September, 1987
                                     ATRAZINE

                                 Health Advisory
                             Office of Drinking Water
                       U.S. Environmental Protection Agency.
DRAFT
I.  INTRODUCTION

        The  Health Advisory (HA) Program,  sponsored by the Office of Drinking
   Water (ODW),  provides information on the health effects, analytical method-
   ology and treatment technology that would be useful in dealing with the
   contamination of drinking water.  Health Advisories describe nonregulatory
   concentrations of drinking water contaminants at which adverse health effects
   would not be  anticipated to occur over specific exposure durations.   Health
   Advisories contain a margin of safety to protect sensitive  members of the
   population.

        Health Advisories serve as informal technical guidance to assist Federal,
   State and local officials responsible for protecting public health when
   emergency spills or contamination situations occur.  They are not to be
   construed as  legally enforceable Federal standards.  The HAs are subject to
   change as new information becomes available.

        Health Advisories are developed for one-day, ten-day,  longer-term
   (approximately 7 years, or 10% of an individual's lifetime) and lifetime
   exposures based on data describing noncarcinogenic end points of toxicity.
   Health Advisories do not quantitatively incorporate any potential carcinogenic
   risk from such exposure.  For those substances that are known or probable
   human carcinogens, according to the Agency classification scheme (Group A or
   B), Lifetime  HAs are not recommended.  The chemical concentration values for
   Group A or B  carcinogens are correlated with carcinogenic risk estimates by
   employing a cancer potency (unit risk) value together with  assumptions for
   lifetime  exposure and the consumption of drinking water. The cancer unit
   risk is usually derived from the linear multistage model with 95% upper
   confidence limits.  This provides a low-dose estimate of cancer risk to
   humans that is considered unlikely to pose a carcinogenic risk in excess
   of the stated values.  Excess cancer risk estimates may also be calculated
   using the One-hit, Weibull, Logit or Probit models.  There  is no current
   understanding of the biological mechanisms involved in cancer to suggest that
   any one of these models is able to predict risk more accurately than another.
   Because each  model is based on differing assumptions, the estimates that are
   derived can differ by several orders of magnitude.

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    Atrazine                                                      August,  1987

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II.  GENERAL INFORMATION AND PROPERTIES

    CAS No.  1912-24-9

    Structural Formula             £|


                                N^^N
                                            H
                        C,H,-I
                               I          I
                               H         H
                2-
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Atrazine                                                   September, 1987

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        Samples were collected at 1,468 surface water locations and 2,123
        ground water locations, and atrazine was found in 36 states.  The
        85th percentile of all non-zero samples was 2.3 ug/L in surface water
        and 1.9 ug/L in ground water sources.   The maximum concentration
        found in surface water was 400 ug/L and in ground, water it was
        1,400 ug/L.

     0  Atrazine has been found also in ground water in Pennsylvania, Iowa,
        Nebraska, Wisconsin and Maryland; typical positives were 0.3 to 3 ppb
        (Cohen et al.,  1986).

Environmental Fate

     0  An aerobic soil metabolism study in Lakeland sandy loam, Hagerstown
        silty clay loam, and Wehadkee silt loam soils showed conversion of
        atrazine to hydroxyatrazine, after 8 weeks, to be 38, 40 and 47% of
        the amount applied, respectively, (Harris, 1967).  Two additional
        degradates,  deisopropylated atrazine and deethylated atrazine, were
        identified in a sandy loam study (Beynon et al., 1972).

     0  Hurle and Kibler (1976) studied the effect of water-holding capacity
        on the rate of degradation and found a half-life for atrazine of more
        than 125 days,  37 days and 36 days in sandy soil held at 4%, 35% and
        70% water-holding capacity, respectively.

     0  In Oakley sandy loam and Nicollet clay loam, atrazine had a half-life
        of 101 and 167 days (Warnock and Leary, 1978).

     0  Carbon dioxide production was generally slow in several anaerobic
        soils:  sandy loam, clay loam, loamy sand and silt loam (Wolf and
        Martin, 1975; Goswami and Green, 1971; Lavy et al., 1973).

     0  14C-Atrazine was stable in aerobic ground water samples incubated for
        15 months at 10 or 25°C in the dark (Weidner, 1974).

     0  Atrazine is moderately to highly mobile in soils ranging in texture
        from clay to gravelly sand as determined by soil thin layer chroma-
        tography (TLC), column leaching, and adsorption/desorption batch
        equilibrium studies.  Atrazine on soil TLC plates was intermediately
        mobile in loam, sandy clay loam, clay loam, silt loam, silty clay
        loam, and silty clay soils, and was mobile in sandy loam soils.
        Hydroxyatrazine showed a low mobility in sandy loam and silty clay
        loam soils  (Helling, 1971).

     0  Soil adsorption coefficients for atrazine in a variety of soils were:
        sandy loam  (0.6), gravelly sand  (1.8), silty clay  (5.6), clay loam
        (7.9), sandy loam (8.7), silty clay loam (11.6), and peat (more than
        21) (Weidner, 1974; Lavy 1974; Talbert and Fletchall, 1965).

     0  Soil column studies indicated atrazine was mobile in sand, fine sandy
        loam, silt loan and loam; intermediately mobile in sand, silty clay
        loam and sandy loam; low to intermediately mobile in clay loam (Heidner,
        1974; Lavy, 1974; Ivey and Andrews, 1964; Ivey and Andrews, 1965).

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     Atrazine                                                   September, 1987

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          0  In a Mississippi field study, atrazine in silt loam soil had a half-
             life of less than 30 days  (Portnoy, 1978).  In a loam to silt loam
             soil in Minnesota, atrazine phytotoxic residues persisted for more
             than 1 year and were detected in the maximum-depth samples  (30 to
             42 inches) (Darwent and Behrens, 1968). In Nebraska, phytotoxic
             residues persisted in silty clay loam and loam soils 16 months after
             application of atrazine; they were found at depths of 12 to 24 inches.
             But atrazine phytotoxic residues had a half-life of about 20 days in
             Alabama fine sandy loam soil, although leaching may partially account
             for this value (Buchanan and Hiltbold, 1973).

          0  Under aquatic field conditions,  dissipation of atrazine was due to
             leaching and to dilution by irrigation water, with residues persisting
             for 3 years in soil on the sides and bottoms of irrigation ditches,
             to the maximum depth sampled, 67.5 to 90 cm (Smith et al., 1975).


III. PHARMACOKINETICS

     Absorption

          0  Atrazine appears to be readily absorbed from the gastrointestinal
             tract of animals.  Bakke et al. (1972) administered single 0.53-mg
             doses of 14c-ring-labeled atrazine to rats by gavage.  Total fecal
             excretion after 72 hours was 20.3% of the administered dose; the
             remainder was excreted in urine (65.6%) or retained in tissues (15.8%).
             This indicates that at least 80% of the dose was absorbed.

     Distribution

          0  Bakke et al.  (1972)  administered single 0.53-mg doses of 1^-ring-
             labeled atrazine to rats by gavage.  Liver, kidney and lung contained
             the largest amounts of radioactivity,  while fat and muscle had lower
             residues than the other tissues examined.

          0  In a metabolism study by Ciba-Geigy (1983a), the radioactivity of
             14C-atrazine dermally applied to Harlan Sprague-Dawley rats at
             0.25 mg/kg was distributed to a minor  extent to body tissues.   The
             highest levels were measured in liver and muscle at all time points
             examined;  2.1% of the applied dose was in muscle and 0.5% in liver
             at 8 hours.

          0  Khan and  Foster (1976)  observed  that in chickens the hydroxy metabo-
             lites of atrazine accumulate in the liver, kidney,  heart and lung.
             Residues  of both  2-chloro and 2-hydroxy moieties were found  in chicken
             gizzard,  intestine,  leg muscle,  breast muscle and abdominal  fat.

     Metabolism

          0  The principal reactions  involved in the metabolism  of atrazine are
             dealkylation  at the  C-4 and C-6 positions of the molecule.   There is
             also some evidence of dechlorination at the C-2 position.   These  data
             were reported by  several researchers as demonstrated below.

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        Bakke et al. (1972) administered single 0.53-mg doses of 1^-ring-
        labeled atrazine to rats by gavage.  Less than 0.1% of the label
        appeared in carbon dioxide in expired air.  Most of the radioactivity
        was recovered in the urine (65.5% in 72 hours), including at least 19
        radioactive compounds.   Approximately 47% of the urinary radioactivity
        was identified as 2-hydroxyatrazine and its two mono-N-dealkylated
        metabolites.  None of the metabolites identified contained the 2-chloro
        moiety (which may have been removed via hydrolysis during the isolation
        technique or by a dechlorinating enzyme as suggested by the in vitro
        studies of Foster et al. (1979), who found evidence for a dechlorinase
        in chicken liver homogenates incubated with atrazine.

        Bohme and Bar (1967) identified five urinary metabolites of atrazine
        in rats:  the two monodealkylated metabolites of atrazine, their
        carboxy acid derivatives and the fully dealkylated derivative.  All
        of these metabolites contained the 2-chloro group.  The in vitro
        studies of Dauterman and Muecke (1974) also found no evidence for
        dechlorination of atrazine in the presence of rat liver homogenates.

        Similarly, Bradway and Moseman  (1982) administered atrazine (50,
        5, 0.5 or 0.005 mg/day) for 3 days to male Charles River rats and
        observed that the fully dealkylated derivative  (2-chloro-4,6-diamino-
        s-triazine) was the major urinary metabolite, with lesser amounts of
        the two mono-N-dealkylated derivatives.

        Erickson et al. (1979)  dosed Pittman-Moore mini-pigs by gavage with
        0.1 g of atrazine  (SOW).  The major compounds identified in the urine
        were the parent compound (atrazine) and deethylated atrazine (which
        contains the 2-chloro substituent).
Excretion
        Urine appears to be the principal route of atrazine excretion in
        animals.  Following the administration of 0.5 mg doses of  14c-ring-
        labeled atrazine by gavage to rats, Bakke et al. (1972) reported that
        in 72 hours most of the radioactivity (65.5%) was excreted in the
        urine, 20.3% was excreted in the feces, and less than 0.1% appeared
        as carbon dioxide in expired air.  About 85 to 95% of the urinary
        radioactivity appeared within the first 24 hours after dosing,
        indicating rapid clearance.

        Dauterman and Muecke (1974) have reported that atrazine metabolites
        are conjugated with glutathione to yield a mercapturic acid in the
        urine.  The studies of Foster et al. (1979) in chicken liver homo-
        genates also indicate that atrazine metabolism involves glutathione.

        Ciba-Geigy (1983b) studied the excretion rate of 14c-atrazine from
        Harlan Sprague-Dawley rats dermally dosed with atrazine dissolved in
        tetrahydrofuran at levels of 0.025, 0.25, 2.5 or 5 mg/kg.  Urine and
        feces were collected from all animals-at 24-hour intervals for 144
        hours.  Results indicated that atrazine was readily absorbed, and
        within 48 hours most of th«.absorbed dose was excreted, mainly in the
        urine and to a lesser extent in the. feces.  Cumulative excretion in

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    Atrazine                                                   September, 1987

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            urine and feces appeared to be directly proportional to the administered
            dose, ranging from 52% at the lowest dose to 80% at the highest dose.

IV. HEALTH EFFECTS

    Humans

       Short-term Exposure

         0  A case of severe contact dermatitis was reported by Schlichter and
            Beat (1972) in a 40-year-old farm worker exposed to atrazine formu-
            lation.  The clinical signs were red,  swollen and blistered hands
            with hemorrhagic bullae between the fingers.

       Long-term Exposure

         0  Yoder et al. (1973)  examined chromosomes in lymphocyte cultures
            taken from agricultural workers exposed to herbicides including
            atrazine.  There were more chromosomal aberrations in the workers
            during mid-season exposure to herbicides than during the off-season
            (no spraying).  These aberrations included a four-fold increase in
            chromatid gaps and a 25-fold increase in chromatid breaks.  During
            the off-season, the mean number of gaps and breaks was lower in this .
            group than in controls who were in occupations unlikely to involve
            herbicide exposure.   This observation led the authors to speculate
            that there is enhanced chromosomal repair during this period of time
            resulting in compensatory protection.

    Animals

       Short-term Exposure

         0  Acute oral LD50 values of 3,000 rag/kg  in rats and 1,750 mg/kg in
            mice have been reported for technical  atrazine by Bashmurin (1974);
            the purity of the test compound was not specified.

         0  Molnar (1971) reported that when atrazine was administered by gavage
            to rats at 3,000 mg/kg, 6% of the rats died within 6 hours, and 25%
            of those remaining died within 24 hours.  The rats that died during
            the first day exhibited pulmonary edema with extensive hemorrhagic
            foci, cardiac dilation and microscopic hemorrhages in the liver and
            spleen.   Rats that died during the second day had hemorrhagic broncho-
            pneumonia and dystrophic changes of the renal tubular mucosa.  Rats
            sacrificed after 24  hours had cerebral edema and histochemical
            alterations in the lungs, liver and brain.

         •  CSE Laboratories (1980) studied the acute oral lethality of atrazine
            in Sprague-Dawley rats dosed at 1,500, 1,700, 1,900, 2,000 or
            5,000 mg/kg.  Deaths occurred within 48 hours in all groups except
            for that given the 1,500-mg/kg dose.   Toxic signs in other groups
            included ataxia, diarrhea, oral discharge and chromorhinorrhea (bloody
            nasal discharge).. After 14 days,  examination of surviving rats

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        revealed that body weights were generally normal,  and gross necropsy
        revealed no abnormalities.

     0  Gaines and Linder (1986)  determined the oral LD50 for adult male and
        female rats to be 737 and 672 mg/kg respectively and 2,310 mg/kg for
        pups.  This study also reflected that the dermal LDso for adult rats
        was higher than 2,500 mg/kg.

     0  An acute dermal 1-05Q value of 7.55 g/kg for technical atrazine applied
        to rabbits has been reported  (Frear,  1969).

     0  Palmer and Radeleff (1964) administered atrazine as a fluid dilution
        or in gelatin capsules to Oelaine sheep and dairy cattle.  Two doses
        of 250 mg/kg atrazine caused  death in both sheep and cattle.  Sixteen
        doses of 100 mg/kg were lethal to one sheep.  At necropsy, degeneration
        and discoloration of the adrenal glands and congestion in lungs,
        liver and kidneys were observed.

     0  Palmer and Radeleff (1969) orally administered 10 doses of atrazine SOW
        (analysis of test material not provided) by capsule or by drench to sheep
        at 5, 10, 25, 50 or 100 mg/kg/day and to cows at 10 or 25 mg/kg/day.
        The number of animals in each dosage group was not stated, and the use
        of controls was not indicated.  Observed effects included muscular
        spasms, stilted gait and stance and anorexia at all dose levels in
        sheep and at 25 mg/kg in cattle.  Necropsy revealed epicardial petechiae
        (small hemorrhagic spots on the lining of the heart) and congestion
        of the kidneys, liver and lungs.  Effects appeared to be dose related.
        A Lowest-Observed-Adverse-Effect-Level (LOAEL) of 5 mg/kg/day in
        sheep and a No-Observed-Adverse-Effect-Level (NOAEL) of 10 mg/kg/day
        in cows can be identified from this study.

     0  Bashmurin (1974) reported that oral administration of 100 mg/kg of
        atrazine to cats had a hypotensive effect, and that a similar dose in
        dogs was antidiuretic and decreased serum cholinesterase activity.
        No other details of this study were reported.

   Dermal/Ocular Effects

     °'  In a primary dermal irritation test in rats, atrazine at 2,800 mg/kg
        produced erythema but no systemic effects  (Hayes, 1982).

     0  In primary eye irritation studies, atrazine was described as irritating
        when applied at an unspecified concentration in rats (Hayes, 1982).

   Long-term Exposure

     0  Hazelton Laboratories (1961)  fed atrazine to male and female rats for
        2 years at dietary levels of 0, 1, 10 or 100 ppm.  Based on the
        dietary assumptions of Lehman (1959), these levels correspond to
        doses of approximately 0, 0.05, 0.50 or 5.0 mg/kg/day.   After 65
        weeks,  the 1.0-ppm dose was increased to 1,000 ppm (50 mg/kg/day) for
        the remainder of the study.  No treatment-related pathology was found
        at 26 weeks, at 52 weeks, at 2 years, or in animals that died and

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        were necropsied during the study.  Results of blood and urine analyses
        were unremarkable.  Atrazine had no effects on the general appearance
        or behavior of the rats.  A transient roughness of the coat and
        piloerection were observed in some animals after 20 weeks of treatment
        at the 10- and 1 00-ppm levels but not at 52 weeks..  Body weight gains,
        food consumption and survival were similar in all groups for 18
        months, but from 18 to 24 months there was high mortality due to
        infections (not attributed to atrazine) in all groups, including
        controls, which limits the usefulness of this study in determining a
        NOAEL for the chronic toxicity of atrazine.

     0  In a 2-year study by Woodard Research Corporation (1964), atrazine
        (SOW formulation) was fed to male and female beagle dogs for 105
        weeks at dietary levels of 0, 15, 150 or 1,500 ppm.  Based on the
        dietary assumptions of Lehman (1959), these levels correspond to
        doses of 0, 0.35, 3.5 or 35 mg/kg/day.  Survival rates, body weight
        gain, food intake, behavior, appearance, hematologic findings,
        urinalyses, organ weights and histologic changes were noted.  The
        15-ppm dosage (0.35 mg/kg/day)  produced no toxicity, but the 150-ppm
        dosage (3.5 mg/kg/day) caused a decrease in food intake as well as
        increased heart and liver weight in females.  In the group receiving
        1,500 ppm (35 mg/kg/day) atrazine,  there were decreases in food
        intake and body weight gain, an increase in adrenal weight, a
        decrease in hematocrit and occasional tremors or stiffness in the
        rear limbs.  There were no differences among the different groups in
        the histology of the organs studied.   Based on these results, a NOAEL
        of 0.35 mg/kg/day can be identified for atrazine.

   Reproductive Effects

     0  A three-generation study on the effects of atrazine on reproduction
        in rats was conducted by Woodard Research Corporation  (1966).  Groups
        of 10 males and 20 females received atrazine at dietary levels of 0,
        50 or 100 ppm.  Based on the dietary assumptions that  1 ppm in the
        diet of rats is equivalent to 0.05  mg/kg/day (Lehman,  1959), these
        levels correspond to doses of approximately 0,  2.5 or 5 mg/kg/day.
        After receipt, animals were fed only half of the dietary levels for
        the first 3 weeks and were then changed to the stated levels for 74
        days.  After 74 days of dosing, rats  within each group were paired
        for mating.  Approximately 13 days  after the first weaning,  the
        females in each group were remated  with different males in the same
        group.  The protocol employed following the first mating was repeated
        with the pups from the second mating.   After the second weaning, the
        parents (F0 generation)  were sacrificed and the weanlings (FI^ genera-
        tion) were used to form  another three  groups.   The entire series of
        tests was repeated following the dosing of the FIO generation with
        50 or 100 ppm (2.5 or 5  mg/kg/day)  atrazine for 105  days.   The F2o
        generation was fed atrazine for 75  days and the entire protocol
        repeated again.  After weaning  of the  F3O  generation,  the study was
        terminated.  There were  no adverse  effects of atrazine on reproduction
        observed during the  course of the three-generation study.   Atrazine
        had no effect on any of  the following  parameters:   mean parental body
        weight,  survival,  appearance, behavior,  number  of litters/group.

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        number of live births,  mean body weights at birth and weaning, and
        percent of pups alive at weaning.  A NOAEL of 100 ppm (5 mg/Jq/day)
        was identified for this study.  However, the usefulness of this study
        is limited due to an alteration of the atrazine content of the diet
        during important maturation periods of the neonates.

   Developmental Effects

     0  In the three-generation reproduction study in rats conducted by
        Woodard Research Corporation  (1966) (described above), atrazine at
        dietary levels of 50 or 100 ppm  (2.5 or 5 mg/Jq/day) resulted in no
        observed histologic changes in the weanlings and no effects on fetal
        resorption.  No malformations were observed, and weanling organ
        weights were similar in controls and atrazine-treated animals.
        Therefore, a NOAEL of 100 ppm  (5 mg/Jq/day) was also identified for
        developmental effects in this study.  However, the usefulness of this
        study is limited due to an alteration of the atrazine content of the
        diet during important maturation periods of the neonates.

     0  Atrazine was administered orally to pregnant rats on gestation days
        6 to 15 at 0, 100, 500 or 1,000 mg/Jq (Ciba-Geigy, 1971).  The two higher
        doses increased the number of embryonic and fetal deaths, decreased
        the mean weights of the fetuses and retarded the sJeletal development.
        No teratogenic effects were observed,  the highest dose  (1,000 mg/Jq)
        resulted in 23% maternal mortality and various toxic symptoms.  The
        100 mg/Jq dose had no effect  on either dams or embryos and is therefore
        the maternal and fetotoxic NOAEL in this study.

     0  In a study by Ciba-Geigy  (1984a), Charles River rats received atrazine
        (97%) by gavage on gestation  days 6 to 15 at dose levels or 0, 10, 70,
        or 700 mg/Jq/day.  Excessive  maternal mortality  (21/27) was noted at
        700 mg/Jq/day, but no mortality was noted at the lower doses; also
        reduced weight gains and food  consumption were noted at  both  70 and
        700 mg/Jq/day.  Developmental  toxicity was also present  at these dose
        levels.  Fetal weights were severely reduced at 700 mg/Jq/day; delays
        in sJeletal development occurred at 70 mg/Jq/ day, and a dose-related
        runting was noted at 10 mg/Jq/day and above.  The NOAEL  for maternal
        toxicity appears to be 10 mg/Jq/day, hower, this is also the  LOAEL
        for developmental effects.

     0  New Zealand white rabbits received atrazine  (96%) by gavage on gestation
        days 7 through 19 at dose levels of 0,  1, 5 or 75 mg/Jq/day  (Ciba-Geigy,
         (1984b).  Maternal toxicity,  evidenced by decreased body weight gains
        and food consumption, was present in the mid- and high-dose groups.
        Developmental toxicity was demonstrated only at  75 mg/Jq/day  by an
        increased resorption rate, reduced  fetal weights, and delays  in
        ossification.  No teratogenic effects were  indicated.   The NOAEL
        appears to be  1 mg/Jq/day.

     0  Peters and Cook  (1973) fed atrazine to  pregnant  rats  (four/group)
        at levels of  0, 50,  100,  200,  300,  400, 500 or  1,000  ppai in the diet
        throughout gestation.  The authors  assumed  a body weight of 300 g  and
        a daily food  consumption  of  12 g (based on  Arrington,  1972);  thus,

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Atrazine                                                   September,  1987
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        these levels correspond to approximately 0, 2, 4,  8,  12,  16,  20  or
        40 mg/Jgg/day.  The number of pups per litter was similar  in all
        groups, and there were no differences in weanling  weights.  This
        study identified a NOAEL of 40 mg/kg/day for developmental effects.
        In another phase of this study,  the authors demonstrated  that sub-
        cutaneous (sc) injections of 50, 100 or 200 mg/kj  atrazine on gestation
        days 3, 6 and 9 had no effect on the litter size,  while doses of 800
        or 2,000 nig/kg were embryotoxic.  Therefore, a NOAEL  of 200 mg/kg by
        the sc route was identified for  embryotoxicity.

   Mutagenicity

      0  Loprieno et al.  (1980) reported  that single doses  of  atrazine
        (1,000 mg/kg or 2,000 mg/kg, route not specified)  produced bone  marrow
        chromosomal aberrations in the mouse.  No other details of this  study
        were provided.

      0  Murnik and Nash  (1977) reported  that feeding 0.01% atrazine to male
        Drosophila melanogaster larvae significantly increased the rate  of
        both dominant and sex-linted recessive lethal mutations.  They stated,
        however, that dominant lethal induction and genetic damage may not be
        directly related.

      0  Adler (1980) reviewed unpublished work on atrazine mutagenicity
        carried out by the European Economic Community.  Mutagenic activity
        was not induced when mammalian liver enzymes  (S-9) were used; however,
        the use of plant microsoraes produced positive results.  Also, in
        in vivo studies in mice, atrazine induced dominant lethal mutations
        and increased the frequency of chromatid breaks in bone marrow.
        Hence, the author suggested that activation of atrazine in mammals
        occurs independently of the liver,  possibly in the acidic part of the
        stomach.

      0  As described previously, Yoder et al. (1973) studied  chromosomal
        aberrations in the lymphocyte cultures of farm workers exposed to
        various pesticides including atrazine.  During mid-season a 4-fold
        increase in chroma tid gaps and a 25-fold increase  in  chroma tid breaks
        was observed.  During the off-season (no spraying), the number of
        gaps and breaks was lower than in controls, suggesting to the authors
        that there is enhanced chromosomal  repair during the  unexposed period.

   Carcinogenicity

      0  Innes et al.  (1969) investigated the tumorigenicity of 120 test  com-
        pounds including atrazine in mice.  Two F^ hybrid  stocks  (C57BL/6 x AnF
        and C57BL/6 x AKR) were used.  A dose of 21.5 mg/kj/day was administered
        by gavage to mice of both sexes  from age 7 to  28 days.  After weaning
        at 4 weeks, this dose level was  maintained by  feeding 82  ppn  atrazine
        ad libitum in the diet for  18 months.  At necropsy, thoracic  and
        abdominal cavities were examined, and histologic studies  were performed
        on all major  organs and grossly  visible  lesions.   Blood smears were
        examined if the mice showed signs of splenomegaly  or  lymphadenopathy.
        The incidence of hepatomas, pulmonary tumors,  lymphomas and  total
        tumors in atrazine-treated mice  was not significantly different  from
        that in the negative controls.

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        0  In data supplied  to EPA (U.S.  EPA,  1986a) in support of pesticide
           registration for  atrazine,  Ciba-Geigy Corporation (1985) submitted
           preliminary summary incidence  information (1-year interim report)
           on the histopathological findings of their 2-year oncogenicity study
           of atrazine in Spraque-Dawley  rats.  The summary tables contained
           indications of increased numbers of tumors in the mammary glands of
           the female rats.   "Hie statistical evaluation of this preliminary
           data raised concerns of a dose-related response for increases in  _
           mammary tumors.  Unfortunately,  the data are of a preliminary nature
           and cannot be used for any  further conclusions in this document before
           the 2-year study  is completed  and evaluated.  However, a subsequent
           briefing paper by Ciba-Geigy (1987) indicated that this study is
           positive.  The evaluation of the recently submitted final report of
           this 2-year rat study will  be  performed at a later date.


V. QUANTIFICATION OF TOXICOLOGICAL EFFECTS

        Health Advisories (HAs) are generally determined for one-day, ten-day,
   longer-term (approximately 7 years) and  lifetime exposures if adequate data
   are available that identify a sensitive  noncarcinogenic end point of toxicity.
   The HAs for noncarcinogenic toxicants  are derived using the following formula:

                 HA =  (NOAEL or LOAEL) x (BW) = 	 mg/L (	 u /L)
                         (UF) x (	 L/day)

   where:

           NOAEL or LOAEL =  No- or Lowest-Observed-Adverse-Effect-Level
                            in mg/kj bw/day.

                       BW -  assumed body weight of a child  (10 kj) or
                            an adult  (70 kj ).

                       UF «=  uncertainty factor  (10, 100 or 1,000), in
                            accordance with NAS/ODW guidelines.

                	 L/day =  assumed daily water consumption of a child
                             (1 L/day)  or an adult  (2 L/day).

   One-day Health Advisory

        No suitable information was found in the available literature for  the
   determination of the One-day HA value for atrazine.  It is, therefore,  recom-
   mended that the Ten-day HA value calculated below for a 10-kj child  of
   0.1 mg/L  (100 ug/L), be used at this time as a  conservative estimate of  the
   One-day HA value.

   Ten-day Health Advisory

        Two  teratology studies by Ciba-Geigy one inthe rat  (1984a) and  one  in the
   rabbit  (1984b) were considered for the calculation  of the Ten-day HA value.
   The rat study reflected a NOAEL of 10 mg/kj/day for maternal  toxicity but this

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Atrazine                                                   September,  1987
                                     -12-
value was also the LOAEL for developmental toxicity while the rabbit study
reflected NOAELs of 5 mg/kg/day for developmental toxicity and  1 .mg/hj/day  for
maternal toxicity.  Thus,  the rabbit appears to  be a more sensitive species  than
the rat for internal toxicity, hence, the rabbit  study with a NOAEL of  1 ing/kg/day
is used in the calculations below.

     The Ten-day HA for a  10  kg child is calculated below as follows:

                      (1 mg/kg/d) x  (10kg)   = n.-i ma/T.  (inn mj/T.j
                       (100 )x (1 L/day)

where:

        1 mg/kg/day = NOAEL, based  on maternal toxicity evidenced by decreased
                      body weight gain and food  consumption.

        10 kj = assumed body weight of a child

        100 = uncertainty  factor, chosen in accordance with ODW/NAS guidelines
              for use with a NOAEL  from an animal study.

        1 L/d = assumed daily consumption for a  child

Longer-term Health Advisory

     No suitable information was found in the available literature for the
determination of the  longer-term HA value for atrazine.  It is,  therefore,
recommended that the  adjusted DWEL  for a 10-kg child of 0.035 mg/L
(35 ug/L) and the DWEL for a 70-Jq  adult of  0.123 mg/L  (123 ug/L) be used at
this time as a conservative estimate of the  Longer-term HA values.

Lifetime Health Advisory

     The Lifetime HA  represents that portion of  an individual's  total  exposure
that is attributed to drinking water and is  considered  protective of noncar-
cinogenic adverse health effects over a lifetime exposure.  The  Lifetime HA
is derived in a three-step process.  Step 1  determines  the Reference Dose
(RfD), formerly called the Acceptable Daily  IntaJe  (ADI).  The  RfD is  an esti-
mate of a daily exposure  to the human  population that is liJely to be  without
appreciable risk of deleterious effects over a lifetime, and is  derived from
the NOAEL  (or LOAEL),  identified from a chronic  (or subchronic)  study, divided
by an uncertainty factor(s).  From  the RfD,  a DrinIcing Water Equivalent Level
(DWEL) can be determined  (Step 2).  A DWEL is a  medium-specific (i.e., drinking
water) lifetime exposure  level, assuming 100% exposure  from that medium, at
which adverse, noncarcinogenic health effects would not be expected to occur.
The DWEL is derived from  the multiplication  of the RfD  by the assumed  body
weight of an. adult and divided by the assumed daily water consumption  of an
adult.  The Lifetime  HA is determined in Step 3  by factoring in  other  sources
of exposure, the relative  source contribution  (RSC).  The RSC from drinking
water is based on actual exposure data or, if data are  not available,  a
value of 20% is assumed  for synthetic  organic chemicals and a value  of 10%

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Atrazine                                                  September, 1987

                                     -13-
is assumed for inorganic chemicals.  If the contaminant is classified as a
Group A or B carcinogen, according to the Agency's classification scheme of
carcinogenic potential (U.S. EPA, 1986b), then caution should be exercised in
assessing the risks associated with lifetime exposure to this chemical.

     The 2-year feeding study in dogs by Woodard Research Corporation
(1964) has been selected to serve as the basis for the calculation of the
Longer-term HA, as well as the DWEL,  and Lifetime HA.  Atrazine (SOW formulation)
was fed to male and female beagle dogs for 105 weeks at nominal doses of 15,
150 or 1,500 ppm; based on measured analytical concentrations of 14.1, 141
and 1,410 ppm, however, these values correspond to approximately 0.35, 3.5
and 35 mg/kg/day (Lehman,  1959).  Survival rate, body weight gain, food
intake, behavior, appearance, hematology, urinalysis, organ weights and
histology were determined.  The 15-ppm dosage (0.35 mg/kg/day) produced no
toxicity,  but the 150-ppm  dosage (3.5 mg/kg/day) caused a decrease in food
intake as well as increased heart and liver weight in females.  In the group
receiving 1,500 ppm (35 mg/kg/day), there were decreases in food intake and
body weight gain, an increase in adrenal weight, a decrease in hematocrit and
occasional tremors or stiffness in the rear limbs.  There were no differences
among the different groups in the histology of the organs studied.  Based on
these results, a NOAEL of  0.35 mg/kg/day was identified for atrazine.  This
NOAEL is supported by the available preliminary data by Ciba-Geigy (1985) on
a new two-year study in the Sprague-Dawley rats that will be completed for
the Agency review in the near future.  This preliminary data reflected adverse
effects (mammary gland tumors) at 70 ppm (3.5 mg/kg/day) but no effects were
were noted at the lower dose level, 10 ppm (0.5 mg/kg/day).  Other studies
(Woodard Research Corporation, 1966; Hazelton Laboratories, 1961) identified
long-term NOAEL values of  5 to 50 mg/kg/day and were not considered to be as
protective as the Woodard Research Corporation  (1964) study in the dog for
use in calculating the HA  values for atrazine.

Step 1:  Determination of the Reference Dose  (RfD)

                  RfD = (0.35 mg/kg/day) . 0.0035 mg/kg/day


where:

        0.35 mg/kg/day = NOAEL, based on the absence of adverse clinical,
                         hematological, biochemical and histopathological
                         effects in dogs.

                   100 = uncertainty factor, chosen in accordance with ODW/NAS
                         guidelines for use with a NOAEL from an animal study.

Step 2:   Determination of  the Drinking Water Equivalent Level (DWEL)

          DWEL = (0.0035 mg/kg/day) (70 kg) = 0.123   /L (123   /L)
                          (2 L/day).

where:
        0.0035 mg/kg/day = RfD.

                    70 kg  = assumed body weight of an adult.

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     Atrazine                                                   September,  1987

                                          -14-


                       2 L/day = assumed  daily water consumption of an  adult.

     Step 3:   Determination of the Lifetime Health Advisory

               Lifetime HA = (0.123 mg/L) (20%)  =  0.0025 mg/L  (3 ug/L)

     where:

          0.123 mg/L  =  DWEL.

                 20%  «  assumed  relative source contribution from water.

                  10  =  additional uncertainty  factor,  according to ODW  policy,
                       to account for possible carcinogenicity.

     Evaluation of Carcinogenic Potential

          0  Preliminary  data  submitted by  Ciba-Geigy  Corporation (1985) in  support
            of the pesticide  registration  of  atrazine indicate that atrazine
            induced  an increased incidence of mammary tumors in female Sprague-
            Dawley rats.  These findings have been  further confirmed in a briefing
            by Ciba-Geigy (1987)  on the  recently  completed study.   An  evaluation
            of this  study will be performed in  the  near future.

          0  The International  Agency for Research on  Cancer has  not evaluated  the
            carcinogenic potential of atrazine.

          0  Applying the criteria described in EPA's  guidelines  for assessment of
            carcinogenic risk  (U.S. EPA, 1986b),  atrazine  may  be classified in
            Group C:   possible human carcinogen.  This  category  is  used for
            substances with limited evidence  of carcinogenicity in  animals  in  the
            absence of human data.  This classification is  considered preliminary
            until the  Office of Pesticide  Program completes a  peer  review of the
            weight of  the  evidence  for atrazine and its analogs.  At present,  ODW
            has determined that at least one  closely  related analog, propazine,
            is a  group C oncogen  based on  an  increased  incidence of tumors in  the
            same  target  tissue (mammary  gland) and animal  species  (rat) as was
            noted for  atrazine.


VI. OTHER CRITERIA, GUIDANCE AND  STANDARDS

         0  Toxicity data on atrazine were reviewed by the National Academy of
            Sciences (NAS, 1977), and the  study by Innes et al.  (1969) was used
            to identify a chronic NOAEL of 21.5 mg/kg/day.  Although at that time
            it was concluded that atrazine has low chronic  toxicity, an uncertainty
            factor of 1,000 was employed  in calculation of the ADI from that
            study, since only  limited data were available.  The resulting value
            (0.021 mg/kg/day)  corresponds to an ADI of 0.73 mg/L in a 70-kg adult
            consuming 2 L of water per day.

         0  Tolerances for atrazine alone and  the  combined residues of atrazine
            and its metabolites in or on various raw agricultural commodities
            have been established (U.S.  EPA,  1986c).  These tolerances range from

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      Atrazine                                                September,  1987

                                           -15-


              0.02 ppm (negligible)  in  animal  products (meat and meat by-products)
              to 15 ppm in various  animal fodders.


 VII. ANALYTICAL METHODS

           0 Analysis of  atrazine  is by  a gas chromatographic (GC)  method applicable
              to the determination  of certain  nitrogen-phosphorus containing pesti-
              cides in water  samples (U.S.  EPA,  1986d).   In  this method,  approximately
              1  L of sample is extracted  with  methylene chloride.  The extract is
              concentrated, and the  compounds  are separated  using capillary column
              GC.  Measurement is made  using a nitrogen phosphorus detector.  The
              method detection limit has  not been determined for this compound,  but
              it is estimated that  the  detection limits for  the method analytes are
              in the range of 0.1 to 2  ug/L.


VIII. TREATMENT TECHNOLOGIES

           0 Treatment technologies which will remove atrazine from water include
              activated carbon adsorption, ion exchange, reverse osmosis,  ozone
             oxidation and ultraviolet irradiation.   Conventional treatment methods
              have been found to be  ineffective for the removal of atrazine from
             drinking water  (ESE,  1984;  Miltner and  Fronk,  1985a).   Limited data
              suggest that aeration  would not  be effective in atrazine removal
              (ESE, 1984;  Miltner and Fronk, 1985a).

           0  Baker (1983) reported  that  a 16.5-inch GAG filter cap using F-300,
              which was placed upon  the rapid  sand filters at the Fremont, Ohio
              water treatment plant, reduced atrazine levels by 30 to 64% in the
              water from the  Sandusky River.   At Jefferson Parish, Louisiana,
              Lykins et al. (1984)  reported that an adsorber containing 30 inches
              of Westvaco  wv-G® 12  x 40 GAG removed atrazine to levels below
              detectable limits for  over  190 days.

           0 At the Bowling  Green,  Ohio  water treatment plant, PAG in combination
              with conventional treatment achieved an average reduction of 41% of
              the atrazine in the water from the Maumee River (Baker, 1983).
              Miltner and  Fronk (1985a) reported that in jar tests using spiked
              Ohio River water with  the addition of 16.7 and 33.3 mg/L of PAC and
              1 5-20 mg/L of alum, PAC removed  64 and  84%,  respectively,  of the
             atrazine.  Higher percent removals reflected higher PAC dosages.
             Miltner and  Fronk (1985b) monitored atrazine levels at water treat-
              ment plants, which utilized PAC, in Bowling Green and Tiffin, Ohio.
              Applied at dosages ranging  from  3.6 to  33 mg/L,  the PAC achieved 31
              to 91% removal  of atrazine, with higher percent removals again
              reflecting higher PAC  dosages.

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Atrazine                                                  September, 1 987

                                     -16-
        Harris and Warren (1964) reported that Amber lite IR-120 cation exchange
        resin removed atrazine from aqueous solution to less than detectable
        levels.  Turner and Adams (1968) studied the effect of varying pH on
        different cation and an ion exchange resins.  At a pH of 7.2, 45%
        removal of atrazine was achieved with Dowex® 2 anion exchange resin
        and with H2PO4~ as the exchangeable ion species.
        Chi an et al. (1975) reported that reverse osmosis, utilizing cellulose
        acetate membrane and a cross-linked polyethelenimine (NS-100) membrane,
        successfully processed 40% of the test solution, removing 84 and 98%,
        respectively, of the atrazine in the solution.

        Miltner and Fronk (1985a) studied the oxidation of atrazine with
        ozone in both spiked distilled and ground water.  Varying doses of
        ozone achieved a 70% removal of atrazine in distilled water and 49 to
        76% removal of atrazine in ground water.

        Kahn et al. (1978)  studied the effect of fulvic acid upon the photo-
        chemical stability of atrazine to ultraviolet irradiation.  A 50%
        removal of atrazine was achieved much faster at higher pH conditions
        than at lower pH conditions.  In the presence of fulvic acids, the
        time needed for ultraviolet irradiation to achieve 50% removal was
        almost triple the time required to achieve similar removals without
        the presence of fulvic acids.  Since fulvic acids will be present in
        surface waters, ultraviolet irradiation may not be a cost-effective
        treatment alternative.

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    Atrazine                                                   September, 1987

                                         -17-
IX. REFERENCES

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    Arrington, L.R.  1972.  The laboratory animals.  In;  Introductory laboratory
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    Baker,  D.   1983.   Herbicide contamination in municipal water supplies in
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    Beynon, K.I., G.  Stoydin and A.N.  Wright.  1972.  A comparison of the
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    Bohme,  E., and  F. Bar.  1967.   Uber  den Abbau von Triazin-Herbiciden in
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    Buchanan,  G.A., and A.E. Hiltbold.   1973.  Performance and persistence of
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Atrazine                                          *         September,  1987

                                      -18-
Ciba-Geigy Ltd.   1984b.   Segment II.   Teratology  study  in  rabbits:   Toxicology/
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Erickson, M.D.,  C.W.  Frank and D.P. Morgan.   1979.  Determination of  s-triazine
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Foster, T.S.,  S.U. Khan  and M.H.  Akhtar.  1979.   Metabolism of atrazine by
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Frear,  E.H., ed.  1969.   Pesticide  index.  State College, PA:  College  Science
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Goswami, K.P., and R.E.  Green.   1971.  Microbial  degradation of the herbicide
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Harris, C.I.   1967.    Fate  of 2-chloro-£-triazine  herbicides in soil.  J. Agric.
     Food Chem.   15:157-162.

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Atrazine                                                   September,  1987

                                     -19-
Hayes, W.J.,Jr.  1982.  Pesticides studied in man.  Baltimore,  MD:  Williams
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Innes, J.R.M., B.M. Ulland, and M.G. Valerio.   1969.   Bioassay of pesticides
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Atrazine                                                   September,  1987

                                      -20-
Miltner,  R.J.,  and C.A.  Fronk.   1985a.   Treatment of synthetic organic contami=
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STQRET.   1987.

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      in soils.  Weeds.   13:46-52.

Turner, M.A., and.R.S. Adams, Jr.  1968.  The  adsorption of  atrazine and
     atratone by anion-  and cation-exchange  resins.   Soil Sci.  Amer. Proc.
      32:62-63.

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Atrazine                                                  September, 1987
                                     -21-
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•Confidential Business Information submitted to the Office of  Pesticide
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