\ I/
                    United States
                    Environmental Protection
                    Agency
 Office of Health and
 Environmental Assessment
 Washington DC 20460
                    Research and Development
 EPA/600/S6-87/007  Mar. 1988
&EPA          Project Summary
                    Investigation  of  Cancer  Risk
                    Assessment Methods
                    Bruce C. Allen, Annette M. Shipp, Kenny S. Crump, Bryan Kilian,
                    Mary Lee Hogg, Joe Tudor, and Barbara Keller
                     The  major focus of this study  is
                    making quantitative  comparisons of
                    carcinogenic potency  in animals and
                    humans for 23  chemicals for which
                    suitable animal and human data exist.
                    These  comparisons are based upon
                    estimates of risk-related doses (RRDs)
                    obtained from both animal and  human
                    data. An RRD represents the average
                    daily dose per body weight of a chem-
                    ical that would result in an extra cancer
                    risk of 0.25. Animal data on these and
                    21  other chemicals of interest to the
                    U.S. Environmental Protection Agency
                    (EPA) and the Department of Defense
                    (DOD) are coded into an animal data
                    base that  permits evaluation  using
                    different risk assessment approaches.
                     The full report  is the result of a two-
                    year study to examine the assumptions,
                    other than those involving  low-dose
                    extrapolation, used  in  quantitative
                    cancer risk assessment. The study was
                    funded by the DOD (through an inter-
                    agency transfer of funds to the EPA),
                    the EPA, the Electric Power Research
                    Institute and, in its latter stages, by the
                    Risk Science Institute.
                     This  Project Summary was  devel-
                    oped by EPA's Office of Health and
                    Environmental Assessment,  Washing-
                    ton, DC, to announce  key findings of
                    the research project that is fully doc-
                    umented in four separate volumes of
                    the  same  title (see  Project Report
                    ordering information at back).


                    Introduction
                     The full report is the  result of a two-
                    year study to examine the assumptions,
                    other than those" involving  low-dose
                    extrapolation, used  in  quantitative
cancer risk assessment. The objectives
of the study are:

  1.  To  identify and express quantita-
     tively  uncertainties  that  are
     involved  in the process of  risk
     estimation, excluding the uncer-
     tainties in the low-dose extrapola-
     tion model;

  2.  To  examine  the  impact of  the
     different assumptions that  are
     made in risk estimation;

  3.  To compare results calculated from
     human and animal data, including
     the identification of the assump-
     tions that produce the best corre-
     lation of  risk estimates between
     humans and animals; and

  4.  To develop guidelines for present-
     ing a range of risk estimates based
     on  different  but scientifically
     acceptable assumptions or  as-
     sumptions that have considerable
     backing   in   the    scientific
     community.

  These  objectives are  pursued using
empirical methods in which carcinogen-
icity data for 44 chemicals are analyzed
systematically  in a  variety of  ways.
Particular attention is placed on those 23
chemicals for which there exist data from
both animal and human studies suitable
for making quantitative comparisons.
  Table 1 lists  components of a quan-
titative  risk  assessment based upon
animal data. Each component requires
a decision on the part of the risk assessor
for which there is no unique "correct"
choice. Also listed in Table 1 are various

-------
possible approaches to each component.
The choices that a risk assessor makes
for these components affect the resulting
estimates of risk. The choices for these
components therefore are related to the
uncertainty in assessment of risk from
animal data.
  Objective 2  is pursued  by  making
different  risk  estimates for the  44
chemicals in the study by systematically
varying  the approaches to  the  compo-
nents listed in Table  1. Examination  of
the distributions  of the changes in the
estimates associated with  different
approaches to the  various components
permits the examination of the impact
of the various approaches (assumptions).
These distributions also  relate to the
uncertainties in  the  process  of  risk
estimation, so this work also applies  to
Objective  1.
  A  major part  of the  study  involves
making  comparisons between risk esti-
mates derived  from  animal  data  and
those derived from human data for those
23  chemicals for which  suitable data
exist for both animals and humans. This
work addresses the question of whether
correlations exist between  animal  and
human  data,  and therefore  is of funda-
mental  importance  to the  scientific
validity  of quantitative risk assessment.
The practice  of  making  quantitative
estimates of human riskfrom animal data
is based upon the hypothesis (heretofore
essentially untested) that such correla-
tions  do  in fact  exist.  If quantitative
correlations can be shown to exist, then
these correlations can provide a stronger
scientific  basis  for  risk assessment.
Further, evaluation of the  correlations
and determination of these approaches
to the components listed in Table 1  that
produce the best correlations can sug-
gest better risk assessment methods and
assist in evaluating and presenting the
uncertainty in  risk estimates  derived
using those methods, in accordance with
Objectives 3 and 4.
Conclusions
  The major focus of this study is making
quantitative comparisons of carcinogenic
potency in animals and humans for 23
chemicals for which suitable animal and
human data exists. These  comparisons
are based upon  estimates of "RRDs"
obtained from both animal and human
data.  An  RRD  represents  the average
daily dose per body weight of a chemical
that would result in an extra cancer risk
of 0.25. Animal data on these  and 21
other chemicals of interest to the EPA
and the DOD are coded into an animal
data base that permits evaluation using
different risk assessment approaches.
  The  major findings of this study are
as follows:

  1.  Animal  and  human RRDs  are
     strongly correlated. The knowledge
that this correlation exists betwee
animal and human carcinogenicit
data should strengthen the scien
tific basis for cancer risk assess
ment and cause increased confi
dence to be placed in estimates c
human cancer risk made  fron
animal data.
Table  1.    Approaches to Risk Assessment Components
  1   Length of experiment
    a^ Use data from any experiment but correct for short observation periods.
    b. Use  data  from experiments which last no less than 90% of the standard expenmen
      length of the test animal.

  2.  Length of dosing
    a^_ Use data from any experiment, regardless of exposures duration
    b. Use data from experiments that expose animals to the test chemical no less than 80°A
      of the standard experiment length.

  3.  Route of exposure
    a. Use data from experiments for which route of exposrue is most similar to that encounterei
      by humans.
    b. Use data from any experiment, regardless of route of exposure.
    c^ Use data from experiments that exposed animals by gavage, inhalation, any oral route.
      or by the route most similar to that encountered by humans.

  4.  Units of dose assumed to give human-animal equivalence
    a. mg/kg body wt/day.
    b. ppm in diet.
    c. ppm in air.
    d. mg/kg body wt/lifetime.
    e^ mg/m2 surface area/day.

  5.  Calculations of average dose
    a^ Doses expressed as average dose up to termination of experiment.
    b. Doses expressed as average dose over the first 80% of the experiment.

  6.  Animals to  use in analysis
    a^ Use all animals examined for the particular tumor type
    b. Use animals surviving just prior to discovery of the first tumor of the type chosen.

  7.  Malignancy status to consider
    a. Consider malignant tumors only.
    b._ Consider both benign and malignant tumors.

  8.  Tumor type to use
    a Use combination of tumor types with significant dose-response.
    b. Use total tumor-bearing animals.
    c. Use response that occurs in humans.
    d^ Use any individual response.

  9.  Combining data from males and females
    §._ Use data from each sex within a study separately.
    b. Average the results of different sexes within a study.

 10.  Combining data from different studies
    a^ Consider every study within a species separately
    b. Average the results of different studies within a species

 11.  Combining data from different species.
    a. A verage results from all available species.
    b. Average results from mice and rats.
    c. Use data from a single, preselected species.
    d^ Use all species separately.

NOTE: Underline indicates approach used in base analysis (Analysis O).

-------
2.  Inthe majority of cases considered,
    analysis methods for bioassay data
    that utilize lower statistical confi-
    dence  limits as  predictors yield
    better predictions of human results
    than do the same methods using
    maximum likelihood estimates.

3.  Analysis methods for animal data
    that utilize  median lower bound
    RRDs detei mined from the ensem-
    ble of data for a chemical generally
    yield  better  predictions of human
    results  than analyses that utilize
    minimum RRDs calculated from all
    the studies available.

4.  Use of the "mg intake/kg body
    weight/day" (body weight) method
    for animal-to-human extrapolation
    generally causes RRDs estimated
    from  animal and human  data to
    correspond  more closely than the
    other methods evaluated, including
    the "mg intake/m2 surface area/
    day" (surface area) method.

5.  The risk assessment approach for
    animal  data that was intended to
    mimic that used by the EPA under-
    estimates the RRDs (equivalent to
    overestimating   human  risk)
    obtained from the human data in
    this study by about an  order of
    magnitude,  on average. However,
    it should be understood  that the
    risk assessment approaches imple-
    mented in this study are computer-
    automated  and  do not  always
    utilize the same data or provide the
    same result as the EPA approach.

6.  Reasonable risk analysis  methods
    can be defined for  the chemicals
    in this study that reduce the resid-
    ual loss (roughly the average mul-
    tiplicative factor by which the RRD
    predictors  obtained  from  the
    animal data are inconsistent with
    the range of human RRDs consist-
    ent with the human data) to 1.7.
    This is  not the same as saying that
    the predictors  are accurate to
    within  a factor of 1.7, because the
    estimated ranges of human RRDs
    that are consistent with the human
    data cover an order of magnitude
    or more for most chemicals.

7.  It has been possible to identify a
    set of analysis  methods using the
    median lower bound estimates that
    are most appropriate for extrapo-
    lating risk from animals to humans.
      given the current state of knowl-
      edge and data analysis. It is pos-
      sible to  use  the information  and
      results presented in this investiga-
      tion to calculate  ranges  of  risk
      estimates that are  consistent with
      the data and also incorporate many
      uncertainties associated with the
      extrapolation procedure.

  8.   The many components  of  risk
      assessment are interrelated  and
      evaluation  of  risk  assessment
      methods should focus on the com-
      plete risk assessment  process
      rather   than   on   individual
      components.

  9.   The data base and method used in
      this study can provide a  useful
      basis for evaluating various  risk
      assessment methods.
This study  only compared human and
animal results for a relatively high risk
level. It did  not examine the uncertainty
inherent  in the low-dose extrapolation
process.
  The animal data base and the methods
used in this study provide a useful basis
for  evaluating  quantitative risk assess-
ment. Their use in the  present context
has  demonstrated  the  strong positive
correlation  between the  animal and
human risk estimates and, hence rele-
vance of animal  carcinogenicity exper-
iments  to  human  risk  estimation.
Moreover, it has been possible to identify
methods of analysis of the bioassay data,
including the choice of the median lower
bound predictor, that satisfactorily pre-
dict risk-related doses in humans. Appli-
cation of these methods has led  to
suggested  guidelines  concerning the
prediction of  human risks  and the
presentation  of ranges  of estimates
incorporating the relevant uncertainties.
  There are, however,  certain  features
of this investigation that should be borne
in mind when evaluating the results of
this study. These are summarized below.
• A risk level of 0.25 is used throughout.

• The bioassay data is rather crude in
   several respects. The data  deficien-
   cies and their impact on the ability to
   perform some analyses are discussed
   in the document.
• The epidemiological data is of variable
   quality. Some degree of subjectivity is
   inherent in the  estimates of uncer-
  tainty associated with the epidemio-
   logical RRDs.
• Different forms (complexes)  of some
   chemicals were grouped together.

• Other approaches to the components
  could be defined and investigated.
• The three loss functions employed in
  the prediction analysis lack an under-
  lying  statistical development and so
  have  been  used merely to  rank the
  analysis methods.
• Many other analysis methods could be
  investigated.
   Bruce C. Allen. Annette M. Shipp,  Kenny S.  Crump, Bryan Kilian, Mary Lee
     Hogg, Joe  Tudor, and Barbara Keller are  with  Clement Associates, Inc.,
     Ruston, LA  71270.
   Chao Chen is the EPA Project Officer (see below).
   The complete report consists of four volumes entitled "Investigation of Cancer
     Risk Assessment Methods:" (Set Order No. PB 88-127 O97/AS; Cost: $80.OO)
     "Summary" (Order No. PB88-127 105/AS; Cost: $14.95)
     "Volume 1. Introduction  and Epidemiology" (Order No. PB 88-127113/AS;
     Cost $32.9 5)
     "Volume2.  Bioassay Data Base" (Order No. PB 88-127121/AS; Cost $25.95)
     "Volume 3.  Analyses" (Order No. PB 88-127139/AS; Cost $19.95).
   The above reports will be available only from: (costs subject to change)
           National Technical Information Service
           5285 Port Royal Road
           Springfield, VA 22161
           Telephone: 703-487-4650
   The EPA Project Officer can be contacted at: .
           Office of Health and Environmental Assessment
           U.S. Environmental Protection Agency
           Washington,  DC 20460

-------
United States
Environmental Protection
Agency
Center for Environmental Research
Information
Cincinnati OH 45268
                                                                                                     ).;:^e
                                                                                                     ' ' - '?a! c  fl
                                                                                                          * ! „.  U
Official Business
Penalty for Private Use $300

EPA/600/S6-87/007

                                                        ^Cl-"1C>/ -1:>rMo:IVJRl
          OOOOS29    PS
                                     IL

-------