3.1.


3.2.


SUBCHRONIC 	
3.1.1. Oral 	
3.1.2. Inhalation 	
CHRONIC 	
3.2.1. Oral 	
3.2.2. Inhalation 	
Page
1
, . . 2
. . . 2
2
, . . 3
3
. . . 3
3
. . . 3
. . . 3
. . . 7
3.3.   TERATOGENICITY AND OTHER REPRODUCTIVE EFFECTS.



4.








5.


3.4.
3.3.1. Oral 	
3.3.2. Inhalation 	 ,
TOXICANT INTERACTIONS 	
CARCINOGENICITY 	 ,
4.1.


4.2.


4.3.
4.4.
HUMAN DATA 	
4.1.1. Oral 	
4.1.2. Inhalation 	 ,
BIOASSAYS 	 ' 	
4.2.1. Oral 	
4.2.2. Inhalation 	
OTHER RELEVANT DATA 	
WEIGHT OF EVIDENCE 	
REGULATORY STANDARDS AND CRITERIA 	
	 7
	 8
	 8
	 11
	 11
	 11
	 11
	 11
	 11
	 17
	 17
	 18
	 19
                                 vll

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                           TABLE  OF  CONTENTS  (cont.)

                                                                        Page

 6.   RISK ASSESSMENT	   20

     6.1.   ACCEPTABLE  INTAKE SUBCHRONIC (AIS) 	   20
     6.2.   ACCEPTABLE  INTAKE CHRONIC (AIC)	   20
     6.3.   CARCINOGENIC POTENCY (q-|*)	   20

            6.3.1.   Oral	   20
            6.3.2.   Inhalation	   26

 7.   REFERENCES	   31

APPENDIX: Summary Table for DOT	   43

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                               LIST OF TABLES

No.                               Title                                Page
3-1     Subchronlc Oral Toxldty of DDT in Rats	    4

3-2     Chronic Oral Toxlclty of DDT	    5

3-3     Reproductive Studies	    9

4-1     Oral Carc1nogen1c1ty of DDT	   12

6-1     Incidence of the Most Commonly Occurring Malignant Tumors
        1n Each of Five Generations of BALB/c Mice Fed DDT	   21

6-2     Incidence of Benign Liver Tumors 1n Each of Six
        Generations of CF-1 Mice Fed DDT	   23

6-3     Incidence of Benign Liver Tumors In BALB/C Mice Fed DDT
        During a 2-Generat1on Experiment	   25

6-4     Incidence of Liver Tumors (Benign and Malignant) In CF-1
        Mice Fed DDT for a Single Generation	   27

6-5     Incidence of Benign Liver Tumors 1n CF-1 Mice Fed DDT for
        15 or 30 Weeks and then Sacrificed at 65, 95 and 120 Weeks.  .   28

6-6     Incidence of Benign Liver Tumors 1n Rats Fed DDT	   29

6-7     Summary of Quantitative Potency Estimates for DDT 	   30
                                     1x

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                             LIST OF  ABBREVIATIONS
ADI                     Acceptable dally Intake
AIC                     Acceptable Intake chronic
AIS                     Acceptable Intake subchronlc
BCF                     Bloconcentratlon factor
bw                      Body weight
CAS                     Chemical Abstract Service
CS                      Composite score
ppm                     Parts per million
SER                     Smooth endoplasmlc retlculum
STEL                    Short-term exposure limit
TLV                     Threshold limit value
TWA                     Time-weighted average

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                      1.   ENVIRONMENTAL CHEMISTRY  AND FATE
    The physical  and  chemical properties  and environmental  fate  of DDT  (CAS
No. 50-29-3 for p.p'-DDT and 789-02-6 for  o.p'-DDT)  are as  follows:
    Chemical class:
    Molecular weight:
    Vapor pressure at  20°C:

    Water solubility at 25°C:
    Log octanol/water
    partition coefficient:
    BCF:
    Half-life 1n
      Water:
      Soil:
pesticide (Callahan et al., 1979)
354.5 (Callahan et al., 1979)
1.5xlO~7 mm Hg for p.p'-DDT
5.5xlO"6 mm Hg for o.p'-DDT
(Callahan, et al., 1979)
1.2-25 yg/8. for p.p'-DDT
26-85 yg/i for o.p'-DDT
(Callahan et al., 1979)

3.98-6.19 (Callahan et al., 1979)
103 to 106 (Callahan et al., 1979)
56-110 days 1n lake water
(Zoeteman et al., 1980)
3-15 years (IARC, 1974)
    The  mobility  of DDT  In soils  has  been studied  by various  authors  (U.S.
EPA, 1980a) and has been  reported  to  be  extremely slow.  Therefore, the leach-
Ing of  DDT from soil  1s  expected to be  very  slow, particularly  1n  soil  with
high  organic  carbon content.   Nevertheless,  leaching  of  DDT  from  soil  Into
groundwater at a frequency of 8-9% has been reported (Page, 1981).
    The  half-life of DDT  In  the  atmosphere 1s  uncertain.   DDT 1s probably lost
from the atmosphere by  ralnout,  fallout  or photochemical  degradation (Spencer,
1975).   The photolytlc  half-life for  the  transformation of  DDT  to DDE  and ODD
1n  the atmosphere can  be  estimated  to be -17 days (Crosby and Mollanen, 1977).
The fact  that DDT has  been  found to participate 1n long distance aerial trans-
port  (Callahan  et  al.,  1979)  Indicates  that  1-t has a long half-life  1n the
atmosphere.

                                      -1-

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            2.  ABSORPTION FACTORS IN HUMANS AND EXPERIMENTAL ANIMALS
2.1.   ORAL
    Jensen  et  al.   (1957)  reported  that  95%  of  the Ingested  DDT  in rats  Is
absorbed  from  the   gastrointestinal  tract.   Over  65% of  the  labeled DOT  was
recovered  in the bile  collected from  rats  for  9 days following  DDT  ingestion
(Jensen et  al.,  1957).   More DDT is absorbed  in  rats when it  is dissolved  in
digestible  vegetable oils  than  when it  is  suspended 1n  water  or dissolved  in
indigestible mineral oils (Keller and  Yeary, 1980).
    In humans,  the  absorption  of DOT  follows  the same pattern as  the  absorp-
tion of dietary  fat, that  is,  absorption is relatively  slow;  however,  absorp-
tion appears to be  complete  after 24 hours (Morgan and Roan,  1977).
2.2.   INHALATION
    Pertinent data   regarding the absorption of  DDT by Inhalation could  not  be
located in the  available literature.
                                     -2-

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                 3.  TOXICITY  IN HUMANS AND EXPERIMENTAL ANIMALS
3.1.   SUBCHRONIC
3.1.1.   Oral.   Laug  et  al.  (1950)  exposed  rats  to different  levels  of  DDT
(1-50 ppm)  1n the  food  and  examined  the  histology of  the liver  15-27  weeks
after the  start of  treatment.   No  effects  were  reported at  an  exposure  of
1 ppm;  however,  at all  the  higher  exposure levels  (5-50 ppm), hepatic  cell
hypertrophy  appeared   to  be  dose-related  and   minimal  alterations  In  Hver
histology were reported at an exposure of  5  ppm (Laug  et  al.,  1950).   Hart and
Pouts (1965)  reported  Increased  liver  mlcrosomal enzyme activity 1n  rats  at  5
and 50 ppm.   Ortega et al.  (1956a,b) reported ultrastructural  changes at  5 and
15 ppm 1n livers of male  rats  (Table 3-1).
3.1.2.   Inhalation.   Pertinent  data  regarding the  inhalation  of  DDT  could
not be located in the  available  literature.
3.2.   CHRONIC
3.2.1.   Oral.   Exposure  of  rats  to  200 ppm  (10  mg/kg/day)  DDT  in the  food
for  2  years   resulted  in  Increased liver weight in  the females  (FHzhugh  and
Nelson,   1947; FHzhugh,  1948).    At  higher  doses  (400-800   ppm),   the  liver
alterations became more severe and were  present in  both  sexes.   Liver  lesions
were present  at  all dose levels  tested,  the lowest of  which  was  10 ppm  (0.5
mg/kg/day)  (Fltzhugh   and  Nelson,  1947;  FHzhugh,  1948)  (Table  3-2).    In
chronic   exposure  studies  with   DDT,  effects appeared  to  be  most  severe  In
offspring exposed to DDT  for  their  entire  Hfespan,  especially during in  utero
development  and  nursing.   This   1s demonstrated  in the  study  of  Treon  and
Cleveland (1955) in which male  rats exposed to  25 ppm  (1.25 mg/kg/day) DDT in
the food for  2  years  and  3 generations had  increased liver weights.   In  mice,
lactation was  decreased   and  the mortality  of   the  offspring  increased at  an
exposure  level  of   100  ppm  (13.0  mg/kg/day) for  6  generations  (Keplinger  et
al.,  1968).   The incidence of  tumors  was increased at  exposure levels of  50

                                     -3-

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                                                                   TABLE 3-1

                                                    Subchrontc Oral Toxlclty of DDT In Rats
Dose*
Isomer
ppm
NR 50
10
5
1
NR 350

i
f NR 50
5
NR 15
5

NR 0.2

rag/kg/day
2.5
0.5
0.25
0.05
17.0


2.5
0.25
0.75
0.25

0.01

Duration of Sex
Exposure
15-27 weeks H/F



33-60 weeks NR


3 months NR

2-18 months NR


1-13 weeks NR

Number
Used
75/75



NR


NR

NR


NR

Effects
Hepatic cell hypertrophy was definitely present at
dose levels of 50 and 10 ppm, and minimally present
at 5 ppm. No effects were reported at 1 ppm.

No htstopathologlc alteration In the exposed as
compared with the control group.

Liver mlcrosomal enzyme activity was Increased at
both exposure levels.
Males had hlstopathologlc alterations (proliferation
of SER and concentric membrane arrays) In the liver
at both exposure levels.
Liver mlcrosomal enzyme activity was not Increased.

Reference
Laug et al.,
1950


Cameron and
Cheng, 1951

Hart and
Fouts, 1965
Ortega et al.,
19S6a,b

Klnoshtta
et al.. 1966
*The fraction of body weight consumed per day  In food,  called  the food factor. Is 0.13 for mice and  0.05  for  rats.   Exposures  given  In  ppm of
 food are converted to mg/kg/day by multiplying the ppm  exposure  level  by  the  food factor.

NR = Not reported

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                                                                            TABLE  3-2

                                                                  Chronic Oral Toxlclty of DDT

Isomer3
ppra
Technical 800
600
400
200
TOO
50
TO
0





Doseb
Duration of
mg/kg/day Exposure
40 2 years
30
20
TO
5
2.5
0.5







Species Sex

rat/ H/F
Osborne- H/F
Hendel H/F
H/F
H
NR
NR
H/F






Number
Used
24/24
24/24
24/12
24/12
T2
NR
NR
24/T2






Effects Reference

At 800 ppm there were Increased Fltzhugh and
mortality and liver lesions. In- Nelson, 1947;
creased liver weight occurred at Fltzhugh, 1948
200 ppm for females and at higher
doses for both males and females.
No second generation offspring
survived In animals exposed to 600
ppm. A reduction In survival of
preweanllng rats occurred at DDT
levels of >50 ppm. Liver lesions
were present at all dose levels,
but no reproductive effects were
reported at exposures of 10 ppm.
         NR
i
en
i
         Technical
         Technical
         Technical
 25
 12.5
  2.5
  0
200
250
 50
 10
250

 20
 1.25
 0.625
 0.125
10
32.5
 6.5
 1.3
32.5

 2.6
2 years/
3 generations
rat
2 generations
2 generations
rat/
Sprague-
Dawley

mouse
4 generations

2 generations
mouse/
BALB/c
mouse/
BALB/c
H/F     40/40      Hales had Increased liver weights
H/F     40/40      at an exposure level of 25 ppm.
H/F     40/40      Although size of the litter and the
H/F     40/40      number of pregnancies remained un-
                   affected by DDT. the mortality of
                   the offspring was Increased at all
                   exposure levels.

NR      NR         Increased liver weight, but no
                   reproductive disturbance, was seen
                   In exposed animals.

NR      NR         There was an Increased Incidence of
                   liver tumors at all exposure levels
                   tested.  At an exposure of 250 ppm,
                   there was Increased mortality In
                   the neonates, and reduced llfespan.
                   Tremors and convulsions occurred In
                   some animals.

NR      NR         Although no effects on reproduction
                   were reported, females suffered re-
NR      NR         duced llfespans In addition to gas-
                   trointestinal bleeding, convulsion
                   and Increased Incidence of tumors.
Treon and
Cleveland, 1955
Ottobonl, 1969
Tomatls et al..
1972
Terraclnl
et al., 1973a,b

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                                                               TABLE  3-2 (cont.)

Isomera
ppm
p.p'-DDT 100
50


Technical 200
p.p'-DDT 200
Technical 3200
2000
400
0
p.p'-DDT 1000

500

0
i
f Technical 1000
500
250

NR 500
250
125
Doseb
Duration of Species
mg/kg/day Exposure
13.0 2 years mouse
6.5


8.0 3.5-7.5 years monkey
8.0
128 39-40 months dog
80
16

80 44/48 weeks hamster

40



80 18 months hamster
40
20

40 llfespan hamster
20
10
Sex
NR



NR

M/F
H/F
H/F
H/F
H/F

H/F

H/F

NR
NR
NR

NR


Number
Used
NR



NR

7/7
2/2
1/1
1/1
25-30/
25-30
25-30/
25-30
79

NR
NR
NR

NR


Effects
The Incidence of liver tumors was
Increased at both exposure levels.


No observed effects reported.

No effects were observed at 400
ppm, but liver damage occurred at
2000 ppm and was more severe at
3200 ppm.
Increased mortality as well as
nervousness and convulsions were
observed In exposed animals.



Increased liver weight and enzyme
(glucose-6-phosphate dehydrogenase)
activity and decreased llfespan
were reported.
No observed effects on growth or
survival .

Reference
Thorpe and
Walker. 1973;
Walker et al..
1972
Durham et al. ,
1963
Lehman. 1952.
1965


Agthe et al..
1970




Gralllot
et al., 1975


Cabral and
Shublk. 1977

technical DDT consists  of  -77.IX p.p'-DDT.  14.9X o.p'-DDT,  0.3X p.p'-DDD, 0.1X  o.p'-DDD,  4.OX p.p'-DDE,  0.1X o.p'-DDE and 3.5X unidentified
 compounds (U.S.  EPA. 1980a).

bThe fraction of  body  weight  consumed  per  day In food, called  the  food factor.  Is 0.13  for mice and 0.05 for  rats.   Exposures  given In ppm
 of food are converted to mg/kg/day by  multiplying the ppm exposure  level by the food factor.

NR = Not reported

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ppm (6.5 mg/kg/day) for 2 years  (Thorpe  and  Walker,  1973;  Walker et a!.,  1972)
and at  20  ppm (2.6  mg/kg/day)   1n  a  2-generatlon  study  (Terraclnl  et  al.,
1973a,b).    The llfespan  of  the  females  that  suffered from  gastrointestinal
bleeding and  convulsions  was  decreased  at  an  exposure level  of 20 ppm  (2.6
mg/kg/day)   for 2-4 generations  (Terraclnl  et  al.,  1973a,b).   Durham et  al.
(1963)  reported  that  there  was  no observed effect  In monkeys  exposed  to  200
ppm (8.0 mg/kg/day) DOT  In  the food  for  3.5-7.5  years;  however, the offspring
of dogs exposed  to 1  ppm  (0.04  mg/kg/day)  DDT  In  the food  for 3 generations
had consistently  Increased  liver  weights (Ottobonl  et al.,  1977).   Hamsters
were exposed to much  higher  levels  of DDT, ranging  from 125 ppm (10 mg/kg/day)
to 1000 ppm (80 mg/kg/day).   At  an  exposure level  of  500  ppm (40 mg/kg/day),
Agthe et al.  (1970)  reported  nervousness, convulsions  and  Increased mortality
1n exposed  animals;  Gralllot  et  al.  (1975)  reported  Increased  liver  weights;
and Cabral  and Shublk (1977)  reported  that  there was no effect on the  growth
or survival of exposed hamsters.
3.2.2.   Inhalation.    Pertinent   data   regarding  the  chronic   toxlclty   of
Inhaled DDT could not  be located In the available literature.
3.3.   TERATOGENICITY AND OTHER REPRODUCTIVE EFFECTS
3.3.1.   Oral.  When  pregnant  mice were exposed  to  1  mg/kg bw  on days  10, 12
and  17  of  gestation, morphologic  changes  were  seen  In   the  gonads and  the
fertility  of   the  female  offspring  was  reduced  (McLachlan and  Dlxon,  1972).
Although no teratogenesls was  observed,  2.5  mg/kg given dally to  pregnant mice
was significantly  embryotoxlc, as well  as blastotoxlc  and  fetotoxlc (Schmidt,
1973).   Similarly 1n rabbits,  Increased resorptlon,  premature  delivery  and
reduced fetal  growth,  but  no  teratogenlclty,  were  caused by  exposure  to 50
mg/kg DDT  on   days 7,  8  and 9 of  pregnancy.  When rats were  exposed  to 7 ppm
DDT 1n  the diet for  60 days  before mating  and for  the duration  of pregnancy,
fertility was  decreased and  the  number  of resorptlons Increased,  but there was

                                      -7-

-------
no evidence of teratogenidty  (Green,  1969)  (Table 3-3).  Although there have
been no reports of any teratogenlc effects of DDT, with  the  possible  exception
of ringtail occurring  1n rats exposed  to  200 ppm DDT  1n  the diet  (Ottobonl,
1969),  DDT has consistently caused a decrease in reproductive  capacity  in mice
(Keplingler et  al.,  1968;  McLachlan  and  Dixon,  1972;  Schmidt,  1973), rats
(Fltzhugh and  Nelson, 1947; FHzhugh, 1948; Treon  and Cleveland,  1955;  Clement
and  Okey,  1974;  Oonsson  et  al.,  1975)  and dogs  (Deichmann et  al., 1971;
Deichmann and  MacDonald, 1971).   Some  studies reported  no observed effects  on
reproduction  1n   rats  (Ware  and  Good, 1967;  Duby  et  al.,  1971)  and dogs
(Ottoboni et al.,  1977)  (see Tables 3-2 and 3-3).
3.3.2.    Inhalation.  Pertinent  data  regarding the  teratogenicity  of  inhaled
DDT were not located 1n  the available literature.
3.4.   TOXICANT INTERACTIONS
    Although there  is widespread concern about the synergistic Interaction  of
DDT with  other  potentially hazardous  chemicals,   the interaction  of DDT with
only a  few  chemicals  has been  studied.   Welsburger   and  Weisburger   (1968)
reported that  10  mg/day  of DDT significantly  increased  the  incidence of hepa-
tomas  In rats, caused by the  ingestlon  of  1 mg/day N-fluorenacetamide (2-AAF).
They postulated  that  DDT  exerted  Us  Influence  by stimulating  the  hepatic
mixed  function oxidase system  (Welsburger  and Weisburger,  1968).  On  the other
hand,  after evaluating the  Interaction  of  DDT, aramite,  methoxychlor, thiourca
and aldrin, Deichmann  et al.  (1967)  concluded  that  the chemicals did  not  act
synergistlcally,  and, in fact, may  have Interacted antagonistically.  Although
there  was  no  Increase  in the overall Incidence of Hver tumors when  mice were
exposed  to 100 ppm DDT and  5  ppm  dleldrln  simultaneously,  the  hlstological
characteristics of  the  liver  tumors  were  more malignant  after  the  mice were
exposed to DDT and dieldrln simultaneously  (Walker  et  al.,  1972).
                                      -8-

-------
                                                                          TABLE 3-3

                                                                     Reproductive  Studies
i
10
Ooseb
Isomera
Technical


p.p'-DDT
o,p'-DDT
Technical
NR
p.D'-DOT
I* • r •*" •





o.o'-DDT
** t r "•* "



NR




NR
ppm
7


15
15
15
1
500
200
20




1000
200
20


150
75



7
0
Duration of Species
mg/kg/day Exposure
0.9 120 days mouse/
BALB/c
and CFW
0.75 2 generations rat
0.75
0.75
0.05 175 days
25 6 months rat
10
1




50 6 months rat
10
1


7.5 8-36 weeks rat
3.75



0.35 2 generations rat
Sex
NR


NR
NR

NR
NR
NR
NR
NR



NR
NR
NR


NR
NR



NR
NR
Number
Used
NR


NR
NR

NR
NR
NR
NR
NR



NR
NR
NR


NR
NR



131
396
Effects
No observed effect on reproduction
was reported.

No effects on reproduction were
reported.


No effects were seen at the 20 ppm
dose level. Growth of offspring
was severely depressed at the 200
ppm dose level, and all offspring
died within 10 days of birth when
the animals were exposed to 500 ppm
p.p'-DDT.
The only effects on reproduction
were seen at the 1000 ppm dose
levels, which caused decreased
fertility and growth In exposed
animals.
An exposure level of 150 ppm caused
reproductive failure. At 75 ppm.
the number of pups/litter was not
changed, but there was a decreased
number of pregnant females.
None of the rats In the second gen-
eration were able to get pregnant.
Reference
Ware and Good,
1967

Duby et al..
1971


Clement and
Okey. 1974





Clement and
Okey, 1974



Jonsson et al..
1975



Green, 1969
        Technical
        NR
200
 25
 12.5
  2.5
  0
10
 1.25
 0.625
 0.125
2 generations
2 years/
3 generations
rat/
Sprague-
Oawley

rat
                   There was decreased fertility and
                   Increased mortality In the first
                   generation.

NR      NR         No reproductive disturbance was
                   seen In exposed animals.
M/F     40/40      Although size of the litter and the
H/F     40/40      number of pregnancies remained un-
H/F     40/40      affected by DDT, the mortality of
H/F     40/40      the offspring was Increased at all
                   exposure levels.
                                                                                                                                       Ottobonl. 1969
Treon and
Cleveland. 1955

-------
                                                                       TABLE 3-3 (cont.)
o
i
Isomera
Technical




Technical



NR







p.p'-DDT





Technical






ppm
250
SO
10


250

20

250
100
25











10
5
1



Doseb
Duration of Species
mg/kg/day Exposure
32.5 2 generations mouse
6.5
1.3


32.5 4 generations mouse/
BALB/c
2.6 2 generations mouse/
BALB/c
32.5 6 generations mouse
13.0
3.25





12 5 times/week, dog
14 months




0.4 3 generations dog
0.2
0.04



Sex Number Effects
Used
NR NR At an exposure of 250 ppm, there
was Increased mortality In the
neonates, and reduced llfespan.
Tremors and convulsions occurred
In some animals.
NR NR No effects on reproduction were
reported.
NR NR

NR NR No reproductive effects were seen
NR NR at exposure levels of 25 ppm. At
NR NR an exposure level of 100 ppm lacta-
tion was reduced and mortality of
the offspring Increased. The
severity of the effects produced
at 100 ppm were greatly Increased
at 250 ppm.
H/F 4/3 Decreased male libido and delayed
female estrus were reported, as
well as Infertility, reduced lacta-
tion and mammary gland development,
and Increased maternal and fetal
mortality.
NR NR Except that estrus occurred earlier
In exposed dogs than In controls,
there were no observed effects on
reproduction. However, liver weights
were consistently higher In pups
exposed to DDT.
Reference
Tomatls et al..
1972



Terradnl
et al.. 1973a,b


Kepllnger
et al.. 1968






Delchmann
et al.. 1971;
Delchmann and
Mac Dona Id. 1971


Ottobonl
et al.. 1977




        aTechn1cal DDT  consists  of  -77.IX p.p'-DDT.  14.9X o.p'-DDT. 0.3X p,p'-DDD.  0.1X o.p'-DDD,  4.OX p.p'-DDE, 0.1X o.p'-DDE and 3.5X unidentified
         compounds (U.S. EPA. 1980a).

        DThe  fraction  of  body weight consumed per day In food, called the food factor,  Is 0.13  for  mice,  0.05 for rats and 0.04 for dogs.  Exposures
         given  In ppm of food are converted to mg/kg/day by  multiplying  the ppm exposure  level  by  the food  factor.

        NR = Not reported

-------
                              4.  CARCINOGENICITY
4.1.   HUMAN DATA
4.1.1.   Oral.  A group of prison volunteers  Ingested  dally doses of DDT  (3.5
mg/man/day  or  35 mg/man/day)  for  21.5 months  (Hayes  et  al.,  1971).  No  111
effects ascribed  to  DDT 1ngest1on were  reported  4-5 years after  the  start  of
the experiment.
4.1.2.   Inhalation.    Human  data  regarding  the  cardnogenlclty  of  DDT  has
been  collected  from  occupational   exposure,  which  occurs  chiefly  through
Inhalation.   In  occupational exposures  where doses  ranged from  an  estimated
10-40  mg/man/day for  1-8 years  (Ortelee, 1958)  and 3-18  mg/man/day for  an
average  of 15 years  (range, 11-19  years)  (Laws  et  al.,  1967),  no  Increased
Incidence of cancer was reported.
4.2.   BIOASSAYS
4.2.1.   Oral.   The  cardnogenlclty  of  DDT  has   been  tested  extensively  1n
mice, rats  and hamsters.   An NCI  study,  reported  by Innes  et al. (1969),  found
Increased  Incidence   of  hepatomas   1n  male  and  female  mice  exposed  to  DDT
beginning  at  7  days  of age.   At first  the  DDT was  Introduced by gavage;  after
weaning at  4  weeks the  DDT was  Incorporated 1n  the diet.  In addition to liver
tumors,  females  had  an Increased  Incidence of  lymphomas  (Innes  et  al.,  1969)
(Table 4-1).
    Tarjan  and  Kemeny  (1969) studied  five generations of  BALB/c  mice exposed
to  DDT  at  a level of 2.8-3.0 ppm  In the diet.   A  variety of tumors accounted
for  the  Increased  Incidence of  cancer  1n exposed  (28.7%)  as  compared with
control  (3.2%)  groups.   Lung  carcinoma,  which  occurred  In  116  of  the 196
animals  with  tumors,   was   the  predominant type.   Leukemia was  found  1n  23
females  and 21  males  of   the 196  animals that  developed  tumors.   Tumors were
also  observed  In the  liver,   kidney,  spleen,  ovary and other  organs.   The
                                     -11-

-------
                                                                               TABLE 4-1

                                                                      Oral CarcinogenicHy of DDT
Vehicle Dose

NR 0 ppm
3.0 ppm





Length of
Treatment
llfespan






Length of Species
Experiment
5 generations mice/
BALB/c





Sex

H/F
N/F





Number
Tested
406
683





Effects

Combined tumor Incidence across 5
generations: lung tumors (16. 9X
treated, 1 .2% control), lymphomas
(4.8X treated, 1.05C control) and
leukemlas (12. 4X treated. 2.5X
control) occurred In the mice exposed
to DDT.
Reference

Tarjan and
Kemeny. 1969





no
I
     Gelatin/
     diet
     Gelatin/
     diet
     NR
     NR
     NR
control                       81  weeks        NR                mlce/Xa      H/F      79/87
46.4 mg/kg/day, days 7-28/                                                M/F      18/18
18.2 mg/kg/day (140 ppm),
4-81 weeks
control                       81  weeks        NR                m1ce/Yb      M/F      90/8?
46.4 mg/kg/day. days 7-28/                                                N/F      18/18
18.2 mg/kg/day (140 ppm),
4-81 weeks


0 ppmc                        llfespan        2 generations     mouse/      H/F     113/111
(0.26 mg/kg/day) 2 ppm                                        CF1          H/F     124/105
(1.3 mg/kg/day) 10 ppm                                                    H/F     104/124
(6.5 mg/kg/day) 50 ppm                                                    M/F     127/104
(32.5 mg/kg/day) 250 ppm                                                  M/F     103/90
0 ppm                         112 weeks       NR                mouse/       M/F      47/47
(6.5 mg/kg/day) 50 ppm                                        CF1          H/F      32/30
(13.0 mg/kg/day)100 ppm                                                   H/F      32/32
0 ppm                         110 weeks       NR                mouse/      H/F      45/44
100 ppro                                                       CF1          H/F      30/30
About 30X of the females died during     Innes
treatment.  Hepatomas occurred In        et al.,  1969
11/18 male and 4/18 female mice
exposed to DDT. whereas only 8/79
male and 0/87 female controls had
hepatomas.

About 30X of the females died during     Innes
treatment.  Hepatomas occurred In 7/18   et al..  1969
male and 1/18 female mice exposed to
DDT. whereas only 5/90 male and 1/82
female controls had hepatomas.

The Incidence of hepatomas was slgnlf-   Tomatts
Icantly Increased (p<0.01) In both       et al.,  1972
males and females exposed to 250 ppm
DDT.  When the animals were aged past
60 weeks, the Increased Incidence of
liver tumors was significant (p<0.01)
at all dose levels In males, but not
females.

Liver tumors In mice on diets con-       Walker
talnlng DDT at a dose of 0. 50 or 100    et al..  1972
ppm occurred In 13, 37 and 53X of the
males, and 17. 50 and 76% of the
females, respectively.

Liver tumors In mice on diets con-       Thorpe and
talnlng 0 or 100 ppm DDT occurred In     Walker,  1983
24 and BOX of the males and 23 and 87X
of the females, respectively.  Malig-
nant liver tumors occurred In 4.4 and
30X of the males and 0 and 40X of the
females.

-------
                                                                           fABLE  4-1  (cont.)
CO
i
Vehicle
NR





NR











NR

Dose
0 ppm
(0.26 mg/kg) 2 ppm
(1.5 mg/kg) 10 ppm
(6.S mg/kg) 50 ppm
(32.5 mg/kg) 250 ppm

0 ppm
(0.26 mg/kg/day) 2 ppm
(2.6 mg/kg/day) 20 ppm
(32.5 mg/kg/day) 250 ppm








0 ppm
(32.5 mg/kg/day) 250 ppm
Length of Length of Species Sex
Treatment Experiment
lifetime 6 generations mouse/ H/F
CF1 H/F
H/F
H/F
H/F

2 generations llfespan mouse/ H/F
CF1 H/F
H/F
H/F








15-30 weeks 65, 95 and mouse/ H/F
120 weeks CF1 H/F
Number
Tested
328/340
354/339
362/355
383/328
350/293

107/131
112/136
106/128
106/121








481
713
Effects
Cumulative Incidence of hepatomas
males: 29.5. 50.5, 50.0. 55.9. 86. OX
for 0, 2, 10, 50 and 250 ppm, respec-
tively. Cumulative hepatomas females:
4.7. 3.5. 9.0, 13.1, 65. 5X for 0. 2,
10, 50 and 250 ppm, respectively.
Only liver tumors occurred more fre-
quently In treated as compared with
control animals. Hale mortality
caused by DDT toxic Hy was Increased
only In the group receiving a dose of
250 ppm. In males, those on diets of
0, 2. 20 and 250 ppm of DDT had Inci-
dences of liver tumors combined across
2 generations of 2/107. 3/112, 1/106.
15/106. For females, the corresponding
Incidences were 0/131. 0/136. 1/128 and
71/121.
Incidence of hepatomas In males
treated for 15 weeks or 30 weeks with
Reference
Turusov
et al.. 1973




Terraclnl et
al., 1973a.b










Tomatls
et al., 1974
     NR
0 ppmd
(3.3 mg/kg/day) 22 ppm
(6.6 mg/kg/day) 44 ppm
0 ppm
(13.05 mg/kg/day) 87 ppm
(26.25 mg/kg/day) 175 ppm
78 weeks
                                                             93 weeks
mouse/
B6C3F1
H
H
H
F
F
F
 20
-50
-50
 20
-50
-50
DDT and killed 65. 95 and 120 weeks
after the start of the experiment was
13/60. 25/60. 25/60 and 38/60. 41/60
and 37/60, respectively.  Corresponding
values for controls, were 12/70, 24/83
and 33/98.  When females were treated
for 15 weeks or 30 weeks with DDT and
killed at 65, 95 and 120 weeks after
the start of the experiment, the Inci-
dence of hepatomas was 3/60, 11/60.
5/60 and 4/54. 11/65 and 11/54, respec-
tively.  Corresponding control values
for females were 0/69. 0/72 and 1/90.

Mortality was significantly Increased
In treated females and the Increase
appeared dose-related.  No other toxic
or carcinogenic effects were seen.
                                                                                                       NCI.  1978

-------
TABLE 4-1 (cont.)
Vehicle
Oil

NR





NR


NR


NR





NR

NR


Dose Length of Length of
Treatment Experiment
0 ppm 18 months NR
5 mg/kg/day (100 ppm)
10 mg/kg/day (200 ppm)
20 mg/kg/day (400 ppm)
30 mg/kg/day (600 ppm)
40 mg/kg/day (800 ppm)
0 ppm 2 years NR
• ** rr* •
80 ppm
200 ppm
•.WU |#f«IH


0 ppm lifetime lifetime
(25 mg/kg/day) 500 ppm

15 rag/rat, 5 days/week 1 year 18 months
by gavage (612.24 ppm)

0 ppm 78 weeks 111 weeks
(16.05 mg/kg/day) 321 ppm
(32.1 mg/kg/day) 642 ppm
0 ppm
(10.05 mg/kg/day) 210 ppm
(21.0 mg/kg/day) 420 ppm
0 ppm lifetime lifetime
(6.25 mg/kg/day) 125 ppm
(12.5 mg/kg/day) 250 ppm
(25 mg/kg/day) 500 ppm

0 ppm NR NR
(10 mg/kg/day) 125 ppm
(20 mg/kg/day) 250 ppm
(40 mg/kg/day) 500 ppm

Species
rats/
Osborne-
Hendel
rats





rat/
Wlstar

rats/
Fischer

rat/
Osborne-
Ncndel



rats/MRC
Portion

hamster


Sex
H/F
M
H/F
H/F
H/F
H/F
H/F
H/F
H/F



H/F
H/F

H/F


H
H
H
F
F
F
H/F
H/F
H/F
H/F

H/F
H/F
H/F
H/F

Number
Tested
24/12
12
24/12
24/12
24/12
36/24
30/30
30/30
30/30



35/32
27/28

15/15


20
-50
-50
20
-50
-50
38/38
30/30
30/30
38/38

40/39
30/28
31/28
39/40

Effects
The authors concluded that there was
an Increased Incidence of liver tumor
formation, but did not relate the
effect to dose levels or sex. and did
not provide any statistical analysis.
Treatment began at weaning.
No difference In tumor Incidence
between treated and control groups,
except for bronchogenlc carcinomas
which occurred In 2/60 controls. 8/60
rats fed DDT at 80 ppm and 0/60 rats
fed 200 ppm.
Increased Incidence of liver tumors
were seen In males (9/27. 35%) and
females (15/28, 56X). No liver
tumors were seen In controls.
No liver tumors were seen.


No Increase In tumor Incidence or
signs of toxlclty were noted for DDT.




The Incidence of hepatomas In males
was 1/38, 0/30, 1/30 and 2/38 for the
0. 125, 250 and 500 ppro groups, re-
spectively. Corresponding Incidences
for females were 0/38. 2/30. 4/30 and
7/30.
No liver tumors were seen In hamsters
at any feeding level. There was a
significant trend In total number of
tumor -bearing females: 7.5. 16.6.
25.8 and 28. 2X for 0. 125. 250 and
500 ppm, respectively.
Reference
Fltzhugh and
Nelson. 1947
Delchmann et
al.. 1967;
Radomskl
et al.. 1965


Rossi
et al., 1977

Welsburger
*n«l
ana
Welsburger,
1968
NCI. 1978





Cabral et
al., 1982b

Cabral et
al.. 1982a


-------
                                                                           TABLE  4-1  (cont.)
Vehicle Dose
NR 0 ppm
(BO mg/kg/day) 1000 ppm
Length of Length of Species Sex Number
Treatment Experiment Tested
NR NR hamster M/F 31/42
H/F 35/36
Effects
An Increased Incidence of liver tumors
was not seen. Incidences of adrenal
adenomas were significantly elevated
In females, but not males. Incidence
for males: 0 ppm. 8/31; 1000 ppm.
14/35 and for females: 0 ppm, 2/42;
1000 ppm, 10/36.
Reference
Rossi
et al., 1983
     aCS7BL/6 females  mated with C3H/Anf  males


     bCS7BL/6 females  mated with AKR  males


     cThe fraction of  body weight consumed per  day  In food, called  the food factor,  Is  0.13 for mice and  0.05  for  rats.  Exposures given  In  ppm  of food are

      converted to mg/kg/day by multiplying  the  ppm exposure  level by  the food  factor.


     dfloses  given are  the TWA dose computed  by NCI.
tn
i

-------
authors emphasized  that the  transplacental  and  translactatlonal  exposure  to
DDT that occurred during the experiment may  have  had  an  Important,  but  unquan-
tlfled, effect upon the results.
    Under   the auspices  of  IARC,   Tomatls   et  al.  (1972),  Terradni  et  al.
(1973a,b), Turusov  et al.  (1973)   and  Shabad  et  al.  (1973)  Investigated  DDT
cardnogenldty  1n  mice.  Several  mult1generat1on studies  were conducted  In
which  mice  were exposed  continuously to  DDT,  Including  transplacentally  and
translactatlonally.   Tomatls  et  al.  (1972) found  that  mice  of  both  sexes
exposed to  250  ppm  DDT  had a  significantly  higher  Incidence of  hepatomas.
When  the  mice exposed  to  lower  doses  of  DDT (2-50  ppm)  were allowed  to  age
past  60  weeks,  the  males, but  not  the  females, had  a  significantly  higher
Incidence  of  hepatomas.   In  another  experiment,  Tomatls et al.  (1974)  demon-
strated that  hepatoma formation was  dose-dependent  and  that  exposure  to  DDT
early  1n  life may  result  In tumor  formation  1n  the  aging animal  even after
removal of  the source of  DDT.   Terradni  et al.   (1973a)  found  that  the Inci-
dence  of  hepatomas  was  Increased 1n BALB/c  mice  exposed to  DDT.   In addition,
the  mice  exposed  transplacentally  and translactatlonally  had an  even  higher
Incidence  of liver  tumors than the mice exposed after  weaning only.
    Walker et  al.  (1972)  and  Thorpe and  Walker   (1973) reported an  Increased
Incidence   of  liver  tumors  1n CF1  mice exposed  to   DDT In their  food  for  2
years.  They  divided the  liver  lesions into  two hlstologlcal  types.   Subse-
quent  analysis  by  Reuber (1974,1976) classified  the  lesions as hepatocellular
carcinomas and preneoplastlc  lesions.
    The NCI (1978) bioassay reported  no carcinogenic  effect  from DDT exposure,
although  the  mortality  of  the  female  mice was  significantly Increased  1n  a
dose-related  manner.   The  dose  levels,  however,   were  low in  comparison with
other bloassays.
                                     -16-

-------
    In rats exposed  to 100-800 ppm  DDT  In the diet  for  18 months,  the  dose-
related changes  Included  hypertrophy of  centrolobular hepatic  cells,  hyalinl-
zatlon of the  cytoplasm  and  focal  necrosis (Fltzhugh and Nelson,  1947).   More
than half (111  out  of  192)  of the rats died during the experiment.   Of  the  81
that remained alive at the end of  the  treatment period.  4  had  Hver  carcinomas
and 11 had  preneoplastlc  hepatic  lesions.   No liver pathology  was observed  1n
the control  animals (Fltzhugh and  Nelson,  1947).   Rossi et  al.  (1977) reported
an Increased incidence of Hver tumors in  rats exposed  to  500  ppm DDT 1n their
diets.  Other  studies  1n rats on  the  carclnogenicity  of DDT 1n  doses  ranging
from  210-642  ppm  (NCI,  1978; Weisburger  and Weisburger,  1968;  Deichmann  et
al.,  1967;  Radomski et  al., 1965)  reported  no  Increased  incidence of  liver
tumors.
    None  of the  bioassays   in  hamsters  revealed  an  increased  Incidence  of
tumors In  DDT  exposed animals  (Agthe  et  al., 1970;  Cabral and  Shubik,  1977;
Graillot  et al., 1975),  and Graillot et  al. (1975)  reported  a marked  dose-
related decrease  In  the  incidence  of lymphosarcoma 1n the  DDT  exposed  animals
as compared with controls.
4.2.2.   Inhalation.  Pertinent data regarding the carclnogenicity of  inhaled
DDT could not be located  In  the available literature.
4.3.   OTHER RELEVANT DATA
    No Increase  in  the number of  reverse  mutants  was  caused by  DDT  in Salmo-
nella  typhimurlum  (strains  TA1535,  TA1536, TA1537 and TA1538)  or  Escherichia
coli  (strains  B/r  try, WP2,  WP2  try and  her), regardless  of   the presence  of
rat  liver  microsomes  (Shirasu  et  al.,  1976;  Marshall  et al.,  1976).   DDT
caused no  significant  Increase in recombination  mutants 1n Bacillus subtilis
(Shirasu  et al.,  1976),  1n recessive  lethal mutants  1n  Neurospora  crassa
(Clark, 1974;  Luers, 1953)  or in mutation frequency in  Salmonella  typhimurlum
                                     -17-

-------
(Buselmaier  et  al.,  1972).   Chromosomal  aberrations  have  been  reported  In
cultivated  rat-kangaroo  cells  (Palmer  et  al.,  1972}  and  human  lymphocytes
(Lessa et al., 1976), but not 1n rat cells  (Legator et  al.,  1973) and In mouse
bone marrow  cells  in vivo (Markaryan,  1966).   An  Increase 1n dominant lethal
mutations  was  caused by  DDT  in  Drosophlla  melanogaster  (Clark,  1974),  the
Swiss mouse  (Clark,  1974)  and the rat  (Palmer  et al., 1972),  but  not 1n the
CF1 mouse (Wallace et al.,  1976) or  the  ICR/Ha mouse (Epstein et al., 1972).
4.4.   WEIGHT OF  EVIDENCE
    DDT  has  been associated  with  liver  tumors  in  mice (Innes et  al., 1969;
Tomatis  et al.,   1972;  Terradni   et  al.,  1973a,b)   and  rats   (Rossi  et  al.,
1977), and  lymphomas  and  pulmonary tumors  (Tarjan  and  Kemeny,  1969) in mice.
Based  on  inadequate  evidence for  cardnogenldty  1n  humans  and   sufficient
evidence  of  cardnogenldty   1n animals  1n  spite  of   inadequate  evidence for
cardnogenldty  1n  short-term tests  (I.e., mutagenldty), DDT  1s  most appro-
priately classified following the scheme proposed by  the Carcinogen  Assessment
Group of  the  U.S.  EPA (Federal  Register,  1984)  as a  Group B2 - Probable Human
Carcinogen.
                                     -18-

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                     5.  REGULATORY STANDARDS AND CRITERIA







    The WHO (1971) recommended a maximum  Interim ADI  1n  food  of 0.005 mg/kg/bw



for DDT.   The  ACGIH (1983)  recommended a  TLV-TWA  of 1  mg/m3 and a  TLV-STEL



of 3  mg/m3,  based on  analogy with  Undane,  which was  judged to be  twice  as



toxic  as DDT (ACGIH,  1980).
                                     -19-

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                              6.  RISK ASSESSMENT
6.1.   ACCEPTABLE INTAKE SUBCHRONIC  (AIS)
    DDT  is  known  to  be an  animal  carcinogen and  data  are  sufficient  for
computing a  q*.   Therefore,  H   Is  Inappropriate  to  calculate  an  oral  or
Inhalation AIS for DDT.
6.2.   ACCEPTABLE INTAKE CHRONIC (AIC)
    DDT Is a  chemical  known to be  an animal carcinogen  and  for  which  data are
sufficient for  computing a  q *.  Therefore,  1t 1s Inappropriate  to  calculate
an oral or Inhalation AIC for DDT.
6.3.   CARCINOGENIC POTENCY (q^)
6.3.1.   Oral.   U.S.  EPA (1985) has  developed  a quantitative estimate  of the
carcinogenic potency of  DDT.  The studies  selected for quantitative evaluation
were:   Tarjan  and  Kemeny  (1969),  Turusov  et  al.   (1973),  Terradnl  et  al.
(1973), Thorpe  and Walker  (1973),  Tomatls and  Turusov (1975),  Cabral  et al.
(1982b) and Rossi et al. (1977).
    The data  used for  estimation of  a q * from the  Tarjan  and  Kemeny  (1969)
study  as  shown  In  U.S. EPA  (1985) are presented  In Table  6-1.   Group sizes
were  considered Inadequate  for evaluation in  the F,  and  F~  generations.   A
potency estimate of 7.27  (mg/kg/day)'1  was estimated  based on  the  geometric
mean of the potencies for generations F~-F5 for lung cancers and leukemia.
    The  data  used  for  estimation  of  a  q *  from the  Turusov  et al.  (1973)
study  as  shown  in  U.S. EPA  (1985) are presented  in Table  6-2.   A  geometric
mean   of  the  potencies  across  six   generations   for   liver  tumors  of  0.80
(mg/kg/day)'1 for males and 0.42 (mg/kg/day)'1 for females was estimated.
    The  data  used  for  estimation   of  a  q * from  the Terradnl  et al.  (1973)
study  as  shown  in  U.S. EPA  (1985) are presented  in Table  6-3.   A  geometric
mean  potency   (q,*)  of  0.082  (mg/kg/day)'1  for  liver  tumors  was calculated
across sexes and two generations.

                                      -20-

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                                                     TABLE  6-1


               Incidence of  the  Host Commonly Occurring Malignant  Tumors  In  Each  of  Five  Generations
                                             of  BALB/c Mice  Fed DDTa
I
ro
Incidence by Generation1* (combined
Site/Dose Group
F!
Lung (carcinomas)
Control 0/3 (00.0)
3 ppm DOTC 2/10 (20.0)
Significance11
qi*e
qi*f
f*
0/39 (00.0)
10/35 (28.5)
p=0.001
18.78
17.20
F3
3/51 (5.9)
13/69 (18.8)
p=0.007
9.09
9.95
male and female) (54)
F4
0/144 (00.0)
41/264 (15.5)
p<0.002
7.45
7.16
F5
2/169 (1
50/305 (16
p<0.001
7.37
7.68

• 2)
.4)



-------
                                                TABLE 6-1 (cent.)
    Site/Dose Group
                                        Incidence  by  Generation0  (combined male  and female)  (%)
Leukemia
Control 2/3 (66.6)
3 ppm DDTC 4/10 (40.0)
Significance*1

-------
                                                    TABLE 6-2


                 Incidence of Benign Liver Tumors In Each of Six Generations of CF-1 Mice Fed DDTa
Benlqn Liver Tumor Incidence by Generation (%)**
Sex/Dose
Group
Hales
Control
2 ppmc
10 ppm
50 ppm
250 ppm
Parental
H/60 (24)
26/60 (44)
32/60 (53)
27/60 (45)
46/60 (76)
F!
13/60 (21)
29/60 (48)
28/60 (47)
35/60 (58)
51/60 (85)
F2
20/60 (34)
38/60 (63)
33/60 (55)
41/60 (69)
53/60 (89)
F3
21/60 (35)
30/60 (50)
36/60 (60)
36/60 (60)
53/60 (89)
F4
16/60 (26)
34/60 (57)
24/60 (40)
32/60 (53)
57/60 (95)
F5
23/60 (39)
25/60 (42)
26/60 (44)
28/60 (47)
48/60 (80)
CO
I
,*d
                    0.572
0.873
0.935
0.878
1.096
0.598

-------
                                             TABLE 6-2 (cont.)
Benign Liver Tumor Incidence by Generation (54)b
Sex/Dose
Group
Females
Control
2 ppmc
10 ppm
50 ppm
250 ppm
qi*d
Parental

3/60
3/60
2/60
8/60
37/60
0.372

(5)
(5)
(3)
(13)
(61)

F!

2/60
1/60
8/60
7/60
43/60
0.471


(3)
(2)
(13)
(12)
(71)

F2

1/60
3/60
8/60
8/60
31/60
0.369

(2)
(5)
(13)
(13)
(52)

FS

2/60
5/60
3/60
9/60
40/60
0.434

(3)
(9)
(5)
(15)
(67)

F4

4/60
0/60
5/60
10/60
48/60
0.526

(7)
(0)
(8)
(16)
(80)

F5

5/60 (8)
0/60 (0)
6/60 (10)
7/60 (11)
38/60 (64)
0.370
aSource: U.S. EPA, 1985

bNumber  of  animals with  tumors/number  of  animals examined  (percent).   The  effective  number of  animals
 was given  by Turusov et al. (1973) as 50-60;  60 has been used  for  every group because the  exact  number
 was not given.

cThe human  equivalent doses are  calculated by  multiplying  the  ppm  values  by 0.13  and  then by  the  cube
 root  of  0.030/70 (=0.0753949).  No  adjustment for  time  was  made because  these  were lifetime  tests  and
 CF-1 mice  were  fed  DDT  continuously  during that time.  For  example, human equivalent doses  are:   2 ppm =
 0.0196, 10 ppm = 0.0980, 50 ppm = 0.4900  and 250 ppm = 2.45  mg/kg bw/day.

dThe qi*s  of  the upper-bound   limits  In  units  of (mg/kg bw/day of dietary  exposure)'1 were  calculated
 using the multistage model.

-------
                                  TABLE 6-3

        Incidence  of  Benign  Liver  Tumors  In  BALB/c  Mice  Fed  DOT  During
                         a  2-Generat1on  Experimenta»b
Incidence of Beniqn Liver Tumors by Generation0
Males
Dose Group
0 ppm
Trendd
2 ppm
20 ppm
250 ppm
qi*e
High dose q-|*
Parental + f-\
2/107
p<0
3/112
1/106
15/106
0.074
0.086
(1.9)
.001
(2.7)
(0.9)
(14.2)



Females
Parental F-j
0/62
p<0.
0/63
1/61
28/63
0.080
0.324
(0)
001
(0)
(1.6)
(44.4)


0/69
p<0.
0/73
0/67
43/58
0.094
0.718
(0)
001
(0)
(0)
(74.1)


aSource: U.S. EPA, 1985

bNumber  of  animals   with   tumors/number   of   animals   examined  (percent).
 Malignant tumors were not observed 1n liver.

cThe  numbers  In  the  grups  of  males were  reduced  by  fighting,  so  the  2
 generations of males  were  pooled.   Each high-dose group  shown  is statisti-
 cally  different  from  Us   control  group  (p<0.001).   Other  palrwlse  tests
 were not significant.

dBeneath  the control   incidence  1s  the p value  for positive  trend  in  Inci-
 dence over the dose levels.

eThe  q-|*s were  calculated  using  the  human  equivalent  dose.    The  "high-
 dose  q-j*"   1s  the  result   of  using  only   the  controls  and the high-dose
 groups  1n  the calculations.  The  human  equivalent doses are calculated by
 multiplying the  ppm values by  0.13  and then  by  the cube  root  of  0.030/70
 (=0.0753949).   For example, 250 ppm = 2.45  mg/kg/day for humans.
                                     -25-

-------
    The data  used  for  estimation of  a  q^ from  the  Thorpe and Walker  (1983)
study as  presented 1n  U.S.  EPA  (1985)  are  shown In  Table  6-4.   q^  values
for  the  Incidence of  malignant  liver   tumors  1n  males  and  females  were
calculated as 0.52 (mg/kg/day)'1 and  0.81  (mg/kg/day)'1, respectively.
    The  data  used  for  estimation  of  a  q *  from  the Tomatls  and  Turusov
(1975)  study as presented  In   U.S.  EPA (1985)  are shown  1n  Table 6-5.   q^
values  for  benign  liver  tumors 1n males  and  females were 1.04  (mg/kg/day)'1
and 0.49 (mg/kg/day)'1,  respectively.
    The  data used  for  estimation  of a  q *  from  the  Cabral  et  al.  (1982b)
study  are  shown 1n  Table 6-6.   A q,  of  0.084  (mg/kg/day)'1 was  calculated
for  liver   tumors  1n  female rats.   The  data   used  for  q^*  estimation  from
Rossi  et al.  (1977)   are also shown  1n  Table  6-6.   q * values  for  liver
tumors  1n male and female rats of  0.16 and 0.27  (mg/kg/day)"1,  respectively,
were calculated.
    Table 6-7 presents  a summary  of  the calculated  potency estimates.   Of
these  values,  the  q *  based on Tarjan  and Kemeny  (1969) was  eliminated based
on  the D1xon  statistical  criterion   for  rejecting outliers  (p=0.01)   and  the
additional considerations that  the  study  was  from  an  unaudited  laboratory and
that  the  feed was  contaminated with DOT.  A  geometric average of  the values
from  the  remaining six  studies resulted  1n  a  final  q *  estimate for  DOT of
0.34  (mg/kg/day)'1:   (0.80  x   0.42  x  0.082  x  0.52  x  0.81  x 1.04  x  0.49  x
0.084 x 0.16 x 0.27)1/10 = 0.34.
6.3.2.   Inhalation.  Pertinent  data  regarding  the cardnogenldty of  Inhaled
DDT could not be located 1n the available literature.
                                     -26-

-------
                                   TABLE  6-4

         Incidence  of  Liver  Tumors  (Benign  and  Malignant)  In CF-1  Mice
                       Fed DDT for a Single Generation3
Dose Group             Incidence of Benign             Incidence of Malignant
                          Liver Tumors^                    Liver Tumors'3
Males

Controls                   11/45 (24%)                       2/45 (4.4%)

100 ppm                    23/30 (80%)                       9/30 (30%)

q-|*                        ND                               0.52


Females

Controls                   10/44 (23%)                       0/44  (0%)

100 ppm                    26/30 (87%)                      12/30 (40%)

qi*                        ND                               0.81


aSource: U.S. EPA, 1985

^Benign Hver  tumors  in this study  were  referred to as  "type  a"  and malig-
 nant liver tumors as "type b."

ND = Not determined
                                     -27-

-------
                                                         TABLE 6-5

                Incidence of Benign Liver  Tumors  In  CF-1  Mice  Fed  DOT  for  15  or  30 Weeks  and  then  Sacrificed
                                               at 65,  95 and  120  Weeksa.°.c
ro
CO
i
        Dose Group
                                        Hales  at Meek
                                         Females at Week
                              65
95
120
65
95
120
0 ppmd
250 ppm for
15 weeks6
250 ppm for
30 weekse
qi*f values
all qi*
30 week
12/70 (17)
13/60 (22)
p=0.142
38/60 (63)
p<0.001
0.36
1.38
24/83 (29)
25/60 (42)
p=0.040
41/60 (68)
p<0.001
1.04
1.43
33/98 (34)
25/60 (42)
p-0.080
37/60 (62)
p<0.001
0.84
1.06
0/69 (0)
3/60 (5)
p=0.097
4/54 (7)
p-0.034
0.19
0.19
0/72 (0)
11/60 (14)
p<0.001
11/55 (20)
p<0.001
0.49
0.79
1/90 (1)
5/50 (10)
p=0.034
11/54 (20)
p<0.001
0.35
0.43
        aSource: U.S. EPA, 1985

        DNumber of animals with tumors/number  of animals  examined  (percent).

        C8orae groups were exposed for 15 weeks;  other  groups were exposed for  30  weeks.   All groups were  sacri-
         ficed serially at 30,  65, 95 and  120  weeks.

        dine human  equivalent  dose for  1  ppm for 15 weeks  Is 0.4084 mg/kg/day and  for  30 weeks Is 0.8168  mg/kg/
         day.  The  human  equivalent  doses are calculated  by multiplying the  ppm  values by 0.13  and  then  by  the
         cube root  of  0.030/70  (=0.0753949).   Adjustments  for  time consist  of  multiplying  the  15-week dose by
         15/90 and the  30-week  exposure  by 30/90.

        eBcneath  each  dosed group  Incidence  Is  the p  value  for  comparison  of the Incidence  In  the dose  group
         with that In the  control  group.
             q^*s were calculated based  on  the  human  equivalent  dose  shown  In  footnote  d.  The  term "all  q^*"  Indi-
         cates that  the dosed  groups  and  the control group  were  used  In  the  calculation.   The  "30 week"  row
         contains the results  of using only the 30-week  exposure cancer  data with  the control cancer  data.

-------
                                  TABLE 6-6

             Incidence of Benign Liver Tumors 1n Rats Fed DDTa»b
Dose Group6
0 ppm
Trendr
125 ppm
250 ppm
500 ppm
qi*9
Cabral et
Males
1/38 (0)
NS
0.30 (0)
NS
1/30 (3.3)
NS
2/38 (5.3)
NS
NDn
al.. 1982bc
Females
0/38 (0)
p=0.003
2/30 (6.7)
NS
4/30 (13.3)
p=0.033
7/38 (18.4)
p=0.005
0.084
Rossi et
Males
0/35 (0)
--
—
9/27 (33.3)
p<0.001
0.16
al.. 1977d
Females
0/32 (0)
—
—
15/28 (53.6)
p<0.001
0.27
aSource: U.S. EPA, 1985

bNumber of animals with tumor/number of animals examined (percent).

cThese were Portion (Wlstar derived) rats.

dThese were Wlstar rats.

eThe  human  equivalent doses  are calculated  by multiplying  the ppm  values
 by  0.0085499,  which  1s  0.05 mg/kg/day  (for rats)  multiplied  by  the  cube
 root  of  0.350/70  (=0.0753949).   No  adjustment  for time  was made  because
 rats were fed continuously for a lifetime.

fBeneath  the control  group  Incidence  1s the p value  for  a  positive  trend
 of  Incidences as  the  dose  Increases,  when  the p  values 1s  less  than p=0.05,
 otherwise NS  (not  significant).   Beneath  each dosed group  Incidence  1s  the
 p  value  for the  comparison  of the  Incidence 1n  the  dosed  group  with  Us
 control group when 1t 1s less than p=0.05,  otherwise NS.

9The  q-]*s  were  calculated  using the  human  equivalent  dose.  For  example,
 500 ppm = 4.275 mg/kg/day for humans.

nNot calculated due to lack of statistical  Increase 1n hepatomas.

NS = Not significant; NO = not determined
                                     -29-

-------
                                  TABLE  6-7



              Summary of Quantitative Potency Estimates for DDT*
Species
Mouse
Mouse
Mouse
Mouse
Mouse
Rat
Rat
Tumor Site
lung/leukemia
liver
liver
liver
Hver
liver
liver
q-j* (mg/kg/day) 1
Males Females
7.27 (combined)
0.80 0.42
0.082 (combined)
0.52 0.81
1.04 0.49
0.084
0.16 0.27
Reference
Tarjan and
Kemeny, 1969
Turusov
et al.. 1973
Terraclni
et al., 1973
Thorpe and
Walker, 1983
Tomatls and
Turusov, 1975
Cabral
et al., 1982b
Rossi et al . ,
1977
*Source:  Adapted from U.S.  EPA,  1985
                                     -30-

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                                 7.   REFERENCES

ACGIH  (American  Conference  of  Governmental  Industrial  Hygienlsts).    1980.
Documentation of  the  Threshold  Limit  Values  for Substances  In Workroom  A1r,
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ACGIH  {American  Conference  of  Governmental  Industrial  Hygienlsts).    1983.
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Agthe, C.,  H.  Garcia,  P.  Shublk,  L.  Tomatls and E.  Wenyon.   1970.  Study  of
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Buselmaler,  W.  and G.  Rohrborn  and C. Propping.  1972.   Mutagenltats-Unter-
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Cabral,  J.R.P.   and  P.  Shublk.    1977.   Lack  of  cardnogenlcity of  DDT  1n
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Cabral,  J.R.P.,  R.K.  Hall,  L.  Rossi,   S.A.  Bronczyk  and K.P.  Shublk.   1982a.
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                                     -31-

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Cabral, J.R.P.,  R.K.  Hall, L.  Rossi,  S.A.  Bronczyk  and K.P. Shubik.   1982b.
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                                     -32-

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Deichmann,  W.B., W.E. MacDonald, A.G.  Beasley  and D. CubH.  1971.   Subnormal
reproduction 1n beagle dogs  Induced  by DDT and aldrin.  Ind. Med.  40:  10-20.
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NIOSH, 1978)

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of  chemical mutagens  by the  dominant lethal  assay in  the mouse.   Toxicol.
Appl. Pharmacol.  23: 288-325.   (Cited in  NIOSH, 1978)

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Fltzhugh,  O.G.  and  A.A.  Nelson.    1947.   The  chronic  oral  toxicity of  DDT
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                                     -33-

-------
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                                     -42-

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                                                     APPENDIX

                                               Summary Table for DDT
                      Species
 Experimental
 Dose/Exposure
      Effect
                                                                                             Reference
    Inhalation

      AIS

      AIC

      Carcinogenic
      potency
CO
1    Oral
AIS

AIC

Carcinogenic
potency
                      mice  and
                      rats
combined data
from six studies
                                             ND

                                             ND

                                             ND
Increased Incidence
of liver tumors
ND

ND

0.34
(mg/kg/day)"
U.S. EPA,  1985
    ND '=  Not  derived

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