297 925
           MERCURY
Ambient Water Quality Criteria
              Criteria and Standards Division
              Office of Water Planning and Standards
              U.S. Environmental Protection Agency
              Washington, D.C.

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                      CRITERION DOCUMENT



                           MERCURY



CRITERIA



                        Aquatic Life



     Inorganic Mercury



          The data base for freshwater aquatic  life  and  in-



organic mercury is insufficient to allow  use of  the  Guide-



lines.  The following recommendation  is inferrred  from toxic-



ity data for saltwater organisms.



          For inorganic mercury the criterion to protect



freshwater aquatic life as derived using  procedures  other



than the Guidelines is 0.064 ug/1 as  a 24-hour  average and



the concentration should not exceed 3.2 ug/1 at  any  time.



          For inorganic mercury the criterion to protect



saltwater aquatic life as derived using the Guidelines is



0.19 ug/1 as a 24-hour average and the concentration should



not exceed 1.0 ug/1 at any time.



     Methylmercury



          For methylmercury the criterion  to protect fresh-



water aquatic life as derived using the Guidelines  is  0.016



ug/1 as a 24-hour average and the concentration  should not



exceed 8.8 ug/1 at any time.



          The data base for saltwater aquatic life  and



methylmercury is insufficient to allow use of the  Guidelines.



The following recommendation is inferred  from toxicity data



for freshv/ater organisms.

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          For methymercury  the  criterion  to  protect saltwater
aquatic life as derived  using procedures  other  than the
Guidelines  is 0.025  ug/1 as  a 24-hour  average and  the  con-
centration  should  not  exceed 2.6 u9/l  at  any time.
                         Human Health
     For the protection  of human health from the toxic prop-
erties of mercury  ingested through water  and through contami-
nated aquatic organisms  the  ambient water criterion  is deter-
mined to be 0.2 ug/1.

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Introduction
     Mercury, a silver-white metal which is a liquid at
room temperature, can exist in three oxidation states: elemental,
mercurous, and mercuric; it can be part of both inorganic
and organic compounds.
     Mercury is a silver-white metal, atomic weight 200.59.
A liquid at room temperature, its melting point is -38.87°C
and its boiling point ranges from 356 to 358°C.  The metal
is insoluble and is not attacked by water.  At 20°C, the
specific gravity is 13.546 (Stecher, 1968), and the vapor
pressure is 0.0012 mm Hg (Stecher, 1968).
     Mercury exists in a number of forms in the environment.
The more commonly found mercuric salts  (with their solubili-
ties in water)  are HgCl2 (lg/13.5 ml water), Hg(N03)  (soluble
in a "small amount" of water), and Hg (CH3COO)250  (lg/2.5
ml water).  Mercurous salts are much less soluble  in water.
HgNo3 will solubilize only in 13 parts water containing
1 percent HNO^.  Rq2^2 *s Practi-caHy  insoluble in water.
Because of this, mercurous salts are much less toxic than
the mercuric forms (Stecher, 1968).
     The Department of the Interior carried out a  nationwide
reconnaissance of mercury in U.S. water in the summer and
fall of 1970 (Jenne,  1972).  Of the samples from the indus-
trial wastewater category,  30 percent contained mercury
at greater than 10 jug/1:  nearly 0.5 percent of the samples
in this group contained more than 1,000 jug/1.  Only 4 percent
of the surfacewater samples contained more than 1,000 jug/1.
The higher mercury concentrations were generally found in
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small  streams.   About half  the 43  samples  from the Mississippi
River  contained  less  than 0.1  jug/1.   The mercury content
of  lakes  and  reservoirs was between  0.1 and  1.8 /ag/1.   With
few exceptions,  the mercury content  of groundwater samples
w,as below detection (O.ljug/1).
     In a survey by the EPA Division of Water  Hygiene,  273
community, .recreations, and federal  installation water  sup-
plies  were  examined.   Of these,  261  or 95.5  percent,  showed
either no detectable  mercury or  less than  1.0 >ug/l in  the
raw and finished water.  Eleven  of the supplies had mercury
concentrations of 1,0 to 4.8jug/l  and one  supply exceeded
5,0/jg/l.   When  this  one supply  was  extensively reexamined,
the mercury concentration was  found  to be  less than 0.8
jug/1  (Hammerstrom,  et al. 1972).
     Seawater contains 0.03 to 2.0jug/l, depending on  the
sampled area, the depth, and the analyst.  In  a study  of
Pacific waters,  mercury concentrations were  found to increase
from .surface  values of near 0.10 jjg/1 to 0.15  to 0.27/ig/l
at  greater  depths.   In an area seriously affected by pollution
 (Minamata B.ay, Japan), values  ranged from  1.6  to 3.6jjg/l.
The National  Research Council  (1977)  has shown typical  oceanic
values for  mercury to be .01 to  .03/ig/1.  Oceanic mercury
is  generally  present  as an  anionic complex (HgCo- ),  which
does not  have as pronounced a  tendency to  bind to particulate
substances  and  then settle  out as  do mercury compounds  found
in  freshwater  (Wallace, et  al.  1971).
     A major  use of mercury has  been as a  cathode in the
electrolytic  preparation of chlorine and caustic soda;  this
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accounted for 33 percent of total demand in the United States
in 1968.  Electrical apparatus (lamps, arc rectifiers, and
mercury battery cells) accounted for 27 percent, and indus-
trial and control instruments (switches, thermometers, and
barometers), and general laboratory applications accounted
for 14 percent of demand.  Use of mercury in antifouling
and mildew proofing paints (12 percent) and mercury formula-
tions used to control fungal diseases of seeds, bulbs, plants,
and vegetation (5 percent) were other major utilizations,
however, mercury is no longer registered by the EPA for
use in antifouling paints or for the control of fungal dis
eases of bulbs.  The remainder (9 percent)  was for dental
amalgams, catalysts, pulp and paper manufacture, Pharmaceuticals,
and metallurgy and mining.
     Several forms of mercury, ranging from elemental to
dissolved inorganic and organic species, are expected to
occur in the environment.  The finding that certain micro-
organisms have the ability to convert inorganic and organic
forms of mercury to the highly toxic methyl or dimethyl
mercury has made any form of mercury potentially hazardous
to the environment (Jensen and Jernelov, 1969).  In water,
under naturally occurring conditions of pH and temperature,
inorganic mercury can be coverted readily to methyl mercury
(Bisogni and Lawrence, 1973).
     Mercury is able to form a series of organometallic
compounds with alkyl, phenyl, and methoxyethyl radicals.
Short-chained alkyl mercurials are toxicologically important
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 because  the carbon-mercury bond can be broken in vivo, with



 the  subsequent disappearance of the organic radical.   In


 humans,  mercurials have been associated with neurological


 disorders,  sensory impairment,  tremors, buccal ulceration,


.gastro-intestinal complaints and multisystem involvement


 due  to general encephalopathy (Matsumoto,  et al. 1965; Chang,


 et -;al. .1973;  Davis,  et al. 1974; Rustam, et al.  1975;  Weiss


-a'nx3-Doherty, ,1976) .   Mercurials will damage the  bronchial


 epithelium -:and interrupt respiratory function in freshwater


 invertebrates.  Rainbow trout will suffer  loss of equilibrium,


 and  ;trout fry ate more susceptible to mercury poisoning


-than finger.lings. Mercurial compounds may  interfere with


 receptor membranes in fish (Kara,  et al. 1976).


      Mercury can be  bioconcentrated many fold in fish  and


.other aquatic organisms because of rapid uptake  and the


 relative inability of fish to excrete methyl mercury from


:their•tissues.  Freshwater values  of 63,000 have been  found


 as-well, as  :sa'ltwater bioconcentration values of  10,000.


      Non-human mammals have been shown to  suffer central


 nervous  system :rdamage as well as teratogenesis and spontaneous


 tumorigenesis (Robbins and Chen, 1951; Spann, et al.  1972;



 Inamoto, et al.  '1976).  There is no data available on  the


.teratogenicity or mutagenicity  of  inorganic mercury in human
      '.                                                 t

 populations  Furthermore, there is no evidence of mercury


.exposure producing carcinogenicity.
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                          REFERENCES







Bisogni, J.J., and A.W. Lawrence. 1973. Methylation of mercury



in aerobic and anaerobic environments. Tech. Rep. 63. Cornell



Univer. Resour. Mar. Sci. Center, Ithaca, New York.







Chang, L.W., et al. 1973. Minamata disease. Acta Neuropathol.



26: 275.







Davis, L.E., et al. 1974. Central nervous system intoxication



from mercurous chloride laxatives. Arch. Neurol. 30: 428.







Hammerstrom, R.J., et al. 1972. Mercury in drinking water



supplies. Am. Water Works Assoc. 64: 60.







Kara, T.J., et al. 1976. Effects of mercury and copper on



the olfactory response in rainbow trout, Salmo gairdneri.



Jour. Fish Res. Board Can. 33: 1568.







Jenne, E.A. 1972. Mercury in waters of the United States,



1970-1971. Open file rep. U.S. Dep. Interior Geol. Surv.



Menlo Park, Calif.







Jensen, S., and A. Jernelov. 1969. Biological methylation



of Nature. 223: 753.
                                 A-5

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Hat sumo to/  H. ,  et al. 1965. Fetal minomata  disease.  A neuro-



pathological. study of two cases of intrauterine  intoxication



by a methyl mercury compound. Jour. Neuropathol.  Exp. Neurol.



24: 563..






National Research: Council. 1977. An assessment of mercury



in the environment. National Academy of Sciences, Washington,



D.C..






Robbi.ns,,. E:..B, ,. .and. R'.,K., Chen. 1951. A new mercurial  diuretic.



Jo.urf.- Am:*- Pharma. Assoc. 40: 249.

                                   (
                                   i



Rastam, H.:,  et  al. 1975. Arch. Environ. Health 30:  190.
     ,, J..W..,,  et al.. 1972. Ethyl mercury p-toluene  sulfonanilide;



l;e-t-ha«i: and  reproductive effects on pheasants.  Science 175:  328.







Ste.eh'er,  PiG'. ,. ed.  1968. The Merck Index. 8th  ed.,  Merck



and Co..,.  Rahway,, New Jersey.




      !


Wallace,  R.A..,  et al. 1.971. Mercury in the  environment:



the human element.  Oak Ridge, Tenn.







Weiss, B,. ,  and R..A. Doherty. 1976. Methylmercury poisoning.
      i


TJer-atology  12.:  311.
                                  A-6

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AQUATIC LIFE TOXICOLOGY*



                         FRESHWATER ORGANISMS



Introduction



     Mercury has long been recognized as  one of  the  more  toxic



metals but only recently was it identified  as a  serious pollutant



in the aquatic environment.  Initially, elemental  mercury which  is



a liquid at room temperature, was considered a relatively inert



heavy metal.  It was thought that it would  quickly settle to the



bottom of a body of water and remain there  in an innocuous state.



However, both aerobic and anaerobic bacteria in  the  sediments are



capable of methylating mercury.  Largely  because of  this  bacterial



methylation process, which is maximum at  a  pH of 6,  elemental mer-



cury can be a serious threat to the aquatic environment.



     The toxicological data base and environmental chemistry of



mercury suggest that monomethyl mercury and divalent inorganic



mercury are the principal environmental concerns for mercury in



aquatic systems.  In the following discussion and  criteria,  the



terms inorganic mercury and methylmercury will be  used  unless re-



ferring to a specific compound.  All data are expressed as mercury,
*The reader is referred to the Guidelines  for  Deriving  Water



Quality Criteria for the Protection of Aquatic Life '[43 FR  21506



(May 18, 1978) and 43 FR 29028 (July 5, 1978)]  in  order to  better



understand the following discussion and recommendation.  The fol-



lowing tables contain the appropriate data that were  found  in the



literature, and at the bottom of each table  are the calculations



for deriving various measures of toxicity  as described  in the



Guidelines.
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     The methylated  form  is  more  water  soluble  than the elemental
form and it  is also  more  biologically active.   Mercury bioconcen-
trates significantly from water and  from food.   Depuration is slow
and the biological half-life of mercury in  aquatic  organisms is
estimated at about two  years.
     Mercury is one  of  the few major pollutants that adversely af-
fects the aquatic environment through both  direct  toxicity and
bioaccumulation.  Bioaccumulation has been  more thoroughly studied
and has raised more  concern.  Methylmercuric  compounds are more
tox.ic than inorganic mercury to mammals as  well as  aquatic life
and most of  the tissue  residue data  reported  are for the organic
form.  There is no known  physiological  function of  mercury and any
mercury added to the aquatic environment may  increase tissue resi-
dues.  The methylation  of mercury in aquatic  systems raises a
question as  to what  basis should  be  used to develop a criterion
for mercury.  Some organic forms  are substantially  more toxic than
other organic forms  and the  inorganic forms.
     Phenylmercuric  acetate  (PMA)  is variable  in formulation, hav-
ing various  levels of active ingredients.   In adjusting the data
in the tables the percentage of active  ingredients  given by the
authors was  used in  converting to metallic  mercury  concentrations.
When the percentage  of  active ingredients was not given, 80 per-
cent PMA was assumed (Allison, 1957).
Acute Toxicity
     Table 1 contains the acute toxicity data for various mercury
compounds and groups these different types  into inorganic mercury
salts, methylmercuric compounds and  others, chiefly organic.  The
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latter information exists principally because  many of  these  com-


pounds have been used for disease treatment  and  parasite  control
                      i
in fish cultural practices.

     The acute toxicity data for inorganic and methylmercuric com-

pounds are probably biased by the lack of data on  other than sal-

monid species.  The single value for the nitrate salt  is  lower


than the values for the chloride salts but no  major significance

can be attributed to the difference since the  work was done  by a

different investigator.  Clearly, however, methylmercuric chloride

is more toxic as shown by the rainbow trout  data.   Brook  trout

appear more resistant than rainbow trout to  methylmercuric


chloride.

     The available data for inorganic mercury  do not give any in-

dication of differences in sensitivity among species of fish.

Since only two species have been tested for  methylmercuric chlo-


ride there is an inadequate data base to draw  inferences.  Phenyl-

mercuric acetate (PMA) is variable in mercury  content  and although

the values have been corrected for mercury content as  indicated

earlier, some variability may be due to the  compounds  used.   Ig-

noring any uncorrected differences in PMA formulations tested, the

differences within species are as great as between species.     ,


     MacLeod and Pessah (1973) reported temperature effects  of

mercuric chloride toxicity to rainbow trout.   At 5, 10, and  15°C,


the unadjusted LC50 values were 400, 280, and  220  ug/lf respec-


tively.  Clemens and Sneed (1958) found that at  temperatures of

10, 16.5, and 24°C, the unadjusted LC50 values for channel catfish

and phenylmercuric acetate were 1,154, 863,  and  233 ug/1,/ respec-


tively.  They also investigated the influence  of life  stage  of
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channel catfish on  its  sensitivity  to  pyridylmercuric acetate.   At
                                             i


23 to 24°C, they  found  about  the  same  influence  of  age between



yolk sac fry  (unadjusted 48-hour  LC50  value  of 374  ug/D  and 3-



inch juveniles  (unadjusted  24-hour  LC50 value of 3,750 ug/D as



they did for  temperature between  10 and 24°C.



     Table 2  contains acute toxicity data  for invertebrate  spe-



cies.  No data  for  organic  forms  of mercury  were found,  probably



because most  of the recent  concerns regarding mercury have  been



with regard to  residues and health  effects.  The adjusted LC50



values for inorganic mercury  range  from 0.02 to  2,310 ug/1.



Again, no judgment  can  be made on the  appropriateness of  the ad-



justment factors  except that  the  adjustment  of 21 is  certainly  not



excessive for differences between species.

                   9

     In summary,  the Final  Fish Acute  Values are 38.0 and 8.8 ug/1



for inorganic mercury and methylmercury, respectively.  No  final



values, will be derived  for  the other mercury compounds  because  of



the wide range  of toxicity  of this  diverse mixture  of compounds.



The Final Invertebrate  Acute Value  is  3.2 ug/1 for  inorganic mer-



cury.  Therefore  the Final Acute Values are  3.2  and 8.8  ug/1 for



inorganic mercury and methylmercuric compounds,  respectively.



Since invertebrate  species  are approximately 12  times more  sensi-



tive than fish  to inorganic mercury, the Final Acute  Values  for



methylmercury would probably be lower  if data were  available for



invertebrate  species.



Chronic Toxicity



     Table 3  contains the chronic toxicity data  for fish.   McKim,



et al. (1976) observed  adverse effects of methylmercuric  chloride



on brook trout at 0.93  ug/1 but not at 0.29  ug/1.   Brook  trout
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were approximately three to four times more resistant  than  rainbow
trout based on acute toxicity.  This is not greatly  different  than
the species sensitivity factor  (6.7) from the Guidelines  and would
tend to support that factor as a minimum.  The geometric  mean  of
these values divided by the species sensitivity  factor (6.7) gives
an estimate of 0.078 ug/1 as the concentration protective of 95
percent of fish species.  The estimate of chronic  toxicity  using
the application factor is 1.8 ug/1.  The Final Fish  Chronic Value
for methylmercury is the lower, or 0.078 ug/1.
     The only chronic data for invertebrate species  are for
Daphnia magna.  The Final Invertebrate Chronic Values  are 0.44 and
0.20 ug/1/ for inorganic mercury and methylmercury,  respectively.
However, the source of the Final Invertebrate Chronic  Value for
methylmercury (0.20 ug/D is a static test with  measured  concen-
trations of methylmercuric chloride (Beisinger,  et al.  manu-
script).  A comparable flow-through test with methylmercuric chlo-
ride by the same authors resulted in an observed effect at  the
lowest measured exposure concentration of 0.04 ug/1-   No  chronic
value could be calculated from this latter test  since  methylmer-
curic chloride could not be detected in the control  test  water
(Beisinger, et al. manuscript).  There was no great  difference be-
tween the static and flow-through tests with measured  concentra-
tions of mercuric chloride (Beisinger, et al. manuscript) with
chronic values of 1.27 anmd 1.87 ug/1/ respectively.
Plant Effects
     A variety of endpoints have been used to measure  the effects
of mercury compounds on plants.  The respective  Final  Plant Values
for inorganic mercury and methylmercury are 60.0 ug/1  and between
2.4 and 4.8 ug/1.
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Residues
     Table 6 contains  bioconcentration  factor (BCF)  data for in-
organic mercury with an  alga  and methylmercuric  compounds with
fish.
     No equilibrium of mercury  in  the  fish  tissues  could be demon-
strated by Reinert, et al.  (1974)  after an  84-day exposure of
juvenile rainbow trout and  the  uptake  of methylmercuric  chloride
by brook trout had not reached  equilibrium  after 273 days (McKim,
et al. 1976).  In the  latter  study,  there was no detectable loss
of mercury from various  tissues after a 16-week  exposure in con-
trol water.  Since whole fathead minnows were only  analyzed once
at the end of a life-cycle  exposure  (Olson,  et al.  1975) no com-
ment can be made with  regard  to equilibrium in this  species.
     Data  (Reinert, et al.  1974) indicate an influence of tempera-
ture on rate of uptake but  was  not considered for BCF calculations
since a steady state was not  achieved even  at the highest tempera-
ture studied.  Tissue  residue concentrations after  12 weeks of ex-
posure followed temperature directly with the lowest bioconcentra-
tion factor (4,525) occurring at 5°C,  and intermediate BCF (6,628)
at 10°C, and the highest BCF  (8,376) at 15°C.
     The contrast between fathead  minnows (Olson, et al. 1975) and
brook trout (McKim, et al.  1976) is  one of  considerable  interest
and potential importance.   Of the  factors that differ between
these tests, the species and  feeding habits,  the latter  is the
most intriguing to consider.  Since  the trout were  fed on pelleted
trout feed, there was  little  opportunity for food chain  input to
the trout.  In contrast, the  fathead minnow,  a browser,  had the
opportunity not only to  feed  on the  introduced food  but  also on
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the Aufwuchs growing within the mercury-enriched  environment of
the exposure chamber.  The higher bioconcentration  factor  for the
fathead minnows, 62,898, may be more representative  of  field data.
     Since the lowest maximum permissible  tissue  concentration
(1.0 mg/kg) is based on the marketability  of  fish and  shellfish,
only data on the edible portion of these organisms may  be  used to
calculate a Residue Limited Toxicant Concentration  (RLTC).   Of the
three tested fish species, the rainbow  trout  and  fathead minnows
were analyzed whole.  Muscle data are available for  the brook
trout.  However, McKim, et al. (1976) concluded that for the brook
trout there was no difference in bioconcentration factors  between
residues in muscle and total body.  Consequently, the highest geo-
metric mean BCF for a single species will  be  used to calculate the
RLTC for methylmercury.  This bioconcentration factor  is 62,898.
The RLTC is, therefore, 0.016 ug/1 to protect the marketability of
fish and shellfish.
     There are no bioconcentration factors  for inorganic mercury
and freshwater fish and shellfish,.  However,  there are  data  for
the American oyster (Kopfler, 1974) that demonstrate the, relation-
ship of uptake between inorganic mercury and methylmercuric  com-
pounds.  The BCF for inorganic mercury  (10,000) is 0.25 of the
comparable value (40,000) for methylmercuric  chloride.   It seems
reasonable to assume that the freshwater BCF  for  edible portions
of fish and shellfish and inorganic mercury should be 0.25 times
62,898 or 15,725.  This BCF results in  a RLTC of  0.064  ug/1  using
the 1.0 mg/kg limit for marketability.
Miscellaneous
     Table 7 contains no additional data that would  alter  the
selection of the RLTCs for the Final Chronic  Value.
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CRITERION FORMULATION


                    Freshwater-Aquatic  Life


Summary of Available Data


     The concentrations  herein  are  expressed  as  mercury.   The


concentrations below have been  rounded  to two significant


figures.


     Inorganic Mercury


          Final Fish Acute Value =  38  ug/1
                                    j

          Final Invertebrate Acute  Value =  3.2 ug/1


               Final Acute Value =  3.2  ug/1


          Final Fish Chronic Value  = not available


          Final Invertebrate Chronic Value  =  0.44 ug/1

       !
          Final Plant Value = 60 ug/1


          Residue Limited Toxicant  Concentration = 0.064 ug/1


               Final Chronic Value  = 0.064  ug/1


               0.44 x Final Acute Value =1.4 ug/1


          The maximum concentration of  inorganic mercury is  the


Final Acute Value of 3.2 ug/1 which is  based  on  the  more acutely


sensitive invertebrate organisms.   The  24-hour average  concen-


tration is 0.064 ug/1 and is based  on  an estimated Residue Lim-


ited Toxicant Concentration.  No important  adverse effects on


freshwater organisms of  inorganic mercury have been  reported to


be caused by concentrations lower than  the  24-hour average con-


centration.


     CRITERION:  For inorganic  mercury  the  criterion to pro-


tect freshwater aquatic  life as derived using procedures other


than the Guidelines is 0.064 ug/1 as a  24-hour average  and the


concentration should not exceed 3.2 ug/1 at any  time.
                              B-8

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     Methylmercury



          Final Fish Acute Value =8.8 ug/1



          Final Invertebrate Acute Value = not available



               Final Acute Value = 8.8 ug/1



          Final Fish Chronic Value = 0.078 ug/1



          Final Invertebrate Chronic Value = 0.20 ug/1



          Final Plant Value = greater than 2.4 ug/1/  less  than  4.8  ug/1



          Residue Limited Toxicant Concentration =  0.016 ug/1



               Final Chronic Value = 0.016 ug/1



               0.44 x Final Acute Value =3.9 ug/1



          The maximum concentration of methylmercury  is the



Final Acute Value of 8.8 ug/1 and the 24-hour average concen-



tration is the Residue Limited Toxicant Concentration of



0.016 ug/1.  No important adverse effects on freshwater aqua-



tic life have been reported to be caused by concentrations



lower than the 24-hour average concentration.



     CRITERION:  For methylmercury the criterion to protect



freshwater aquatic life as derived using the Guidelines is



0.016 ug/1 as a 24-hour average and the concentration should



not exceed 8.8 ug/1 at any time.
                              B-9

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                                Table I.  Freshwater fish acute values for morcury
Organism
Bloassay    Test        Chemical
Method*     Conc.»»     Description
                    Adjusted
Time     LC50       LC50
(hrs)    (ug/l)"»  (ug/1)***
Reference
Rainbow trout (juvenile),
Salmo gairdneri
Rainbow trout (juvenile),
Salmo gairdneri
Rainbow trout (juvenile),
Salmo galrdneri
Rainbow trout (juvcnl le),
Salmo galrdnerl
Rainbow trout (juvenile),
Salmo gulrdnori
Rainbow trout (juvenile),
m Salmo galrdneri
1
o
Rainbow trout (larva),
Salmo gairdnerl
Rainbow trout (juvenile),
Salmo gairdneri
Rainbow trout (juvenile),
Salmo galrdneri
Hrook trout (juvenile),
Salvellnus fontlnalls
Brook trout (yearling),
Salvollnus fontlnalis
Rainbow trout (juvenile),
Salmo galrdnerl
•Rjlnbo* trout (juvenile).
Sol mo rjcilrriner i
Inorganic Mercury
KT U Mercuric %
ch 1 or i de
FT U Mercuric 96
chloride
rT U Mercuric 96
ch 1 or i de
R U Mercuric 96
ch 1 or 1 de
R U Mercuric 24
ct> 1 or 1 de
FT 11 Mercuric 96
nitrato
Methy Imercuric Compounds
R U Methy Imurcuric 96
ch 1 or 1 do
R U Methy Imercuric 96
ch lorlde
R U Mothy Imercuric 96
chloride
FT 11 Methy Imercuric 96
chloride
FT M Methy Imercuric 96
ch lorlde
Other Mercury Compounds
R U Ethyl mercury 4fl
phosphate
R U Pheny Imorcury 96
acetate
400 300 MacLeod &
Pessah, 1973
260 216 MacLeod &
Pessah, 1973
220 169 MacLeod &
Pessah, 1973
155 05 Mat! da, 1971
903 326 Wobesor, 1973
33 33 Hale, 1977
24 1J Wobesor, 1973
42 23 Wobesor, 1973
25 14 Mat Ida, et al
1971
04 04 McKim, et al.
1976
65 65 McKim, et al.
1976
43 19 Mat Ida, et al,
1971
5.1 2.0 Matlda, et al,
1971

-------
                                                     Table I.   (Continued)
CD
Organ Ism

Rainbow trout (juvenile),
Salmo galrdnerI

Rainbow trout (juvenile),
Salmo galrdnorl

Rainbow trout (juvenile).
Salmo galrdnerI

Brown trout (juvenile),
Salmo trutta

Brown trou t (j uven iIe),
Salmo trutta

Brook trout (juvenile),
Salvellnus fontlnalls

Brook trout (juvenile),
SaIve11nus font i naI Is

Lake trout (juvenile),
Salvellnus namaycush

Lake trout (juvenile),
Sal veilnus namaycush

Goldfish,
Carassius auratus

Channel  catfish (juvenile),
I eta Iurus punctatus

Channel  catfish (juvenile),
Ictalurus punctatus
    Channel  catfish (juvenile),
    Ictalurus punctatus

    Channel  catfish (juvenile),
    Ictalurus punctatus
                                    Bloassay    Test
                                    Method*     Cone."
FT
S
S
S
S
S
S
S
S
S
S
S
U
U
U
U
U
U
U
U
U
U
U
U
Chemical
Description
Phenylmercury
acetate
Phenylmercury
acetate
Merthlolate
Pyr Idy Imercury
acetate-
Merthlolate
Pyr Idy Imercury
acetate
Merthlolate
Pyr Idy Imercury
acetate
Merthlolate
Phenylmercury
lactate
Ethy Imercury
phosphate
Ethy Imercury
p-to 1 uene
sulfonanl 1 Ide
Phenylmercury
acetate
Phenylmercury
acetate
Time
(hrs)
24
48
48
48
48
48
48
48
48
96
96
96
96
96
LC50
25
1,781
10,505
2,954
26,760
5,082
39,910
3,610
1,055
82
50
51
35
1,154
Adjusted
LC50
'•• (ug/l)»»«
12.8
789
4,652
1 ,308
1 1 .850
2,250
16,345
1,599
467
45
27
28
19
635
Reference
MacLeod &
Pessah, 1973
Wlllford,
1967
Wlllford,
1967
Will ford ,
1967
Wlllford,
1967
Wll Iford,
1967
Wlllford,
1967
Wlllford,
1967
Wlllford,
1967
Ellis, 1947
Clemens &
Sneed, 1959
Clemens &
Sneed, 1959
Clemens 4
Sneed, 1959
Clemens &
Sneed, 1958

-------
                                                            Table  I.   (Continued)
OJ
 I
t~-
1-0
Organism

Channel cafflsh (juvenile),
I eta I urus punctatus

Channel" catfish (juvenile),
I eta Iurus punctatus

Channel catfish (yolk sac  fry),
I eta Iurus punctatus

Channel catfish (I wk-6ld),
I eta Iurus punctatus

Channel catfish (juvenile  3")
Ictalurus punctatus

Channel catfish,
Ictalurus punctatus

Channel catfish,
Ictalurus punctatus

Blueglll (Juvenile),
Lepomls macroch I ru's

Blueglll (juvenile),
Lepomls macrochIrus
                                           Bloassay
                                           Method*
                                            Test
0


U


U


U


U


U


U


U


U
Chemical
pfocfjpttdn

 PhenyImercufy
 acetate

 Pheny(mercury
 acetate

 PhenyImercury
 acetate

 PhenyImercury
 acetate

 PhenyImercury
 acetate

 Pheny Imercury
 acetate

 Merthlolate
 PyrIdyImercury
 acetate

 Merthlolate
Time
(hrs)

 72
                                                                                       48
                                                                                       48
                                                  Adjusted
                                       LC50       LC50
                                       (ug/f )'»'••  (ug/l)*«»
                                                                                                863'
          233
          374
                                                                                       48      1,373
434
103
                                                                                       24      2,180         340


                                                                                       24      3,750         585
                     608
                                                                                       48     2j800       1,240
                                                                                       48     7,600       3,365
 48    31,960     14i152
Reference

Clemens &
Sneed, 1958

Clemens &
Sneed. 1958

Clemens &
Sneed, 1958

Clemens &
Sneed, 1958

Clemens &
Sneed, 1958

Will ford,
1967

Will ford.
1967

Will ford,
1967

Will ford,
1967
*   S = static, R = renewal, FT = flow-through

»•  0 = unmeasured, M = measured  '

*** Reported as concentration of mercury.

    Geometric mean of adjusted LC50:   Inorganic mercury = 147 ug/l
                                                                                        = 38 ug/l
                                      Methyl mercuric compounds = 34.5 ug/l
                                                                                                 = 8.8  ug/l
               Lowest LC50 value with measured Inorganic mercury concentration and flow-through exposures = 33 ug/l

-------
                               Table 2.  Freshwater Invertebrate acute values for norcury
Organ Ism
                                                               Adjusted
Bloassay    Test        Chemical           Time     LC50       LC50
Method*     Cone."     Description        (hrs)    (ug/l)"**  (ug/l)*«»
Reference
Rotifer,
Ph 1 1 od 1 na acut i corn 1 s
Kotlfur,
Philodlna acut 1 corn Is
Sludge worm,
Tubifex tub! f ex
Sludge worn,
Tubifex tub! fox
Daphnld,
Oaphn la maqna
Crayfish (nixed agos),
I Faxonella clypcata
U) Crayfish (mixed ages),
Faxonellij clypeata
Crayf isli,
Orconcctcs 1 Imosus
Crayfish (mixed ages),
Procnmbarus cl.irkl
Crayfish (mixed ages),
Proconibrirus clarki
Hay fly,
Ephumcrello subvaria
Stoncf ly,
Acroncuria lycorius
Inorganic Morcury
S U Morcurlc
ch 1 or i do
S U Mercuric
ch 1 or 1 do
R U . Mercuric
chloride
R U Mercuric
ch 1 or 1 do
R U Mercuric
chloride
R U Mercuric
chloride
R U Mercuric
ch 1 or 1 de
S U Mercuric
ch 1 or 1 do
R U Mercuric
ch 1 or i de
R U Mercuric
chloride
S U Mercuric
chloride
S U Mercuric
ch 1 or 1 de
96 518 439 Bulkoma. et
at. 1974
% 1,105 1,004 Hulkoma, ot
al. 1974
48 82 30 Brkovlc-
Popovlc &
Popov ic, 1977*-
48 100 36.4 Drkovlc-
Popovic &
Popov Ic, 19771
48 5 4 Bleslnger &
Christenson,
1972
96 0.02 0.02 Holt &
Finrjorman, 1977
72 10 5 Kelt &
Fingerman, 1977
% 50 42 Boutet 4
Chalsemart In,
1973
72 0.2 0.1 Holt &
Flngorntan, 1977
72 10 5 Holt &
Flngorman, 1977
96 2,000 1,694 Warnick &
Dell, 1969
96 2,000 1,694 Warnick i
fJoll, 1969

-------
                                                              Tab 10 2.  (Continued)
00
                                                                                                          Adjusted
Organism
Caddlsf ly,
Hydropsyche bettenl
Br 1st leworm,
Nals sp.
Snail (egg),
Amnlcola sp.
Snail (adult).
Amnlcola sp.
Scud,
Gammarus sp.
Midge,
Chlronomus sp.

Bloassay
Method**
S

S

S
S

S

S

Test
Cone.**1
U

M

M
M

M

M

Chemical
Description
Mercuric
chloride
Mercuric
nitrate
Mercuric
nitrate
Mercuric
nitrate
Mercuric
nitrate
Mercuric
nitrate
Time
{hrs)
96

96

96
96

96

96

LC50
(ug/l)"»
2,000

1 ,000

2,100
80

10

20

LC30

-------
                 Table 3.  Freshwater fish chronic values for mercury (McKIm, et al.  1976)

                                                        Chronic
                                            Limits      Value
Organism                        Test*       (up/I)"    (ug/l)««


                                           Methylmercuric chloride

Brook trout,                     LC        0.29-0.93     0.52
Salvellnus fontlnalls


*  LC = life cycle or partial life cycle

** Reported as concentration of mercury.

   Geometric mean of chronic value = 0.52 ug/l       0.52   _ Q.078 ug/l
                                                     6.7

   Lowest chronic value = 0.52 ug/l

                                          Application Factor Values

                                96-hr LC50           MATC
Species                           (ug/l)            (ug/l)           AF
Brook trout,                        75               0.52          0.007
Salve IInus fontlnalIs


Geometric mean AF = 0.007                                                      Geometric mean LC50 « 75 ug/l
                                  3.007 |/ 75 u
g/l x 8.8 ug/l = 1.8 ug/l

-------
                                 Table 4»  :Fr,es:hw.$ter Invertebrate ^chronic values for mercury
03
 I
Organ 1 sm
Cladoceran,
Daphnla magna
Cladoceran,
Daphnla magna
Cladoceran,
Daphnla magna
Cladoceran,
Daphnla magna
Cladoceran,
Daphnla magna
Cladoceran,
Daphnla magna
Chronic
Limits Value
Test? Jug/!)" 
-------
                                        Table 5.  Freshwater plant effects for mercury
00
I
Organ 1 sra
Alga,
Anklstrodesmus braunll
Alga,
Chlorella pyrenoldosa
Alga,
Chlorella pyrenoldosa
Alga,
Effect

Concentration
(ug/l)
Inorganic Mercury
Mercuric chloride
Enzyme 2,590
Inhibition
Growth 100
Retarded growth 150
(12 hrs)
Inhibited rates 2,006
Reference
Mat son, et al. 1972
Hannan & Patoul 1 let,
Kamp-Nlelsen, 1971
DeFlllppIs & Pallaghy
1972
, 19
          Chlorella sp.  Emerson strain
Alga,
Chi orel la vulgar Is

Alga,
Summer assemblage

Water milfoil,
MyrIophy11 urn spIcatum
          Alga,
          Anklstrodesmus braunll

          Alga,
          Coelastrum mlcroporum
          Alga,
          Florida Lake assemblage
of chlorophlll
synthesis,
respiration, and
photosynthesis

Growth
Photosynthetlc
activity
                                                              1,030
60
Growth Inhibition,  1,200
50 percent

          Methylmercuric Compounds

           Methylmercuric chloride

Enzyme Inhibition   1,598
                                Growth  Inhibition,     >2.4-<4.8
                                50 percent
                Rosko & Rachlln, 1977
Bllnn, et al. 1977
                                                                                 Stanley, 1974
                                                                       Matson, et al.  1972
                                       Holderness, et al. 1975
                                           Other Mercury Compounds

                                         Methylmercuric dlcyandlamlde

                                Growth                 <0.8            Harrlss, et al.  1970

-------
                                                      Table 5.  (Continued)
00
 I
M
00
           Organism
                                Effect
  Concentration
  (ug/l)
Reference
                     N-Methylmercurlc-1,2,3,6-tetrahydro-3,6-methano-3,4>5t6,7,7-hexachlorophthalImlde
           Alga,                           Growth
           Florida Lake assemblage
           A|ga,                           Nuisance
           Cladophoraceao                  control

           Alga,                           Nuisance
           Ulothrlchaceae                  control
           Alga,
           Chlorella sp. Emerson strain
                                       Ethylmercuric phosphate

                                                    38.6
                                                    38.6
                                        PhenyImercuric acetate

                                Inhibited rates    200.6
                                of chlorophllI
                                synthesis, respiration,
                                and photosynt hesIs
           Alga,                           Growth
           Florida Lake assemblage
Alga,                           Growth
Florida Lake assemblage
       <0.6


Diphenyl mercury

      <28.3
                                                                       Harrlss, et al. 1970
                         Burrows & Combs,  1958
                         Burrows & Combs, 1958
                         OeFlllppIs iPallaghy, 1976
                                                                       Harrlss, et al. 1970
Harrlss, et al.  1970
           Final plant value:  Inorganic mercury = 60 ug/l

                               Methylmercuric compounds = >2.4, <4.8 ug/l

-------
Organ Ism
Table 6.  Freshwater residues  for mercury


 Bloconcentratlon Factor
 Time
(days)    Reference
Inorganic Mercury
Mercuric chlorldo
Alya,
Syncdra ulna

33,800 0.29
Mo thy liner cur ic Compounds
Fujlta 4 Hashlzume. 1972
Kethy Imorcurlc chlorldo
Rainbow trout (juvenile),
Salmo galrdneri
Rainbow trout (juvenile),
Salmo gairdnerl
Rainbow trout (juvenile),
Salmo galrdneri
Brook trout,
Salvelinus fontirialls
03 Brook trout,
1 Salvelinus fontlnalls
Fathead minnow,
Plmophales promelas
Organism
Man
Mink
Mustcla vlson

4,532
6,622
8,049
20,000
12,000
62,890
Maximum Permissible Tissue
Action Level or Effect
edible fish or shot If Ish
hlstological evidence
of Injury
84
84
84
273
756
336
Concentration
Concentration
(mg/kg)
1.0
1.1
Re inert, et al. 1974
Ro Inert, et al . 1974
Ue Inert, et al . 1974
McKim, et al . 1976
McKIm, ot al . 1976
Olson, ot al. 1975
Reference
44 Fl< 4012
Wobosor, 1973
Highest geometric mean edible  tissue  bloconcentrat Ion factor for methyl mercury and a  single  spades =  62,898

Lowest miixlrnun permissible  tissue  concentration = 1.0 mg/kg,      ....... = 0.000016 mg/kg =  0.016  ug/l

-------
Organism
Table 7.  Other freshwater  data for mercury


               Effect
Test
Duration
                                        Result
                                        (ug/l)
                                               Inorganic Morcury

                                               Miircur Ic tlilor I do
           community
(pr Imnry  produi.ur1.,,
horbl vfMjrs ami
carnivorous midges)
Oayflsh  (odult),
Orconoctci  I Imosus
 1  yr
                        lrjdl  mmibors,
              !>t), 96 hrs LC50
(blastula embryo), 96 hrs LC'JO
(gastrula embryo), 96 hrs LCbO
(nuurula embryo), 96 hrs LCt>0
(tall bud embryo), 96 hrs LC50
(larva), 5 days LCbO
(adult), 96 hrs LC50
2
<2
>1.0-<10
>l.0r<10
>0.l-<10
1,000
>7,500-
-------
                                               Table 7.  (Continued)
Organism
Rainbow trout (juvenile),
Salmo galrdneri
Rainbow trout (juvenile),
Salmo gairdnerl
Brook trout,
Salvelfnus fontlnalls
Carp (embryo),
Cyprlnus carplo
White sucker (adult),
Catostomus commersonl
White sucker (adult),
Gatostomus commerson 1
Threesplne stickleback,
Gasterosteus aculeatus
Threesplne stickleback,
03 Gasterosteus aculeatus
1
Rainbow trout,
Salmo galrdneri
Rainbow trout,
Salmo gairdnerl
Rainbow trout,
Salmo gairdnerl
Test
Duration
2 hrs
>64 days
48 hrs
60-72 hrs
6 mln
16 mln
10 days
110 mln
>64 days
120 days
269 days
Effect
Depressed ol factor
bulbor response
Growth
Increased cough
frequency
Reduced hatching
success
Blood enzyme (LDH)
Inhibition 20*
Blood enzyme (GOT)
Inhibition 20*
LCO
Death
Methyl mercuric Compounds
Methyl mercuric chloride
Growth Inhibition
Loss of appetite (as ug
of Hg In total ration
consumed, 1/3 as CH^ngCI
Loss of nervous control
(as ug/l of Hg In total
Result
(ug/l)
74
>3
>3,000
8,000
10,000
>8
4,018
>0.04
860
1,600
Reference
Mara, et al. 1976
Matlda, et al. 1971
Drummond, et al . 1974
Huckabee & Griffith, 1974
Chrlstensen, 1971/72
Chrlstensen, 1971/72
Jones, 1939
Jones, 1947
Matlda, et al. 1971
Matlda, et al . 1971
Matlda, et al. 1971
Rainbow trout,
Salmo gairdnerl

Brook trout (embryo),
SalvolInus fontlnalls

Brook trout (a lev In),
SalvelInus fontlnalls
       30 mln
    16-17 days
Incubation period
+ 21 days
ration consumed, 1/3 as
CH3HgCI)

Reduced  vlabl I Ity         1,000
of sperm - EC50

Decreased enzyme              0.88
(GOT) activity

Reduced  growth                 0.79
Mclntyre, 1973
Chrlstensen, 1975
Chrlstensen, 1975

-------
                                                    ":'.-  .'  •  „•.   41  iC.*t- ij'.v* *
                                                    Table 7.   (Continued)
CD
1
NJ
to
Organ 1 sm
Brook trout (a lev In),
Sa 1 vo 1 1 nus font 1 na 1 is
Brook trout (juvenile),
Salvellnus tonti nails
Brook ;trout,
Salvellnus (ontlnalls
Newt,.
Triturus vlridoscens
Newt,.
Triturus virldescens
Newt, , . .
Triturus virldescens
Leopard frog (tadpole) '',
Rana plpiens
Leopard frog,
Rana plpiens
>':.,!: . '..'
Leopard frog (blastula embryo),
Rana plpiens
Leopard frog (gastrula embryo),
Rana plpiens
Leopard frog (neural plate
embryo) , .
Rana piplens
Leopard frog (blastula embryo),
Rana plpiens
Leopard frog (gastrula embryo),
Rana plpiens
Leopard frog (neural plate
Test ..
Duration
38 days
14 days
8 days
>2 days
17 days
8 days
48 hrs
<4 mos
5 days
5 days
5 days
96 hrs
96 hrs
96 hrs
Effect
{ •'•>
Increased enzyme
(GOT) activity
Increased blood
plasma chloride
Increased, cough
frequency
Delayed limb
regene'rat ion
Death
Death
Lciod
Fa i 1 ure to
metamorphose
LC50
LC50
LC50
Teratogenesis EC50
Teratogenes 1 s EC50
Teratogenesis EC50
Resui.t
(ug/l)'
0.79
2.93
>3
8
24
8
50
1
12-16
8-12
12-16
4-8
12-16
12-24
Reference
Christonsen, 1975
Christensen; et al. 1977
Drummond,* et al. 1974
Chang, ot al. 1976
Chang, et al . 1976
Chang, et a'l.' 1976
Chang, et al . 1974
Chang, et al . 1974
Dial, 1976
Dial, 1976
Dial, 1976
Dial, J976
Dial, 1976
Dial, 1976
embryo),.
Rana  plpiens

-------
                                               Table 7.   (Continued)
Organism
Mink (ailult),
Mustola vlscn
Mink (adult),
Mustola vlson
Mallard duck,
Anas platythynclos
Lous 1 ana red crayfish
(juveni le),
Procambarus clarkl
Chinook salmon (finger) Ing),
Oncorhynchus tshawytscha
1 Chinook salmon,
t>o Oncorhynchus tshawytscha
OJ 	
Sockeye salmon (juvenile),
Oncorhynchus nerka
Sockeye salmon (juvenile),
Oncorhynchus nerka
Sockeye salmon (juvenile),
Oncorhynchus nerka
Rainbow trout (juvenile).
Sal mo galrdnerl
Rainbow trout (juvenile).
Test
Duration
93 days
93 days
2
generations
110 hrs
1 hr
20 hrs
1.5 hrs
1 'hr
1 hr
1 hr
i
l^hr
Effect
Hlsto logic evidence of
Injury
LC50 In brain tissue
Other Mercury Compounds
Methyl mercuric dicyandl amide
Reduced fortuity and
food conversion
off Iclency
LC50
Ethyl mercuric phosphate
Distress
Safe for disease control
Pyr Idyl mercuric acetate
LC50
Safe for disease
control
; Safe for dlsoase
control
j LCI 00
!LCO
Result
(ug/l)
1,100
11,900
0.1
mg/kg
In food
53.6
77
39
10,560-
15,840
<954
<4,752
1,034
967
Reference

Woboser, 1973
Wobeser, 1973
Heinz, 1976
Hendrlck & Everett, 1965
Burrows A Combs, 1958
Burrows & Combs, 1958
Burrows 4 Palmer, 1949
Rucker, 1948
Ruckor 1 Hhlpple, 1951
Allison, 1957
Allison, 1957
Salmo galrdnerl

-------
Table 7.  (Continued)
'33
1
M
Organism
Rainbow trout (juvenile),
Salmo galrdnerl
Rainbow trout (juvenile),
Salmo galrdnerl
Rainbow trout (a lev In),
Salmo galrdnerl
Rainbow trout (juvenile),
Salmo galrdnorl
Rainbow trout,
Salmo galrdnerl
Brown trout (juvenile),
Salmo trutta
Brook trout (juvenile),
Salvellnus fontlnalls
Brook trout (juvenile),
Salvellnus fontlnalls

Test
Duration
1 hr
1 hr
1 hr
1 hr
>64 days
1 hr
1 hr
1 hr
Effect
LC50
LC18
Safe for disease
control
LC60
Phenyl mercuric acetate
Growth
Safe for disease control
Safe for disease control
Safe for disease control
Result
(ug/l)
4,752
2,376
<4,752
517
0.11-1.1
4,752
2,067
4,752
Reference

Rodgers, et al. 1951
Rodgers, et al. 1951
Rucker & Whlpple, 1951
Allison, 1957
Matlda, et al.' 1971
Rodgers, et al..-1951
AHUon, .19.57, .
Rodgers, et al . 1951

-------
                       SALTWATER ORGANISMS



Acute Toxicity



     In static  tests of 96-hour duration  (Table  8),  adjusted LC50



values for mercuric chloride and the mummichog are  437 ug/1



(Eisler and Hennekey, 1977) and 1,093  ug/1  (Klaunig,  et al.  1975).



Extended exposure for 168 hours did not increase toxicity (Table



13).  When the  geometric mean of 691 ug/1  is  adjusted for species



sensitivity, it results in a Final Fish Acute Value  of 190 ug/1



for mercuric chloride.



     The data for saltwater invertebrate  species are  more abundant



(Table 9) and encompass various life stages of annelids,  bivalve



and gastropod molluscs, crustaceans, and  echinoderms.  Early life



stages were more sensitive to mercuric chloride.  Embryos of the



clam, Mercenaria mercenaria, and oyster, Crassostrea  virginica,



had adjusted LC50 values of 4.1 and 4.7 ug/1/ respectively



(Calabrese, et  al. 1977).  Among crustaceans, larval  stages  were



also more sensitive.  Larvae of the shrimp, Palaemonetes  vulgaris,



had an adjusted LC50 value of 3.6 ug/1 (Shealy and Sandifer,



1975).   Similar sensitivity was shown by juvenile mysid shrimps



Mysidopsis bah ia.  Under flow-through conditions  with measured



concentrations, the 96-hour LC50 values were  3.6  and  .3.9  ug/1



(Sosnowski, et  al. 1979).  The value for larval  Carcinus  maenas  is



5.1 ug/1 (Conner, 1972) while adults of this  species  were less



sensitive with  adjusted LC50 values of 364 ug/1  (Portmann, 1968)



and 437 ug/1 (Connor, 1972).



     Among the microcrustaceans tested, the calanoid  copepods,



Acartia tonsa and Acartia clausi,  were the most  sensitive to



mercuric chloride.  The adjusted 96-hour LC50 values  for  these
                              B-25

-------
species ranged  from  8.5  to  17  ug/l«   The  harpactacoid copepod,


Tigriopus japonicus,  was  the most  resistant  with  a LC50  of  189


ug/1.


     The adjusted  LC50 values  for  polychaete annelids ranged  from


12 ug/1 for larval Capitella capitata and 19 ug/1  for adult


Nean.thes arenaceodentata  to 85 ug/1  for juvenile N.   arenaceo-


dentata (Reisch, et  al.  1976).   Eisler and Hennekey (1977)  ob-


served ah LC50  of  59  ug/1 for  adult Nereis virens.   Among  the


echinoderms tested,  the  LC50 value for the adult  starfish,


Asterias. forbesi,  was 51  ug/1  (Eisler and Hennekey,  1977).


     Application of  the  Guidelines to the invertebrate acute  data


for mercuric chloride results  in a geometric mean  of 49  ug/1  and


when adjusted for  species sensitivity, produces a  Final  Inverte-

    !»'
brate Acute Value  of  1.0  ug/1  for  mercuric chloride.  Of the  re-


ported studies, none  had  values  lower than this,  indicating that


guideline procedures  are  protective  of at least 95  percent  of the


invertebrate' species.


     There was  only  one  study  reported on the acute toxicity  of


methylmercuric  compounds  to a  saltwater invertebrate species. The


adjusted 96-hour LC50 value was  127  ug/1  for methylmercuric chlo-


ride and the amphipod, Gammarus  duebeni  (Lockwood  and Inman,


1975).  This results  in  a Final  Invertebrate Acute  Value of 2.6


ug/1 for 'methylmercury.


Chronic
     The  chronic  toxicity  of  mercuric  chloride  has  been determined


 (Table  10)  based  upon  a  flow- through,  life-cycle  exposure  of  the


 mysid shrimp,  Mysidopsis bahia  (Sosnowski,  et al.  1979).   In  this


 experiment,  groups  of  30 juvenile  shrimp  were reared  in each  of
                               B-26

-------
four concentrations and a control for 36 days at 21°C and  a  salin-
ity of 30°/oo.  Responses examined  include time of appearance of
first brood, time of first spawn, productivity, and growth.  All
of these responses were significantly (P<0.05) affected  at a con-
tinuous mercury concentration of 1.65 ug/1.
     The highest concentration of mercuric chloride tested having
no effect on growth and reproductive parameters was 0.82 ug/l«
This no-observed-effect concentration is approximately 0.22  times
the mean 96-hour LC50  (3.75 ug/1) determined for juveniles.  The
chronic value, calculated as the geometric mean of the chronic
limits, for Mysidopsis bahia exposed to mercuric chloride  is 1.2
ug/1.  Because Mysidopsis bahia is  among the most sensitive  to
mercuric chloride (Table 9) it is not appropriate to correct for
species sensitivity.  Therefore, in the absence of any other suit-
able chronic data, the Final Invertebrate Chronic Value  becomes
1.2 ug/1.
Plant Effects
     Inorganic mercury compounds at concentrations as low  as 1.0
ug/1 (Kayser, 1976) have affected several species of saltwater
algae (Table 11).  Growth inhibition was observed among  18 species
of saltwater algae between 5 ug/1 (the lowest concentration
tested) and 15 ug/1 (Berland, et al. 1976).  Similar results were
observed for various mercury compounds including mercuric  acetate,
mercuric cyanide, ethymercuric phosphate, phenylmercuric iodine,
and n-alkyl mercuric chlorides.
     The work of Harriss, et al. (1970) convincingly demonstrates
that various organomercurial fungicides at concentrations  as low
as 0.1 ug/1 reduced photosynthesis  and growth in laboratory  cultures
                              B-27

-------
of the saltwater  diatom, Nitzchia  delicatissima,  and several natu-
     i
ral .phytoplankton communities  from Florida  lakes.   The  Final Plant.

Values are  1.0  and 100  ug/1  for  inorganic mercury and methylmer-
     1
cury.

Residues

     The rapid  accumulation  of inorganic and  organic mercury com-

pounds by.various species of saltwater  biota  is  summarized  in

Table 12..   Inorganic  mercury is  rapidly accumulated by  a variety

of. saltwater phytoplankton  (Hannan,  et  al.  1973a,b;  Laumond, et
     !
al.  1973; Parrish and Carr,  1976).   The lobster,  Homarus

americanus, when  exposed to  6  ug/1  mercuric chloride for 30 days,

had  a bioconcentration  factor  (BCF)  of  129  and mean tissue  residue

of 1.00 mg/kg wet weight (Thurberg,  et  al.  1977)  which  is the

lower limit of  the current FDA guideline.

     Cunningham and Tripp  (1973) exposed oysters  to seawater con-

taining 10  ug Hg/1 (as  mercuric  acetate).   Whole  body residues of

2.8  mg/kg were  obtained after  a  45-day  exposure  resulting in a BCF

of 2., 800.   Kopfler (1974) exposed  oysters to  1.0  ug Hg/1 (as mer-

curic chloride) for 74  days.   Whole  body residues  of approximately

10 mg/kg were obtained  resulting  in  a BCF of  10,000.  The depura-

tion of inorganic mercury occurred  during the first 18  days post

exposure and resulted in a 21  percent decline in  tissue residues.

No significant  decreases in  residue  concentrations were recorded

for  the remainder of  the 160-day depuration period (Cunningham and

Tripp, 1973).   These  studies indicate that  inorganic forms  of mer-

cury are rapidly  bioaccumulated, result in  tissue  residues  in ex-

cess of regulatory guidelines, and  are  not  rapidly or completely

depurated after several months.
                               B-28

-------
      Kopfler  (1974) determined  the  rate  of  bioaccumulation  and



equilibrium residue concentrations  in oysters  for  both  methyl and



phenylmercuric chloride exposed at  1.0 ug Hg/1 for 74 days.  There



were  no significant differences in  the rate of accumulation  nor



the final residues  (40 mg/kg).   This resulted  in  a BCF  of 40,000



compared to the 10,000 value determined  for the inorganic form of



mercury (Kopfler, 1974).  Therefore, the form  of  mercury had a



significant effect on bioconcentration.



      The Residue Limited Toxicant Concentration (RLTC)  for  mer-



curic chloride is calculated by dividing the maximum permissible



tissue concentration  (1.0 mg/kg) by the  highest geometric mean of



the bioconcentration  factors for the lobster  (129) and  for  the



oyster (2,800 and 10,000).  The oyster geometric  mean of 5,291



results in a RLTC for inorganic mercury  of  0.19 ug/1.



     The RLTC for methylmercuric chloride is calculated by  divid-



ing the maximum permissible tissue  concentration  by the geometric



mean of the oyster BCF of 40/000.   Therefore,  the  RLTC  for  methyl-



mercury chloride is 0.025 ug/1.



Miscellaneous



     For several groups of saltwater organisms, mercury concentra-



tions of 10 ug/1 and  lower reportedly interfere with or impair



various metabolic processes considered essential  for normal



growth, survival, reproduction,  and well-being (Table 13).



     Weis and Weis (1977) show  that embryonic  Fundulus  hetero-



clitus exposed to concentrations as low  as  10  ug/1 for  3 days  ex-



hibit some developmental abnormalities as fish larvae.   Winter



flounder adults exhibit decreased respiration  and  changes  in



various blood chemistry values  after exposure  for  60 days  to
                              B-29

-------
10 ug/1  (Calabrese, et  al. 1975).  Adult  striped  bass  also exhibit



decreased respiration 30 days after  immersion  in  5  ug/1  mercury



for 30 days (Dawson, et al.  1977).   Protozoans  showed  reduced



growth during immersion in 2.3 ug/1  for 8 days  (Gray and Ventilla,



1973), or 2.5 to 5.0 ug/1 for 12 hours  (Gray,  1974).   Some deaths



were observed among adult clams exposed to  4.0  ug/1 for  168 hours



(Eisler and Hennekey, 1977)  and among oyster embryos subjected  to



3.3 ug/1 for 12 days and clam larvae exposed to 4.0 ug/1 for 8  to



10 days  (Calabrese, et  al. 1977).  Inorganic mercury concentra-



tions that did not produce significant mortality  include 1.0 ug/1



(43 hours) for oyster embryos (Calabrese, et al.  1973),  2.5 ug/1



(42 to 48 hours) for clam larvae (Calabrese, et al. 1973),  and  1.0



ug (168 hours) for adult softshell clams  (Eisler  and Hennekey,



1977).  Exposure to 10  ug for less than 2 hours interferes with



the ability of barnacle cyprids to attach to the  substrate



(Pyefinch and Mott, 1948).   Copepods show a decrease in  egg and



faecal pellet production after exposure to  2.0  ug and  higher for



10 days  (Reeve, et al.  1977), growth inhibition after  exposure  for



70 days,  to 5 ug  (Sonntag and Greve,  1977),  and  no growth inhibi-



tion during a 70-day period  to 1.0 ug  (Sonntag  and  Greve,  1977).



Signigicant mortality was observed among  crab  larvae in  47 hours



at 10.0 ug (Connor, 1972) and at 1.8 ug for 8  days  (DeCoursey and



Vernberg, 1972).  Crab  larvae also demonstrate  increased metabolic



rate after 24 hours in  1.8 ug and increased swimming activity in  5



days, at  1.8 ug  (DeCoursey and Vernberg, 1972).  Grass  shrimp lar-



vae, exhibit abnormal development after exposure for 48 hours to 10



to 18 ug  (Shealy and Sandifer, 1975).  However, no  measurable ef-



fect on  respiration, growth  or molting of 'Shrimp  adults  was ob-
                               B-30

-------
served at 1.0 ug after 60 days  (Green, et  al.  1976),  on  mortality
of adult hermit crabs exposed for 168 hours  to 10.0 ug/1 (Eisler
and Hennekey, 1977), and on mortality of grass shrimp larvae  after
48 hours to concentrations lower than 5.6  ug  (Shealy  and Sand ifer,
1975).  Among echinoderms, adult starfish  exhibited no change in
survival patterns after exposure to 10.0 ug  for 168 hours (Eisler
and Hennekey, 1977), but mercury did retard  growth  and development
of larvae after exposure for 40 hours to 3.0  ug (Soyer,  1963).
All of the data listed thus far in this section apply to inorganic
mercury compounds.  Within the  10 ug constraint,  there is only  one
observation with organomercury  compounds,  that of Cunningham
(1976).  She demonstrates that  adult oysters  held 12  hours daily
for 15 days in 10 ug, as mercuric acetate, showed a reduction in
shell growth.
                              B-31

-------
 CRITERION FORMULATION



                    Saltwater-Aquatic Life



 Summary of Avialable Data



      The concentrations herein are expressed as mercury.   The



 concentrations below have been rounded to two significant



 figures.



      Inorganic Mercury



           Final Fish Acute Value = 190 ug/1



           Final Invertebrate Acute Value = 1.0 ug/1



                Final Acute Value = 1.0 ug/1



           Final Fish Chronic Value = not available



           Final 'Invertebrate Chronic Value =1.2 ug/1



           Final 'Plant Value = 1.0 ug/1



           Residue Limited Toxicant Concentration = 0.19 ug/1 *



                Final Chronic Value = 0.19 ug/1



                0.44 x Final Acute Value = 0.44 ug/1



           .The  maximum concentration of inorganic mercury is



•the  Fi'na.! -Acute Value of 1.0 ug/1 which is based on  the more



 acutely sensitive invertebrate species.  The 24-hour average



•conj&entration  is the Residue Limited Toxicant Concentration



of .0...19 ug/1.   No important adverse effects have been re-



ported  to be  caused by concentrations lower than the 24-hour



-.average .concentration.



      CRITERION:  For inorganic mercury the criterion to pro-



tect  .saltwater aquatic  life as derived using the Guidelines



 is 0.. 19 .ug/1  as a 24-hour average and the concentration



 should  not exceed 1.0 ug/1 at any time.
                               B-32

-------
     Methylmercury
          Final Fish Acute Value = not available
          Final Invertebrate Acute Value = 2.6 ug/1
               Final Acute Value =2.6 ug/1
          Final Fish Chronic Value = not available
          Final Invertebrate Chronic Value = not  available
          Final Plant Value » 100 ug/1
          Residue Limited Toxicant Concentration  = 0.025  ug/1
               Final Chronic Value = 0.025 ug/1
               0.44 x Final Acute Value =1.1 ug/1
     No saltwater criterion can be derived for methylmercury
using the Guidelines because no Final Chronic Value  for
either fish or invertebrate species or a good substitute  for
either value is available.  However, results obtained with
methylmercury and freshwater organisms indicate how  a cri-
terion may be estimated.
     For methylmercury and freshwater organisms the  Residue
Limited Toxicant Concentration is lower than either  the Final
Fish or Final Invertebrate Chronic Value.  Therefore, it
seems reasonable to estimate a criterion for methylmercury
and saltwater organisms using the Residue Limited Toxicant
Concentration.
     The maximum concentration of methylmercury is the Final
Acute Value of 2.6 ug/1 and the 24-hour average concentration
is the Residue Limited Toxicant Concentration of  0.025 ug/l«
     CRITERION:  For methylmercury the criterion  to  protect
saltwater aquatic life as derived using procedures other  than
the Guidelines is 0.025 ug/1 as a 24-hour average and the
concentration should not exceed 2.6 ug/1 at any time.
                              B-33

-------
             «  S = static


             ** U = unmeasured
                                             Table 8*   Marine fish acute values for mercury
                                                                                                             Adjusted
Organ 1 sm
Muntnlchog (adult),
Fundulus heterocl Itus
Mummlchog (adult),
Fundulus heterocl Itus
. .
Blpassay Test
Method*' OpfiCif!1
S U
S U
Chemical
Description
Inorganic Mercury
Morcurlc
ch 1 or 1 do
Mercuric
chloride
Time
(hrs)
96
96
LC50
(ug/l)
aoo
2,000
LC50
(ug/l)
- ^ f- ;-
43?
1.093
Reference
Elsler &
1977
Klaunlg,
Hennekey*
et al. 1975

                Geometric mean of adjusted  values  for  mercuric  chloride - 691  ug/l    -^-~- = 190 ug/l
                                                                                       3 •/
03
 I
U)

-------
Table 9.  Marine Invertebrate acute values for mercury
03
1
CO
Ul
Organism
Polychaete (larva),
Capital la capltata
Polychaete (adult),
Neanthes arenacoodentata
Polychaete (juvenile),
Noanthes arenaceodentata
Sandworm (adult).
Nereis vlrens .
Bay scallop (Juvenile),
Argopecten Irradlans
Oyster (embryo),
Crassostrea virgin lea
Soft-shell clam (adult),
Mya arenarla
Hard-shell clam (embryo),
Merconarla mercenarla
Mud snal 1 (adult),
Nassarlus obsoletus
Clam (adult),
Rangla cuneata
Mysld shrimp,
Mysldopsls bah la
Mysld shrimp,
Mysldopsls bah la
Copepod,
Acartla tonsa
Copopod,
Acartla tonsa
Copepod ,
Acartla tonsa
Bloassay
Method*
S
S
S
S
S
S
S
S
S
S
FT
FT
S
S
S
Test
Cone.**
U
U
U
U
U
U
U
U
U
U
M
M
U
U
U
Chemical
Description
Inorganic Mercury
Mercuric
ch 1 or 1 de
Mercuric
ch 1 or 1 de
Mercuric
chloride
Mercuric
chloride
Mercuric
ch 1 or 1 de
Mercuric
chloride
Mercuric
chloride
Mercuric
chloride
Mercuric
ch 1 or 1 de
Mercuric
chloride
Mercuric
chloride
Mercuric
chloride
Mercuric
chloride
Mercuric
chloride
Mercuric
chloride
Time
(hrs)
96
96
96
96
96
48
96
48
96
96
96
96
96
96
96
LC50
(ug/l)
14
22
100
70
89
5.6
400
4.8
32,000
5,100
3.9
3.6
to
14
15
Adjusted
LC50
(ug/l)
12
19
85
59
75
4.7
339
4.1
27,104
4,320
3.9
3.6
8.5
12
13
Reference
Relsh, et al. 1976
Relsh, et al. 1976
Relsh, et al. 1976
Eisler & Hen nek ey,
1977
Nelson, et al . 1976
Calabrese, et al .
1977
Eisler & Hennekey,
1977
Calabrese, et al .
1977
Eisler & Hennekey,
1977
Olson & Harrel, 1973
Sosnowskl, et al .
1979a
Sosnowskl , et al .
1979a
Sosnowskl and
Gentile, 1978
Sosnowskl and
Gentile, 1978
Sosnowskl and
Gentile. 1978

-------
                                    Table 9.   (Continued)
Organism
Copepod ,
Acartla tonsa
Copepod ,
Acartla clausl
Copepod ,
PsQudodlaptomus coronatus
Copopod,
Eurytemora af finis
Copopod ,
Tlgrlopus japonlcus
Crab (adult),
Carclnus maenas
Crab (adult),
Carclnus maenas
Crab (larva),
00 Carclnus maenas
1
w Hermit crab (adult),
°^ Pagurus long 1 carpus
Grass shrimp (larva),
Palaemonetes vulgar Is
White shrimp (adult),
Peneus setllerus
Starfish (adult),
Ast.erlas forbesl
Amphlpod (adult),
Gammarus duebenl

Bloassay
Method"
S
S
S
S
S
S
S
S
S
S
S
S
S
Tost
Cone."*
U
U
U
4J
U
:U
U
U
U
U
U
U
U
Chemical
Description
Tlirso
thrs)
Mercuric 96
c.hlorldo
Mercuric 96
chloride
Mercuric 96
chloride
Mercuric 96
chloride
Mercuric 96
chloride
Mercuric 48
chloride
Mer.curl.c 48
chloride
Mercur 1 c 48
chloride
Mercuric 96
chloride
Mercur 1 c 48
chloride
Mercur l.c 96
chl or 1 de
Mercur 1 c 96
ch 1 or 1 de
Methyl mercuric Compounds
Methy (mercuric
ch 1 or 1 do
%
LC50
(ug/l)
20
'0
79
158
223
1,000
1 ,2.00
14
50
10
... - '7
60
150
LC50

-------
tn
 I
U)
•-J
                             Table  10.  Marine  Invertebrate chronic values for mercury (Sosnowskl, et al. I979a)
            Organism
Test*
 Limits
 (ug/l)
Chronic
Value
(ug/l)
                                                           Mercuric chloride
            Mysld shrimp,
            MysIdopsls bah I a
 LC
0.82-1.65
 1.2
            *  LC = life cycle or partial  life cycle

               Geometric mean of chronic values -  1.2  ug/l,  since this species Is among the most sensitive (Table 9) no
                                                             species  sensitivity  factor will be used.

               Lowest chronic value-  1.2  ug/l

-------
                                Table iii  Marine plant effects for mercury

Organ 1 sm
Concentration
Effect (iig/l)
Reference
Inorganic Mercury
Mercuric chloride
CO
1
OJ
00
Alga,
Chaetoceros costatum
A 1 ga ,
Chaetoceros galvestonensls
Alga,
Chaetoceros galvestonensls
Alga,
Chi orel la sp.
Alga,
Cyclotel la sp.
Alga,
Dunal lei la sp.
Alga,
Dunal lei la ter.tlolecta
Alga,
Dunal lei la tertlolecta
Alga,
Dunal lei la tertlolecta
Alga,
Isochrysls galbana
Alga,
Isochrysls galbana
Kelp (zoospores, gameto-
phytes; sporophytes),
Laminar la hyperborea
Accumu 1 at 1 on
after death
Reduced growth
No growth
66% reduction
In CC>2
Reduced growth
75? reduction
In C02
Chlorophy 1 l-a
decrease
Decreased growth
No effect on
growth
Accumulation
No growth
Growth Inhibition
10
100
2,500
100
2,500
143
10
2
10
2,000,000
to
Glooschenko, 1969
Hannan, et al . 1973b
Hannan, et al . 1973b
Mills & Col well, 1977
Hannan 1 Patoul 1 let, 1972
Mills & Colwell, 1977
Betz, 1977
Da vies, 1976
Da vies, 1976
Da vies, 1974
Da vies, 1974
Hopkins 4 Kaln, 1971
Kelp (zoospores, gameto-
  phytes, sporophytes).
Laminar Ia hyperborea
Lethal
10,000
Hopkins & Kaln, 1971

-------
Table 11.  (Continued)
Organ 1 sm
Giant Kelp,
Macrocystls pyrlfera
Alga,
Phaeodacty lum trlcornutum
Alga,
Phaeodacty lum tr icornuluni
Red alga (spore ling),
(' lunar la e logons
Pod a (go (spore ling),
. Plumarla olcgans
Hod alga (spore ling),
Plumarla elegans
Rod alga (spore ling),
6 species
03
I Algae,
W |fl species
Algao,
16 species
Algae,
3 species
Algae,
3 species
Algae,
3 species
Dlnof lagol late,
Gymnodinlum splondcns
Dlnof lagol late,
Scrippslul la fnuroense
Concentration
Effect (ug/l)
Decreased 50
photosynthesis
Reduced growth 50
No growth 120
Growth Inhibition 40-1,000
Abnormal 1,000
development
LC50 13
Lethal 3,000-8,000
Growth inhibition <5-l5
Lethal
Depressed growth
No further
bioaccunu 1 at ion
Changes in eel 1
chemistry
Morcur ic
Reduced growth
Reduced growth,
morphological
_ » _ *•
10-50
30-350
40
30-350
acetate
10
1-10
Reference
Clendennlng & North,
Hannan, et al. I973a
tlannan, ot al. I973a
Boney, 1971
Boney, 1971
Donoy, ct al. 1959
Bonoy & Corner, 1959
Borland, et al. 1976
Borland, ot al. 1976
Sick & Windom, 1975
Sick & Windom, 1975
Sick & Windom. 1975
Kaysor, 1976
Kayser, 1976

-------
Organism

Dlnoflagcllate,
Scrlppsleila  faeroense
Alga,
Dunallolja tertjolecta

Alga,
Phaoodactylum trlcornutum
Alga;
Cyclotella sp.
table 1U  (Continued)


Effocf
     GohcontratIon
     jug/I)
Photosy ht hes is     >2,000


              Dimethyl mercury
Reduced growth
                                                      100
                                           Other Mercury Compounds
Roforonco'
No growth            1^000              Kayser^ 1976

          Methylmercuric Compounds

           MothyImercuric chIor I do

Photosynthesis     >2jOOO              Overnelj, 1975
                            Overnell, 1975
                            Hannan i Patoulilot, 1972
                         N MethyImercurIc-1,2,3,6-tetrahydro-3,6-methano-3,4,5^6,7,
                                           7-hexachloropFTthai (mine
Diatom,
Nltzchla delIctlsslma
Algae,  .
§ species

Algae,
5 species
DI atom,
Nltzchla delicatlsslma
Red alga (sporcllng),
Plumarla elegans
Reduced
photosynthesis
             0.1
           Ethyl mercuric phosphate

Lethal                 60


Growth Inhibition    0.6-60
Reduced
photosynthesis
PhenyImercuric acetate

             OJ
LC50
 PhenyImercuric Iodine

            13
Harrlss, et al. 1970




Ukeles, 1962


Ukeles, 1962




Harrlss, et al. 1970




Boney, et al. 1959

-------
         Organ Ism
         Diatom,
         Nltzchla del I cat IssIma
         Red alga  (sporolIng),
         Plumarla  olegans

         Red alga  (sporellng),
         Plumarla  elegans

         Red alga  (sporellng),
         Plumarla  elegans

         Red algae (sporellng),
         6 species
Table 11.  (Continued)


Effect
                Concentration
                (ug/l)
              PI phony I  mercury

                        0.1
Reduced
photosynthesis
         n-Alkyt mercuric chlorides

Growth Inhibition    40-1,000
Abnormal
development

LC50
Lethal
                    1,000
                       13
                     12-80
Reference
Harrlss, et al. 1970
                                       Boney, 1971
Boney, 1971
Boney, et al. 1959
Boney & Corner, 1959
00
I
         Lowest plant value:   Inorganic morcury = 1.0 ug/l

                               methy(mercuric compounds =  100 ug/l

-------
                                               Table 12.  Marine residues  for  mercury
DO
             Organism
             A,l,ga,
             Chaetoceros galvestonensls

             Alga,
             .Croomonas sallna

             AJga .(mixed),
             Aster .lone 1:1 a' J apon I ca p I us
             U;l,P9enos~sp7 "

             Alga,
            .Phaeodjacty I urn fr I cor nutum

             Lobster  (adult),
            Komarus  amerlcanus

             Oyster  (aduTt),
             Crassostrea v.lrglnlca

            Oyster  (adult),
            Q"assQStr,ea virgin lea
            Oyster  (adult),
            Crassostrea  virgin lea
            Oyster  (adult),
            Crassostrea virgin lea
B.loconcentratlon factor

            •I norga.nj c Mercury
 Time
(days)    Reference
                                                                  c ,chlor;lde
, 7,400


   853


 3,467



 7,120


   129


 2,8.00


10,000
                                         Hannan,  et a,l . ,1973J»
                                        Par.rlsh A Carr, J-976
                                 8        Laumond,  et at. 1973
                                4


                               30


                               45


                               74
        Methylmercuric Compounds

         Methylmercuric chloride

       40,000                  74

                               •
         Other Mercury Compounds

         PhenyImercuric chloride

       40,000                  74
          Han.nan, et al. ,1973 «
          Thurberg, et al. 1977
          Cunningham & Trlpp, 1973
          Kopfler, J974
          Kopfler, 1974
          Kopfler, 1974

-------
                                               Table 12.  (Continued)



Organ ism                                  Bioconcentration Factor          (days)           Reference

                                          Maximum Permissible Tissue  Concentration

                                                                      Concentration
Organism                                  Action Level or Effect         (mg/kg)            Reference

Man                                       edible fish and shellfish        1.0              44  FR  4012




Geometric mean edible tissue bioconcentration factor = 5,291 for mercuric  chloride  and  40,000 for  methyl-
mercuric chloride.
Lowest maximum permissible tissue concentration =  1.0 mg/kg
13
I
4-
Ul

                                1.0
  mercuric chloride •= '   = 0.00019 mg/kg = 0.19 ug/1

  methylmercuric chloride        = 0.000025 mg/kg =  0.025  ug/1

-------
03
I
Organism
Shiner perch,
Cymatogast.er aggregata

Mufnnicftog  (adult),
Fundulus heteroclltus

Mummlchog  (adult),
Fundulus heteroclltus

Mummlchog  (adult),
Fundulus heteroclltus

Mummlchog  (adult),
Fundulus heteroclltus

Mummlchog  (adult),
FunduI us heteroc11tus

Mummlchog  (embryo),
FunduI us heteroc11tus

Mummlchog  (ombryo),
Fundulus heteroclltus

Munmlchog  (embryo),
Fundulus heteroclltus

Mummlchog  (adult),
Fundulus heteroclltus
            Mummlchog (adult),
            Fundulus heteroclltus

            Mummlchog (adult),
            Fundulus heteroclltus

            Mummlchog (adult),
            Fundulus hetoroclltus
Test
Ouretlon
                                     Table 13,  ipthpr marine data ;for mercury


                                               Effect
                                 168 hrs


                                 168 hrs


                                 168 hrs


                                  24 hrs


                                  28 days


                                   3 days


                                   3 days


                                  12 hrs
                                  96 hrs


                                  48 hrs


                                  96 hrs
                                                                                     Result
                                                                                     (ug/l)
   rlnorganjc Mercury

   Mercuric chloride

Brain chplInesterase
Inhibition

LCO
              LC50
              LCI 00
                                                                                     33,900


                                                                                        100


                                                                                        800
                                      Reference
                                                                                     Abou-Donla & Menzel , 1967
                                                    Elsler & Hennekey, 1977
                                      Elsler & Hennekey, 1977
                                                                                      1,000      Elsler & Hennokey, 1977
              Disrupted osmoregulatlon     125      Renfro, et al. 1974
              Enzyme Inhibition
              Many developmental
              abnormal Itles

              Some developmental
              abnormal Itles

              Some developmental
              abnormal Itles
                                                                                         12
                                      Jacklm, 1973
                            30-40     Wels & Wels, 19773


                            10-20     Wols 4 Wels, 1977a


                            30-40     Wols & Wols, 19773
                                               Mercury redistribution   1,000 ug/Hg  Shellne & Schmidt Nielsen,
                                               among organs following   kg body wt   1977
                                               Se pretreatment          plus 400 ug
                                                                        Se/kg body wt
              Hlstopathology
              LCI 00
              Aberrant behaviour
                           250-5,000  Gardner, 1975
                           2,000      Elsler, et al. 1972
                           1,150      Klaunlg, et al. 1975

-------
                                     Table  13.   (Continued)
Organ 1 sm
Mummlchog (adult),
Fundulus hcteroclltus
Munmlchog (adult),
Fundulus hoterocl Itus
Stickleback (adult),
Gastorosteus aculeatus
W inter flounder (adult),
Pseudoplcuronectes americanus
Winter flounder (adult),
Pseudopleuronectes amerlcanus
Striped bass (adult),
Morono saxat ills
Protozoan,
Crlstlgera sp.
03
1 Protozoan,
•^ Crlstlgera sp.
Protozoan,
Crlstigera sp.
Protozoan,
Euplotes vannus
Protozoan,
Cup lotos vannus
Polyctiacte (adult),
Ctonodilus sorrntus
Polycluiote (adult),
Ctenotlllus r.(;rratus
Polychnoto (ydult),
Ctcnodllus sorratus
Sandworm (adult).
Test
Duration
10.5 days
96 hrs
950 mlns
24 days
60 days
30 days
8 days
12 hrs
7 hrs
48 hrs
48 hrs
96 hrs
96 hrs
21 days
16U hrs
Effect
LCIOO
Reduction In enzyme
activity
LCIOO
Increased enzyme
activity of bladder
and kidney
Decreased respiration,
blood chemistry changes
Decreased respiration
30 days post-exposure
Reduced growth
Reduced growth
Death
Reproduction Inhibition
No effect on reproduction
LC62
LCIOO
Reprodud Ion Inhibited
LCO
Result
(ug/l)
too
170
1,000
Injections
of 1,000 ug
Hg/kg body
10
5
2.3
2.5-5
20
1,000
100
50
100
>50
25
Reference
Weis 4 Wels, 1976
Jackim, ct al. 1970
Boetlus. 1960
Schmidt-Nielsen, et al. 1977
wt
Calabrese, et al. 1975
Dawson, et al. 1977
Gray 4 Vent ilia, 1973
Gray, 1974
Cray 4 Ventilla, 1971
Persoone 4 Uyttersprot, 1975
Persoono 4 Uyttcrsprot, 1975
Relsh I. Carr, 1978
Relsh 4 Carr, 1970
Relsh 4 Carr, 1970
Elsler 4 Hennnkey, 1977
tlerels v I runs

-------
                                     Table  13.   (Continued)
Organism
Sand worm (adult).
More is v Irons
Sandworm (adult),
Nereis V irons
Polychaoto (adult),
Ophryotrocha dladena
Polychaete (adult),
Ophryotrocha diadcma
Polychocto (adult),
Ophryotrocha dladema
Polychacto (adult)j
Ophryotrocha diadcma
Polychacte (adult),
Ophryotrocha labronlca
Oyster (larva),
, Crassostroa gigns
•u

Crassostrea virginica
Oyster (embryo),
Crassostroa virginica
Oyster (mlult),
Crassostren virginica
Hard-shell clam (larva),
Mcrccnarla morconnrla
Test
Duration
168 hrs
160 hrs
96 hrs
96 hrs
96 hrs
21 days
0.5 hrs
24 hrs
12 days
12 days
12 days
40 hrs
19 days
8-10 days
E100
1,000
32
3.3
12
20
1
50
4
Reference

Elslcr 4 Honftekey, 1977
Elslor 4 Honnekoy, 1977
Rolsh 4 Carr, 1978
Relsh & Carr, 1978
Rolsh & Carr; 1978
Relsh A Carr, 1978
Brown & Ahsanullah, 1971
Okubo & Okubo, 1962
Calabreso, et al. 1977
Calabrose, et al. 1977
Calabreso, et al. 1977
Calabroso, et al. 1973
Kopfler, 1974
Calabreso, et al. 1977
Hard-she 11 clam (larva),        8-10 days
Mcrconarla mercenarla
LC50
"14  "    Calabrese, ot al. 1977

-------
                                      Table 13.  (Continued)
Organism
llard-sholl clam (larva),
Morconarl;» mcrcenarla
Hard-sholl clan (larva),
Mcrconaria norcenarla
Soft-she 1 1 clan (adult),
Mya arcnaria
Soft-sholl clan (adult),
Mya arcnaria
Soft-sholl clam (adult),
Mya arenarla
Uluo mussel (larva),
Mytl lus edul Is
riud snal 1 (adult),
Ucissarlus obsoletus
G> Mud snai 1 (adult),
^ Nassarius obsoletus
Mud snal 1 (adu It),
Nassarius obsolotus
Barnacle (cyprid),
Halanus Improvlsus
Fiarnacle (adult),
Ftalanus balanoidcs
(iarnacle (cyprid),
Balanus bctlanoldcs
I'iarnacle (cyprid),
Ralanus balanoidcs
Barnacle (naupllus).
Test
Duration
C-IO days
42-48 hrs
160 hrs
160 hrs
160 hrs
24 hrs
168 hrs
168 hrs
160 hrs
40 hrs
48 hrs
<2 hrs
6 hrs
6 hrs
Effect
LC95
LCO
LCO
LC50
LCI 00
Abnormal development
LCO
LC50
LCI 00
Abnormal development
LC90
Substrate attachment
inhibition
LC50
LC50
Result
(ug/l)
25
2.5
1
4
30
32
100
700
5,000
16,600
1,000
10
90
60
Reference
Calabrose, et al. 1977
Calabroso, et al. 1973
Elslor 4 Honnekey, 1977
Eisler 4 Honnekey, 1977
Elsler 4 Hennekoy, 1!»"
Okubo 4 Okubo, 1962
Elslor 4 Honnekey, 1977
Elsler & Hennekoy, 1977
Eisler 4 Hennokoy, 1977
Clarke, 1947
Clarke, 1947
Pyof inch I Mott, 1948
Pyef inch 4 Mott, 1948
Pyof inch & Mott, 1948
Ralanus cren^itus

-------
                                          Tiibib 13;   icbhtliiuoc
Ofcjaffli/ii
Copcpods (adult),
5 fjoridr<»
CbpcpbiJs (adult),
5 rjbhera
Copejibd (adu'ltJ;
Acaftia fclausl
Copcpod (adult),
Pscudbca'tarius nilriutus
fcbpopod (ridult);
Pscudpcaianus nl.hutus
Isopod (adult),
Jacra alb'l.frohs
Isopod (adult);
Jaora nordriiarin I.
ro Isopod (adult);
1 Jacrn alblfrohs sorisu
CO Iscpod (adult);
Idotoa noglbcla
Isopod (adult),
idotea' fcnnrfjiriafa
Crab ( larva);
Care inns nabrias
Crab (larva),
Carclnus maona's
Crab ( larva),
Corclnus mannas
Cral) (larva),
Carclnus irnr-nns
Crali (larva).
JO days
48 hrs
1.9 hrs
70 days
70 days
5 days
57 hrs
<24 hrs
<24 hrs
<24 hrs
47 hirs
20^30 hrs
4i3-J3.5 hrs
2.7 hrs
0.55 Hrs
Decrease In ^tja and ( ,
faecal pel'ibt product Ifari
ii(j-Cu interact Ions oV)
survival
LC50
Growth inhibition
tto growth inhibition
Osradregu'iatldh disruption
LC95
LCI 00
LCI DO
LC90
LWO
LC50
LC50
LC50
IC50
50
5
i
100
100
100
100
100
10
33
100
l;000
3,300
Rbbve> et ai. 1977
Rcbvb,* et ai; 1977
Cbrfler & Sparrow; 1956
Sbnritag £ Grieve, 1977
Sonhtat) 4 Greve; 1977
Jones; 1975
Jones; 1973
Jonos; J973
Jbnbs, 1973
Jones, J973
Connor; 1972
Connor, 1972
Conner, 1972
Conner; 1972
Connor, 1972

-------
                                     Table 13.  (Continued)
Organism
Crab (larva),
Carcinus maenas
Whlto shrimp (adult),
Peneus setlferus
Hermit crab (adult),
Pagarus longlcarpus
Hermit crab (adult),
Pagarus longlcarpus
Hermit crab (adult),
Pagarus longicarpus
Grass shrimp (larva).
Pa 1 aemonetes vulgar Is
Grass shrimp (larva),
Palacmonotes vulgar is
W Grass shrimp (larva),
J^ Palaemonotos vulgar is
Fiddler crab (adult),
Uca pugl lator
Fiddler crab (adult).
Oca pugi lator
Fiddler crab (adult),
Uca pugi later
Fiddler crab (zoea),
Uca pugl Ifitor
Fiddler crab (zoea),
Uca pugl lator
Fiddler crab (zoea).
Test
Duration
0.22 hrs
60 days
168 hrs
168 hrs
168 hrs
24 hrs
48 hrs
-18 hrs
28 days
6 days
24 hrs
8 days
24 hrs
5 days
Effect
Result
(ug/l)
LC50 10,000
No effect on respiration, 1
growth, or molting
LCD 10
LC50 50
LC100 125
LCI 00 56
LCD <5.6
Abnormal development 10-18
Low survival, Inhibited 1,000
1 Imb regeneration
Decreased survival 180
Increased oxygen 180
consumption
Decreased survival 1.C
Increased metabolic rate 1.8
Increased swimming activity 1.8
Reference
Conner, 1972
Green, et al . 1976
Elsler 4 Hennekcy, 1977
Eislor 4 Hennekoy, 1977
Elsler 4 Hennekey, 1977
Shealy 4 Sandifer, 1975
Shealy 4 Sandifer, 1975
Shealy 4 Sandifer, 1975
Weis, 1976
Vernberg 4 Vernberg, 1972
Vernberg 4 Vernberg, 1972
DeCoursey 4 Vornberg, 1972
DeCoursoy 4 Vernberg, 1972
DeCoursey 4 Vernborg, 1972
Uca pugllator

-------
                                     Table  13.   (Continued)
03
1
cn
0
Organ 1 sm
Sea urchin (spormatazoa),
Arbacla punctulata
Sea urchin {spormatazoa),
Arbacla punctulata
Starfish (adult).
Aster las forbosl
Starfish (adult).
Aster las forbosl
Starfish (adult).
Aster las forbesl
Sea urchin (embryo),
Arbacia punctulata
Echlnoderm (larva),
Paracentrotus llvldus
Oyster (adult),
Crassostrea virgin lea
Oyster (adult),
Crassostrea virgin lea
Copepod (adult),
Acartla clausl

Test
Duration
0 rains
24 mlns
168 hrs
168 hrs
168 hrs
13 hrs
40 hrs
Result
Effect (ug/l)
Increased swimming 20
spood
Decreased swimming 2,000
speed
LCO 10
LC50 20
LC100 125
Abnormal development 92
Retarded growth and 3
development
Mercuric acetate
15 days Reduction In shell growth
12 hrs dally
60 days LC55
1.9 hrs LC50
Methyl- and Ethylmercury Compounds

Methyl mercuric chloride
10
100
50

Reference

Young 4 Nelson, 1974
Young & Nelson, 1974
Elsler & Hennekey, 1977
Elslor & Hennekey, 1977
Elsler & Hennekey, 1977
Waterman, 1937
Soyer, 1963
Cunningham, 1976
Cunningham, 1976
Corner & Sparrow, 1956
Mumrnlchog (adult),
Fundulus heteroclltus

Oyster (adult),
Crassostrea vlrglnlca
24 hrs
Disrupted osmoregulatlon     125      Ronfro, et al.  1974
19 days      Trace metal upset
                              50
Kopfler, 1974

-------
                                                Table 13.  (Continued)
           Organ Ism

           Amphi pod (adult),
           Gammarus duebenI

           Fiddler crab (adult),
           Uca spp.

           Fiddler crab (adult),
           Uca spp.
           Blue mussel  (adult),
           Mytil us edulls
                                 Test
                                 Duration

                                   3 days
Effect

Diuresis
                                  32 days      No  limb regeneration


                                  32 days      Melanin absent In
                                               regenerated IImbs

                                               Methylmercuric acetate

                                  24 hrs       Reduced feeding
Result
(ug/l)      Reference
    56
                             100
                             400
Lockwood & Inman, 1975
                           300-500    WeIs, 1977
            WeIs, 1977
            Dorn, 1976
CO
 I
Ul
           Copopods (adult),
           Acartla clausl
Oyster (adult),
Crassostrea virgin lea
           Stickleback (adult),
           Gasterosteus aculeatus
           Sockeye salmon (juvenile),
           Oncorhynchus nerka
           Sockeye salmon (adult),
           Oncorhynchus nerka
           Sockeye salmon (adult),
           Oncorhynchus nerka
                                 1.9 hrs
                                             19 days
                                 370 mlns
                               12-15 wks,
                               1  hr wkly
                               12-15 wks,
                               hr wkly as
                               juvenlles

                               12 1-hr
                               exposures
                               as Juveniles
Ethylmercuric chloride

LC50                          50


Other Mercury Compounds

Phenylmercurlc chloride

Trace metal upset             50


Phenylmercurlc acetate

LC100                        100


PyrIdylmercuric acetate

1.2 mg Hg/kg wet wt        1,000
muscle 12 weeks post-
exposure

0.24 mg Hg/kg wet muscle   1,000
3 yrs post-exposure
0.04 mg Hg/kg wet muscle   1,000
4 yrs post-exposure
            Corner & Sparrow, 1956
            Kopfler, 1974




            Boetlus, 1960




            Amend, 1970



            Amend, 1970



            Amend, 1970

-------
                                             Table 13,  (Continued)
        Organism

        Silver salmon (adult),
        Oncorhynchus klsutch
        Chinook salmon (adult),
        Oncorhynchus tshawytscha
    Test
    Duration

  12-15 wks
as juventIcs
  1  hr wkly

  35 wks as
  juvaniles
  I  hr wkly
Effect

0.03 m1t)/kg wet muscle
2 yrs post-exposure
up to 0.12 mg Hg/kg wt
muscle 4 years  later
Result
(ug/l)

 1,000
 1,000
                                                                                             Reference
Amend, 1970
Amend, 1970
08
I
tn

-------
                           MERCURY



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-------
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-------
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-------
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                                               -/


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-------
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-------
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                            B-feV

-------
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-------
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Mammalian Toxicology and Human Health Effects
     Human beings are exposed to a variety of physical and
chemical forms of mercury.  Since these forms differ  in
their toxicity and in the hazard they present to human health
it will be necessary in many parts of this document to treat
these forms separately from the point of view of hazard
evaluation.  The situation is made even more complicated
by our lack of knowledge of the forms of mercury in water.
Thus/ the approach being taken is to discuss the most impor-
tant forms of mercury to which humans are exposed, and from
this to evaluate the importance of intake from the water
supply..
     At this point, it is useful to give at least general
definitions of the usual forms that mercury can take. It
is customary (Maximum Allowable Concentrations Committee,
               t
1969) to consider three broad categories of the physical
and chemical forms of mercury.  These categories are  selected
mainly because of the difference in their toxic properties
and in the hazards they present to human health.  The first
category consists of metallic mercury.  Mercury in the zero
oxidation state  (Hg°) is usually referred to as mercury
vapor when present in the atmosphere or as metallic mercury
when present in  its liquid form.  The second category compris-
es the inorganic compounds of mercury, which include  the
salts of the two oxidation states of mercury, Hg2"l"+  (mercurous
salts), and Hg++ (mercuric salts).  The third major category
                              C-l

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contains the so-called organic mercurials or organic mercury


compounds.  These are defined as those compounds of mercury


in which mercury is attached to at least one carbon atom


by a covalent bond.  The toxic properties in this third


category, however, vary enormously.  The most  important


sub-group in the organo-mercurials category is comprised

of the methyl mercury and related short-chain  alkyl mercurial


compounds.  From the point of view of environmental exposures,


the methyl mercury compounds are the ones of greatest concern.

The other organo-mercurials may take the form  of aryl and
   ' *,
alkoxy-aryl mercurials as well as a wide variety of other

organo-mercurials used in medicine and agriculture.  In


general these organic forms of mercury are much less toxic

   I    -                                              !
than the short-chain alkyl mercurials.


     The main sources of human 'mercury exposure are methyl


mercury compounds in the food supply and mercury vapor in


the atmosphere of occupational settings.  Other sources
   i
of exposure to a wide variety of mercury forms result from


occupational, medicinal, or accidental circumstances.  As


will be discussed later, the water supply probably contains


mercury mainly in the form of Hg   salts complexed with
   i
a variety of constituents in water.


     The topics of mercury in the environment, human expo-


sure to mercury, and an estimate of health effects and hazards


o'fr mercury have been the subject of many reviews by expert


committees and individual authors over the past ten years.


Included are reviews by the Swedish Expert Group  (1971);


Study Group on Mercury Hazards (1971); WHO (1972, 1976);
                              C-2

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Miller and Clarkson (1973); Friberg and Vostal  (1972); Nordberg
(1976); and The National Academy of Sciences  (1978).  Addit-
ional references are Hartung and Dinman  (1972) , and Buhler
(1973).
     The source material for this document comes primarily
from original scientific publications, but the  reviews ment-
ioned above have also been of inestimable value in  the prepara-
tion of this document and in developing an overall perspec-
tive of the mercury problem.  Special mention should be
made of the review prepared by the WHO (1973) where the
recommended safe levels of mercury in water are discussed.
                           EXPOSURE
Introduction
     A variety of original articles and reviews have dealt
with sources, pathways and mechanisms of transport and sinks
of mercury in the environment.  These include Wallace, et
al. (1971); D'ltri (1972); Friberg and Vostal (1972); Gar-
rels,  et al. (1973); Kothny (1973); WHO  (1972,  1976); Heindryckx,
et al. (1974);  Korringa and Hagel (1974); Wollast, et al.
(1975); Abramovskig, et a.". (1975); and National Academy
of Sciences (1978).  In view of the number of recent reviews,
and the fact that a review has just been completed by a
National Academy of Sciences Panel, no attempt will be made
in this section to deal with this subject in detail except
to emphasize those data that deal directly with human uptake
of mercury from the water supply.
     The dynamics of mercury in the environment may be viewed
in the context of a global cycle.  This cycle presents a
general perspective within which man's contribution to the
                              C-3

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environmental mercury  burden may be  viewed.  However,  before



quoting numbers related  to  the global  turnover of  this element,



several caveats are  in order.  Many  of  the calculations



involve assumptions  for  which supporting  experimental  evidence



is tenuous, to say the least.  Concentrations of mercury



in certain environmental samples  (e.g., in fresh water  and



ocean water) are so  low  as  to challenge the skill  of the



best analyst using the most sophisticated modern equipment.



Matsunaga, et al.  (1979) have recently reviewed the methodo-



logical errors involved  in  the measurement of mercury  in



seawater..  These analytical figures  are multiplied by  huge


                                           12   2
numbers (e.g.  the area  of  oceans  (361 x  10  ) m   and  the


                                     17    2
precipitation over oceans  (4.11 x  10   1/m  yr) to  calculate



the "mercury budgets"  for the global cycle.  Authorities



differ in their interpretation of  certain environmental



samples and the most recent data seem  to  conflict  with  earlier



data (N'atl. Acad. Sci. 1978; Korringa  and Hagel, 1974).



It is likely, therefore, that the  "up-dating" of the global



cycle and other more localized cycles will continue.   Never-



theless, certain general conclusions have survived the  test



of time and are useful in developing a perspective with



regard to human exposure to mercury  and the possibilities



of control.



     The Global Cycle  of Mercury:  The atmosphere  is the



major pathway for distribution of  mercury.  Most reviewers



are in good agreement  that  the total entry into the atmosphere



ranges from 40,000 to  50,000 tons* per year (Table 1)  on




     i


*"tons" are metric tons, ie. 1,000 kg,  in this text.




                              C-4

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                                 TABLE 1

                   Entry  of  Mercury into  the Atmosphere
               Source                    Annual input (metric tons)

                                    Ref.  (1)        (2)             (3)


Natural
     Continental degassing           17,800                      50,000
     Oceanic emission                 7,600
     Coastal emission                 1,420
     Emission from land biota             40
     Volcanic                        	20
     Total                           26,880        25,000
Anthropogenic                        10,000        16,000
     Total                           36,880        41,000


   (1)  National Academy of Sciences  (1978)

   (2)  Korringa and Hagel  (1974)

   (3)  Heindryckx, et al.  (1974)
                                 C-5

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a worldwide basis.   The main input to the atmosphere is



from  natural sources.   Emission (degassing)  from continental



land  masses accounts for about 66  percent of the total natural



input.  Emission from the ocean surface is next in importance,



whereas emission from land biota and volcanoes seems to



be  negligible.



      Manmade (anthropogenic)  release, although less than



'tha't  due  to natural causes,  is substantial,  accounting for



•about one third  of  total input.



      The  amount  of  mercury contained in the  atmosphere .is



tine subject of widely divergent figures (Table 2) .   The



main  point of contention is  the assumption with regard to



the change of atmospheric mercury  concentration with height.



The most  recent  review of the'subject (Natl. Acad.   Sci.



-'1978) assumed an exponential decline with increasing altitude,
    i

whereas others have assumed  that mercury mixes to a height
    i

•'Q'f  1  kilometer  (Heindrykx, et al.  1974) .  This wide range




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                                 TABLE  2

             The Amount of Mercury  in some  Global Reservoirs
     Reservoir                         Mercury Content   (metric  tons)


                                       (1)           (2)


     Reservoir
Atmosphere                               850
Fresh water                            2000
Fresh water biota                        400
Ocean Water  ,                            41 x  106      70 x 106
Oceanic Biota                         200,000


   (1)  National Academy of Sciences  (1978)

   (2)  WHO  (1976)

   a  Only living biota

      Living and dead biota
                                 C-7

-------
lead to substantial  local pollution..


     Most of the atmospheric  transport  goes to the oceans


(Table 3).  Figures  vary widely.   The earlier  estimates


gave numbers of about  40,000  to  50,000  metric  tons/year.


However, the most recent estimates indicate deposition from


the atmosphere to be about  11,000  metric  tons/year.   The


entry of: mercury into  the ocean  from all  known sources seems


not to exceed about  50,000  metric,  tons/year although  the


contribution from hydrothermal sources  is unknown  and may


be important (U.K,.. Dep. Environ. 19-76).


     'The amount of mercury  contained in the oceans is-extreme-


ly; large compared with the  known inputs.   Most estimates


(see Table 2) fall in  the range of 41 million  to 70 million


tons..*  Based on the  figures given  in Tables 2  and  3,  it


is. clear that mercury  concentrations: in the open oceans
       •

(a.s- opposed to coastal and  inland  waters)  have not changed


significantly over recorded history.  Oceanic  fish levels


most probably have remained unchanged by  man's activities,
                                                       i

especially in wide ranging  oceanic, fish such as shark, sword-


fish,, and tuna fish..


     The amount of mercury  dissolved in ocean  water  is ex-


tremely large as. compared to  the amount in oceanic biota


(Table 2).  On the other hand, mercury  in living biota ac-


counts for abo.ut one^half of  the total  mercury in  freshwater.


The figures in Table 2 are  expressed, in, terms  of total mercury.

    I
If expressed in terms  of methyl mercury,  the amount of mercury
    i

in biota would considerably exceed that in fresh water.


     Data on concentrations of mercury  in the-  lithos.phere
                               C-8

-------
                                 TABLE 3
                     Entry of Mercury into the Ocean
     Source
  Annual input (metric tons)
(1)           (2)             (3)
Atmospheric deposition
Open Ocean and Polar
Coastal waters
Land run-off
Soluble
Particulate
Hydrothermal

7,600
3,600

1,600
3,700
?
41,000

5,000


5,000
?
50,000

5,000


5,000
?
(1)  National Academy of Sciences, 1978
(2)   Korringa and Hagel, 1974
(3)   Heindryckx,  et al.  1974
                                 C-9

-------
 have been reviewed by several expert groups  (World Health


.Organ.,  1976; U.K. Dep. Environ., 1976; Natl.  Acad.  Sci.,


.1978).   Mercury concentrations in nonmineralized soils vary


.over two. orders of magnitude, the average  concentration


.bel'ng .about 0.07 pg Hg/g.  Freshwater sediments  in non-pollut-


-xed .rivers and lakes in the United States usually contain


."less than 0.1 A9/9 (wet sediment).  Insufficient data exist


 .to  calculate average values .and ranges of .mercury concentra-


 tions .in oceanic sediments.


      Mercury is strongly bound to soil and is  predominantly


 .attached to organic matter (Andersson, 1976; Keckes and


 Mlet.tinen,  1970.; Landry, et al. 1978) .  Kimura and Miller

     i
 .(.1970) .reported that mercury mobility is minimal even in


 soils con.taminated by mercury fungicides.  However, Fuller


 (-1,977(, 1978) has reported that the mobility of mercury in
     i
 soils i's increased in the presence of leachates  from municipal
     i

.lanrTfl.lls.
     i

      Chemical and 'Physical Forms of Mercury in the Environ-


ment .awd Theix Transformation:  Mercury occurs in a variety
     i

JQ£ ^physical and chemical forms in nature.  Mercury is mined


;;as  cinnabar  (:Hg,s) but in some areas  (Almaden,  Spain)  the


..ore  is BO rich that metallic mercury is also present.


      Human  activities ;have resulted in the release of a
     t

.wide .variety of both inorganic and organic forms of mercury


 '(-Table 4)..   The electrical and chloralkali industries and
     i

'the  burning .of fossil fuels ..release mercury to the atmosphere


ma.rn.l-y as Hg°.  Release to water via direct discharge involves


rEg    and Hg° (e.g. chloralkali).  Methyl mercury compounds


 have been .released to fresh and oceanic water  in Japan as


                             C-10

-------
       Patterns  of Mercury Consumption in the United  States
     End use
                      Annual Consumption (% total)
                             1970
                                    1973
               1985'
Electric Apparatus
Caustic Chloride
(chloralkali)
Paints
Industrial Instruments
Dental
Catalysts
Agriculture
Laboratories
Pharmaceuticals
Others
26

25
17
7.9
3.7
3.7
3.0
3.0
1.1
9.6
33

24
14
13
4.9
1.2
3.4
1.2
1.1
4.2
32

23
5.1
21
6.2
0.8
1.1
7
0.8
9.8
 Total consumption
 (metric tons)
                   2100
1867
2091
 This table is adapted  from table 1.3  in  the report of the
     National Academy of  Science (1978) and  from figures
     derived from U.S.  EPA.  (1975a).

3The percentages were estimated under  the  assumption that consumption
     by laboratories was  negligible.
                               (CH3)2Hg
                  Fish
      Hg°-»
                   j
                                Shellfish
                                  \
                               CH3SHgCH3
•	CH.Hg*	*-(CH,),Hg    CH.S-HgCH,
Bacteria    3 >^  Bacteria     4 •*      VJ     J
                                        Bacteria
                            v..
                                            Air
                                                      Water
                                                      Sediment
  Figure 1.   The mercury  cycle demonstrating  the bioaccumulation
  of  mercury in fish and  shellfish.

  Taken from Figure 3.1  in the National Academy of Sciences
  (1978).
                               C-ll

-------
 a byproduct of the manufacture of aceteldehyde  and  vinyl


 chloride.  Other anthropogenic sources have  resulted in

                                                       i
 release of aryl and alkoxy-aryl compounds  as well as methyl


 and ethyl mercury compounds used as fungicides.


      The inorganic forms of mercury may undergo oxidation


—-reduction reactions in water as indicated  by  the  equations:


           2 Hg° = Hg+* + 2 i . . .....  (1)
                                        (.2).
;;Stock (193-4)  has demonstrated that Hg° can be oxidized  to


-Hg   r in water in the presence of .oxygen.  The reaction  prob-


 ably "fakes "place in rain droplets during removal  of  Hg°


•from 'the ratmosphere by precipitation.  Wallace, et al.  (1971)

     i
 have noted tha.t mercury concentrations as high  as 40 g/1


;can be attained when water .saturated with oxygen  is  exposed


-.to  .mercury vapor.  The mercurous form of mercury  (Hg7  )
     i                                                 * •

 undergoes .disproportionation to Hg° and Hg   in the  presence


,:o"f  rsulf.ur ligands  (Cotton and Wilkinson, 1966) .   Jensen
                                                       i

:arid 'Jerne.lov (1972) have noted that -the presence  of  organic


substances in water facilitates .the transformation of Hg°


 to  Hg  .  "The mercuric ion, Hg   is the substrate for the


"biomethylation reaction that occurs in microorganisms present


..in  .aquatic sediments (Figure 1) .


      In -a recent review by the National Academy of Sciences


 (197.8), it was noted -that the main pathway of methylation


"o;f  soluble Hg   involved --a transfer of methyl groups from
     i

.'methyl cobalamine  (methyl-B12) and that the  rate  of  formation


;of  methyl mercury  is largely determined by the  concentra-


tions x>f soluble Hg   and methyl B,--
                                C-12

-------
     Both dimethyl mercury and monomethyl mercury may be
formed by bacteria present in sediments.  The formation
of dimethyl mercury is favored by a high pH.  Dimethyl mercury
is volatile and may enter the atmosphere, where it may undergo
decomposition to yield Hg° (Wood, 1976).  It may also be
converted to monomethyl mercury in rainfall especially in
acid rains containing Hg  .  In the presence of Hg   , one
molecule of dimethyl mercury is converted to two molecules
of monomethyl mercury (Cotton and Wilkinson, 1966).
     A variety of bacterial and fungal organisms have the
capacity to methylate Hg  . Jensen and Jernelov (1972) have
pointed out that conditions which promote bacterial  growth
will enhance methylation of mercury.  Thus, the highest
rates of methylation in the aquatic environment are  seen
in the uppermost part of the organic sediments and in suspend-
ed organic material in water.  Furthermore, those microorgan-
isms able to methylate mercury at high rates are also, usually
resistant to the toxic effect of Hg
     Microorganisms are also capable of demethylating methyl
mercury compounds and of splitting the carbon-mercury bond
in a variety of other organic mercurials.  This process
involves, first, the cleavage of the carbon-mercury  bond
to release Hg   and, second, the reduction of Hg   to Hg°.
Both processes are enzyme-mediated (Natl. Acad.  Sci. 1978).
Microorganisms capable "of demethylation reactions have been
shown to occur in aquatic sediments, soils and human fecal
material.  Microbial resistance to methyl mercury correlates
                              013

-------
with the capacity to convert methyl mercury to Hg  •  Both



methylation and demethylation rates have been measured in



aquatic sediments in the laboratory (for review, see Natl.

     I

Acad. Sci. 1978).  In general, methylation and demethylation



account for the conversion of a small fraction of  the total



mercury in the sediment on an annual basis  (probably 5 percent



or less).  The total production of methyl mercury  in fresh



water on a global scale was estimated to be about  10 metric



tons/year per year and in the oceans to be about 480 metric



tons/year.


     I                              ++
     Divalent inorganic mercury (Hg  ) may undergo reduction



to Hg°.  Certain widely occurring bacteria such as Pseudomonas



have been shown to be capable of this reduction (Magos,



et al.  1964; Furukawa, et al. 1969).  Yeast cells  also carry



out this reaction and the capacity to do this correlates



with a resistance to the toxic effects of Hg    (Singh and



Sherman, 1974).



     In addition to being a substrate for both methylation



and reduction reactions in microorganisms, Hg   is avail-



able to form a variety of precipitates, complexes, and chelates



in water.  A stable precipitate is formed with the sulfide



ion S~.  The latter is usually present in anaerobic aquatic



environments.  The formation of HgS may limit the  amount



of mercury available for methylation reactions  (Jensen and



Jernelov, 1972).  However, our knowledge of the chemical



forms of mercury in natural waters is incomplete.  For theore-



tical reasons, the degree of oxygenation, pH, and  the presence



of inorganic  (e.g. Cl~) and organic (e.g.-S~f C00~, and



N in organic matter in water) ligands are probably important




                              C--14

-------
 factors in determining the chemical species of mercury in
'water.   On thermodynamic grounds,  one would expect inorganic
 mercury to be present mainly as Hg   compounds in well-oxy-
 genated water and an increasing fraction of mercury as Hg°
 or HgS  in reducing conditions (Natl.  Acad. Sci.  1978).
 In view of the high concentrations of chloride and, to a
 lesser  extent, bromide anions in sea water, inorganic mercury
 should  be present as various halide complexes  (HgCl4~, HgCl-jBr"
 HgCl.,~, HgCl2Br~, HgCl2)  in marine water.
      Methyl mercury compounds readily pass across cell mem-
 branes  and bind to tissue ligands.  Thus, methyl mercury
 tends to be removed from water by  living biota.  Unfortu-
 nately, little information is available on concentrations
 of methyl mercury in fresh or marine water.  Chau and Saitoh
 (1973)  were unable to detect methyl mercury (detection limit
 0.24 ng Hg/1) in unfiltered Great  Lakes water, and measured
 0.5 to  0.7 ng Hg/1 in four small mercury-polluted lakes.
 Andren  and Harriss (1975)  could not detect methyl mercury
 in samples of river and coastal waters of the Eastern Gulf
 of Mexico.
      Wood (1976)  has pointed out that, as a result of meth-
 ylation and demethylation reactions,  the concentrations
 of methyl mercury will approach a  steady state in any given
 ecosystem.  The steady state concentration will be affected
 by any  environmental factors that  influence either or both
 reactions.  Many factors may be involved, some of which
 have been mentioned above.  However,  there is a need for
 further studies on the dynamics of methyl mercury in the
 environment.
                               C-15

-------
found that 153 samples out of  a  total  of  193  had values



below 0.25 jug/1.  No  value above 0.8 jug/1 was detected.



The U.S. EPA  (1975b)  established that  only 2.5 percent of



512 drinking water  samples had mercury levels which exceeded



the proposed 1975 Federal standard  for drinking water  of



2,000 ng Hg/1.  A geological survey of mercury in U.S. rivers



and estuaries reported by Wers.haw (1970)  found that more



t.han half of the 73 rivers that  were sampled  had mercury



Concentrations low.er  than 1,000  ng  Hg/1 and 34 of the  rivers



had concentrations  of less than  100 ng Hg/1.   windom in



1973, reporting on  measurements  of  the Savannah estuary



fo.und. that concentrations ranged up to 450 ng Hg/1.



     Levels of- mercury in ocean  waters are usually below



3QQ ng Hg/1.  Stock and Cucuel in 1934 reported a mean value



of 30 ng Hg/1.  Hosohara  (1961)  recorded  mercury levels



a,t different depths in the Pacific; values on the surface



were about 80 to 150  ng Hg/1,  and values  at a depth of 300



meters were found to  range between  150 and 270 ng Hg/1.



Further details on  the ocean mercury- levels have been  given



in the publication  by the U.K. Department o.f  the Environment



(•1976,).  Matsunaga, et al. (1979),  in  the most recent  report



on mercury in waters, claim that 5  to  6 ng Hg/1 "may be



a reliable value for  baseline  of mercury  in unpolluted oceans,"



which is roughly 10. to 100 times lower than concentrations



reported above.  The  authors (Matsunaga,  et al.  1979)  attribute



the wide scatter in previously reported values to problems



in analytical techniques  (i.e. contamination).
                               C-1.6

-------
     Most samples of drinking water obtained in the United
States and Europe have mercury levels below 50 ng Hg/1.
Assuming a daily consumption of 2 liters of water by the
70 kg standard man, this would correspond to a daily intake
of 100 ng Hg.  Values up to 200 ng Hg/1 have been reported
in water in areas with minerals rich in mercury.  This concen-
tration would indicate an intake of 400 ng Hg/day.  Most
mercury in fresh water is probably in the form of complexes
of Hg  .  Gastrointestinal absorption of this form of mercury
is less than 15 percent.  Thus, an intake of 400 ng Hg/day
would correspond to a retained dose of less than 100 ng
Hg/day.  The current drinking water standard in the United
States is 200 ng Hg/1.  This corresponds to a daily intake
of 400 ng Hg or an estimated retained dose of 600 ng Hg.
Ingestion from Foods
     The U.K. Department of the Environment (1976) and the
National Academy of Sciences (1978) have reviewed the results
of a large number of surveys of merury concentrations in
food.  These surveys uniformly indicate that a distinction
must be made between fish and non-fish food.  In foodstuffs
other than fish and fish products, the concentrations of
mercury are so low as to be near or below the limit of detec-
tion of mercury of the analytical methods used in reported
studies.  In the United States, figures from surveys carried
out by the Food and Drug Administration indicate that most
foodstuffs have total mercury levels below 20 ng Hg/g.
Meat and poultry may contain levels up to 200 ng Hg/g  (quoted
in Nat. Acad. Sci. 1978).  In view of the uncertainties
in these numbers, it is impossible to calculate average
                              C-17

-------
daily intakes for non-fish food  in the United States.  An

extensive study in Sweden noted  that dietary mercury from

non-fish sources was about 5,000 ng Hg/day, and that the

methyl mercury content was not known.  A low intake of mercury

from non-fish sources is consistent with the finding that

non-fish eaters have the lowest  blood concentrations of

mercury.

     A variety of surveys have been carried out in the United


States of concentrations of mercury and the forms of mercury

in fish  (for review, see Natl. Acad. Sci., 1978).  These

surveys  indicate that the average concentration of mercury


in most  fish is less than 200 ng/g, with virtually all the
                                                    i
mercury  in fish muscle in the form of methyl mercury compounds.

However, certain large carnivorous oceanic fish can regularly


develop much higher levels.  In  general, over 50 percent

of swordfish tested had values more than 1,000 ng/g.  Observa-

tions on 3,000 samples of canned tuna indicated an average


total mercury concentration of approximately 250 ng/g, with

.four percent of the samples being above 500 ng/g.  Concentra-

tions much higher than these, ranging to over 20,000 ng/g,


have been reported in freshwater fish caught in heavily

polluted areas  (Fimreite and Reynolds, 1973).  The oceanic

fish in Minamata Bay in Japan also had values of this order

of magnitude.

     The age or length or weight of the fish appears to

be an important factor in determining the mercury concen-


tration  in fish muscle for both  freshwater and marine fish;
                               C-18

-------
 the older the fish, the higher the mercury concentration.
 This is consistent with the report that the half-time of
 methyl mercury in fish is of the order of 1,000 days  (Miettinen,
 et al. 1969; Miettinen, 1972).  Thus, accumulation might
 be expected to occur throughout the life of these species.
 In general, fish that are carnivorous and are at the end
 of a food chain tend to have the highest concentrations.
 Thus, freshwater fish such as the northern pike and oceanic
 fish such as the shark and swordfish have elevated mercury
 levels compared to other fish.  Marine mammals can also
 accumulate mercury.  For example, the livers of seal may
 attain very high concentrations of total mercury in the
 order of 340,000 ng/g, but over 90 percent of this is in
 the form of inorganic mercury probably combined in an inert
 form with selenium (Koeman, et al.  1973).  Nevertheless,
^-sufficient amounts of methyl mercury are found in seal tissue,
 including liver, so that individuals consuming seal meat,
 such as Eskimo, may develop high blood concentrations of
 methyl mercury (Galster, 1976).
      Observations on museum specimens of tuna fish and sword-
 fish suggest that the concentrations of mercury have not
 changed throughout this century.  For example, Miller, et
 al. (1972) found mercury concentrations in tuna ranging
 from 180 to 640 ng/g, which may be compared with present
 values in tuna ranging roughly from 200 to 1,000 ng/g wet
 weight.  The lack of observable change in mercury levels
 in tuna and other oceanic fish is consistent with the large
 reservoir of mercury in the oceans.
                                C-19

-------
     The U.S. Department of Commerce  (1978) has published

data relating to the  intake of mercury  from fish  in  the

diet of the U.S. population.  Mercury analyses were  made

on the edible tissues of 19,000 samples of fish representing
   i
all major and recreational species of the U.S. collected

in 1971-73.  Information on seafood consumption was  obtained

from a survey of 25,647 panelists who maintained  a diary

of their fish consumption.  One-twelfth of the panelists

recorded consumption  each month for one year  from September,

1973 to August 1974.  The selected data from  these studies

are given in Table 5.  Approximately 95 percent of the panel-

ists reported eating  fish.  Tuna fish was by  far  the most

popular item with 68  percent of the fish eaters reporting

they ate tuna fish.   Since 20 percent did not report the

species of fish consumed, and assuming  that a high proportion

of this group in fact consumed tuna, the proportion  eating

tuna would be about three-quarters of the test population.

By comparison, the next most popular species  of fish was

flounder, eaten by only 13 percent.

     The average concentration of mercury in  tuna is one

of the highest in the group of fish species consumed by

more than five percent of the panelists.  It  is clear, there-

fore, that the consumption of tuna fish in the United States

accounts for most of  the dietary intake of methyl mercury,

as this form of mercury accounts for more than 90 percent

of the total mercury  in tuna and most other species  of fish.
   i

     The data in Table 5 do not allow an estimate of the

average daily intake.  However, if we assume  (a)  F.D.A.

                               020

-------
                           TABLE 5

    Average and Maximum Mercury Levels in Species of Fish
          Eaten by 2% or More of 24,652 Panelists3.
Species



Tuna (light)

Shrimp
Flounder
Perch (marine)
Salmon
Clams
Cod
Pollock
Haddock
Herring
Oysters
Mercury concentration0
jug Hg/g fresh weight

Panelists
(%)
68

21
13
10
10
9
6
5.9
5.8
5.1
5.0

Average

0.14 (skipjack)
0.27 (yellow fin)
0.05'
0.10
0.13
0.05
0.05
0.13
0.14
0.11
0.02
0.03

Max imum

0.39
0.87
0.33
0.88
0.59
0.21
0.26
0.59
0.95
0.37
0.26
0.45
Number
of
Fish in
sample
70
115
353
1179
268
806
584
134
227
88
272
260
Data from U.S. Dept of Commerce, 1978.

Approximately 21% of the panelists did not report the
species of fish consumed.  Approximately 6.1% of the
panelists consumed other species of finfish.

Numbers are rounded to two decimal places.

The fish were sampled at source and are not samples of
the fish consumed by the panelists.
                             C-21

-------
figure of 27 g fish/day  as  the  upper  95  percent  of  fish

intake in the U.S. population;  (b) an average  value of 220

ng Hg/g for mercury  in tuna;  and  (c)  that  75 percent of

the fish consumption is  tuna, it  follows that  95 percent

of the population consumes  less than  4,500  ng  Hg/day as

methyl mercury from  tuna.   Contributions from  other fish

listed in Table  5 would  be  less than  1,000  ng  Hg/day assuming

an- average concentration of 100 ng Hg/g  fish.  Thus, it

seems, likely that 95 percent of the population will consume

Less than 5,000  ng Hg as methyl mercury  per day  from fish.

If- the averag.e, daily fish consumption in the United States

is taken, as: 17 g instead of 27  g  (Food Agric.  Organ. 1946-

196,6 quoted in Table 5.2 in the Natl.  Acad. Sci. 1978),

the; average methyl mercury  consumption from fish would be
                                                     i
3,000.-ng Hg./day/70 kg person.

     The U.S. Department of Commerce  Report  (1978)  did not

give estimates of, daily  intakes of mercury  from  fish.   The

report did-, however,  calculate  the probability of individuals

exceeding an average daily  intake of  30,000 ng Hg/70 kg

body weight.  It concluded  that,  under the  previous FDA

guideline of 500 ng  Hg/g fish,  99.89  percent of  the U.S.

population would have a  daily intake  of  less than 30,000

ng Hg/70 kg body weight.  The report  also  estimated that

99.87 percent would  be below this intake figure  under  the

current. F.D.A., guideline of 1,000 ng  fish.

     The National Academy of Sciences (1978) criticized

the. U.S. Department  of Commerce Report (1978)  because  "consump-

tion rates were  figured  at  less than  normal portions and

a.t minimum mercury levels."  They noted  that Weight WatchersR


                              C-22

-------
diet portions of fish are larger than the values of portions
of fish used in the U.S. Department of Commerce  (1978)  study.
McDuffie (1973) has reported intakes of mercury by 41 dieters
in New York State.  He reported that 25 percent consumed
between 9 and 16 jug Hg/day, the second quartile between
17 and 26,  the third quartile between 27 and 38, and the
highest quartile from 40 to 75 /ag Hg/day.
     Given the difficulties in accurately estimating dietary
j^ntakes of mercury, it is surprising that no comprehensive
surveys have been reported on blood concentrations of mer-
cury in representative samples of the U.S. population.
In McDuffie's study (1973) on Weight Watchers,R two of  the
41 dieters had maximum blood concentrations between 50  and
100 ng Hg/ml, which is consistent with a daily intake in
the range 50 to 100 ug Hg (using the model discussed in
the next section).  Gowdy, et al. (1977) reported that  9
of 210 subjects whose blood was collected for health reasons
showed total mercury levels above 50 ng Hg/ml, and four
were above 100 ng Hg/ml.  The form of mercury was not identi-
fied so that these high values may not have been due to
the intake of methyl mercury in fish.  However, the relation-
ship between inorganic and methyl mercury may be more complica-
ted than previously suspected because of a recent report
on dentists in which methyl mercury levels were found to
be five times higher in dentists than in controls not exposed
to inorganic mercury (Cross, et al.  1978).
     A bioconcentration factor (BCF) relates the concentration
of a chemical in water to the concentration in aquatic  organ-
                              C-23

-------
isms.  Since bioconcentration  tests  have  not  been  conducted

to steady-state for  all  four major groups of  aquatic  organisms

consumed in the United States, some  BCF values  have to  be

estimated.  A recent survey on fish  and shellfish  consumption

in the United States (Cordle,  et al.  1978)  found that the

per capita consumption is 18.7 g/day.  From the data  on

the 19 major species identified in the survey,  the relative

consumption of the four  major  groups  can  be calculated.

     Pentreath  (1976a) found a BCF of about 250 for the

muscle of plaice, whereas Kopfler  (1974)  obtained  a value

of about 10,000 for  oysters.   Since  these values are  0.21

ancf 0.33, respectively,  of the comparable values for  methyl

rneEcury, it seems reasonable to assume that the BCF values

for mercuric chloride should be 0.27  times  those for  methyl

mercury, on the average.
   !
                          Consumption         Bioconcentration
          group             (Percent)          	factor	

Freshwater fishes              12                    6,000

ga.ltw.ater fishes               61                      310

Saltwater molluscs             9                    8,000

S.altwater decapods             18                      310

Using the data for consumption the BCF for  mercuric chloride

is 'estimated to be 1,700 for consumed fish  and  shellfish.

     Tests with freshwater fish have  obtained BCF  values

for methyl mercury up to 8,400 for rainbow  trout  (Reinert,

et al> 1974), 20,000 for brook trout  (McKim,  et al. 1976),

and; 63,000 for fathead minnows (Olson, et al. 1975) for

a geometric mean of  22,000.  For saltwater  fish, a steady-

state BCF of about 1,200 was predicted for  the  plaice (Pentreath,


                               C-24

-------
1976a) and a value of 1,100 was found for skate  (Pentreath,

1976b) for a geometric mean of 1,150.

     Kopfler (1974) found that oysters achieved  BCF  values

up to 30,000 for methyl mercury, although many of  the  animals

died in the 60-day exposure.  No data are available  concerning

BCF values for decapods, but they would probably have  values

similar to those of saltwater fishes.

                          Consumption        Bioconcentration
     Group                  (Percent)         	factor	

Freshwater fishes             12                   22,000

Saltwater fishes              61                     1,150

Saltwater molluscs             9                   30,000

Saltwater decapods            18                     1,150

Using the data for consumption and BCF for each  of these

groups, the weighted average BCF for methyl mercury  is esti-

mated to be 6,200 for consumed fish and shellfish.

Inhalation

     In 1934, Stock and Cucuel reported average  air  concentra-

tions in the general atmosphere in Germany to be 20  ng Hg/m  .

Swedish and Japanese findings made 30 years later  were similar

(Fujimura, 1964; Eriksson, 1967).  Sergeev (1967)  reported

concentrations averaging 10 ng Hg/m  in the USSR.  McCarthy,

et al. (1970), working in Denver has documented  the  lowest

reported findings - 2 to 5 ng Hg/m .  In the San Francisco

area, concentrations were in the range of 0.5 to 50  ng Hg/m  ,

according to Williston (1968).

     Isolated "hot spots" having unusually high  concentrations

of mercury in the atmosphere have been reported  near suspected

points of emissions.  For example, air levels of up  to 10,000


                              C-25

-------
ng Hg/m  near  rice  fields  where  mercury fungicides had been



used and values  of  up to 18,000  ng  Hg/m  near a busy super-

   I

highway in Japan have been reported by Fujimura (1964).



Maximum air concentrations of  600 and 15,000 ng Hg/m  near



mercury mines  and refineries,  respectively,  were reported


by McCarthy, et  al.  (1970).  The highest reported levels
   5

of. mercury in  the atmosphere come from a study by Fernandez,



et. al.,  (1966)  who found values of up to 800,000 ng Hg/m3



in a village near a  large  mercury mine in Spain.  The remark-



ably high mercury vapor levels reported by these authors



indicate a need  for  further investigations into localized



high concentrations- of mercury in the atmosphere.



     Many of these  authors have  suggested that elemental



mercury vapor  is the predominant form of mercury in the



atmosphere (for  review, see Natl. Acad.   Sci., 1978).  Obser-



vations by Johnson  and Braman  .(1974)  at a suburban site



in Florida indicate  that approximately 60 percent of the



mercury in the atmosphere  is in  the form of  vapor, 1.9 percent



is; inorganic',  and 14.9 percent occurs as methyl mercury


compounds;.  Mercury  present in a particulate form accounted
                                                      i

for less than  one percent.  The  amount of mercury bound



to. particulate:s  s.eems to be related to area  of industrializa-



tion; and urbanization.  For example,  Heindryckx, et al.



(.1.974) found that aerosol  mercury levels corresponding to



remote background levels in Norway  and Switzerland were



ajs- low as: 0..02 ng Hg/m .   In1 a heavily industrialized area



of Belgium near  Liege the  aerosol levels noted were as high



as; 7.9- ng Hg/m .. In New York  City  (Goldwater, 1964)  and



Chicago. (B-rar, et al.  1969) , concentrations  of particulate-



bound; mercury  of up  to 41  and  14. ng Hg/m , respectively,



                               C-26

-------
were observed.  However, as pointed out by the National



Academy of Sciences (1978), considerable technical difficul-



ties present themselves in the attempt to measure particulate-


bound mercury; methods development and more reliable data



are needed in this area.



     The average concentration of mercury in the ambient



atmosphere appears to be about 20 ng Hg/m .  Assuming a



daily ventilation of 20 m  for the "standard 70 kg man,"



and assuming that 80 percent of the inhaled vapor, is retained,


the average daily retention should be 320 ng Hg/70 kg body



weight.  In urban and industrialized areas, it seems unlikely



that the mercury concentration in the atmosphere will regular-


ly exceed 50 ng/m , corresponding to 800 ng Hg daily retention.



The contribution of inhalation where people may be living


near "hot spots" is impossible to assess without further



information on air concentrations and the time of residence



of individuals in these areas.



     Occupational exposure to mercury vapor occurs in this


country (Smith, et al. 1970).  The current threshold limit



for occupational exposures is 0.05 mg Hg/m .  Assuming a



ventilation of 10 m  during the working day, a 5-day per


week exposure, and an average time-weighted air concentra-



tion which does not exceed 0.05 mg Hg/m , then the maximum
                                                 t


daily retention from occupational sources should not exceed


286 ;ug/70 kg for a seven-day week.



Dermal



     In general, absorption of mercury through the skin


is not a significant route of human exposure.  However,



under certain circumstances, such as occupational and medici-



nal exposure, it may be significant (see Absorption section).


                              C-27

-------
                        PHARMACOKINETICS


      The disposition  of  mercury in the body was reviewed


 •by a Task Group on Metal Accumulation (1973) and more  recent-
   i      '
 •ly .by :a -WHO Expert Committee (World Health Organ., 1976).


 i'Since the disposition of mercury in the body is highly depen-


 .•deht upon the physical and  chemical .forms of .this metal,


 ,-iit-.will .;be necessary  in  this .section to consider them  sepa-
   i                                                  t
irately.  Most information with regard to disposition in
   I
:;man ,and ^animals is available for methyl mercury compounds

   i               +                                   *
 .and inorganic  (Hg ) .complexes  of mercury ingested in the


 adiet -and :for ..the inhalation of •••mercury vapor.

      •'In general, insufficient  information is available on


-oithver compounds of mercury, except for the mercurial diuretics,


 »to allow .an extensive discussion.   .Because mercurial diuretics


-,;ar-e .now virtually obsolete  .for therapeutic use a complete


 review of this topic  is  not called for.
                                                      i

      •Nordberg  (197-6)  and the Task Group on Metal Accumulation


 .(.Ii973) have reviewed  evidence  for -suitable indicator media


;:for . me.thyl mercury.   The evidence reviewed below indicates


 •;t;hat :th.e blood .concentration of methyl mercury is a measure

.-.of -:'the .accumulation in the  body and the concentration  in


-the tar.get organ, the brain.   Urinary excretion is a poor


 .indicator o'f body bur,den as -most of the mercury is excreted

 .-via .the .feces.  The hair is probably the indicator medium


 of choice ..as 
-------
 as to whether the brain concentration exactly parallels
 the blood concentration in man.   Secondly, the blood con-
 centration could undergo a transient increase in individuals
 who have recently consumed a large amount of methyl mercury.
 The hair sample has to be analyzed in a special way and
 has to be collected,  transported, and stored under special
 conditions,  as discussed by Giovanoli and Berg (1974), to
 avoid the appearance  of artifacts.
      There is no satisfactory indicator medium for assessment
 of mercury vapor exposure, body  burdens, and concentration
 in the target organ.   It is the  practice in industry to
 use urinary  concentrations on a  group basis to give an indi-
 cator of exposures and body burden.  However, it seems likely
 that urinary concentrations may  reflect kidney levels rather
vthan concentrations in the target tissue of the brain.
      Since several exponential terms are required to describe
 the blood curve following a brief mercury vapor, multi-compart-
 ment pharmacokinetics are implied for man.  Thus, an isolated
 blood sample will not provide any information regarding
 exposure or  body burden.  Serial samples, however, may indi-
 cate the existence of a steady state or give limited informa-
 tion about recent exposure.  If  individuals are in steady-
 state, correlation between time-weighted average air concen-
 trations and blood concentration should be expected.  This
 was confirmed by Smith, et al. (1970) in chronically exposed
 workers.  The authors observed about a 49 microgram per
 100 ml increase -in the steady-state blood level for each
 1 mg/m  increase in the blood exposure concentration.
                               C-29

-------
     The same considerations with  regard  to  indicator  media


apply to inorganic mercury as  to inhaled  mercury  vapor.


It is. likely that urinary mercury  excretion  primarily  reflects


the accumulated amount  in kidney tissue.  Conclusions  about


the role of blood as  an  indicator  medium  cannot be  made,


since, little is known about the biological half-times  of


mercury in. the. blood  compartment versus other  tissues.


Absorption


     Methyl. Mercury and  Other  Short Chain Alkyl Mercurials:


No, quantitative information is available  on  the absorption


of the. short-chain alkyl mercurial compounds through human

   !
s.kin.-  However, cases of severe poisoning have occurred


fol.lowing  the topical application, for medicinal  purposes,


o,f. methyl mercury compounds (Tsuda, et al. 1963;  Ukita,


et al. 1.963; Okinata, et al. 1964; Suzuki and  Yoshino, 1969).
__

Although,,  in these cases, the  main pathway of  intake was


pr.ob.ably through skin,  the possibility of some inhalation


exposure- cannot be excluded.


     Likewise, no specific data are available  on  the inhala-


tion of alkyl mercurial  compounds.  The Task Group  on  Metal
   i                                                  :

Accumulation (1973) suggested  that the retention  of the


inhaled mercurials would probably  be on the  order of 80


percent..  These conclTusions were based mainly  on  the diffusi-


bility and the lipid  solubility of many of the compounds


of methyl mercury.  Furthermore,; no quantitative  information


Is: available on d.usts and aerosols of the alkyl mercurial


compounds.  Many of these compounds have  been  used  in  the


past as fungicides, resulting  in occupational  exposures


o£ workers.  Since some  of these occupational  exposures


                               C-30

-------
 have led to severe poisoning and death?S^!se)eihs" likely
 lung retention would be high, although  both  skin  absorption
 and gastrointestinal absorption might also have played a
 ,role._                      "•• '._• •.   ..,'_  ''   _' _'"'"' "'" '•':' . .
      Several quantitative measurements  have  been  made on
 the absorption of methyl mercury compounds in the gastro-
 intestinal  (G.I.) tract.  Experiments on. volun.teers by Aberg,
 et al.  (1969) and Miettinen  (1973). have demonstrated  virtually
 complete absorption in the G.I. tract whether the methyl
. mercury is administered as a simple  salt in  solution  or
 whether it is bound to protein.  The findings of: the  tracer
 studies have been confirmed  in observations  on.volunteers
 who ingested tuna fish for several days .(Turner,  et al...
 1974, 1975).  Shahristani.and cowprkers. (1976)/ in studies
 of the dietary intake of methyl mercury in homemade bread
 contaminated, with a fungicide, obtained results consistent
 with a high degree of absorption from the.diet.
      No quantitative information is  available on  the  other
 short-chain alkyl mercurials.  However, the  fact  that several
 outbreaks of poisoning have  occurred due to  the consumption
 .of homemade bread contaminated with  ethyl mercury fungi-
 cides suggests that this form of mercury is  also  well absorbed
 from the G.I. tract.               .
     .Age and sex differences in G.I., absorption of methyl
 mercury compounds have not been reported. However, the
 fact that very high blood concentrations of  methyl mercury
 were attained in infants who had ingested methyl  mercury
 solely  in their mothers' milk suggests  that  absorption in
 the very young is also substantial  (Amin-Zaki,  et al. 1974b).
                               C-31

-------
      Mercury Vapor and Liquid Metallic Mercury:   About 80
 percent  of  inhaled mercury vapor  is  retained as  evidenced
 by  observations of humans  (Teisinger and Fiserova-Bergerova,
 1965;  Neilsen-Kudsk/  1965a;  Hursh, et al.  1976).   Teisinger
 and Fiserova-Bergerova (1965)  proposed that the  vapor was
 absorbed across the walls  of the  bronchioles and  larger
 airways  of  the  lung/  but subsequent  evidence points strongly
 to  the alveolar regions as the predominant site of absorption
 into the blood  stream (Berlin,  et al.  1969).
      The importance of skin  as a  pathway for transport of
 metallic mercury into the  blood stream is  debatable.   Julius-
 berg (1901)  and Schamberg, et al, (1918)  indicated that
 appreciable skin absorption  of metallic mercury  takes place
 in  animals.   However/ the  possibility cannot be  excluded
 that some inhalation  'exposure also occurred in these  experi-
_
 ments.
      The gastrointestinal  absorption of metallic  mercury
 in  the liquid form is believed to be very  small.   Bornmann,
 et  al.  (1970) administered gram quantities orally to  animals,
 and Friberg and Nordberg (1973) calculated that  less  than
 0.01 percent of the administered  dose of metallic mercury
 was in fact absorbed.  Persons  have  accidentally  ingested
 several  grams of metallic  mercury and showed some increase
 in  blood levels (Suzuki and  Tanaka,  1971).   However,  there
 are many case reports in the literature of individuals con-
 suming,  accidentally  or otherwise, gram quantities of liquid
 metallic mercury and  the metal passing through the G.I.
 tract  into  the  feces  without any  ill effects.
                               C-32

-------
     Salts of Inorganic Mercury:  No quantitativ'&-'i^ipirm9't'i-.0.n'
is available on the absorption of mercury  in  the  form of
                      _L 1.                    .'.-',.,
inorganic mercuric  (Hg  ) salts by human  skin.   However,
solutions of mercuric chloride have been  shown  to be absorbed
by guinea pigs; five percent of the mercury  in  a two percent
solution of mercuric chloride was absorbed across the intact
skin of these animals over a five-hour  period  (Friberg,
et al. 1961; Skog and Wahlberg, 1964).   If such a rate of
penetration applied to  human skin, one  might expect substan-
tial absorption of mercuric chloride  salts in man.
     Information on the pulmonary deposition and absorption
of inorganic mercury aerosols is lacking  except for the
experimental work on dogs by Morrow,  et al.  (1964).  This
group reported that 45  percent of mercury administered as
mercuric oxide aerosol  having a mean  diameter of 0.16 urn
was cleared within 24 hours; the remainder cleared with
a half-time of 33 days.
     Rahola, et al. (1971) reported findings on the G.I.
absorption of inorganic mercury given to  ten volunteers.
Eight of the volunteers, five males and three females, received
a single dose of mercuric nitrate bound to calf liver protein,
containing approximately 6 ug of inactive mercury per dose.
The other two volunteers received an  acid solution of mercuric
nitrate.  During the four to five days  following treatment,
an average of 85 percent of the dose  was  excreted in the
feces; urinary excretion was only 0.17  percent  of the dose.
These findings suggest  that G.I. absorption  of  inorganic
-.-,-,-
mercury by humans is less than 15 percent, which correlates
with studies on experimental animals  (Clarkson, 1971).
                              C-33

-------
Experiments on animals indicate that G.I. absorption is
greater in suckling animals than in mature ones  (Kostial,
et al. .1978).
     Other Compounds of Mercury:  The aryl and alkoxyaryl
mercurials are used as fungicides and slimicides, and as
such occupational exposures to these compounds probably
still occur.  To what extent these mercurials reach the
water supply is not known.  In general/ the aryl mercurials
are well absorbed from the G.I. tract, as evidenced by animal
experiments (Clarkson, 1971).  Most classes of these organo-
mercurial compounds undergo rapid conversion to  inorganic
mercury in body tissues.
                              C-34

-------
Distribution and Metabolism
                                                •r.

     Methyl Mercury and Other Short-Chain Alkyl Mercurials:


  Details on the distribution and retention of methyl mercury


in man and animals were reviewed by Friberg and Vostal  (1972),


by the Task Group on Heavy Metal Accumulation  (1973), and


by a WHO Expert Committee (1976) .  The general picture which


emerges is that methyl mercury compounds, after absorption


from the G.I. tract, distribute readily to all tissues  in


the body.  Unlike inorganic mercury, large concentration


differences in various tissues are not seen.  Methyl mercury


is characterized by its ability to cross diffusion barriers


and cell membranes without difficulty.


     Tracer studies in volunteers have revealed that about


five percent of the ingested dose is deposited in the blood


compartment after tissue distribution is completed.  About


90 percent of the methyl mercury in blood is associated


with the red blood cells.  Thus/ the red cell to plasma


ratio is between 10:1 and 20:1.  The mercury in the red


blood cells is almost entirely  (more than 90 percent) in


the form of methyl mercury compounds.  However, in plasma


approximately 25 percent can be in the form of inorganic


mercury that has been produced by cleavage of the carbon


mercury bond (Bakir, et al. 1973).  The rate of decline


in blood concentration of methyl mercury after cessation


of exposure can be well described by a single biological


half-time as evidenced by both tracer experiments in volunteers


and also in people who had ingested methyl mercury in substan-


tial amounts from.either fish or contaminated food  (see


Table 6).  The tracer experiments reveal a half-time of


                              C-35

-------
approximately  50  days.   However,  the  range  of  half-times


reported  in  both  tracer  experiments and  in  people  having


substantial  exposures covers  a  very wide range.  Whether


this range of  values  is  due to  individual differences  or


to experimental or  observational  inaccuracies  in the measure-
                         >„

ments  is  not clear.



     Based on  observations in animals, the  entry of the


mercury into the  brain is delayed  by  a few'  days as compared


to entry  into  other tissues (Norseth  and Clarkson, 1971).


According to observations on  volunteers,  the amount trans-


ferred to the  head  region following the  ingestion  of a single


dose of radioactive tracer is about 10 percent of  the  body


burden after tissue distribution  is complete.  However,


only three subjects were involved  in  this study  (Aberg,
                      i-

et al.  1969).  There is a great need for more data which


would allow estimation of the .amount  of  mercury that enters


this critical  organ (the brain) .-   In  man, the brain to blood


ratio is  in a  range of 5:1 or 10:1.   The biological half-


time of methyl mercury in the brain is not  well described


in man but the observations by  Aberg, et al.  (1969) of three


volunteers indicate a half-time in roughly  the same range


as that observed  in blood and in the  whole  body  (see Table


6).  Whether or not the  half-times in brain and blood  are


identical is an important consideration  in  the decision


to use blood as an  indicator  medium for  brain concentrations.


     The concentration of methyl mercury in other  tissues


such as muscle', liver, and kidney  usually does not vary


by more than a factor of 2 or 3, with the highest  concentra-


tions being found in the kidney cortex.   In muscle, the



                              C-36

-------
                                           TABLE  6

                                 Mercury Intake and Clearance
Clearance half-times (days)










o
i
co
«J
NO. Of
subjects
5
15

5
5

16

48

Hg intake
C/ug/kg/day)
tracer :
tracer

up to 5
up to 5

up to 50

up to 50


Body
70
76
(52-93)
—
— . .

• - . —

—


Blood
_._
50

— .
seea
(58-164)
65
(45-105)
—


Hair References
s -'•
— Aberg, et al. (1969)
• — Miettinen (1973)
••' ' ' • .
(33-120) Birke, et al. (1967)
Skerfving (1974)
' - '-"' • • ' '•.... ::
— . Bakir, et al. (1973)
K
72° Shahristahi & Shihab (1974)
(35-189)
One person had a biological half-time of 164 days.  The other  four  were  in the  range of
  58-87 days.

 The data were distributed bimodally.  One group accounting  for  89% of the samples  had
  a mean value of 65 days and the other group had a mean  value of 119 days.

-------
mercury is usually almost entirely in the  form of methyl
mercury but in liver and kidney a substantial proportion
can be present as inorganic mercury.  Most of this evidence
is based on studies using animals. Autopsy data  in Iraq
indicate a substantial proportion present  as inorganic mercury
in liver (Magos, et al. 1976).
     Methyl mercury is readily transferred from  mother to
fetus across the placenta.  At birth the concentration in
the umbilical cord or infant  blood is usually slightly higher
than that observed in maternal blood.  In  observations on
women having normal pregnancies and on a low to  moderate
fish intake, Tejning (1970) reported that methyl mercury
in the fetal blood cells was  about 30 percent higher than
in the maternal cells.  Suzuki, et al. (1971) confirmed
the finding of higher fetal blood concentrations.  The studies
on the outbreak of methyl mercury poisoning in Iraq  (Bakir,
et al. 1973; Amin-Zaki, et al. 1974a, 1976) also showed
that methyl mercury was readily transferred across the placen-
ta, resulting in higher concentrations in  fetal  blood at
the time of delivery.  Apparently the differences between
fetal and maternal blood are  due to differences  in concentra-
tion in the red blood cells rather than to differences in
plasma concentrations.
     Methyl mercury is secreted in mother's milk.  The studies
of the Iraqi outbreak revealed the close correlation between
maternal milk and blood concentrations, with the milk concen-
tration on the average being  about 5 percent of  the  simul-
                               038

-------
taneous blood concentration (Bakir, et al. 1973).  About
40 percent of the mercury in milk was found to be in the
inorganic form.  Skerfving (1974), in a study of 15 lactating
females following intake of methyl mercury from fish, also
noted a correlation with blood concentrations but found
a smaller percentage (approximately 20 percent) of mercury
in the form of methyl mercury in the milk.
     Mercury is accumulated in head hair after exposure
to methyl mercury compounds. , A variety of observations
(see Table 7) indicate that the hair to blood concentration
ratio is about 250:1 with considerable variation from one
study to another.  Mercury is accumulated in the hair at
the time of its formation and, thus, in freshly formed hair,
the concentration in hair is proportional to that in blood.
Once incorporated into the hair sample the concentration
of mercury is stable and thus, as the hair is examined longitu-
dinally, a history is obtained of previous blood concentrations
(Clarkson, et al. 1976).  Hair grows at approximately 1
cm per month (Shahristani and Shihab, 1974) so that the
measurement of each 1 cm segment corresponds to the average
blood concentration during a particular month-  The hair
is therefore a very useful medium to recapitulate past ex-
posures as well as to "give information on current exposure
to methyl mercury.  An example of the close parallel between
concentration in hair and blood is shown in Figure 2 (Amin-
Zaki, et al.  1976).
     Methyl mercury is metabolized to inorganic mercury
in animal tissues (Gage, 1961; Nors.eth and Clarkson, 1970).
                                C-39

-------
                      BOTH
                       MOTHtt'MC-OO
                                  o MQTHfIfS 81000
                                  4 MOTHERS HAIR
                                  * MOTHEfS MUK
                                  • BAST'S 81000
'3009
2000

1000

200


200

 100 "*

 50 |


• 20 5

. „ I

•  3 i
    Figure 2.  Concentration of total mercury in 1  cm  segments
    of  sample of mother's  hair, whole blood, and milk,  and baby's
    blood (postnatal exposure).  Concentrations in  milk and blood
    are plotted according  to dates of collection.   This figure
    is  taken from Figure 4  of the report of Amin-Zaki,  et al.  1976
                                    TABLE 7

Relationship between Concentrations of Mercury in Samples  of Blood and Hai;
       in  People having Long-term Exposure to Methyl Mercury from Fish
No. Of
subjects
12
51
50
45
60
0
0
0
0
0
Whole blood
(x)
.004
.004
.005
.002
.044
(mg/kg)
- 0.
- 0.
- 0.
- 0.
- 5.
65
11
27
80
5
Hair
(y)
(mg/kg)
1 -
1 -
1 -
20 -
1 -
180
30
56
325.
142



Linear regression
y =
y =
y =
y =
y =
280x-l.
230x+0.
140X+1.
260x+0
230x-3.
3
6
5

6
This Table  is adapted from  Table  1 in the report
of the WHO,  1976.

                                     C-40

-------
In man, conversion to inorganic mercury is an important



process in excretion, as shall be discussed later:



     Mercury Vapor and Liquid Metallic Mercury:  Approximately



2 percent of an inhaled dose of radioactive mercury vapor



was found to be deposited in 1 liter of whole blood after



tissue distribution was complete  (Hursh, et al. 1976).



The concentration in the red blood cells of these volunteers



was higher than that seen in plasma.  The half-time in blood



was estimated to be about 4 days, accounting for at least



60 percent of the mercury deposited in the blood volume.



     An accidental mercury vapor exposure of a family has



supplied some additional information concerning half-times



(Figure 3).   The major portion of the exposure probably



occurred within a half-hour peri'od with a smaller protracted



exposure over the duration of an evening.  It appears that



there was an early rapid decline over the first few days



post exposure, and by about days five to seven, the mercury



in blood was decreasing with an approximate 15-day half-



time which was maintained for the remainder of the first



month's post exposure.  Another family's exposure to mercury



vapor involved a husband and daughter who were exposed for



six to eight months in the home.  The wife had experienced



a prior exposure for about 18 months in her workplace.



Samples of blood were collected starting about one month



after cessation of exposure.  Therefore, an early and rapid



fall in blood conentration due to short half-time components



was missed.   The blood concentration of mercury in the wife



declined, with a half-time of 30 days.  The other two family






                              C-41

-------
              160-1
             120-
              80-
n


a
o
o
              40-
              0-r
             200-
          ee
          ui
          z

          **  30
          C  3°
          ce
          O
          Z
          -  20H
                 25   30

                  Oct.
                    9   14   19

                   November
24
Figure 3.  The  fall  in mercury concentrations in blood in two

adult females following a brief exposure (less than 3 hr) to

mercury vapor.   Upper  graph has a linear scale on the ordi-

nate.  The lower graph has a logarithmic scale and curve

stripping procedures were used to estimate a component with

the different half-time (slow component, 14.9 days; fast com-

ponent, 2.4  days).   Data from Clarkson, 1978. (unpublished data)
                                 C-4.2

-------
members had longer half-times but their blood levels were
sufficiently low that dietary mercury might have influenced
the results.
     Evidence from animal experiments and from  isolated
suspensions of human blood indicate that mercury vapor,
once absorbed into the bloodstream, can undergo oxidation
to divalent mercury (Hg  ).  The red cells are  an  important
site of this oxidation process, which is believed  to be
mediated by the hydrogen peroxide catalase pathway  (for
review, see World Health Organ. 1976; Clarkson, et  al. 1978).
However, the oxidation in the red blood cells is not suffic-
iently rapid to prevent some of the dissolved mercury vapor
from persisting in the blood stream for sufficient  periods
of time to reach the blood-brain barrier.  Here it  is believed
to rapidly cross into brain tissues where it is again subject-
ed to oxidation processes.  A scheme for the pathway of
inhaled mercury vapor reaching the brain is given  in Figure
4.  Hursh, et al. (1976) made regional body counts  on volunte-
ers who had inhaled a tracer dose of radioactive mercury
vapor.  They found that approximately seven percent of the
inhaled dose was absorbed into the head region  following
completion of tissue distribution.  The half-time  in the
head region was found to be 21 days  (Table 8).  This half-
time was considerably shorter than that seen in other tissues
in the body with the exception of blood.
     The main site of accumulation of mercury in the body
after inhalation of mercury vapor is the kidney.   In fact,
animal experiments indicate that as much as 90  percent of
                              C-43

-------


Figure 4.  A diagrammatic  representation  of  the  pathway of in-
halgd mercury vajj>or  (Hg  )  to  the  brain.   The oxidation process
(Hg  —	^ Hg   )  is depicted  as occurring  in  the  red blood
cells and brain  tissue.++0xidation  also occurs  in other areas.
The ligands to which Hg    attaches  have not  been identified
(depicted as S and X) but  sulfhydryl groups  are  suspected to
be involved.  Taken from Clarkson (1974).
                             .;-44

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                                          TABLE 8

                     Summary of Half-Times'o£ Mercury  in Human Tissues

Tissue
Exposure
Conc~
Duration
First Component
% deposited
mg/m





0
i
*>•
tn

Blood3
Bloodb
Bloodb
Lung°
Kidney0

Head0

Whole Body0
0.
0.
0.
0.
o.

0.

0.
1
1
05
1
1

1

1
20
min
few hours
60
90
T 1/2
Second Component
% deposited
days
4
2
.0
.0
months ? ?
20
20

20

20
min
min

min

min
100
100

100

100
1
64

21

58
.7
.0

.0

.0
not
10
100
not
not

not

not
detected


detected
detected

detected

detected
T 1/2
days

20
|0






|* Cherian et al., 1978
D Hursh, et al.  (1976).
  Observations made at Rochester but not published.  For details,  see  text,

-------
 the  total  body  burden can be  found  in  kidney tissues  (Rothstein



 and  Hayes,  1964).



     Mercury  can penetrate into  the  fetus  after  maternal



 exposure to mercury  vapor.  This  rate  of transfer  appears



 to be considerably greater than  that seen  for  the  inorganic



 species of mercury  (Clarkson,  et  al. 1972).   However,  no



 published  information is  available with regard  to  human



 exposures.  Observations  on a  family accidentally  exposed



 for  a brief period of time to  mercury  vapor  indicated  that



 the  mercury concentration at delivery  of the baby  was  the



 same as that  in the  mother.



     A summary of the estimated  biological half-times  of



mercury in the body  following  exposures to mercury vapor



 is given in Table 8.   Most  of  the information  in this  table



comes from tracer" experiments  of  Hursh, et al.  (1976)  and



 from unpublished observations  of  people who  were accidentally



exposed for brief periods of time.  The whole body half-



 time and the  half-time in kidney  seem  to be  approximately



the  same as that of  methyl  mercury in  man.



     Salts of Inorganic Mercury:  Studies using  a  variety



of animal species have shown that, in  general,  the distribu-



tion of mercury after  doses of mercuric salts or inorganic



mercury bound to protein  is similar to the distribution



observed after exposure to  mercury vapor (for review,  see



Clarkson, 1972a,b; Friberg  and Vostal, 1972).  However,



there are important  differences.  The  red cell  to  plasma



ration has been reported  to be 0.4 in  humans exposed to



a tracer dose of Hg"1"1" (Rahola, et al.  1971)  whereas the



amount in the red cells is  considerably higher  after exposure



                               C-46   :''. '

-------
to mercury vapor (Cherian, et al.  1978).  The most dramatic
differences lie in the ability to penetrate across the blood-
brain and placental barriers.  Relatively small amounts
of the mercuric ion penetrate the brain or the fetus follow-
ing exposure to inorganic salts as compared to mercury vapor
and alkyl mercury compounds.  Jogo (1976) has reported that
the blood-brain barrier of suckling rats i.s more permeable
to inorganic mercury than' that of adults.
     Inorganic Mercury Accumulates in the Kidneys:  Animal
experiments have shown that as much as 90 percent of the
body burden can be found in this organ.  Inorganic mercury
has the ability to induce the synthesis of metallothionein
or metallothionein-like proteins in kidney tissue  (Piotrowski,
et al. 1974a, 1974b) .   This ability is shared with inhaled   »
mercury vapor (Cherian and Clarkson, 1976).
     The retention of mercury by five human volunteers after
a single dose of inorganic mercury has been reported by
Rahola, et al.  (1971).  The whole body biological half-time
averaged 45 days and was significantly greater than the
biological half-time observed for plasma  (24 days) or for
the red blood cells (28 days).  Rahola, et al.  (1971) reported
that 0.2 to 0.4 percent of the ingested dose was found in
the blood volume one day after dosing.
     Other Compounds of Mercury:  The conversion of organo-
mercurial compounds to inorganic mercury results in a pattern
of distribution that eventually is similar to that obtained
                              C-47

-------
after  exposure  to  inorganic  salts.  The kidney  is  the main



organ  of  accumulation  in  all cases.



Excretion



     Methyl Mercury  and Other Short-Chain Alkyl Mercurials:



The excretion of mercury  from the body in humans exposed



to methyl mercury  occurs  predominately by the fecal  route.



Less than ten percent  of  excretion occurs in the urine.



The form of mercury  in feces is almost completely  the inorgan-



ic form  (Turner, et  al. 1974) and about 90 percent of the



mercury in urine is  also  inorganic (Bakir/ et al.  1973).



These  observations indicate that, in man, an important step



in the excretion process  is the cleavage of carbon - mercury



bond.



     The site of the cleavage of this carbon-mercury bond



in the body is not known.  Animal experiments indicate there



is a substantial biliary  secretion of methyl mercury raising



the possibility that biotransformation to the inorganic



form might be affected by micro flora in the gut (Norseth



and Clarkson, 1971).



     Mercury Vapor and Liquid Metallic Mercury:  Urine and



feces  are the main pathways of excretion after exposure



to mercury vapor, although exhalation of vapor and excretion



in saliva and sweat may contribute (Lovejoy, et al.  1974;



Joselow, et al. 1968).  Animal data indicate that, shortly



after  exposure, the G.I.  tract is the predominant pathway



of excretion but as  the kidney becomes more and more the



predominant site of  storage of mercury, urinary excretion



takes over (Rothstein  and Hayes, 1964).  In humans,  following



a brief exposure, urine accounted for 21 percent of  the
                       i




                              C-48

-------
total urine and fecal excretion, but after a long term occupa-
tional exposure, urine contributeded 58 percent  (Table 9).
Tracer experiments using human volunteers indicated that
the specific activity of mercury in'urine was unrelated
to the specific activity -;in.plasma  (Cherian, et al. 1978).
This observation suggests that urinary mercury originates
from a-large pool of mercury in the kidney rather than from
glomerular filtration of plasma mercury.
     Approximately seven percent of an inhaled dose of mercury
vapor was shown to be excreted in the expired air of humans.
The great majority of this came out within seven days and
comprised 37 percent of the first week's excretion  (Table 9).
     .Quantitative information on the excretion via .sweat
and saliva is not available.  In workers experiencing profuse
perspiration, amounts of mercury excreted in the sweat may
exceed those of urine (Lovejoy, et al. 1974) .
     High individual variation and great day-to-day fluctu-
ation were the principal features of urinary mercury excretion
by workers under similar exposure conditions (Jacobs, et
al. 1964).  Copplestone and McArthur  (1967) found no cor-
relation between urinary excretion and air concentrations.
They noted that some individuals excreted extremely large
amounts of mercury, some in excess of 1,000 /ig/1  without
apparent ill effects.  Their own findings and their review
of the literature (Jacobs, et al. 1964; Neal, et al. 1941)
led Copplestone and McArthur (1967) to propose that "mercu-
                              C-49

-------
                            TABLE 9

           Parameters of Excretion of Mercury in Man
              Following Exposure to Mercury Vapor.
Excretion
Medium
Urine
Urine
Feces
Feces
Expired air
Exposure
Cone. 3 Duration
(rag Hg/m )
0.1 20 minutes
0.05 - 0.2 (years)
0.1 20 minutes
0.05 - 0.2 (years)
0.1 20 minutes
Percent of
Total Observed
Excretion
13a
58b
49a
42b
37a
a
et al. 1976;  Cherian, et al. 1978).

Combined urine and 'feces  (Tejning and Ohman, 1966).
                              C-50

-------
rialism might be due to an inability to excrete  absorbed
mercury rather than simply to exposure."
     Piotrowski, et ail. (1973) observed workers  following
exposure to mercury vapor, arid reported that  urinary  excretion
could be described'by a two-term exponential  equation equi-
valent to-half-times at 2 and 70 days.  The authors claimed
that individual variations in urinary excretion  are minimized
when urine samples are collected at the same  time  each morning.
     Lundgren, et al.  (1976), Smith, et al.  (1970), and
Hernberg -and Hassanan  (1971)  have reported generally  similar
relationships between steady-state urinary excretion  and
blood levels.  Averaging their results, one would  expect
a 0.06; mg/r  "increase in 'the urinary excretion rate for
each .10"0 ug/100 ml change in the blood mercury level.   These
results can be combined with the data on blood levels versus
exposure concentration 'reported by Smith, et  al.  (1970)
to predict a '2.9 mg/1 change in the urinary excretion for
each 1 mg/m  change in the time-weighted air  concentration.
     Tejriing and Ohman (1966) cited steady-state urine and
fecal excretion rates which can be interpreted to  mean that
urinary excretion will account for approximately 57 percent
of combined urinary and fecal excretion when  the exposure
concentration, is between 0.05 and 0.2 mg/m .  When these
excretion rates arer compa'red to those predicted  above a
discrepancy of a :factor of two to three is found1;  with the
predicted rates being greate'r than those observed  by  Tejriing
and Ohman (1966).
                              C-51

-------
     Several factors might contribute to the daily vari-
ability of urinary mercury concentrations.  Daily changes
in urinary specific gravity, problems with analytical metho-
dology, volatilization of mercury from urine (Magos, et
al.  1964) , absorption of mercury to glassware, the diffusion
of mercury out of plastic bottles, and the entrainment of
mercury into the particulate fraction of urine, all make
the analysis of urinary mercury extremely difficult (Greenwood
and Clarkson, 1970).
     In conclusion, although correlation of urine mercury
concentrations with blood or time-weighted air concentration
may yield consistent results when the data are averaged
over large groups of people, no explanation is at hand for
the large fluctuations in daily excretion by individuals.
However, few longitudinal studies have been made, and all
measurements to date on exposed workers with one exception
have measured concentrations of total mercury.  Recently,
Henderson and co-workers  (1974) have pointed to the importance
of identifying chemical forms of mercury in urine.  They
concluded that dissolved elemental vapor in urine might
be a better indicator than total mercury.
     The exhalation of mercury in expired air is a recent
finding in humans  (Hursh, et al. 1976).  The short half-
time reported by these workers following brief exposure
to the vapor suggests that mercury in expired air would
indicate only recent exposure.  However, experiments on
animals given mercuric salts (Clarkson and Rothstein, 1964;
Dunn, et al. 1978) reported a close correlation between
                                C-52

-------
the rate of exhalation and the body burden of divalent mercury
    *) .   During chronic exposures to mercury vapor, the
body burden of Hg   may reach levels at which reduction
of this form of mercury can make a significant contribution
to loss by exhalation.  Thus, sampling of expired air at
appropriate times after inhalation of vapor may provide
information on both recent and long term exposure.
     Salts of Inorganic Mercury:  Studies by Rahola, et
al. (1971) on volunteers who ingested tracer doses of inorganic
mercury revealed that urine and fecal excretion were approx-
imately equal .after the unabsorbed oral dose was cleared
by the G.I. tract.  The whole body half-time of 45 days
observed in these volunteers is consistent with excretion
in urine and feces, amounting to a total of 1.5 percent
of the dose per. day.
     It is possible that urinary excretion could be increased
by kidney damage.  For example, Cember (1962) reported that
cytotoxic doses of inorganic mercury could lead to desquamation
of renal tubular cells, resulting in a sharp increase in
mercury excretion.  Magos (1973) has reviewed other studies
where agents producing kidney damage leading to desquamation
of cells cause an increase in urinary mercury excretion.
     Other Compounds of Mercury:  Retention .half-times of
the aryl and alkoxy-aryl mercurials in man are generally
not known.  Their rapid conversion to inorganic mercury
would suggest that their half-times would not exceed those
reported in volunteers discussed above.  The mercurial diuretics
generally have half-times considerably shorter than that
                                C-53

-------
reported  for  inorganic  mercury  because of  the  rapid
excretion of  the  intact mercurial.
     Mathematical Models of Accumulation of Methyl Mercury
in Man:  The  body will  continue to  accumulate  methyl mercury
so long as  intake is greater  than excretion  until a steady-
state is obtained where intake  and  excretion balance.  A
common way  to describe  the progress of accumulation in the
body is in  terms of the biological  half-time.  This concept
is useful,  provided that the  processes of  transport and
distribution  in the body occur  more rapidly than  the elimina-
tion step.  Thus, the single  biological half-time can then
describe the decline in not only the amount in the body
but also in the concentration in various tissues.  As pointed
out by the  WHO Expert Committee (1976), if tissue compartments
retain mercjary with widely differing retention half-times,
then the whole body biological  half-time would not be useful
and could give misleading information toxicologically.
     However, this evidence indicates that the rate of decline
of mercury  in the whole body  and in various tissues including
the target  organ can be described by a single  biological
half-time.
     The WHO Expert Committee has summarized the mathema-
tical expressions relating daily intake to biological half-
time and accumulation in man. These derivations are quoted
below.
     In cases where the elimination of a metal such as methyl
mercury follows a single exponential first order  function,
the concentration in an organ at any time can  be  expressed
by the following equation:
                              ' C-54  '  •''.-'• -.

-------
          c =C  e~b-fc                              „.,,,:,,,•..,,,.,,...
          c  *-o*e    ...........  *  *  *  •••••'--'"•  •
          . . .(1)
where     C =concentration in the organ at  time t
          C concentration in the organ at  time p
          b =elimination constant, and
          t =time.
The relation between the elimination constant and the biolo-
gical half-time is the following:
          T =ln2/b
where:    T =biological half-time, and
          In2 (natural lo garithm of 2) = 0.693
     If data on exposure and absorption of  the metal are
known, then it is possible to predict the body burden of
the metal at constant exposure over different time periods.
If a constant fraction of the. intake is taken up by a certain
organ,*' the accumulated amount in that organ can also be
calculated.  The  following expression gives the accumulated
amount' of metal in the total body  (or organ):
          A =(a/b) (l-exp(-b.t) ) . . . .  .  .  .  .  .  . . .  .
          . . . .  (2)
where     A =accumulated amount, and
          A =amount taken up by the body  (or  organ)  daily.
At steady-state the following applies:
          A =a/b  ...............  ......
     In other words, the steady-state  amount in the -body
 (or organ) A is proportional  to  the  average daily intake
and inversely proportional  to the  elimination rate.  The
latter point will be discussed in  a  later  section in relation
to human hazards, as large  individual  variations in elimi-
nation rates imply large individual  variations in steady-
                                 C-55

-------
            1000
                                            Exposure pwidd

                                            Body burdtn & blood

                                            KUir
                                                     7.0
                                                        0
                                                        E

                                                     •1JJ -
Figure 5.  The  changes in the body burden  and  hair and blood
concentrations  of mercury during constant  daily  exposure
(shaded area) and after exposure.  This calculation was
based on a daily  intake of 10 /ag of methyl mercury during
the exposure period,  an elimination half-time  of 69 days,
and a hair to blood concentration ratio of 250.   This
figure is taken from Figure 1 of WHO  (1976).
                               056

-------
state body burden, even in people having the same average
daily intake.
     Equations (1), (2), and  (3) are illustrated graphically
in Figure 5.  During the period of steady daily intake  (assumed
to be 10 jug/70 kg body weight) , the amount in the body  rises
rapidly at first, reaching half its maximum  (steady-state)
value in a time equivalent to one elimination half-time
(assumed to be 69 days for methyl mercury in man).  After
an exposure period .equivalent to five elimination half-times
(approximately one year for methyl mercury), the body is
within three percent of its final steady state value.  The
steady-state body burden is 100 times the average daily
intake assuming an elimination half-time of 69 days.  Upon
cessation of exposure, the body burden will immediately
begin to fall, following an exponential^curve that is an
inverse  .mage of the accumulation curve.  Thus the body
burden will have returned to within three percent of pre-
exposure values in five half-times.
     In this example,  it is assumed that the hair-to-blood
ratio is constant and equal to 250 and that one percent
of the body burden is found in 1 liter of blood in a 70 kg
man.
     Equation 3 is useful in that it predicts a relationship
between long-term dietary intake and the concentrations
of mercury in such indicator media as blood and hair.   It
is thus possible to test the predictive value of equation
3 by carrying out dietary studies on exposed populations
and measuring concentrations of methyl mercury in blood
                              C-57

-------
and hair.  A prediction of equation 3 is that once  the  indi-
vidual has attained steady-state, the concentration in  blood
should be directly proportional to the average daily intake.
This prediction was confirmed in a study by Skerfving  (1974)
in a group of fish eaters in Sweden.  Results of Skerfving's
study, along with studies on other fish eating populations,
are summarized in Table 10.  In some cases, observations
were made on concentrations in hair, and in others,  measure-
ments of blood concentrations were made.  All have  been
converted into blood concentrations for comparative purposes.
Furthermore, it is possible to predict the steady-state
concentration in blood from a given dietary intake  with
the kinetic parameters given in the studies by Aberg, et
al. (1969), and Miettinen (1973) on volunteers.  This estimate
is also given in Table 10.  The calculation involves the
assumption that 95 percent of the methyl mercury was absorbed
from the diet, that one percent was distributed in  1 liter
of blood, and that the biological half-time in blood was
approximately 50 days.  In general, the factor relating
the steady-state blood concentration to the average daily
intake (the coefficient of x; Table 10) varies from a value
of 0.3 to 1.0.  The low values for this coefficient have
been attributed to the difficulty of an accurate estimate
of dietary intake and to the possibility that in some of
the populations studied the individuals had not attained
a true steady-state.  Nevertheless, equation 3 seems to
be useful in that it allows comparison of the results of
various types of studies, including both exposed populations
and volunteers.  A recent study of five volunteers  ingesting
                              C-58

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                            TABLE  10
No. of
subjects
h
6+26°
139+26°
6+14^
725C
22
15

Time of
exposure

years
years
years
years
years
single tracer
dose
Ave. Hg. intake
Oug/day/70 kg B.W.)
(x)
0-800
0-400
0-800
0-800
0-800


Steady blood
concentration
(ng/ml)
(y)
y=0.7x+l
y=0.3x+5
y=0.8x+l
y=0.5x+4
y=0.5x+10

y=1.0x
For details of these calculations, see text.
is adapted from Table 3 of WHO (1976).
This table
None or low fish consumers.

Estimated from data on hair concentrations and daily intake.
The hair to blood concentration ratio was assumed to be
250 and the average body weight of the population under
study to be 60 kg.
                             C-59

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contaminated freshwater  fish yielded a coefficient of about
0.8, close to the  tracer prediction of 1.0  (Kershaw, et
al. 1978).  Quantitative accuracy in relating dietary intake
to steady-state blood levels is of considerable importance
to estimates of hazard to human health from dietary intake
of methyl mercury, as will be discussed later.
     Thus far, the discussions have employed average values
for various parameters used in mathamatical modeling of
accumulation of methyl mercury in man.  In fact, there are
substantial differences. The biological half-time in man,
as indicated in Table 6, actually varies over a wide range
of values.  Shahristani and Shihab (1974) have published
the observation that there is a bimodal distribution of
biological half-times as calculated from analysis of hair
samples in the Iraqi outbreak.  As shown in Figure 6, these
authors found that the majority of a population of 48 people
studied had half-times distributed around the normal value
of about 65 days, but about nine percent of the population
had a significantly different distribution of half-times,
averaging about 119 days.  Greenwood, et al.  (1978) have
noted that the half-time in blood of lactating females (average
42 days) is significantly lower than that of non-lactating
adult females (average 74 days).  The excretion of methyl
mercury in milk is not sufficient to explain the reduced
biological half-time in blood of lactating females.
     Experiments on mice by Doherty, et al. (1977) have
revealed that methyl mercury is not eliminated from mice
throughout their suckling period.  Observations by Landry,
                              C-60

-------
              20
40      60       80      100

  Biological Half-Life. Days
120
Figure 6.  Population distribution curve  of  methyl mercury
(Shahristani  &  Shihab,  1974).  For details,  see text.
                             C-61

-------
et al.  (1978) revealed  that changes in the diet of mice
can also lead to large  changes in the biological half-time
of methyl mercury.
     There are  important  species differences in the kinetics
and distribution of methyl mercury.  For example, the blood
to plasma ratio, which  is about ten to one for man and other
primates, is as high as 300 to 1 in rats.  The blood to
brain ratios exhibit substantial species differences with
man and other primates  having a ratio of about one to five,
most laboratory animals having ratios of one to one, and
the rat having a ratio  of ten to one.  The biological half-
times may be as short as  seven days in the mouse or as high
as 700 days or more in  certain marine species  (for review,
see Clarkson, 1972a).


                           EFFECTS
     Greatest emphasis  will be placed on those effects occur-
ring at the lowest levels of exposure to mercury and to
the target systems that suffer effects most hazardous to
the animal at the lowest  exposure.  Greater weight will
be given to human data  when reliable; otherwise, animal
data will be used.
     This section gives separate treatment to the physical
and chemical forms of mercury that are toxicologically dis-
tinct.  The short-chain alkyl mercurials, mercury in the
zero oxidation state (mercury vapor and liquid metallic
mercury) and the compounds of divalent inorganic mercury
(Hg  ) will receive the most attention as these are the
forms of mercury to which man is most frequently exposed.
                                062

-------
Acute, Sub-acute,  and Chronic Toxicity



     Methyl Mercury and Other Short-Chain Alkyl Mercurials:



The toxic effects  of methyl mercury have been described



in several recent  reviews (Swedish Expert Group, 1971; Study



Group on Mercury Hazards, 1971; World Health Organ. 1972,



1976; Miller and Clarkson, 1973; Friberg and Vostal, 1972;



Nordberg, 1976; Natl. Acad.  Sci., 1978).  A major conclusion



of these reviews is that prenatal methyl mercury poisoning



differs qualitatively and probably quantitatively from postna-



tal poisoning.  These two situations will be treated separate-



ly in this section.



     Effects on Adults:  Prior to the major outbreaks in



Japan in the 1950's and 1960's, cases of poisoning due to



occupational and accidental methyl mercury exposure had



already indicated  the principal signs and symptoms of severe



poisoning.  The first recorded poisoning took place in 1863



(Edwards, 1865).  In that year, three young laboratory workers



developed neurological symptoms three months after they



were first exposed; two of them died.  Four cases of methyl



mercury poisoning  were described by Hunter, et al.  (1940).



The patients had worked in a factory that manufactured methyl



mercury compounds  for use as a seed grain fungicide.  They



were asymptomatic  during the initial three to four months



of exposure and then contracted symptoms that were confined



to the nervous system.  The presenting symptoms were par-



esthesia of the extremities, impaired peripheral field of



vision, slurred speech, and unsteadiness of gait and of



limbs.  Examination showed that all four had ataxia, con-



striction of visual fields,  and impaired stereognosis, two-



                              C-63

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point discrimination  and joint position sensation  in  the
fingers.  Three had dysarthria.   In all cases,  the maximum
severity of symptoms  occurred several weeks after  exposure
to the poison had ceased.  The degree of  improvement  varied,
and persisting neurological signs were found in all four
cases.  Twelve co-workers remained asymptomatic.  One of
the patients died in  1952 and the neuropathological findings
were reported by Hunter and Russell (1954).  These authors
correlated the ataxia with cerebellar atrophy that parti-
cularly affected the  granule cell layer,  and related  the
visual signs to focal atrophy of  the calcarine cortex.
     In 1956, four patients were admitted  to the hospital
attached to a factory in Minamata, Japan  exhibiting a neuro-
logical disorder of unknown etiology.  Within a few weeks
about 30 individuals  with similar complaints were  identi-
fied in the Minamata  area.  Faculty from Kumamoto University
carried out investigations and by 1959 it  became clear that
Minamata disease was  the Hunter-Russell syndrome of methyl
mercury poisoning (Katsuna, 1968), which  resulted from the
consumption of fish from Minamata Bay that were contaminated
by methyl mercury. The latter was discharged into the bay
via the local factory effluent, but may also have been pro-
duced by biomethylation of Hg   released  from the factory.
Hair and brain of victims contained elevated concentrations
of methyl mercury.  Similar cases appeared in.Niigata, Japan
in 1965 (Tsubaki and  Irukayama, 1977).  The total number
of Japanese cases was recently reported to be at least 1,224
(Tsubaki and Irukayama, 1977).  A poison  that had previously
                               C-64

-------
been recognized as an occupational hazard had become identi-



fied as an environmental risk to public health.



     In the late 1960's a Swedish Expert Group (1971) con-



ducted an exhaustive review of toxicological and epidemio-



logical data related to methyl mercury poisoning in man



and animals.  This review was initiated as a result of the



discovery that widespread mercury pollution existed in Swedish



lakes and rivers, that all forms of mercury were subject



to biomethylation by microorganisms present in sediments



in both fresh and oceanic water, and that fish readily accumu-



lated and concentrated methyl mercury in their edible tissues.



The main purpose of the group was to assess the margin of



safety in the Swedish population with respect to dietary



intake and risk of poisoning from methyl mercury in fish.



Their st ^tegy was to obtain information on two relationships:



(1) the relationship between blood concentrations and risk



of poisoning (frequency of signs and symptoms) from methyl



mercury and (2) the relationship between long-term dietary



intake and steady-state blood concentrations.  By combining



these two relationships they obtained estimates of risks



to various groups in the Swedish populations classified



according to their fish consumption.  Ultimately this infor-



mation was used by the Swedish government to set regulations



on maximal permissible concentration of methyl mercury in



fish.



     For information on blood concentrations and health



effects, the Swedish group had to rely on limited data from



the Niigata outbreak.  Blood samples had been collected
                                 C-65

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from only 17 patients  (Figure 7); these data were insufficient
to establish a statistical relationship between blood con-
centration and frequency of cases of poisoning  (blood con-
centration-response) .  Consequently, they attempted to iden-
tify the lowest blood concentration associated with the
onset of signs and symptoms of poisoning.  In patients from
whom several blood samples had been collected, the methyl
mercury concentration fell exponentially with time, corre-
sponding to a half-time roughly in the range of 70 days.
Where sufficient data points were available, the blood concen-
tration was extrapolated back to the time of onset of symptoms.
The group concluded  that the lowest concentration in blood
associated with the  onset of symptoms in the most sensitive
individual was 200 ng Hg/ml whole blood.  They calculated
the maximum safe blood concentration to be 20 ng Hg/ml,
using a safety factor of 10.  The safety factor took into
account, among other things, the greater sensitivity of
the fetus as compared to adults (see Effects of Prenatal
Exposure).
     Information on  the relationship between average daily
intake and steady-state blood concentration came from two
sources:  radioactive tracer experiments using volunteers
and dietary studies  on individuals eating fish over long
periods of time.  Information was available on three volunteers
who received an oral dose of radioactive methyl mercury
(Aberg/ et al.  1969).  Gastrointestinal absorption was
virtually complete  (about 95 percent of the dose) and the
                              C-66

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          100

        1
        3 50
        ^


        1 20

         
         ffl
         o
                                    \
                     100       200       300
                     Days after appearance of symptoms
400
Figure 7.  Concentration  of  mercury in samples of blood
collected from patients suffering from methyl mercury  poison-
ing in the Niigata outbreak.   Samples from the same patients
are connected by a straight  line.  The arrow indicates the
estimated time of onset of symptoms.   The units of mercury
concentration in blood are /ag  Hg/100  ml.  The numbers  on
the ordinate should be multiplied by  ten to convert to ng
Hg/ml.  Data is taken from   Swedish Expert Group  (1971).
                               C-67

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whole body half-time was about 70 days,  roughly  in agreement
with the half-times observed  in blood  in the Japanese patients.
     Mathematical models of accumulation of methyl mercury
in man have been discussed previously.  The accumulated
amount in the body, A, would  be related  to the average daily
amount taken up by the body,  a, by the expression:
             .  A= (a/b)  (1 -  exp(-b.t)	(1) ,
where t is the time of exposure and b  is the elimination
constant, which is related to the whole body half-time T,
by the expression:
               T = In 2/b	(2) .
     Equation (1) is depicted diagrammatically in Figure
5.  The steady state body burden, A    , would be closely
attained after exposure for a period of time equivalent
to five half-times. A     would be given by:
               A    « a/b		(3) .
     The tracer experiments indicated  two  important criteria
that might be applied to dietary studies on steady-state
relationship:  1) individuals should be receiving a steady
daily intake for about one year, and two)  the accumulated amount
in the body A   should be linearly related to the average
daily intake (equation 3).  If the blood compartment equili-
brates relatively rapidly with other compartments, steady-
state blood concentrations should- also be proportional to
daily intake.
     Dietary studies were conducted with Swedish  fishermen
and their families whose.regular diet  contained  fish.  Blood
concentrations were compared  to the average estimated dietary
intake of methyl mercury.  The latter  was estimated from
                              C-68

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measurements of mercury in the fish muscle and the results
of careful questioning about dietary intake of fish.  The
results of two studies are given in Figure 8.  Both studies
appear to confirm a linear relationship but the slopes of
the lines differ greatly.  Despite the fact that the regres-
sion line of the Birke, et al. (1967) study depended heavily
on one high data point, the authors rejected the other data
on the basis of inaccurate dietary information.  They conclud-
ed that an average daily intake of 300 ug Hg as methyl mercury
would yield a steady-state blood concentration of 200 ng
Hg/ml and that the maximum safe daily intake would be 30
ug Hg.  These conclusions were endorsed by the World Health
Organization (1972) which recommended a tolerable weekly
intake arithmetically equivalent to the Swedish maximum
safe daily intake.
     Despite the excellence of these in-depth reviews, the
conclusions were necessarily limited by the quality of the
data available at that time.  In fact, the Swedish Expert
Group (1971) pointed to several weaknesses and uncertainties
in the data:  1) No information was available on the accuracy
of the analytical methods used to detect mercury during
the Niigata outbreak.  The dithizone procedure used for
the blood and hair analyses has a low sensitivity and high
background.  Large volumes of blood  (up to 50 ml) must have
been used.  In several patients, the hair to blood ratio
departed from what is now believed to be the true ratio
(see World Health Organ, 1976).  2) The patients were admitted
to the hospital after the appearance of signs and symptoms.

                              C-69

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                Hg IN BLOOD CELLS
                09/9
               1200
               1000
                800
               600
               400-
               200
                                           0.5       0.8
                                  M«Hg-|NTAKE THROUGH FISH
                                                 mg HO/DAY
               EXTREME
               FISH CONSUMERS    BIRKE ET AC 1987   n. (I

              ONON F.SH CONSUMERS  TEJN.NC 1*89 A«0 ,970 n. J.
              ABNORMAL SUBJECTS*    -   1B87       /a
              A FISHERMEN         -   ,,59     H*"

              O FISHERMEN OF LAKE     • '  1M7     „"«,
                                   ^w *  .   n • 9 A
—— y « 1*00 x . 3
   ••.
	y . »oox. 11
Figure  8.   Relation between total mercury  concentrations
in blood  cells and exposure to methyl mercury through fish.
The  figures in the ordinate should be divided by two to
convert the concentration units to ng Hg/ml whole blood.
The  regression equations of Birke, et al.  and of Tejning
quoted  above are the  same as those quoted  in Table 1.2 except
the  units of Y and X  have been changed.  Taken from Figure
11.2  in Swedish Expert  Group (1971).
                                   C-70

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It was necessary to extrapolate the observed blood concentra-
tions (based on samples collected in the hospital) back
to the time of onset of symptoms.  The statistical uncertainty
in the linear regression extrapolation was high.  3) The
Swedish data relating dietary intake to blood concentration
are also fraught with uncertainty.
     By the time more recent major reviews appeared  (Nordberg,
1976; World Health Organ. 1976), several studies had been
published on fish-eating populations and preliminary reports
had appeared on the large outbreak of poisoning in Iraq.
Miettinen (1973) had completed his study on 14 volunteers
taking radioactive methyl mercury.  His data, along with
observations of exposed populations in Iraq and elsewhere,
allowed development of a compartmental model for uptake,
distribution, and excretion of methyl mercury in man.  The
World Health Organization review adopted a similar approach
as the Swedish Expert Group in defining relationships:
1) between symptoms and blood concentration, and 2) between
daily intake and steady-state blood concentrations.
     A World Health Organization Committee examined the
Iraqi data on adults (World Health Organ. 1976).  The outbreak
in Iraq occurred in the winter of 1971-1972 among people
living in rural areas.   These people consumed homemade bread
prepared from seed grain that had been treated with a methyl
mercury fungicide.  There were 459 deaths among 6,540 hospi-
talized cases; many others were not admitted to the hospitals
(Bakir,  et al.  1973).   Cases of severe poisoning and fatal-
ities that occurred outside of hospitals may have been consider-

                              C-71

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ably greater.  The  Iraqi data derive from three studies:
1) a preliminary report based on 120 patients  (Bakir, et
al.  1973); 2) an epidemiological survey by a WHO  team  involv-
ing 956 persons in  a  heavily affected rural village and
1,014 persons  in a  control village  (Mufti, et al.  1976);
and 3) an Iraqi study by Shahristani, et al.  (1976) of  184
persons in rural areas, 143 of whom consumed  the contaminated
bread.
     Using the data of Bakir, et al. (1973), Clarkson,  et
al. (1976) compared the frequency of paresthesia with mercury
concentrations in blood  (Figure 9).  Frequencies of paresthesia
(five to ten percent) observed at low Hg concentrations
were interpreted to be background values for  the population
and unrelated  to methyl mercury.  The point of intersection
of the two lines representing parasthesia frequencies and
Hg concentrations was taken to indicate the blood  Hg con-
centration at  which paresthesias due to methyl mercury  emerge
above the background  frequency.  This blood Hg concentration
is 290 ng Hg/ml.  However, the Hg concentrations were those
existing 65 days after cessation of exposure  to methyl  mercury
and, in view of the reported blood Hg half-times of 65  days
in these patients,  the maximum blood Hg concentration was
probably about 480  ng Hg/ml whole blood at the end of exposure.
     The Shahristani, et al. (1976) study reported no cases
of methyl mercury poisoning occurring below a hair concentra-
tion of 120 ug Hg/gm  hair, equivalent to about 480 ng Hg/ml
whole blood.   The World Health Organization study  (Mufti,
et al.  1976)  measured total dose according to the amount
                              C-72

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  1001
   80-
3  60-
.5
*3»
u
o>
IB
   20-
                       10      30        TOO


                   Mercury in blood (pg/IOOml)
300
   Adapted  from Figure 3  of Clarkson,  et al.  (1976).



                          C-73

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of contaminated bread consumed.  The relationship between
frequency of paresthesia and total dose of methyl mercury
had the same general relationship as that shown  in Figure
9.  The background parasthesia frequency was estimated to
be about four percent (World Health Organ. 1976), and the
total dose at which paresthesias due to methyl mercury emerged
above the background frequency was approximately 37 mg.
Since the average body weight in the group was 50 kg, this
dose would correspond to 50 mg in a 70 kg standard man.
The equivalent blood concentration would be approximately
500 ng Hg/ml whole blood.
     The Iraqi studies failed to identify a diagnosed case
of methyl mercury poisoning at 200 ng Hg/ml whole blood.
If such cases existed, they could not be differentiated
from individuals having non-specific signs and symptoms.
The Iraqi studies clearly show a need for more specific
tests for effects of methyl mercury at low doses.
     Several studies of fish-eating populations were also
reviewed by the World Health Organization (1976).  Findings
in Peru (Turner, et al. 1974) and Samoa (Marsh, et al.
(1978)  agreed with those from other fish-eating populations.
No adverse health effects in adults could be associated
with exposure to methyl mercury from fish.  However, only
about 15 people had blood levels in the range of 200 to
400 ng Hg/ml.
     As noted previously, a wide individual variation exists
in blood half-times.  A study by Shahristani and Shihab
(1974)  indicates a bimodal distribution in 48 Iraqis.  One
                              C-74

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group, accounting for 89 percent of the samples, had a mean
half-time value of 65 days, while the other group had a
mean value of 119 days.
     The significance of individual variation in half-times
is demonstrated by the report of Nordberg and Strangert
(1976).  The steady-state blood concentration for any given
dietary intake of methyl mercury is directly related to
the biological half-time (see equations 2 and 3).  These
authors realized that the bimodal distribution of half-times
reported by Shahristani and Shihab (1974) predicted that
a subgroup of the population (the group with the 119-day
average half-time) would attain steady-state blood concentra-
tions almost double those of the group having the 65 day
half-time.  Nordberg and Strangert (1976) went on to calculate
the overall risk of poisoning from dietary methyl mercury
by combining the relationships of the blood concentration
versus frequency of paresthesia (reported by Bakir, et al.
1973) with the bimodal distribution of half-times.  A result
of their calculation is given in Figure 10, which shows
that, for example, a daily intake of 280 pg Hg/70 kg man
(close to the minimum toxic intake calculated by the Swedish
Expert Group, 1971)  would yield a risk of paresthesia of
about eight percent based on the Bakir, et al.  (1973) data
and of three to four percent based on data from the WHO
study in Iraq (Mufti, et al.  1976).
     Several important conclusions may be drawn from these
studies of adult poisonings:  (1)  More data are needed on
the prevalence of effects at the lower regions of the dose-
response relationships. (2) More individuals should be identi-
                                C-75

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          A Probability of
           poisoning, P
                     0.5  1.0   1.5   2.0    2.5 mg daily dose
               'JO' .01~-02'.T>3- .'OS'   ;OX      .I'D


                            DOSE (mg/day)
Figure 10.   Dose-response curve for long-term  exposure to
methyl mercuric compounds in human beings  (50  kg  body wt).
A, whole dose-response curve; B, detailed presentation of
the curve  representing lower doses.  a, daily  dose  of Hg
in the form  of  MeHg ;  P(a),  probability of poisoning  calculated
for the total population; P.,(a), probability of poisoning
for the part of the population with biological half-time
of 64 days.  Probability P = 1.0 corresponds to 100%.  (From
Nordberg and Strangert, 1976).
                                C-76

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fied in fish-eating populations having blood concentrations
in excess of 200 ng Kg/ml.  Even negative results would
be most helpful in setting the upper limits of risk, assuming
that selection processes can be eliminated. (3) Objective
methods are needed to detect the first effects of methyl
mercury exposure.  Paresthesia and other subjective com-
plaints are the first effects associated with methyl mercury
poisoning, but are not good for detecting these first effects
because of the high background, i.e., high frequency in
non-exposed individuals.  At present, no biochemical, neuro-
physiological, or other objective test serves as an early
warning sign (Nordberg, 1976).  (4)  The bimodal distribu-
tion of half-times reported by Shahristani and Shihab (1974)
needs confirmation and further refining through observation
of larger numbers of people.   (5)  Further data are needed
on the relationship between long-term dietary intake and
steady-state blood concentrations in order to test the model
for both long and short half-time groups.  The tentative
blood level limits based on the data from Iraq also need
verification in another population because dietary or genetic
factors may be important.
     A statistical relationship has been suggested by Skerfving
et al. (1974)  between frequency of chromosomal aberrations
and blood concentration of methyl mercury.  This report
was based on 37 people exposed to methyl mercury through
intake of various amounts of fish.  The highest exposure
group had blood concentrations in the range of 14 to 116
ng Hg/ml and the non-exposed group showed concentrations
                           C-77

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in the range of 3  to  18 ng Hg/ml.  However, a  study made
a few months after  the outbreak  in Iraq could  find no corre-
lation between chromosomal damage and exposure to methyl
mercury  (Firman, 1974).
     Bakir, et al.  (1973) found  few clinical effects associated
with damage to non-nervous tissue in the victims of methyl
mercury poisoning.  An earlier outbreak of ethyl mercury
poisoning revealed  cardiovascular effects due  to renal and
cardiac damage  (Jalili and Abbasi, 1961).
     The Swedish Expert Group  (1971) reviewed  case reports
of dermatitis due  to  occupational skin contact with, alkyl
mercurials used as  fungicides.   Jalili and Abbasi  (1961)
and Damluji, et al.  (1976) have  reported exfoliative dermatitis
resulting f ronv oral ingestion of methyl and ethyl mercury
compounds.
     Effects of Prenatal Exposure:  The earliest mention
in the literature  of  psychomotor retardation caused by fetal
exposure to methyl mercury was by Engleson and Herner (1952) .
A Swedish family had  eaten porridge made from  methlymercury
treated grain.  The asymptomatic mother gave birth to a
daughter who appeared  to be normal at birth and in the first
two months of life.   It later became clear that the child
was mentally and physically retarded.  Upon further examina-
tion a year or two  later, she continued to have marked psycho-
motor retardation  and  the authors (Engelson and Herner,
1952) postulated that  "mercury intoxication, perhaps during
early fetal life,  seems to us to be a possible cause."
Her father and brother were diagnosed as having mercury
posioning.  Urinary mercury concentrations were elevated
                               C-78

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in the mother; no blood or hair analyses were performed.
     Harada (1968) reported on 22 children from Minamata,
Japan who had severe psychomotor retardation which he conclud-
ed was due to fetal methyl mercury poisoning.  All children
came from families in which at least one other member had
been diagnosed as having methyl mercury poisoning, with .
fatal results in 13 families.  Five of the mothers had experi-
enced transient paresthesia during pregnancy but had been
well otherwise.  The childrens' ages ranged from one to
six years at the time of initial examination and at those
ages it was not possible to determine their degree of exposure
to methyl mercury in utero.  Two of these children died
and neuropathological studies were reported by Takeuchi
(1968).  He concluded that there was evidence of a disturbed
brain development and that the cerebral and cerebellar lesions
were the same as those found in kittens that had been exposed
to methyl mercury iri utero.
     In August 1969 a family in New Mexico began to eat
pork from a hog that had been fed methyl mercury-treated
seed grain (Snyder, 1971; Pierce, et al.  1972).  At that
time the mother was three months pregnant and ate the con-
taminated pork regularly for the following three months.
She remained asymtomatic but delivered a severely brain-
damaged infant who, at eight months of age, was blind and
hypo-tonic.  Some other members of the family suffered severe
methyl mercury poisoning.  This was the first report of
methyl mercury toxicity from eating contaminated meat and
the only published fetal case in the United States  (Snyder,
1971).
                              C-79

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     The Iraqi outbreak offered an excellent opportunity
to develop quantitative information with regard to prenatal
exposures to methyl mercury.  Large numbers of the popula-
tions, of both sexes, were exposed to a wide range of dietary
intake of methyl mercury within a period of a few months.
Thus, pregnant females could have been exposed to a pulsed
dose of methyl mercury at any time during pregnancy, and
might have consumed a very wide range of doses.  Early studies
on 15 mother-infant pairs identified infants who were prena-
tally exposed to and severely poisoned by methyl mercury
(Amin-Zaki, et al. 1974a).  Choi, et al. (1977) reported
abnormal neuronal migration in a human infant prenatally
poisoned with methyl mercury in Iraq.  A group of infants
                                                      i
was also identified that had been exposed to methyl mercury
primarily by sucking  (Amin-Zaki, et al. 1974b).
     Follow-up neurological and pediatric studies by a Univer-
sity of Rochester team  obtained dose-effect relationships
between prenatal exposure and effects on the infants  (Marsh,
et al.  1978).  Ten infants of mothers who had maximum hair
concentrations in the range of 99 to 384 ppm  (ug/g) differed
from two groups having lower maternal hair concentrations
(12 to 85 ppm and 2 to 11 ppm, Table 11) in the mean age
of walking and talking and in mean heights.  The high mercury
group also differed from the other two groups in the number
of infants having multiple signs and of poisoning symptoms
(Figure 11). For example, all the infants in the high exposure
                             i
group except two had three or more adverse health effects
per infant.  In contrast, the two groups with lower exposures
consisted mainly of infants having one or no adverse effects.
                              C-80

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                             TABLE 11

       Maternal Hair Hg and Symptoms in Children and Mothers
Exposure Groups3
Maternal hair peak Hg
ug Hg/g
29 Children
Walking, mean age (months)
Talking, mean age (months)
height at 54-60 months (cm)
29 Mothers
Asymptomatic in pregnancy
Paresthesias in pregnancy
I
0-11
16.4
20.5
100.5
78%
22%
II
12-85
15.8
21.9
97.8
60%
40%
III
99-384
29.1
33.9
85.5
20%
80%
3 The ranges for hair concentrations were chosen to give
  as near as possible the same number of infants in each
  group - Group 1,9;  Group II, 10 and Group III, 10.  The
  student "t" test revealed no significant differences in
  mean ages of walking and talking and mean heights between
  Groups I and II.  Group. Ill differed significantly from
  Group I and II (walking P < 0.001, talking P< 0.005, height P<
  0.05).  The chi-square test revealed no difference in
  frequency of maternal paresthesia between Groups I and
  II.  Group III differed significantly from the two lower
  groups (P < 0.015)  (Marsh, et al. 1978).
                              C-81

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                     E3 MATER/AL PEAK HAIR
                        Hg CONCENTRATION


1
m
i?l
no$
II
27?
^
^xl
|i




i&
                                               %
                                                      Uj
                                              0.5-
                                             11 ppm
                                         22°-o
§  1-^
                            ,
                          ',$2'.
                                          10
 12-   30c-o
85 ppm
                                          10
                                   99-
                                 334 ppm
       80°
            NO. OF ABNORMALITIES/INFANT
Figure 11.  The  number  of abnormalities in each infant are
compared  in three  groups of infants.  The infants are grouped
according to peak  (maximal)  maternal hair concentrations
during pregnancy.   The  maximum concentration, ppm (jig Hg/g) ,
is given  as a number  in each shaded square.  More abnormalities
were found in infants in the high exposure group  (maternal
hair 99^-384 ppm) as compared to the two lower exposure groups
(12-85, 0.5-11 ppm).  The frequencies of maternal paresthesia
are also  listed  (Marsh, et al. 1978).
                                C-82

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A statistical analysis revealed a highly significant  (P
005, chi square test) difference in distribution between
the high exposure and the two lower exposure groups.
     The small number of infant-mother pairs in this  study
does not allow us to identify a specific threshold maternal
hair concentration below which adverse effects do not occur
in both mother and infant.  A high risk of adverse effects
appear to exist at maternal hair concentrations in the range
of 99 to 384 ppm.  However, in the next lower concentration
range (12 to 85 ppm)  the frequencies have fallen dramatically
and do not differ significantly from those seen in the lowest
range (0.5 to 11 ppm).  Thus, adverse effects seen in maternal
hair concentrations up to 85 ppm may have been due to causes
other than methyl mercury exposure.  Unfortunately, only
four infant-mother pairs were available between 25 and 50
ppm maximum maternal hair concentration.
     An epidemiological study of school children living
in the Minamata area of Japan has recently been reported
(Med. Tribune, 1978).  Children suspected of prenatal and
early postnatal methyl mercury exposures (age group 8 to
16)  exhibited a higher incidence of neurological deficits,
learning difficulties, and poor performance on intelligence
tests than children of similar age in a control area.  These
findings confirm predictions from studies of animals  prenatal-
ly exposed to methyl mercury (Spyker, et al. 1972), in which
a variety of behavioral and neurological tests revealed
deficits only after the animals had reached maturity.
                              C-83

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     In summary/ our knowledge is still limited  in perhaps

the most critical area of methyl mercury toxicity in man.

A study on a fish-eating population is needed to complement

the Iraqi program to test if methyl mercury ingested from

contaminated bread  is equivalent toxicologically to methyl

mercury chronically ingested from fish. The on-going Iraqi

study has demonstrated the feasibility of relating the dose

of the mother during pregnancy to effects seen in the infant

during the first six years of life.  Other effects may mani-

fest themselves in  later years as the child matures.

     Effects on Animals:  Animal studies reveal  that effects

on non-human primates are similar to those on man  (Berlin,

et al. 1973).  Neurological damage has also been reported

in various -other species (Swedish Expert Group,  1971; World

Health Organ. 1976).  In general, effects manifest themselves

at the same brain concentrations but corresponding blood

concentrations may  differ widely due to species  differences

in blood to brain ratios (Figure 12).

     The rat appears to experience effects not seen in man.

Kidney damage has been reported by several investigators

(Klein, et al. 1972, 1973; Fowler, 1972a; Magos  and Butler,

1972). Damage to the peripheral nervous system has been

reported in rats (Somjen, et al. 1973a,b; Chang  and Hartman,

1972a,b), whereas neurological signs in man appear to be

due mainly to damage to the central nervous system  (Von

Burg and Rustam, 1974).  However, effects on the neuromuscular
                               ..         N
junction have been  found in severe cases of poisoning in

Iraq (Von Burg and  Landry, 1976).
                              C-84

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     0-
             10   20   30   40'   50   60  -70   80

                                SlOOD(ppm)
90   ICO
Figure 12.   Comprehensive brain/whole blood regression lines
in four species  orally dosed with methyl nercury.   The shaded
areas correspond to  the onset of the first detectable signs
and symptoms of  poisoning.

Figure by courtesy of Weiss, Laties and Wood.   Environmental
Health Sciences  Center, Univ. of Rochester.
                              C-35

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     The first  effects of methyl mercury  as  evidenced  by  ani-


mal experiments are  on protein  synthesis  in  neurons  (Yoshino


et al. 1966; Cavanagh and Chen, 1971; Chang  and  Hartmari,


1972a,b; Syversen, 1977).  The  effects of methyl mercury


on the neuromuscular junction are due to  a highly  selective


interaction with the acetyl choline receptor  (Shamoo,  et


all. 1976).                                             !


     Ganther, et al.  (1972) reported a sparing effect  of


dietary selenium on methyl mercury toxicity  in rats  and


Japanese quail.  Subsequent animal studies have  confirmed


Ganther's findings  (World Health Organ. 1976; Nordberg,


1976).  However, the concentrations of methyl mercury  or


selenium added  to the diet have been higher  than those found
  '"'*•**•„          '                            ' • -

in human diets.  Following the  observation of Garither, et


al. (1972)  that selenium salts, added to the diet,  delayed


the onset of toxic effects, due  to methyl  mercury in  Japanese


quail, several publications have appeared in the literature


on selenium-mercury  interactions  (for review, see  World


Health Organ. 1976; Nordberg, 1976).  However, in  the  most


recent evaluation of experimental data, it was concluded


that there is insufficient evidence to conclude  that selenium


in the human diet would protect against the  toxic  effects


of methyl mercury (Permanent Comm.Int. Assoc. Occup. Health,,


1977):.                                       .        • -.



     Effects on Adults of Mercury Vapor and  Liquid Metallic


Mercury:  The effects of inhaled mercury  vapor on  human


health have been known since ancient times.  Recently, several


reviews have dealt with this topic (Friberg  and  Vostal,
                              C-86

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1972; Natl.  Inst. Occup. Safety Health, 1973; Friberg and
Nordberg, 1973; Nordberg, 1976; World Health Organ. 1976).
Health effects have not been associated with oral  ingestion
of liquid metallic mercury.
     Exposure to extremely high concentration of mercury
vapor (greater than 1 mg Hg/m ) can damage lung tissue,
causing acute mercurial pneumonitis (Milne, et al. 1970).
Exposure to lower levels results in signs and symptoms indica-
ting effects primarily on the central nervous system.
     Most of our knowledge derives from studies of occupa-
tional exposures.  These reviews listed above refer to observa-
tions of more than 1,000 individuals and indicate  that the
classical signs and symptoms of mercury vapor poisoning
(mental disturbances, objective tremors, and gingivitis)
occur in workers following chronic exposures to average
air concentrations above 0.1 to 0.2 mg Hg/m  (Neal, et al.
1937, 1941; Bidstrup, et al. 1951; Friberg, 1951;  Rentes
and Seligmann, 1968).
     In a comparative study of over 500 workers, Smith,
et al. (1970)  reported effects on the nervous system that
were related to the time-weighted average air concentration
of mercury.  Objective tremors were found at air concentra-
tions above 0.1 mg Hg/m .  Nonspecific symptoms such as
loss of appetite, weight loss and shyness seem to  occur
at a greater frequency than in the control group at average
air concentrations in the range of 0.06 to 0.1 mg  Hg/m .
     Extensive Russian studies on occupationally exposed
workers have been reported in a monograph by Trachtenberg
                              C-87

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(1969) and reviewed by Friberg and Nordberg  (1973).  A  syn-


drome involving  insomnia,  sweat-ing,  and emotional  lability


was claimed to occur at  a  higher  frequency as compared  to


controls in workers exposed  at high  ambient  temperatures


(40 to 42°C in summer and  28  to 38°C in winter)  to mercury concen-


trations in the  range of 0.006 to Q..1 mg Hg/m .


     Considerable uncertainty still  exists with  regard  to


health effects at concentrations  below 0.1 mg Hg/m .  Friberg


and Nordberg  (1973) point  to  the  possibility of  "interviewer"


effects in occupational  studies in which the factory physician


is aware of the  mercury  concentration to which the workers


are exposed.  The Russian  "analytical methods seem to be


crude, being  based on subjective  evaluation of color shades."


     In the study of Trachtenberg (1969), uptake of  iodine


by the thyroid was significantly  greater in a mercury-exposed


group of workers than in a control group.  However,  Kazantzis


(1973) has suggested that  these studies should be  repeated


and should include measurements of serum thyroxin.   He  pointed


out that increased uptake of  radioactive iodine  will occur


if the store  of  iodine in  the thyroid gland  is low and  need


not necessarily  be associated with increased secretion  of


thyroxin.


     Four cases  of proteinuria were  reported in  workmen


exposed to mercury vapor (Kazantzis,  et al. 1962).   Exposure
    ;

levels were probably high, as urinary concentration  was


in excess of  i,000 pg Hg/1.   Increased urinary excretion


of protein in exposed versus  non-exposed workers was reported


by Joselow and Goldwater (1967).  Ashe, et al.  (1953) found




                              C-88

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morphological evidence of kidney damage in rabbits exposed
to mercury vapor.
     Few biochemical changes have been reported due to inhala-
tion of mercury vapor.  Wada, et al.  (1969) noted that blood
cholinesterase activity was decreased when urinary mercury
excretion was greater than 200 ug Hg per gram of urinary
creatinine.  This rate of excretion should correspond to
an average air concentration (eight hrs/day, five days/week)
in the range of 0.05 to 0.1 mg Hg/m .
     Table 12, which summarizes data from animal and human
studies, shows that the earliest effects of mercury vapor
appear at roughly similar brain concentrations in a variety
of species.  Because of species differences in ventilation
rates and pharmacokinetics parameters of inhaled mercury,
the same brain concentrations in various species would not
                                                      i
necessarily correspond to the same average air concentration.
     Effects of Prenatal Exposure:  Little information is
available on biological effects in humans due to prenatal
exposure to mercury vapor.  Studies carried out early in
this century suggest that women chronically exposed to mercury
vapor experienced increased frequencies of menstrual distur-
bances and spontaneous abortions; also, a high mortality
rate has been observed among infants born to women who dis-
played symptoms of mercury poisoning  (Baranski and Szymczyk,
1973).  However, the degree of exposure of these women to
mercury vapor is unknown.  In 1967, an epidemiological survey
in Lithuania called attention to an increased incidence
of abortion and mastopathy related to duration of time on
                              C-89

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                                TABLE 12

         Estimated Average Brain Concentrations at which Toxic
               Effects  Appear  in Adult Humans and  Animals
Species    Brain Cone.    Severity of
            Hg/g wet wt.  effects
Reference
Rabbit

Rat
Rat
Human
1.0
(approx. )
2.8
1.9
0.85
mild3

mild3
mild3
mildb
Ashe, et al. (1953)
'
Rothstein & Hayes (1964)
Berlin, et al. (1969)
Estimated0 from
                                            Hursh, et al.  (1976)
                                            Smith, et al.  (1970)
    The animals were described as irritable.

    Subjective, symptoms such as complaints of loss of appetite.

    The steady-state brain concentration was estimated from
    the data of Hursh, et al.  (1976), which show that 7% of
    an inhaled dose is deposited in the brain, and that the
    half-time in brain is 21 days.  Brain weight was assumed
    to be 1.5 kg, and the time-weighted average air concentration
    associated with mild effects to be 0.1 ng Hg/m , according
    to data of Smith, et al. (1970).  Workers were assumed
    to inhale 10 m  air during an 8-hour occupational exposure,
    to retain 80% of the inhaled mercury, and to work for
    5 days per week.
                                  C-90

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the job among women working in dental offices where mercury
vapor concentrations ranged up to 0.08 mg/m  (Baranski and
Szymczyk, 1973).  Another report described the case of a
woman chronically intoxicated by mercury vapor in whom two
pregnancies ended unfavorably.  After recovery from overt
mercury poisoning, this woman gave birth to a healthy child
(Derobert and Tara, 1950).
     In summary, little is known about the reproductive
  i
effects of inhaled mercury vapor.  In view of the observed
reproductive effects of other forms of mercury, studies
are urgently needed in this area.
     Salts of Inorganic Mercury:  The lethal oral dose in
man of HgClj has been estimated to be between 1 and 4 grams
(Gleason, et al.  1957).  Death is due to acute renal failure.
The effects of chronic exposure to salts of inorganic mercury
have not been described in man.   Long-term occupational
exposure to HgfNO^)^ must have occurred in the felt hat
industry (Neal, et al. 1937).  However, poisoning was believed
to be due to inhalation of mercury vapor produced from HgfNO^
during the procedure of treating the felt.
     Fitzhugh, et al.  (1950)  treated rats with HgCl2 added
to the food for periods of up to two years.  Morphological
changes were induced in kidney tissue at dietary concentra-
tions of 0.5 pg Hg/g food.  However, these studies have
been criticized by Goldwater  (1973) who noted that no effects
   I
were produced in other groups of rats receiving much higher
dietary levels of mercury (2.5 to 10 /ag Hg/g).
     Compounds of inorganic mercury have been shown to be
diuretic in dogs (Mudge and Weiner, 1958).  The nature of
   !
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the anion is important.   Inorganic mercury complexed with
cysteine is a more potent diuretic than HgCl2-
     Piotrowski, et al.   (1973) have discussed the role
of metallothionein in controlling the toxic action of Hg
on the kidney.  The authors pointed out that the toxic effects
on the kidney following a single dose of Hg   salt appear
when the metallothionein  binding capacity is exceeded.
Repeated daily doses of Kg"1"* cause induction of metallothionein
synthesis.  Consequently, much higher concentrations of
inorganic mercury may be  tolerated by the kidney after chronic
exposures (Clarkson, 1977).
     Aryl Alkoxy-aryl, and Other Organic Compounds of Mercury:
Despite the widespread usage of phenyl mercury compounds,
little information is available regarding their effects
on human health.  Since Goldwater's review (1973), new infor-
mation has come to light.  No evidence of adverse health
effects could be found in 67 workers occupatibnally exposed
to phenyl mercury compounds.  Air concentrations were generally
below 0.1 mg Hg/m .  Elemental vapor was the principal form
of mercury in air.
     A'case of acrodynia  has been reported in a child allegedly
exposed to mercury after  the bedroom had been painted with
paint containing phenyl mercury compounds.  The form of
mercury in the air was not identified but it is likely that
mercury vapor was the principal component (Hirschman, 1963).
     Goldwater  (1973) referred to seven workers who had
spent about six weeks working with material containing methoxy-
                              C-92

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ethyl mercury chloride.  Remarkably high blood levels were
reported (range 34 to 109, average 65 jug Hg/100 ml) four
weeks after the end of exposure.  No adverse health effects
could be detected.
     Rats exposed for two years to phenyl mercury acetate
in the diet exhibited morphological changes in the kidneys
'(Fitzhugh, et al. 1950).  As pointed out by Goldwater  (1973),
a dose-response relationship was not established, as animals
receiving higher doses showed no effect.
Teratogenicity
     Methyl Mercury and Other Short-Chain Alkyl Mercurials:
Although brain damage due to prenatal exposure to methyl
mercury has occurred in human populations, no anatomical
defects have been reported.  However, adequate epidemiological
studies have not been performed and the possibility of  terato-
                                                       \
logical action of methyl mercury in human subjects cannot
be dismissed at this time.
                                                       !
     Embryotoxicity and teratogenicity of methyl mercury
in animals have been reported by several authors.  Oharazawa
(1968) noted an increased frequency of cleft palate in mice
treated with an alkyl mercury compound.  Fujita  (1969)  treated
mice .to daily administration of 0.1 mg Hg/kg as methyl mercury
and found that the offspring had significantly reduced birth
weight and possible neurological damage.  No gross terato-
logical effects were noted.  Histological evidence of damage
to the brain as a result of prenatal exposure to methyl
mercury has been reported on several animal species  (Matsumoto,
et al. 1967; Nonaka, 1969; Morikawa, 1961).  Non-lethal

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anatomical malformations  in  animals prenatally  exposed  to
methyl mercury  have  also  been  reported by  Spyker and Smithburg
(1972) and Olson  and Massaro (1977).  Effects due  to prenatal
exposure  in mice  were found  to be about  twice as great  as
those induced by  postnatal exposure and  were greater when
the methyl mercury was administered late in the period  of
brganogenesis.
     Mercury Vapor and Liquid  Metallic Mercury:  Although
the syndrome of mercury vapor  poisoning  has long been known
in adults, practically nothing is known  about prenatal  damage.
Rats exposed prenatally to mercury vapor are reported to
have died within  six days after birth.   In one  experiment,
where exposures were continued throughout gestation, all
of the pups died; some of the  deaths could be attributed
to a failure of lactation in the dams.   A second part of
the experiment  exposed the dams only prior to the  time  of
impregnation. In  this case,  during lactation and nursing
viable pups appeared normal, yet 25 percent of  these pups
died before day six.   No  teratological effects were observed,
birth weights were reportedly within the normal range,  and
histopathologic findings were  negative,  although the concen-
trations of vapor were high  (LC25 for the adult females)
(Baranski and Szymczyk, 1973).
     Salts of Inorganic Mercury:  Teratological effects
of HgCl, have been reported  in animals (Gale and Perm,  1971).
However, no data  are available on the teratogenicity of
inorganic mercury in human populations.
                              C-94

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Mutagenicity
     Methyl Mercury and Other Short-Chain Alkyl Mercurials:
No mutagenic effects have been reported in human populations
due to exposure to methyl mercury.  However, a statistical
relationship was found between the frequency of chromosome
breaks and blood concentrations of methyl mercury  in 23
Swedish fish eaters.  The mercury concentration in the
blood of the exposed group ranged from 14 to 116 ng Hg/ml,
and in the non-exposed group from 3 to 18 ng/ml  (Skerfving,
et al. 1974).
     Khera  (1973)  has reported that, in rats, alkyl mercury
compounds may damage gometes prior to fertilization.  Similar
experiments in mice failed to demonstrate statistically
significant effects.  Studies by Ramel (1972) and Suter
(1975) have revealed damage to reproduction resulting from
exposure to alkyl mercurials during adult life.  Methyl
mercury has been shown to block mitosis in plant cells,
human leukocytes treated in vivo, and human cells  in tissue
culture, and to cause chromosome breakage in plant cells
and point mutations in Drosophila (Swedish Expert Group,
1971; Ramel, 1972).
     Mercury Vapor and Liquid Metallic Mercury:  Nothing
has been reported on the mutagenic effects of mercury vapor
in humans, animals, or in vitro tests.
     Salts of Inorganic Mercury:  Reversible inhibition
of spermatogonial cells has been observed in mice treated
with HgCl   (Lee and Dixon, 1975).  No evidence has been
                              C-95

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published concerning the rautagenicity of mercury salts in
humans.
Carcinogenicity
     When metallic mercury was injected intraperitoneally
into rats, sarcomas were observed only at those tisues that
had been in direct contact with the metal (Druckrey, et
al. 1957).
     No other evidence exists that links exposure to mercury
with cancer.
                                C-96

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                    CRITERION FORMULATION

Existing Guidelines and Standards
     A World Health Organization expert group has recommended
an international standard for drinking water of 1 ug Hg/liter
(World Health 0, 1971); the U.S. Environmental Protection
Agency has recommended a standard of 2 jug Hg/liter  (U.S.
EPA, 1973) .
Current Levels, of Exposure
     Evidence reviewed in the Exposure section indicates
that the predominant form of mercury in freshwater  (and
probably marine water also) is Hg  , present as chelates
and complexes with a variety of inorganic and organic ligands.
However, the data are not sufficiently detailed or accurate
to exclude the possibility of the presence of other forms
of mercury,  especially in contaminated areas.  Methyl mercury
compounds may be present due to biomethylation of inorganic
mercury in sediment, elemental mercury (Hg°) due to discharge
from industry, and aryl and alkoxy mercurials due to their
use in the paint industry.  Although it is highly probable
that the proportions of organo-mercurials and elemental
mercury vapor are small compared to inorganic divalent mercury
(Hg  )  compounds, it will be assumed that the species most
toxic to man accounts for 100 percent of the total mercury
in water because methyl mercury compounds are the forms
of mercury which are most toxic to man and present the greatest
risk of irreversible functional damage.  (See Effects section.)
                              C-97

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Special Groups at Risk
     The evidence presented in this document indicates that
intake of mercury from drinking water is toxicologically
negligible.  Human exposure to the most hazardous form of
this metal, methyl mercury, is almost exclusively via consump-
tion of fish.  Thus, the population most likely to be at
risk is heavy consumers of fish containing the highest
mercury concentrations.  The stage of the human life cycle
subject to the greatest hazard from mercury intake is probably
prenatal.
     Other forms of mercury probably do not present a signifi-
cant risk, except in the case of mercury vapor.  The latter
may present a health risk if occupational exposures are
not maintained below acceptable limits.  Unfortunately,
the stage of the life cycle most susceptible to the toxic
effects of mercury vapor has not yet been identified.
     An unusual and rare reaction to inorganic mercury forms,
called acrodynia or "Pink's Disease," has been described.
This disease has occurred in children receiving oral doses
of medications containing inorganic mercury, or inhaling
mercury vapor.  Only a small number of children develop
acrodynia when exposed to mercury.  It is unlikely that
a small amount of inorganic mercury ingested in drinking
water would cause this disease.
Basis and Derivation of Criterion
     From a health effects perspective and recognition of
exposure potential the organo mercury compounds are the
most important especially methyl mercury.  However, inorganic
compounds of mercury should also be recognized because of
                               C-98

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their toxicity potential but perhaps more importantly because
with alkylation from environmentally present biological
systems the inorganic mercury can be converted to methyl
and dimethyl mercury.
     The approach that has been adopted by this criterion
document involves the following steps:  (1) identify those
organs or tissues most sensitive to damage by the different
chemical and physical forms of mercury, damage being defined
as an effect that adversely changes normal function or dimin-
ishes an individual's reserve capacity to deal with harmful
agents or diseases;  (2)  determine the lowest body burden
known to be associated with functional damage in man and,
if possible, determine the highest body burden tolerated
by man;  (3) estimate the potential human intake from ingest-
ing water and eating contaminated fish products; and (4)
estimate the effect on body burden of mercury by establishing
a criterion for mercury in ambient water based on human
health effects.
     Table 13, taken from the review by the World Health
Organization expert group (1976), indicates long-term daily
intakes of methyl mercury which relates to the earliest
effect on the central nervous system.  This system is more
sensitive to damage from methyl mercury than other functional
systems in the human body.  The conclusions represented
in Table 13 were recently endorsed by the National Academy
of Sciences (1978).
     Evidence reviewed in the Effects section of this document
is essentially the same as the evidence reviewed by the
WHO group with regard to adult exposures to methyl mercury.
                               C-99

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                                TABLE 13

         The Concentrations of Total Mercury in Indicator Media
          and the Equivalent Long-Term Daily Intake of Mercury
         as Methyl Mercury Associated with the Earliest Effects
        in the Most Sensitive Group in the Adult Population ''
Concentrations in indicator media
BloodHairEquivalent long-term daily  intake
(jug/100 ml)          (pg/g)         (jug/kg body weight)


20-50                50-125        3-7
  a The risk of  the earliest effects can be expected  to be
    between 3 to 8%.

    The table should not  be considered  independently  of the  text,

  0 This table is adapted from Table 6  in WHO, 1976.


  Effects on the adult nervous system have been estimated

  to occur at blood concentrations  in the range of  200 to

  500 ng Hg/ml,  corresponding to a  long-term daily  intake

  of methyl mercury in the diet of  3 to 7 /ag/kg body  weight.
                                ^>N
  The risk of effects at  this intake level is probably less

  than eight percent  (1 in 12 chances).

       Since the WHO  (1976) criteria document was written,

  new evidence has been documented.  As reported in the Effects
                                 C-100

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section, females who had experienced maximum hair concentra-



tions during pregnancy in the range of 99 to 384 jug Hg/g



had a high probability of having children liable to retarded



development.  Unfortunately, the population size was too



small to establish a lower limit to effects of prenatal



exposure.  A hair concentration of 99 jug/g is equivalent



to a blood concentration of about 400 ng Hg/ml.



     The most recent information on effect of mercury on



human health has come from the study of the Iraq outbreak



of 1971-1972.  The follow-up of the cases of prenatal ex-



posure is still in progress.  As noted by the National Academy



of Sciences  (1978), "continued careful evaluation of this



very important cohort of pre-natally exposed individuals



will provide the most sensitive assessment of human methyl-



mercury toxicity."



     Thus, at this stage of knowledge of the dose-effect



relationship of mercury in man, it appears that the earliest



detected effects in man are at blood concentrations between



200 and 500 ng Hg/ml, for both pre-and post-natal exposures.



Blood concentrations of methyl mercury correspond to body



burdens in the range of 30 to 50 mg Hg/70 kg body weight,



and to long-term daily intakes in the range of 200 to 500



jug Hg/70 kg.



     Mercury intake from drinking water, according to data



reviewed in the Exposure section of this document, is less



than 1 jug Hg/day, and is considerably less than the diet por-



tion (Table 14).  Assuming that the concentration of methyl



mercury in all samples of drinking water is at the current
                               C-101

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                              TABLE  14
      Estimate  of Average and  Maximum Daily Intakes  of  Mercury
       by  the  "70 kg standard  Adult"  in  the U.S.  Population3,
Mercury intake pg/day/70kg. Predominate form
Media
Air
Water
Food
Average
0.3
0.1
3.0
Maximum
0.8 Hg°
0.4 Hg
5.0 CH-.Hg"1'
     aFor details on the calculation of these numbers, see
       the Exposure section of this document.
      These are approximate figures indicating that 95%
       of the population have intakes less than these figures.
       Occupational exposures are not included.

U.S. EPA standard of 2 jug Hg/1, the maximum daily iatake
would only be 4 jug Hg, assuming 2 liters of drinking water
are consumed per person each day.  This maximum intake would
amount to only about one to two percent of the minimum toxic
intake given in Table 14.  Thus, from the toxicological
standpoint, exposure to mercury via drinking water only
would be negligible.
     The ingestion of water has been assumed to be the main
pathway of direct intake of mercury from water.  The transport
of mercury through skin is another possible route of intake.
Indirect transfer of mercury from water to man is much more
important than transfer from direct routes.  This conclusion
is based on the assumption that fish bioaccumulate a signifi-
cant amount of methyl mercury from water.  In theory, it
should be possible to calculate the maximum concentration
                               C-102

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of methyl mercury in water which would assure that concen-
trations in edible tissues of fish do not exceed the Food
and Drug Administration Guidelines of 1.0 jug Hg/g fresh
tissue.  Thus, if the bioaccumulatiori factor is known for
each species of edible fish, it is arithmetically simple
to estimate the maximum concentration of methyl mercury
in water.  For example, the U.S. EPA (1978) calculated bio-
concentration factors  (concentration in fish/concentration
in water) 'for methyl mercury compounds based on literature
reports.  These factors are for edible fish species:  4,525
to 8,376 for rainbow trout Salmo gardineri, 20,000 for
brook trout Salvelinus fontinalis, and 900 to 1,640 for
clams Anodanta grandis, Lampsitis radiata, Lasmigona complanta.
Thus, if the maximum bioaccumulation factor of 20,000 is
adopted, the maximum concentration of methyl mercury in
freshwater that would prevent fish from exceeding the current
FDA guideline would be 0.05 jug/1.
     Unfortunately, both practical and theoretical difficul-
ties thwart any accurate calculation.  First, quantitative
information is inadequate with regard to the role of direct
uptake from water versus accumulation from food chains as
contributors to the total amount of methyl mercury in fish.
Differences may be expected between fish at lower and upper
ends of the food chain.  Second, the accumulation factors
for methyl mercury uptake by fish are only known for few
species.  Third, the concentration of methyl mercury in
water is probably a variable fraction of total mercury in
water.  The proportion of methyl to total mercury will prob-
ably vary in different bodies of water, being influenced
                              C-.103

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by such factors as water pH, degree of oxygenation, the
amount of biota and the sedimentary concentrations of mercury.
Fourth, in most cases, the concentration of methyl mercury
in water will be so low as to defy accurate measurement
even by the most modern technology.
     When more information is available on the behavior
of mercury in aquatic environments, it might be possible
to calculate a reliable criterion based on acceptable concen-
trations of mercury in fish.  In the meantime, a more pragma-
tic approach will have to be used.  The discharge of mercury
into bodies of water must be carefully controlled.  Those
bodies of freshwater supporting edible fish with mercury
concentrations above the acceptable levels will have to
be identified, and anthropogenic discharge of mercury curtail-
ed.  It is also possible that non-anthropogenic sources
are predominant (for example, in ocean waters) so that control
is not possible.  This empirical approach, although the
only one available, is unsatisfactory as it allows mainly
after-the-fact corrections.  Development of procedures for
estimating maximum safe concentrations of mercury in ambient
water that will prevent unacceptable bioaccumulation of
methyl mercury by fish is clearly desirable.
Methyl Mercury
     Two approaches could be used to derive a criterion
for methyl mercury.  One approach is to use the existing
U.S. drinking water standard of 2 >ug/l and the typical water
quality exposure assumptions (2 1 water/day, 0.0187 kg fish
products/day) along with an estimated fish/shellfish biocon-
                               C-104

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centration factor of 6,200 to calculate a potential uptake.
This can then be compared to the lowest Observable Effect
Level (LOEL)  to determine the range of safety.  A second
approach is to use the LOEL as a basis for establishing
an acceptable daily intake (ADI) and calculate a criterion
level using the typical water quality assumptions.
Given: fish/shellfish consumption = 0.0187 kg fish/person/day
bioconcentration factor for methyl mercury = 6,200 = ^
          water consumption = 2 I/person/day
(1)  Assume criterion = 2 jug/1
      Human exposure  = (2 I/day + (6,200 x 0.0187)
                      = 2  (2 + 115.9)
                      = 235.8 pg/day
     Recognizing that the LOEL range is 200 to 500 ug Hg/day,
we could hypothesize that there is little or no margin of
safety at the 2 jug/1 criterion level especially where realiz-
ing that dietary sources other than fish products may be
contributing to the body burden.
(2)  Derive ADI using typical water quality exposure and LOEL
     LOEL range = 200-500 pg Hg/day
                  Use 220 jjg Hg/day to assure marginal safety
            ADI = 200 pg/day
                = C  2 I/day +  (6,200 x 0.0187)
            200 = C (2 + 115.9)
     200/117.9  = C
     1.7 pg/1   = C
     According to the National Academy of Science  (1977)
an uncertainty factor of ten can be applied to the ADI as
                              C-105

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the 200 to 500 data results from studies on prolonged inges-
tion by man, with no indication of carcinogenicity.
       200/10   = C (2 + 115.9)
     0.17 jjg/1  = C
     0.2 jjg/1  "-• C
     Whereas, approach #1 has an estimated narrow margin
of safety if any and given that LOEL's do exist it is reason-
able to focus on the ADI based criterion with an uncertainty
factor as the preferred basis for establishing a criterion.
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