vvEPA
           United States
           Environmental Protection
           Agency

           Research and Development
           Health Effects
           Laboi ato' •/
           Research Triar.iie Park NC 27711
                                  EPA-600/4-79-077
A One Step
Method for the
Determination of
Carbamate
Pesticides by
Derivatization with
a-Bromo-2,3,4,5,
6-Pentafluorotoluene

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                RESEARCH REPORTING SERIES

Research reports of the Office of Research and Development, U S  Environmental
Protection Agency, have been grouped into nine series  These nine broad cate-
gories were established to facilitate further development and  application of en-
vironmental technology  Elimination of traditional grouping  was  consciously
planned to foster technology transfer and a maximum interface in related fields
The nine series are

      1   Environmental  Health Effects Research
      2   Environmental  Protection Technology
      3   Ecological Research
      4   Environmental  Monitoring
      5   Socioeconomic Environmental Studies
      6   Scientific and Technical Assessment Reports (STAR)
      7   Interagency Energy-Environment Research and  Development
      8   "Special" Reports
      9   Miscellaneous Reports

This report has been assigned to the ENVIRONMENTAL MONITORING series
This series describes research conducted to develop new  or improved methods
and instrumentation for the identification and quantification of environmental
pollutants at the lowest conceivably significant concentrations  It also includes
studies to determine the ambient concentrations of pollutants in the environment
and/or the variance of pollutants as a function of time or meteorological factors
This document is available to the public through the National Technical Informa-
tion Service, Springfield, Virginia  22161

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                                                     EPA-600/4-79-077
                                                  September 1979
A ONE STEP METHOD FOR THE DETERMINATION  OF  CARBAMATE PESTICIDES
  BY DERIVATIZATION WITH o-BROMO-2,3,4,5,6-PENTAFLUOROTOLUENE
                              by

   Merrill D. Jackson, Stephen D. Soileau,  G.  Wayne Sovocool
                   and Richard A. Sachleben
               Environmental Toxicology  Division
              Health Effects Research  Laboratory
         Research Triangle Park, North Carolina   27711
              HEALTH EFFECTS RESEARCH  LABORATORY
              OFFICE OF RESEARCH AND DEVELOPMENT
             U.S. ENVIRONMENTAL PROTECTION  AGENCY
         RESEARCH TRIANGLE PARK, NORTH CAROLINA  27711


                             U.S. Environmental Protection ARency
                             Region 5, Library (PL-12J)
                             77 West Jackson Boulevatd. 12th Floor
                             Chicago, IL 60604-3590

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                               DISCLAIMER
     This report has been reviewed by the Health Effects Research
Laboratory, U.S. Environmental  Protection Agency, and approved for
publication.   Approval does not signify that the contents necessarily
reflect the views and policies  of the U.S.  Environmental Protection
Agency, nor does mention of trade names or commercial products consti-
tute endorsement or recommendation for use.

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                                FOREWORD

     The many benefits of our modern, developing,  industrial  society are
accompanied by certain hazards.   Careful assessment of the relative risk
of existing and new man-made environmental  hazards is necessary for the
establishment of sound regulatory policy.   These regulations  serve to
enhance the quality of our environment in order to promote the public
health and welfare and the productive capacity of our Nation's population.

     The Health Effects Research Laboratory, Research Triangle Park,
conducts a coordinated environmental health research program  in toxicology,
epidemiology, and clinical studies using human volunteer subjects.
These studies address problems in air pollution, non-ionizing radiation,
environmental carcinogenesis and the toxicology of pesticides as well as
other chemical pollutants.  The Laboratory participates in the development
and revision of air quality criteria documents on pollutants  for which
national ambient air quality standards exist or are proposed, provides
the data for registration of new pesticides or proposed suspension of
those already in use, conducts research on hazardous and toxic materials,
and is primarily responsible for providing the health basis for non-
ionizing radiation standards.  Direct support to the regulatory function
of the Agency is provided in the form of expert testimony and preparation
of affidavits as well as expert advice to the Administrator to assure
the adequacy of health care and surveillance of persons having suffered
imminent and substantial endangerment of their health.

     Pursuant to the mission of the laboratory to investigate the effects
of pesticide and toxic substances on human health, this project was
undertaken to investigate an analytical method which would permit the
analysis of many of the carbamate pesticides using the standard Environ-
mental Protection Agency gas chromatographic parameters already set for
the organochlorine pesticides.  The method and analytical parameters for
the carbamate pesticides tested by this method are presented.
                                           F. G. Hueter, Ph.D.
                                                Director
                                   Health Effects Research Laboratory

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                                ABSTRACT







     A procedure was developed for the determination of trace quantities



of a broad range of carbamate pesticides.   The carbamates were hydrolyzed



and derivatized in a single step, using alkali and orbromo-2,3,4,5,6-



pentafluorotoluene (PFBB), and were subsequently analyzed using electron



capture gas chromatography.  This one step derivatization method created



a novel derivative in which one fluorine on the PFB ring was displaced



by an ethoxide ion via aromatic nucleophilic substitution.
                                     IV

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                                CONTENTS



                                                                     Page



DISCLAIMER	ii



FOREWORD	iii



ABSTRACT	iv



LIST OF FIGURES	vi



LIST OF TABLES	v.i



ACKNOWLEDGMENTS 	  vii



SECTIONS



I.    CONCLUSION	1



II.   INTRODUCTION	2



III.  EXPERIMENTAL	4



IV.   DISCUSSION	8



V.    REFERENCES	20



APPENDIX	23

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                             LIST OF FIGURES

No.                                                                  Page

 1.   General Mechanism of Fluorine Displacement by
     Ethoxide Ion	14

 2.   Thiophanate Methyl Derivative	16

 3.   General Derivatization Route of Substituted Phenoxide
     Forming Carbamates	17

 4.   Aldicarb Derivative	19
                             LIST OF TABLES

No.                                                                  Page

 1.  Carbamate Pesticides Evaluated 	  9

 2.  PFBB Reaction Products and Major MS Fragments	13
                                    VI

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                             ACKNOWLEDGMENTS



     The cooperation of Dr.  Lynn Wright in running the CI mass spectra



and Dr.  Dan Zehr for helpful suggestions is gratefully acknowledged.

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                                SECTION I
                               CONCLUSIONS

     A method has been evaluated for the general  analysis of carbamate
pesticides.   This method involves the hydrolysis  of the intact carbamate
pesticide to a substituted phenoxide ion which is then derivatized by
the addition of crbromo-2,3,4,5,6-pentafluorotoluene (PFBB).   The method
provided chromatographiable peaks using the standard EPA gas chromatographic
parameters with 18 of the 23 carbamate pesticides tested.
     Mass spectra were run on selected carbamate  derivatives.   It was
determined from these that those carbamates which would hydrolyze to
form phenolic intermediates formed derivatives with one fluorine displaced
by an ethoxy group in the PFBB characterized by an abundant fragment ion
of m/z 179,  while those carbamates which would not form the phenolic
irtermediates followed no discernible pattern.

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                               SECTION II



                              INTRODUCTION







     Since the introduction of carbaryl  in 1956,  carbamate pesticides



have become widely used in agricultural  pest control  programs.   With the



advent of this wide use, problems of analysis have become evident.



Carbamates generally give poor electron capture response and are too



thermally unstable to be analyzed by conventional gas chromatography.



However, many methods have been developed to overcome these problems.  A



large number of these methods involve some type of chemical derivatization.



Three basic types of derivatization procedures have been developed;



derivatization of the intact carbamate, derivatization of the subsequent



substituted phenol or phenol analog generated through hydrolysis, or



derivatization of the subsequent amine generated through hydrolysis.



     There have been several methods developed for the direct conversion



of carbamates to chromatographiable compounds.  Silylation,  acetylation,



alkylation,    transesterification,   '   and perfluorination  '   of



various carbamates have been accomplished.  Other methods involve hydrolysis


                                                           14
of phenol generating carbamates and subsequent bromination,   chloro-


            15~20                     21               23
acetylation,      thiophosphorylation,   and silylation  '  of the phenolic



intermediates.  Other reagents used for the derivatization of phenolic


                                             22~25
intermediates include dinitrophenyl reagents,      and crbromo-2,3,4,5,6-


                                               26~ 30
pentafluorotoluene (pentafluorobenzyl bromide).       Not all carbamates



form phenols during hydrolysis.  For  those carbamates which hydrolyze to



give amines, methods have  been developed for derivatization of the

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                     31            32                        33
amines.   Bromination,   iodination,   and p-bromobenzoylation   of the



intermediate amines are several of the methods used.  Also, as with the


                                                           34 35
phenolic intermediates previously mentioned, dinitrophenyl,  '   and



pentafluorobenzyl  '    reagents have been used.



     While all of these methods are relatively sensitive by electron



capture detection, no single procedure covered a wide range of carbamate



pesticides.


                                        39
     The EPA Pesticide Analytical Manual   contains general procedures



for the organochlorine and organophosphorus pesticides.  The purpose of

                          i»

this study was to determine if one of the carbamate derivatization



methods could be extended to a wide range of carbamate pesticides at the



residue level and still use the standard gas chromatographic columns and


                                                 39
operating conditions described in the EPA manual.

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                               SECTION III



                              EXPERIMENTAL







Reagents and Solvents



     Alcoholic potassium hydroxide:   Dissolved 1.0 g of solid potassium



hydroxide in 100 ml of 95% ethanol (1% w/v).



     Derivatizing reagent:   Diluted 0.1 ml of a-bromo-2,3,4,5,6-penta-



fluorotoluene (Aldrich Chemicals,  Milwaukee,  WS) in 10 ml of 95% ethanol



(CAUTION:  This reagent is a strong lacrymator).



     Carbamate Standards:   Analytical grade pesticides (Pesticide Repository,



U.S.  Environmental Protection Agency, Research Triangle Park, NC) were



dissolved in either benzene, n-hexane or toluene (1 mg/ml).   Appropriate



dilutions were prepared.



     n-Hexane:  pesticide quality



     Benzene:  pesticide quality



     Toluene:  pesticide quality



     Ethanol:  95%



Equipment



     Gas chromatograph:  Model MT-220 equipped with a nickel   electron



capture detector (Tracer, Inc., Austin, TX).   Glass columns (182 x 0.2



cm i.d.) containing either 1.50% 0V-17/1.95% OV-210 or 4% SE-30/6%



OV-210 on Gas Chrom Q, 80-100 mesh were used.  All columns were pre-



conditioned at 225°C for 24 hours prior to use.  Operating parameters



were:  inlet, 220°C; column oven, 220°C; detector, 350°C; nitrogen



carrier gas,  100 ml/min.

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     Mass spectrometers:   Model  HP-5930A equipped with an HP-5700A gas



chromatograph and a 5933A data system was used in the electron impact



mode (Hewlett Packard, Palo Alto, CA).   Standard 70 eV conditions were



used with a filament emission of 120 pa and an ion source temperature of



190°C.   All samples were scanned from m/z 50 to 550 at m/z 160 per sec.



The gas chromatograph was equipped with a 182 x 0.2 cm i.d.  glass column



packed with 1.50% 0V-17/1.95% OV-210 on Gas Chrom Q, 80-100 mesh.  The



operating parameters were:   helium flow, 40 ml/min; inlet temperature,



200°C;  transfer line temperature, 210°C; and the oven and membrane



separator were temperature programmed from 80°C (2 min) to 230°C at



8°C/min.  Model 3200 quadrupole mass spectrometer equipped with a CI



source, Model 9500 gas chromatograph and Model 6100 data system (Finnigan



Corp.,  Sunnyvale, CA).  The experimental conditions were:  ionization



source temperature 120°C; source pressure 130 Pa; reagent and carrier



gas, (ultra pure) methane, 20 ml/min; separator oven 220°C and transfer



lines 200°C; injection port temperature 225°C.  The 182 x 0.2 cm i.d.



glass GC column contained 1.50% 0V-17/1.95% OV-210 on Gas Chrom Q,



80-100 mesh and was operated at 210°C.



     Tube block heater:  CRC Rubber Co., Cleveland, OH



     Tube rotator:  Kraft Apparatus, Inc., Mineola, NY



     Culture tube:  15 ml, screw capped, teflon lined caps



     Centrifuge tube, 15 ml graduated, glass stoppered



     Teflon tape, 1 cm wide

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Procedure

     Pipet 1 ml of alcoholic potassium hydroxide, 0.1 ml  of derivatizing

reagent and 1 ml of carbamate standard into a 15 ml  culture tube with a

teflon lined screw cap.   Place the culture tube in a pre-heated (95 ±

1°C) tube block heater for two hours.   The length of time and temperature

are critical, for overheating can cause an increase in the formation of
                                     OO
extraneous gas chromatographic peaks.     Remove, allow to cool at room

temperature, and add 5 ml of distilled water and 4 ml of n-hexane to the

culture tube.  Place the culture tube on the tube rotator (60 rpm) for

two minutes and at the end of this time transfer the n-hexane layer to a

15 ml centrifuge tube.  Add an additional 4 ml of n-hexane to the culture

tube, and place in the tube rotator for an additional two minutes.

Combine the n-hexane layer with the previous n-hexane extract.  Bring

the final volume of the centrifuge tube to 10 ml with n-hexane.  The

sample is now ready for further cleanup or gas chromatographic analysis.

Characterization

     The PFB derivative was characterized by electron capture gas chroma-

tography and the derivatization procedure evaluated utilizing the following

criteria:

     1.   G.C.  Retention Time Relative to Aldrin

     2.   Derivatization Linearity.  Linearity was checked over a concen-

          tration range from 0.1 ng/pl to 1,000  ng/ul, if possible, or

          to the limits of detection.  Allowances of ± 15% were tolerated

          in determining the range of derivatization  linearity.

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3.    Linearity of Electron Capture Detector Response.  The response



     linearity of the derivatives were determined on two gas chroma-



     tographic columns.   A concentration of the derivative was



     selected so that a 5 [jl injection would produce a peak height



     of approximately 40-45% full scale deflection (FSD).  Injections



     of 2 to 8 ul» at 1 pi increments, were made, with an allowance



     of ± 10% tolerated in determining linearity.



4.    Minimum Detectable Level.   Minimum detectable level was defined



     to be 10% full scale deflection, provided that this was at



     least twice the background noise.  (This might be a combination



     of gas chromatographic baseline and background from the derivati-



     zation procedure.)  The theoretical concentration for this



     response was calculated and the proper concentration prepared.



5.    Quantity p_f Derivative Required to Give 50% Full Scale Deflection.



     This quantity is not necessarily five times the minimum detectable



     level, since this level was determined using a "clean" baseline.



     A clean baseline was achieved by preparing a derivative at a



     sufficient concentration such that dilution by a factor of 100



     was necessary to bring the derivative peak(s) on scale.  In



     this way, blank interference peaks were negated.



6.    Storage of Derivatized Samples.  One sample was stored at 4°C



     (refrigeration) and a second sample was stored in the dark at



     ambient conditions.  These samples were chromatographed at 0,



     1, 2, 4, and 8 days to determine their stability under storage



     conditions.

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                               SECTION IV



                         RESULTS AND DISCUSSION






Derivatization



     The derivatization procedure used is similar to that of Coburn and


     40
Chau.     The hydrolysis and the derivatization steps have been combined



into one step, to save time and minimize chances for error.



     All of the pesticides which were tested with this method are given



in Table 1.  Of the 23 carbamate pesticides tested,  only five (asulam,



pebulate, propham, trial late and vernolate) did not form a gas chromato-



graphable derivative.



     The characterization data on the derivatives is located in the



appendix.  During the course of the characterization of the carbamate



derivatives, two main difficulties were encountered.  These difficulties



were a decrease in the extent of reaction at low concentrations (i.e.,



> 10 ng/ul) and large background interference caused by the derivatization



reagent  (this interference is discussed in the Mass Spectrometric Identifi-



cation section).  It is not clear why the extent of the reaction decreases



at low concentrations, but it could be caused by competing reactions of



the PFBB with ethoxide ions, or a small loss of derivative in the extrac-



tion procedure, which becomes a large percentage of the derivative at



low concentrations.  With some of the carbamate derivatives, the back-



ground  interference was so great that dilution of the final extract by a



factor of  100 to  quantitate the gas chromatographic peaks was required.
                                   8

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Table 1.  Carbamate Pesticides Evaluated

                        Chemical Name
Common Name

Aldicarb (Temik)


Aminocarb (Matacil)


Asulam (Asulox)


Barban (Carbyne)


Benthiocarb (Bolero)


Carbaryl (Sevin)

Carbofuran (Furadan)


CDEC (Sulfallate)


Chlorpropham (CIPC)


Desmedipham (Betanex)


Formetanate Hydrochloride (Carzol SP)



Kabutilate (Tardex)


Meobal

Methiocarb (Mesurol)
                        2-Methyl-2-(methylthio)propional=
                        dehyde-0-(methylcarbamoyl)oxime

                        4-Dimethylamino-m-tolyl methyl
                        carbamate

                        Methy1(4-amino benzenesulfonyl)
                        carbamate

                        4-Chlorobut-2-ynyl-3-chloro-
                        phenyl carbamate

                        S-4-Chlorobenzyl diethyl-
                        thiocarbamate

                        1-Naphthyl N-methylcarbamate

                        2,3,-Dihydro-2,2-dimethylbenzo=
                        furan-7-yl methylcarbamate

                        2-Chlorallyl diethyldithio-
                        carbamate

                        Isopropyl N-(S-chlorophenyl)
                        carbamate

                        3-Ethoxy carbonyl amino-phenyl
                        phenylcarbamate

                        m-((Dimethyl amino)methylene)
                        amino)phenyl methylcarbamate
                        hydrochloride

                        m-(3,3-Dimethylureido)phenyl
                        tert-butylcarbamate

                        3,4-Dimethylphenyl N-methylcarbamate

                        4-(Methylthio)-3,5-xylyl
                        N-methylcarbamate

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                Table 1.


Common Name

Methomyl (Lannate)


Pebulate (Tillam)

Phenmedipham (Betanal)


Promecarb (Carbamult)


Propham (IPC)

Propoxur (Baygon)


Thi ophanate-Methyl


Trial!ate


Vernolate (Vernam)
Carbamate Pesticides Evaluated
    (Continued)

              Chemical Name
              S-Methyl N-((methylcarbamoyl)
              oxy)thioacetimidate

              S-Propyl butyl ethylthiocarbamate

              3-Methy1oxy-carbony1 ami no-pheny1 N-
              (3'-methylphenyl)carbamate

              3-Isopropy1-5-methy1phenyl
              methylcarbamate

              Isopropy1-N-pheny1carbamate

              o-Isopropoxyphenyl N-methyl-
              carbamate

              1,2-Di(3-methoxycarbony1-2-
              thioureido)benzene

              S-(2,3,3-Trichloroallyl)di=
              i sopropylthi ocarbamate

              S-Propyl-N,N-dipropylthiocarbamate
                                    10

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This interference was especially troublesome when retention times of the



derivatives were short (less than 0.6 relative to aldrin), or when



retention times were near 1.2.   The level of interference can be expected



to increase when samples from environmental media are used instead of



analytical standards.  Hence, the value of this method is limited unless



a suitable cleanup procedure can fie found.  Another limiting factor was



that unless the carbamate can form a substituted phenoxide ion in the



alkaline reaction mixture, the structure of the derivative may be difficult



to determine.  However, this appears to be a fairly sensitive method for



the determination of carbamates which can form a substituted phenoxide



ion in the reaction mixture.



     During the course of this project, it was found that the sensitivity



of the carbamate derivatives fell into two categories.  One group had



minimum detectable levels of approximately 200 pg, while the other group



generally had minimum dectable levels of greater than 5 ng.  This suggested



that there were multiple routes of derivatization.



Mass' Spectrometric Identification



     Carbaryl, meobal, promecarb, thiophanate-methyl, CDEC, aminocarb,



and barban derivatives were analyzed by gas chromatography-mass spectrom-



etry.   The mass spectra of these derivatives along with the spectra of



the reagent blank products are located in the appendix.



     In many of the recorded mass spectra (exceptions--CDEC, aldicarb



and two minor peaks which appear in the spectra of carbaryl and aminocarb),



two ions were found; m/z 207 and m/z 179.  The pentafluorobenzyl (PFB)



ion at m/z 181, found by Coburn et aj_.   to be the significant fragment



in the mass spectrum of the normal unsubstituted PFB derivative of mobam
                                   11

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(4-Benzothienyl-N-methylcarbamate) and which would be expected in all
unsubstituted derivatives, was not generally found.   The exceptions were
the presence of this ion in the mass spectra of the minor (ca 10% based
on peak heights) gas chromatographic peaks in the chromatograms of
carbaryl and aminocarb and the main peak of the aldicarb derivative.
     The m/z 207 fragment, assigned as an ethoxytetrafluorobenzyl ion,
was designated as originating in the mass spectral fragmentation reactions
of an ethoxide displacement product of PFB, with one of the fluorines
being displaced.  A logical ethylene loss of 28 mass units from the m/z
207 fragment yielded the intense m/z 179 fragment, and in certain cases,
a further loss of CHO yielded a m/z 150 fragment, and a further fluorine
loss yielded a m/z 131 fragment.  These fragments were initially recognized
in the gas chromatographic-mass spectrometric analysis of a reagent
blank.  See Table 2 for the structures of the compounds formed in the
reagent blank mixture.
     Considering the alkalinity of the reaction mixture and the electro-
negativity of the fluorines, the likely mechanism for the ethoxide
displacement of the fluorine is aromatic nucleophillic substitution.
This mechanism  involves attack by the nucleophile CpHrO , upon the  PFB
ring to form a  carbanionic intermediate, and subsequent expulsion of the
corresponding fluoride ion from the carbarn'on to yield the final product.
The outline for this mechanism  is found in Figure 1.
     Of the carbamates analyzed, four (carbaryl, promecarb, aminocarb,
and meobal) are capable of forming the substituted phenoxide  ions in the
alkaline reaction mixture.  The mass spectra of the  resulting products
are consistent  with the expected ether derivative.
                                   12

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      Table 2.   PFBB Reaction Products and Major  MS Fragments
Mass
Structure
Mass
Structure
 179
                     207
                                                          OC2H5
 224
                     226
                                                           OC2H5
                                                       Product ill
252
                        C2H5
                   Product II
                                                H5C20
                     278
                                       OC2H5
                                     Product IV
    (The exact position of the OC2H5 group on the ring is not known. The
    ethoxy groups are placed arbitrarily.)
                                    13

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                                 0-Ar
                                F   OC2H5
     Ar=Aromatic ring system
       of carbamate pesticide
The position of the ethoxy group
on the ring is not known
OC2H5
  Figure 1. General mechanism of fluorine
  displacement by ethoxide ion.
                  14

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     The derivative resulting from the reaction of thiophanate-methyl,
although the most sensitive of the carbamate derivatives analyzed, did
not follow this route of derivatization.   The derivative, of mass 414,
was determined to be a di-ethoxytetrafluorobenzyl sulfide (see Figure
2).  It should be noted that thiophanate-methyl cannot form a phenoxide
ion, and hence does not form a derivative consistent with Figure 3.  The
structure of what we call the thiophanate-methyl derivative was confirmed
by independent synthesis through reaction of sodium sulfide and PFBB in
alcoholic KOH.  The gas chromatographic retention times, and mass spectrum
of the synthesized compound were identical to that of the thiophanate-
methyl derivative.  Thiophanate-methyl may be degraded to yield the
sulfide ions for the reaction mixture, or the sulfide may have come from
an impurity in our thiophanate-methyl standard..
     The spectra of aminocarb and carbaryl proved to be particularly
interesting.  Two derivatives were found; the minor (approximately 10%
by relative peak height) derivative formed contained the m/z 181 penta-
fluorobenzyl fragment, while the major (90%) derivative formed contained
the m/z 207 fragment from the ethoxy substituted PFBB.  This could mean
that the replacement of a fluorine by the ethoxy group takes place after
formation of the ether linkage between the substituted phenoxide ion and
pentafluorobenzyl group.  The general scheme of the derivatization route
of substituted phenoxide ion forming carbamates is located in Figure 3.
     The derivatization of aldicarb proved to be another exception of
the scheme outlined in Figure 3.  Although it is impossible for aldicarb
                                   15

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        F      F
                               F     F
C2H50
CH2-S-CH2
2H5
         F     F
                               F      F
      Figure 2. Thiophanate-Methyl Derivative.
      Di-ethoxytetrafluorobenzyl sulfide
                      16

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The position of the ethoxy group
on the ring is not known
  Figure 3. General derivatization route of
  substituted phenoxide forming carbamates.
                    17

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to form a substituted phenoxide ion,  aldicarb cleaved at the C-0 ester
linkage and formed the normal  PFB type derivative (unsubstituted by an
ethoxide ion).   The structure  of the  aldicarb PFB derivative is given in
Figure 4.
     Certain carbamates wnich  had the ability to form substituted phenoxide
ions did not form derivatives  which were very sensitive to gas chromatog-
raphy (i.e. karbutilate, desmedipham).  Possible reasons for this were a
very slow rate of formation or rapid  destruction of substituted phenoxide
ions, attack of substituent groups on the phenolic ring by PFBB, resulting
in derivatives with prohibitively long retention times, or competing
reactions of the carbamate with ethoxide ions.
     The mass spectra of barban derivative seems to support some of
these hypotheses.  Several compounds  were created in the derivatization
reaction.  Of these, two were found to be ethoxy replacement products of
barban and one was found to be the m/z 207 ethoxy PFB addition derivative
of 3-chloroaniline (which was formed during hydrolysis).
     The structure of the CDEC derivatives proved to be the most difficult
to determine.  Three peaks were found in the total ion chromatogram, the
largest  of which was determined to be underivatized CDEC.  Structures
(see Appendix) have been proposed which seem to fit the mass spectra of
the remaining two peaks.
                                   18

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       CH3

        I
CH,S — C — C = I
  3     I    I
       CH3  H
                       F      F
           — O — CH2
                       F     F
Figure 4. Aldicarb derivative.
                19

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                                SECTION V
                               REFERENCES

1.    Fishbein, L. , and Zielinski, W. L. Jr., J. Chromatog.,  20,  9,  1965.
2.    Bache, C. A., and Lisk, D. J., J. Gas Chromatog., 6,  301,  1968.
3.    Khalifa, S., and Mumma, R. 0., J. Agr. Food Chem., 20,  632  (1972).
4.    Seiber, J. N. , J. Agr. Food Chem., 20, 443, 1972.
5.    Butler, L. I., and McDonough,  L. M., J. Agr.  Food Chem.,  16,  403,
     1968.
6.    Sullivan, L. J., Eldridge, J.  M., and Knaak,  J.  B., J.  Agr.  Food
     Chem., 15, 927, 1967.
7.    Lawrence, J. F. , and  Laver, G. W., J. Agr. Food  Chem.,  23,  1106,
     1975.
8.    Lawrence, J. F., JAOAC, 59, 1061, 1976.
9.    Greenhalgh, R., and Kovacicova, J., J. Agr. Food Chem., 22, 325,
     1975.
10.  Van  Middelem,  C. H.,  Moye, H.  A., and Janes,  M.  J., J.  Agr. Food
     Chem., 19,  459, 1971.
11.  Moye,  H.  A., J. Agr.  Food Chem.,  19, 452,  1971.
12.  Walker, G., Winterlin, W., Fouda, H., and  Seiber,  J., J.  Agr.  Food
     Chem., 22,  944, 1974.
13.  Lau,  S.  C. , and Marxmiller,  R.  L., J. Agr.  Food  Chem.,  18, 413,
     1970.
                                     20

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14.   Rails, J.  W.,  and Cortes, A., J. Gas Chromatog.,  2,  132,  1964.



15.   Miller, C. W., Shafik, M. T., and Biros, J. J., Bull  Environ.



     Tontam. Toxicol., 8, 339, 1972.



16.   Butler, L.  I., and McDonough, L. M., JAOAC, 53, 495,  1970.



17.   Stanley, C. W., Thornton, J. S., and Katague,  D.  B.,  J.  Agr.  Food



     Chem., 20,  1265, 1972.



18.   Argauer, R. J., J. Agr.  Food Chem., 17, 888,  1969.



19.   Stanley, C. W., and Thornton, J. S., J. Agr.  Food Chem.,  20,  1269,



     1972.



20.   Butler, L.  I., and McDonough, L. M., JAOAC, 54, 1357,  1971.



21.   Bowman, M.  C.  , and Beroza,  M.   JAOAC,  50,  926,  1967.



22.   Caro, J. H., Glotfelty,  D.  E.,  Freeman, H.  P.,  and Taylor,  A.  W.,



     JAOAC, 56,  1319, 1973.



23.   Cohen, I.  C., Norcup,  J., Ruzicka,  H.  A.,  and Wheals,  B.  B.,  J.



     Chromatog., 49, 215, 1970.



24.   Holden, E.  R., JAOAC,  56, 713,  1973.



25.   Holden, E.  R., JAOAC,  58, 526,  1975.



26.   Seiber, J.  N., Crosby, D. G., Fouda, H.,  and  Soderquist,  C.  J.,  J.



     Chromatog., 73, 89, 1972.



27.   Kawahara,  F.  K., Anal. Chem., 40,  1009, 1968.



28.   Johnson,  L. G., JAOAC, 56,  1503, 1973.



29.   Kawahara,  F.  K., Environ. Sci.  Techno!.,  5,  235,  1971.



30.   Coburn, J.  A., Ripley, B. D., and  Chau, A.S.Y., JAOAC,  59,  188,



     1976.
                                     21

-------
31.   Gutenmann, W. H., Lisk, D. J., J. Gas Chromatog., 4, 424,  1966.
32.   Baunok, I., and Geissbuehler, H., Bull. Environ. Contain. Toxicol.,
     3, 7, 1968.
33.   Tilden, R. L., and Van Middelem, C. H., J. Agr.  Food Chem.,  18,
     154, 1970.
34.   Holden, E. R., Jones, W. M.,  and Beroza, M., J.  Agr. Food  Chem.,
     17, 56, 1969.
35.   Cohen, I. C., and Wheals, B.  B., J. Chromatog.,  43, 233, 1969.
36.   Moffat, A. C., and Hornig, E. C., Anal. Letters, 3, 205, 1970.
37.   Hartvig, P., and Vessman, J., Anal. Letters, 7,  223, 1974.
38.   Agemian, H., and Chau, A.S.Y., Analyst, 101, 733, 1976.
39.   Thompson, J. F., Analysis of  Pesticide Residues  in Human and
     Environmental Samples, U.S.  Environmental  Protection Agency,
     Research Triangle Park, NC,  1977.
40.   Coburn, J. A. and Chau, A.S.Y.,  Environm.  Letters, 10,  225,  1975.
                                     22

-------
                                APPENDIX







     For each carbamate pesticide,  the following information is given:



     1.    Gas chromatographic retention time (aldrin = 1)



     2.    Derivatization Linearity



     3.    Linearity of electron capture detector response



     4.    Minimum Detectable Level



     5.    Quantity of derivative required to give 50% full scale deflection



     6.    Storage of derivatized samples



     7.    Mass spectra and comments as applicable







                                                               Page



Aldicarb	25



Aminocarb	29



Barban	34



Benthicarb	40



Carbaryl	43



Carbofuran	48



CDEC	50



Chloropropham 	 56



Desmedipham	59



Formetanate Hydrochloride 	 62



Karbutilate	65



Meobal	68



Methiocarb	72
                                    23

-------
                                                               Page
Methomyl	75
Phenmedipham	78
Promecarb	81
Propoxur	85
Thiophanate-methyl	88
Reagent blank (mass spectra)	92
                                     24

-------
                                ALDICARB








DERIVATIZATION LINEARITY



Linear from 1 to 100 (jg



AMOUNT NEEDED TO PRODUCE 10% FSD



          OV-17/OV-21Q                       SE-3Q/OV-210



             0.080 ng                           0.040 ng



AMOUNT NEEDED TO PRODUCE 50% FSD



          OV-17/OV-210                       SE-30/OV-210



             0.080 ng                           0.070 ng



RELATIVE RETENTION TIME (ALDRIN = 1.00)



          OV-17/OV-210                       SE-30/OV-210



             0.56                               0.60



COMMENTS



Must be diluted 100 fold due to background interference





DECAY



Stable under test conditions
                                    25

-------
    12.0
    10.0
E
u

I-'
I
1    6.0
UJ

Q.
     2.0
0    .010
                                                       .070
                      .030          .050




                    AMOUNT INJECTED, ng




Column Linearity Check of Aldicarb Derivative on OV-17/OV-210.
                                  26

-------
    14,0
    12.0
    10.0
E
o

h-"
I
LU
CL
8.0
     6.0
     4.0
     2.0
      0
        0     .010           .030           .050           .070



                             AMOUNT INJECTED, ng



       Column Linearity Check of Aldicarb Derivative on SE-30/OV-210.
                                   27

-------
 MO     CO  E
X     I     X  (o
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      CO
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                                                28

-------
                                AMINOCARB








DERIVATIZATION LINEARITY



Linear from 1 to 100 jjg



AMOUNT NEEDED TO PRODUCE 10% FSD



          OV-17/OV-210                       SE-30/OV-210



             1.6 ng                             0.49 ng



AMOUNT NEEDED TO PRODUCE 50% FSD



          OV-17/OV-210                       SE-30/OV-210



             2.7 ng                             2.6 ng



RELATIVE RETENTION TIME (ALDRIN = 1.00)



          OV-17/OV-210                       SE-30/OV-210



             2.0                                1.9



COMMENTS



The standard is very light sensitive.  Must handle with care.





DECAY



Stable under test conditions.
                                    29

-------
       01234



                        AMOUNT INJECTED, ng





Column Linearity Check of Aminocarb Derivative on OV—17/OV—210.
                               30

-------
      01            234



                       AMOUNT INJECTED, ng





Column Linearity Check of Aminocarb Derivative on SE— 30/OV—210.
                               31

-------
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                                                  32

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                                                      33

-------
                                 BARBAN

DERIVATIZATION LINEARITY
Linear from 100 to 1000 \iq
AMOUNT NEEDED TO PRODUCE 10% FSD
          OV-17/OV-210
             20 ng
AMOUNT NEEDED TO PRODUCE 50% FSD
          OV-17/OV-210
             34 ng
RELATIVE RETENTION TIME (ALDRIN = 1.00)
          OV-17/OV-210
             2.0
COMMENTS
None.
DECAY
Stable under test conditions.
SE-30/OV-210
   33 ng
SE-30/OV-210
   100 ng
SE-30/OV-210
   3.0
                                     34

-------
       0    33   67   100   133  167  200   233   267   300




                     AMOUNT INJECTED, ng




Column Linearity Check of Barban Derivative on OV—17/OV—210.
                               35

-------
   0     33    67   100  133   167   200   233   267  300




                 AMOUNT INJECTED, ng





Column Linearity Check of Barban Derivative on SE—30/OV—210.
                           36

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                                                37

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-------
                               BENTHIOCARB







DERIVATIZATION LINEARITY



Linear from 10 to 1000 ug



AMOUNT NEEDED TO PRODUCE 10% FSD



          OV-17/OV-210                       SE-30/OV-210



             0.65 ng                            0.48 ng



AMOUNT NEEDED TO PRODUCE 50% FSD



          OV-17/OV-210                       SE-30/OV-210



             1.8 ng                             2.0 ng



RELATIVE RETENTION TIME (ALDRIN = 1.00)



          OV-17/OV-210                       SE-30/OV-210



             0.91                               1.00



COMMENTS



Must be diluted 100 fold due to background interference.





DECAY



Stable under test conditions.
                                    40

-------
    14


    13



    12


    11


    10


     9



o    8

I
LU
Q.
     6


     5


     4


     3



     2



     1


     0
                0.25        0.5        0.75        1.0        1.25        1.5        1.75       2.0


                                        AMOUNT INJECTED, ng


                Column Linearity Check of Benthiocarb Derivative on OV—17/OV—210.
                                                 41

-------
    16


    15


    14


    13



    12


    11


    10


     9
O    8
ui
X
     6


     5


     4


     3



     2



     1


     0
                0.25        0.5       0.75        1.0        1.25


                                       AMOUNT INJECTED, ng
1.5
1.75
2.0
                 Column Linearity Check of Benthiocarb Derivative on SE—30/OV—210.
                                                 42

-------
                                CARBARYL
DERIVATIZATION LINEARITY



Linear from 1 to 1000 (jg



AMOUNT NEEDED TO PRODUCE 10% FSD



          OV-17/OV-21Q                       SE-30/OV-210



             0.20 ng                            0.18 ng



AMOUNT NEEDED TO PRODUCE 50% FSD



          OV-17/OV-210                       SE-30/OV-21Q



             1.0 ng                             0.89 ng



RELATIVE RETENTION TIME (ALDRIN = 1.00)



          OV-17/OV-210                       SE-30/OV-210



             4.7                                3.6



COMMENTS



None.






DECAY



Stable under test conditions.
                                    43

-------
0.2
0.6
                   0.3        0.4       0.5




                     AMOUNT INJECTED, ng





Column Linearity Check of Carbaryl Derivative on OV-17/OV-210.
0.7
0.8
                    44

-------
   10
u
LLJ
               0.1        0.2
0.6        0.7        0.8
                  0.3        0.4        0.5




                       AMOUNT INJECTED, ng





Column Linearity Check of Carbaryl Derivative on SE—30/OV—210.
                                               45

-------
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                                               47

-------
                               CARBOFURAN



DERIVATIZATION LINEARITY

Linear from 2 to 1000 ug

AMOUNT NEEDED TO PRODUCE 10% FSD

          OV-17/OV-210

             0.70 ng

AMOUNT NEEDED TO PRODUCE 50% FSD

          OV-17/OV-210

             3.1 ng

RELATIVE RETENTION TIME (ALDRIN = l.QO)

          OV-17/OV-210
             2.1
COMMENTS
SE-30/OV-210

See comments
SE-30/OV-210
SE-30/OV-210
Must be diluted 100 fold due to background interference.  Characteri-
zation was not attempted on the SE-30/OV-210 column due to high
background interference.
DECAY

Stable under test conditions.
                                    48

-------
     0      0.5   1.0   1.5   2.0    2.5   3.0   3.5    4.0   4.5




                    AMOUNT INJECTED, ng





Column Linearity Check of Carbofuran Derivative on OV—17/OV—210.
                            49

-------
                                  CDEC



DERIVATIZATION LINEARITY

Linear from 0.1 to 1000 |jg

AMOUNT NEEDED TO PRODUCE 10% FSD

          OV-17/OV-210

             0.024 ng

AMOUNT NEEDED TO PRODUCE 50% FSD

          OV-17/OV-210

             0.15 ng

RELATIVE RETENTION TIME (ALDRIN = 1.00)

          OV-17/OV-210
             0.64
COMMENTS
SE-30/OV-210

   0.024 ng
SE-30/OV-210

   0.15 ng
SE-30/OV-210

   0.62
The derivative was difficult to quantitate due to the variability of
length of derivatization time.  This made decay studies impossible and
the error was greatly increased in the other studies.
DECAY
Not applicable.
                                    50

-------
0.025
0.05
0.15
                  0.075       0.1      0.125




                    AMOUNT INJECTED, ng





Column Linearity Check of CDEC Derivative on OV-17/OV-210.
0.175
0.2
                               51

-------
0.025
0.05
0.075       0.1       0.125




    AMOUNT INJECTED, ng
0.15
0.175
    Column Linearity Check of CDEC Derivative on SE—30/OV—210.
                                52

-------
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                              CHLOROPROPHAM

DERIVATIZATION LINEARITY
Linear from 10 to 1000 |jg
AMOUNT NEEDED TO PRODUCE 10% FSD
          OV-17/OV-210
             0.72 ng
AMOUNT NEEDED TO PRODUCE 50% FSD
          OV-17/OV-210
             3.1 ng
RELATIVE RETENTION TIME (ALDRIN = 1.00)
          OV-17/OV-210
          0.39*, 2.9
COMMENTS
SE-30/OV-210
   0.72 ng
SE-30/OV-210
   3.0 ng
SE-30/OV-210
   0.40*, 3.0
Must be diluted 100 fold due to background interference.

DECAY
Stable under test conditions.
*Major peak
                                    56

-------
    17

    16


    15

    14


    13

    12

    11
£   10
u
LU
I
     0      0.5   1.0   1.5   2.0    2.5   3.0   3.5   4.0  4.5

                    AMOUNT INJECTED, ng

Column Linearity Check of Chlorpropham Derivative on OV—17/OV—210.
                              57

-------
    12
    11
    10
u
2
Hi

X


<    6
LLJ
O_
                                  1      T
       0     0.5     1.0     1.5     2.0     2.5    3.0    3.5     4.0    4.5



                            AMOUNT INJECTED, ng




    Column Linearity Check of Chlorpropham Derivative on SE—30/OV—210.
                                     58

-------
                               DESMEDIPHAM
DERIVATIZATION LINEARITY



Linear from 100 to 1000 pg



AMOUNT NEEDED TO PRODUCE 10% FSD



          OV-17/OV-210                       SE-30/OV-210



             6. 3 ng                             8.4 ng



AMOUNT NEEDED TO PRODUCE 50% FSD



          OV-17/OV-210                       SE-30/OV-210



             32 ng                              42 ng



RELATIVE RETENTION TIME (ALDRIN = 1.00)



          OV-17/OV-210                       SE-30/OV-210



             2.8                                1.8



COMMENTS



None






DECAY



Stable under test conditions.
                                    59

-------
    12


    11


    10


     9
CM

 §   7
in
 LU
 Q.
     4


     3



     2



     1


     0
                5.6       11.1       16.7        22.2       27.8       33.3       38.9       44.4


                                        AMOUNT INJECTED, ng


                   Column Linearity Check of Desmedipham Derivative on OV—17/OV—210.
                                               60

-------
    15




    14




    13





    12




    11




    10
I    9






I    8
LLJ

X
HI

Q.
7





6




5




4




3





2





1




0
                5.6        11.1      16.7       22.2       27.8       33.3       38.9       44.4



                                       AMOUNT INJECTED, ng




                   Column Linearity Check of Desmedipham Derivative on SE—30/OV—210.
                                               61

-------
                            FORMETANATE, HCL







DERIVATIZATION LINEARITY



Linear from 100 to 1000 pg



AMOUNT NEEDED TO PRODUCE 10% FSD



          OV-17/OV-21Q



             4.7 ng



AMOUNT NEEDED TO PRODUCE 50% FSD



          OV-17/OV-210



             23 ng



RELATIVE RETENTION TIME (ALDRIN = 1.00)



          OV-17/OV-210
             1.7
COMMENTS



None
DECAY



Stable under test conditions.
SE-3Q/OV-210



   4.1 ng
$E-30/OV-210



   20 ng
SE-30/OV-210



   2.2
                                    62

-------
                   24
28
                     12        16        20




                        AMOUNT INJECTED, ng





Column Linearity Check of Formetanate-HCI Derivative on OV—17/OV—210.
32
63

-------
    2.5        5.0        7.5        10.0      12.5       15.0       17.5




                            AMOUNT INJECTED, ng





Column Linearity Check of Formetanate-HCI Derivative on SE-30/OV-210.
20.0
                                    64

-------
                               KARBUTILATE
DERIVATIZATION LINEARITY



Linear from 100 to 1000 pg



AMOUNT NEEDED TO PRODUCE 10% FSD



          OV-17/OV-210                       SE-30/OV-210



             9.7 ng                             9.9 ng



AMOUNT NEEDED TO PRODUCE 50% FSD



          OV-17/OV-210                       SE-30/OV-210



             49 ng ,i                            49 ng



RELATIVE RETENTION TIME (ALDRIN = l.OQ)



          OV-17/OV-210                       SE-30/OV-210



             2.5                                2.1



COMMENTS



None





DECAY



Stable under test conditions.
                                    65

-------
10
20
70
              30        40        50        60




                     AMOUNT INJECTED, ng




Column Linearity Check of Karbutilate Derivative on OV-17/OV-210.
80
                             66

-------
    24


    22


    20


    18


    16


i   14
H
I
2   12
LLJ
LU
Q.
     6


     4


     2


     0
                10        20        30         40         50         60        70


                                         AMOUNT INJECTED, ng


                  Column Linearity Check of Karbutilate Derivative on  SE-30/OV-210.
80
                                               67

-------
                                 MEOBAL
DERIVATIZATION LINEARITY

Linear from 10 to 1000 pg

AMOUNT NEEDED TO PRODUCE 10% FSD

          OV-17/OV-21Q                       SE-30/OV-210

             0.091 ng                           0.096 ng

AMOUNT NEEDED TO PRODUCE 50% FSD

          OV-17/OV-210                       SE-30/OV-210

             0.46 ng                            0.48 ng

RELATIVE RETENTION TIME (ALDRIN = 1.00)

          OV-17/OV-210                       SE-30/OV-210

             1.2                              1.0, 1.2*

COMMENTS

Confirmation of derivatization linearity below 10 |jg was impossible
because of background interference.


DECAY

Stable under test conditions.

*Major peak
                                    68

-------
0.07       0.13      0.20       0.27       0.33        0.40      0.47




                       AMOUNT INJECTED, ng





  Column Linearity Check of Meobal Derivative on OV-17/OV-210.
0.53
                                69

-------
u
I
UJ
I
<
a.
15

14

13

12

11

10

 9

 8

 7

 6

 5

 4

 3

 2

  1

  0
                0.07       0.13       0.20        0.27       0.33       0.40        0.47
                                       AMOUNT INJECTED, ng

                   Column Linearity Check of Meobal Derivative on SE—30/OV—210.
                                                                                   0.53
                                               70

-------
71

-------
                               METHIOCARB







DERIVATIZATION LINEARITY



Linear from 1 to 1000 pg



AMOUNT NEEDED TO PRODUCE 10% FSD



          OV-17/OV-210                       SE-30/OV-210



             0.35 ng    »'                       0.30 ng



AMOUNT NEEDED TO PRODUCE 50% FSD



          OV-17/OV-210                       SE-30/OV-210



             1.8 ng                             1.5 ng



RELATIVE RETENTION TIME (ALDRIN = 1.00)



          OV-17/OV-210                       SE-30/OV-210



             3.7                                3.1



COMMENTS



None.
                              «




DECAY



Stable unaer test conditions.
                                     72

-------
   10

LU
CC.
LLJ
a.   4
0        0.25        0.50       0.75        1.0       1.25        1.50       1.75


                                   AMOUNT INJECTED, ng



           Column Linearity Check of Methiocarb Derivative on OV-17/OV-210.
                                                                                         2.0
                                                73

-------
0.25       0.50
0.75        1.0       1.25




 AMOUNT INJECTED, ng
1.50       1.75
 Column Linearity Check of Methiocarb Derivative on SE—30/OV— 210.
                                74

-------
                                METHOMYL








DERIVATIZATION LINEARITY



Linear from 1 to 100 pg



AMOUNT NEEDED TO PRODUCE 10% FSD



          OV-17/OV-210                       SE-30/OV-210



             0.031 ng                           0.026 ng



AMOUNT NEEDED TO PRODUCE 50% FSD



          OV-17/QV-210                       SE-30/OV-210



             0.16 ng                            0.13 ng



RELATIVE RETENTION TIME (ALDRIN = 1.00)



          OV-17/OV-210                       SE-30/OV-210



         0.37, 0.71, 1.3*                   0.25, 0.40, 1.5*



COMMENTS



Measurements were made on the third peak.





DECAY



Stable under test conditions.



*Major peak
                                    75

-------
0.025       0.05      0.075       0.1       0.125      0.15      0.175       0.2




                         AMOUNT INJECTED, ng





  Column Linearity Check of Methomyl Derivative on OV—17/OV—210.
                                 76

-------
0.025
0.15      0.175
        0.05      0.075        0.1       0.125




                    AMOUNT INJECTED, ng




Column Linearity Check of Methomyl Derivative on SE—30/OV—210.
0.2
                                77

-------
                              PHENMEDIPHAM







DERIVATIZATION LINEARITY



Linear from 100 to 1000 ug



AMOUNT NEEDED TO PRODUCE 10% FSD



          OV-17/OV-210                       SE-30/OV-210



             18 ng                              14 ng



AMOUNT NEEDED TO PRODUCE 50% FSD



          OV-17/OV-210                       SE-30/OV-210



             88 ng                              68 ng



RELATIVE RETENTION TIME (ALDRIN = 1.00)



          OV-17/OV-210                       SE-30/OV-210



         1.8,2.3*, 2.8                      1.5, 1.6*, 1.8



COMMENTS



Measurements were made of the second peak.





DECAY



Stable under test conditions.



*Major peak
                                    78

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u


SE
o

LLJ
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12




11




10




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 7




 6




 5




 4




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 0
            10         20        30        40        50        60       70        80




                                  AMOUNT INJECTED, ng





            Column Linearity Check of Phenmedipham Derivative on OV—17/OV—210.
                                          79

-------
10       20        30        40        50        60       70       80




                     AMOUNT INJECTED, ng





Column Linearity Check of Phenmedipham Derivative on SE—30/OV—210.
                             80

-------
                                PROMECARB

DERIVATIZATION LINEARITY
Linear from 10 to 1000 pg
AMOUNT NEEDED TO PRODUCE 10% FSD
          OV-17/OV-210
             0.14 ng
AMOUNT NEEDED TO PRODUCE 50% FSD
          OV-17/OV-210
             0.68 ng
RELATIVE RETENTION TIME (ALDRIN = 1.00)
          OV-17/OV-210
             1.4
COMMENTS
SE-30/OV-210
   0.14 ng
SE-30/OV-210
   0.70 ng
SE-30/OV-210
   1.4
Confirmation of derivatization linearity below 10 ug was impossible
because of background interference.
DECAY
Stable under test conditions.
                                    81

-------
16




15




14





13





12




11





10





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 8





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 6





 5




 4





 3





 2





  1




  0
            0.1         0.2        0.3        0.4        0.5        0.6        0.7        0.8




                                   AMOUNT INJECTED, ng





              Column Linearity Check of Promecarb Derivative on OV—17/OV—210.
                                           82

-------
   15




   14




   13





   12




   11




   10
E   9
u
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    4




    3





    2





    1




    0
               0.1         0.2        0.3        0.4        0.5         0.6        0.7       0.8



                                      AMOUNT INJECTED,ng





               Column Linearity Check of Promecarb Derivative on SE—30/OV—210.
                                              83

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                                PROPOXUR







DERIVATIZATION LINEARITY



Linear from 10 to 1000 |jg



AMOUNT NEEDED TO PRODUCE 10% FSD



          QV-17/OV-210                       SE-3Q/QV-210



             0.080 ng                           0.081 ng



AMOUNT NEEDED TO PRODUCE 50% FSD



          OV-17/OV-21Q                       SE-30/OV-210



             0.24 ng                            0.24 ng



RELATIVE RETENTION TIME (ALDRIN = 1.00)



          OV-17/OV-210                       SE-30/OV-210



             1.2                                1.2



COMMENTS



Must be diluted 100 fold due to background interference.





DECAY



Stable under test conditions.
                                    85

-------
        0    .04    .08   .12   .16   .20   .24   .28   .32   .36




                        AMOUNT INJECTED, ng





Column Linearity Check of Propoxur Derivative on OV—17/OV—210.
                                86

-------
  LLJ
  Q.
      16


      15


      14


      13


      12


      11


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7



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5


4


3


2


1


0
                    I
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        0    .04    .08  .12   .16   .20    .24   .28   .32  .36

                        AMOUNT INJECTED, ng


Column Linearity Check of Propoxur Derivative on SE—30/OV—210.
                                 87

-------
                           THIOPHANATE METHYL

DERIVATIZATION LINEARITY
Linear from 10 to 100 pg
AMOUNT NEEDED TO PRODUCE 10% FSD
          OV-17/OV-210
             0.0087 ng
AMOUNT NEEDED TO PRODUCE 50% FSD
          OV-17/OV-21Q
             0.044 ng
RELATIVE RETENTION TIME (ALDRIN = 1.00)
          OV-17/OV-210
             3.0
COMMENTS
SE-30/OV-210
   0.012 ng
SE-30/OV-210
   0.057 ng
SE-30/OV-210
   3.3
Confirmation of derivatization linearity below 10 ug was impossible
because of blank peak interference.
DECAY
Stable under test conditions.
                                    88

-------
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     6


     4


     2


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                0.01
                      0.02
0.06
0.07
                    0.03        0.04       0.05


                        AMOUNT INJECTED, ng


Column Linearity Check of Thiophanate Methyl  Derivative on OV—17/OV—210.
0.08
                                                89

-------
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               0.01       0.02       0.03       0.04      0.05       0.06       0.07      0.08



                                         AMOUNT INJECTED, ng




           Column Linearity Check of Thiophanate Methyl Derivative on  SE—30/OV—210.
                                               90

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                                   TECHNICAL REPORT DATA
                            (Please read Instructions on the reverse before completing)
  REPORT NO.
    EPA-600/4-79-077
 . TITLE AND SUBTITLE
                             2.
                                                           3. RECIPIENT'S ACCESSIOP+NO
    A  One Step Method for  the  Determination of Carbamate
    Pesticides by Derivatization  with a-Bromo-2,3,4,5,6-
    Pentafluorotoluene
             5. REPORT DATE
                 September 1979
             6. PERFORMING ORGANIZATION CODE
  AUTHOFUS)
    Merrill  D.  Jackson, Stephen  D.  Soileau, G. Wayne
    Sovocool  and Richard A. Sachleben
                                                           8. PERFORMING ORGANIZATION REPORT NO.
9 PERFORMING ORGANIZATION NAME AND ADDRESS
    Analytical  Chemistry Branch
    Environmental  Toxicology Division
    Health Effects Research Laboratory
    Research  Triangle Park. NC   27711
                                                           10. PROGRAM ELEMENT NO.
                1EA615
              11. CONTRACT/GRANT NO.
                N/A
12 SPONSORING AGENCY NAME AND ADDRESS
    Health  Effects  Research Laboratory
    Office  of Research and Development
    U. S. Environmental Protection  Agency
    Research  Triangle Park, NC   27711
                                                            13. TYPE OF REPORT AND PERIOD COVERED
RTP, NC
Final
              14. SPONSORING AGENCY CODE
                EPA 6007*11
15. SUPPLEMENTARY NOTES
16. ABSTRACT
    A procedure was developed for  the  determination  .     \ce q'
-------