&EPA
            'Jnited States
            Environmental Protection
            Agency
            Office of
            Pesticides and Toxic Substances
            Washington OC 20460
September 1980
            Pesticides
0,0,0,0-Tetrapropyl
    dithiopyrophosphate
          Aspon
Pesticide Registration
Standard

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  0,0,0,0-TETRAPROPYL DITHIOPYROPHOSPHATE

                  ASPOIT*

      Pesticide Registration Standard
 Patrick Miller
 John Bascietto
 Charlotte Blalock
 Padma Datta
 Roland Gessert
 Steve Hopkins
 William Miller
 Randall Norris
 Ingrid Sunzenauer
Project Manager (SPRD)
Wildlife Biologist (BED)
Residue Chemist (BED)
Environmental Chemist (BED)
Toxicologist (BED)
Plant Physiologist (BED)
Product Manager (RD)
Writer/Editor (SPRD)
Entomologist (BFSD)
              September 1980

Office of Pesticides and Toxic Substances

     Environmental Protection Agency
     401 M Street, SW
     Washington, DC  20460

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          REGISTRATION STANDARD  FOR  ASPO

                       CONTENTS

                                                     Page
How to Register Under a Registration Standard	   1

Regulatory Position	   9

MANUFACTURING-USE ASPON®
I.  Regulatory Position	   25
  A.  Regulatory Decision	   25
  B.  Criteria for Registration  Under  the
      Standard	   25
  C.  Acceptable Ranges and Limits	   26
      1.  Product Composition Standards	   26
      2.  Acute Toxicity Limits	   27
      3.  Use Patterns	   27
  D.  Data Gaps	   27
  E.  Required Labeling	   29
      1.  Product Chemistry	   29
      2.  Human Hazard - Precautionary Labeling....   30
      3.  Environmental Hazards	   30
      4.  Physical or Chemical Hazards	   30
      5.  Use Patterns	   31

II.  Regulatory Rationale	   33
  A.  Regulatory Decision	   33
  B.  Acceptable Ranges and Limits	   33
      1.  Product Composition Standards	   33
      2.  Acute Toxicity Limits	   34
      3.  Use Patterns	   34
  C.  Data Gaps	   34
  D.  Required Labeling	   35

III.  Product Chemistry	   37
 DISCIPLINARY REVIEW
  Chemistry Profile	   38
  Data Gaps	   38
  Required Labeling	   39
 TOPICAL DISCUSSIONS
  Chemical Identity	   40
  Manufacturing Process	   41
  Formation of Unintentional  Ingredients	   41
  Ingredients in Pesticide Products	   42
  Product Analytical  Methods  and Data	   42
  Physical/Chemical Properties	   42
  B i bl i og r aphy	   45

IV.  'Environmental Fate."	   47
 DISCIPLINARY REVIEW
  Environmental Fate Profile	   47
  Data Gaps	   47

                       -i-

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                                                    Page
V.  Toxicology	  49
 DISCIPLINARY REVIEW
  Toxicology Profile	  49
  Data Gaps	  49
  Required Labeling	  50
 TOPICAL DISCUSSIONS
  Acute Effects	  51
  Local Irritation	  52
  Dermal Sensitization	  53
  Subchronic 21-Day Dermal	  53
  Subchronic Neurotoxicity	  53
  Teratology	  53
  Mutagenicity	  54

VI.  Residue Chemistry	  57

VII.  Ecological Effects	  59
 DISCIPLINARY REVIEW
  Ecological Effects Profile	  59
  Data Gaps	  59
  Required Labeling	  59
 TOPICAL DISCUSSIONS
  Microbes	  60
  Birds	  60
  Aquatic Invertebrates	  61
  Freshwater Fish	  62
  Bibliography	  63
                         ASPON®
EMULSIFIABLE CONCENTRATE 	
I.  Regulatory Position	  65
  A.  Regulatory Decision	  65
  B.  Criteria for Registration Under the
      Standard	  65
  C.  Acceptable Ranges and Limits	  66
      1.  Product Composition Standards	  66
      2.  Acute Toxicity Limits	  67
      3.  Use Patterns and Application Methods	  68
  D.  Data Gaps	  69
  E.  Required Labeling	  70
      1.  Product Chemistry	  70
      2.  Human Hazard - Precautionary Labeling....  71
      3.  Environmental Fate	  73
      4.  Environmental Hazards	  73

II.   Regulatory Rationale	  75
  A.  Regulatory Decision	  75
  B.  Acceptable Ranges and Limits	  75
      1.  Product Composition Standards	  75
      2.  Acute Toxicity Limits	  75
      3.  Use Patterns and Application Methods	  77
  C.  Data Gaps	  77
  D.  Required Labeling	  78

                       -ii-

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                                                     Page
III.  Product Chemistry	   81
 DISCIPLINARY REVIEW
  Chemistry Profile	   81
  Data Gaps	   81
  Required Labeling	   82
 TOPICAL DISCUSSIONS
  Chemical Identity	   82
  Manufacturing Process	   82
  Formation of Unintentional Ingredients	   83
  Ingredients in Pesticide Products	   83
  Product Analytical Methods and Data	   83
  Physical/Chemical Properties	   83
  Bibliography	   84

IV.  Environmental Fate	   85
 DISCIPLINARY REVIEW
  Environmental Fate Profile	   85
  Exposure Profile	   85
  Required Labeling	   86

V.  Toxicology	   87
 DISCIPLINARY REVIEW
  Toxicology Profile	   87
  Toxicology Hazard Assessment	   87
  Data Gaps	   88
  Required Labeling	   90
 TOPICAL DISCUSSIONS
  Acute Effects	   92
  Local Irritation	   93
  Bibliography	   96

VI.  Ecological Effects	   97
 DISCIPLINARY REVIEW
  Ecological Effects Profile	   97
  Required Labeling	   97
 TOPICAL DISCUSSIONS
  Terrestrial Plants	   97
  Aquatic Invertebrates	   98
  Freshwater Fish	   98
  Bibliography	   99
GRANULAR ASPO
I.  Regulatory Position	   101
  A.  Regulatory Decision	   101
  B.  Criteria for Registration Under the
      Standard	   101
                       -111-

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                                                    Page
  C.  Acceptable Ranges and  Limits	   102
      1.  Product Composition Standards	   102
      2.  Acute Toxicity Limits	   103
      3.  Use Patterns and Application Methods	   104
  D.  Data Gaps	   104
  E.  Required Labeling	   106
      1.  Product Chemistry	   106
      2.  Human Hazard - Precautionary Labeling....   106
      3.  Environmental Fate	   106
      4.  Environmental Hazards	   107

II.  Regulatory Rationale	   109
  A.  Regulatory Decision	   109
  B.  Acceptable Ranges and  Limits	   109
      1.  Product Composition Standards	   109
      2.  Acute Toxicity Limits	   109
      3.  Use Patterns and Application Methods	   Ill
  C.  Data Gaps	   Ill
  D.  Required Labeling	   112

III.  Product Chemistry	   113
 DISCIPLINARY REVIEW
  Chemistry Profile	   113
  Data Gaps	   113
  Required Labeling	   113
 TOPICAL DISCUSSIONS
  Chemical Identity	   114
  Manufacturing Process	   114
  Formation of Unintentional Ingredients	   114
  Ingredients in Pesticide Products	   114
  Product Analytical Methods and Data	   115
  Physical/Chemical Properties	   115

IV.  Environmental Fate	   117
 DISCIPLINARY REVIEW
  Environmental Fate Profile	   117
  Exposure Profile	   117
  Required Labeling	   117

V-  Toxicology	   119
 DISCIPLINARY REVIEW
  Toxicology Profile	   119
  Toxicology Hazard Assessment	   119
  Data Gaps	   120
  Required Labeling	   122
 TOPICAL DISCUSSIONS
  Acute Effects	   122
  Local Irritation	   124
  Bibliography	   127

                       -iv-

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VI.  Ecological Effects	
 DISCIPLINARY REVIEW
  Ecological Effects Profile	   129
  Required Labeling	   129
 TOPICAL DISCUSSIONS
  Terrestrial Plants	   129
  Freshwater Fish	   130
  Bibliography	   131

BIBLIOGRAPHY	   133

APPENDIX A - Toxicity Category Warning and
First Aid Statements	   147
                       -v-

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                                   Chapter  1

                               HOW TO REGISTER
                        UNDER A REGISTRATION STANDARD
Organization of the Standard
Purpose of the Standard
Requirement to Re-register Under the Standard
"Product Specific" Data and "Generic" Data
Data Compensation Requirements under FIFRA 3(c)(1)(D)
Obtaining Data to Fill "Data Gaps"; FIFRA 3(c)(2)(B)
Amendments to the Standard
Organization of the Standard

    This first chapter explains the purpose of a Registration Standard and
summarizes the legal principles involved in registering or re-registering under
a Standard.  The second chapter sets forth the requirements that must be met  to
obtain or retain registration for products covered by this particular
Registration Standard.  In the remaining chapters, the Agency reviews the
available data by scientific discipline, discusses the Agency's concerns with
the identified potential hazards, and logically develops the conditions and
requirements that would reduce those hazards to acceptable levels.


Purpose o: the Standard

    Section 3 of the Federal Insecticide, Fungicide, and Rodenticide Act
(FIFRA) provides that "no person in any State may distribute, sell, offer for
sale, hold for sale, ship, deliver for shipment, or receive (and having so
received) deliver or offer to deliver, to any person any pesticide which is not
registered with the Administrator [of EPA]."  To approve the registration of  a
pesticide, the Administrator must find, pursuant to Section 3(c)(5) that:
    "(A) its composition is such as to warrant the proposed claims for it;
     (B) its labeling and other material required to be submitted comply with
         the requirements of this Act;
     (C) it will perform its intended function without unreasonable adverse
         effects on the environment; and
     (D) when used in accordance with widespread and commonly recognized
         practice it will not generally cause unreasonable adverse effects on
         the environment."
    In making these findings, the Agency reviews a wide range of data which
registrants are required to submit, and assesses the risks and benefits
associated with the use of the proposed pesticide.  But the established
approach to making these findings has been found to be defective on two counts:
    First, EPA and its predecessor agency, the United States Department of
Agriculture (USDA), routinely reviewed registration applications on a 'product
by product' basis, evaluating each product-specific application somewhat
independently.'  In the review of products containing similar components, there
was little opportunity for a retrospective review of the full range of
pertinent data available in Agency files and in the public literature.  Thus
the 'product by product1 approach was often inefficient and sometimes resulted
in inconsistent or incomplete regulatory judgments.

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    Second, over the years, as a result of inevitable and continuing advances
in scientific knowledge, methodology, and policy, the data base for many
pesticiaes came to be considered inadequate by current scientific and
regulatory standards.  Given the long history of pesticide regulation in
several agencies, it is even likely that materials may have been lost from the
data files.  When EPA issued new requirements for registration in 1975  (40 CFR
162) ana proposed new guidelines for hazard testing in 1978 (43 FR 29686, July
10, 1973 and 43 FR 37336, August 2, 1973), many products that had already been
registered for years were being sold and used without the same assurances of
human and environmental safety as was being required for new products.  Because
of this inconsistency, Congress directed EPA to re-register all previously
registered products, so as to bring their registrations and their data bases
into compliance with current requirements [See FIFRA Section 3(g)l-
    Facing the enormous job of re-reviewing and calling-in new data for the
approximately 35,000 current registrations,  and realizing the inefficiencies of
the 'product by product' approach, the Agency decided that a new, more
effective method of review was needed.
    A new review procedure has been developed.  Under it, EPA publishes
documents called Registration Standards, each of which discusses a particular
pesticide active ingredient.  Each Registration Standard summarizes all the
data available to the Agency on a particular active ingredient ana its current
uses, and sets forth the Agency's comprehensive position on the conditions and
requirements for registration of all existing and future products which contain
that active ingredient.  These conditions and requirements, all of which must
be met to obtain or retain full registration or re-registration under Section
3(c)(5) of FIFRA, include the submission of needed scientific data which the
Agency does not now have, compliance with standards of toxicity, composition,
labeling, and packaging, and satisfaction of the data compensation provisions
of FIFRA Section 3(c)(1)(D).
    The Standard will also serve as a tool for product classification.  As part
of the registration of a pesticide product,  EPA may classify each product for
"general use" or "restricted use" [FIFRA Section 3(d)].  A pesticide is
classified for "restricted use" when seme special regulatory restriction is
needed to ensure against unreasonable adverse effects to man or the
environment.  Many such risks of unreasonable adverse effects can be lessened
if expressly-designed label precautions are strictly followed.  Thus the
special regulatory restriction for a "restricted use" pesticide is usually a
requirement that it be applied only by, or under the supervision of, an
applicator who has been certified by the State or Federal government as being
competent to use pesticides safely, responsibly, and in accordance with label
directions.  A restricted-use pesticide can  have other regulatory restrictions
[40 CFR 162.11(c)(5)] instead of, or in addition to, the certified applicator
requirement.  These other regulatory restrictions may include such actions as
seasonal or regional limitations on use, or a requirement for the monitoring of
residue levels after use.  A pesticide classified for "general use," or not
classified at all, is available for use by any individual who is in compliance
with State or local regulations.  The Registration Standard review compares
information about potential adverse effects of specific uses of the pesticide
with risk criteria listed in 40 CFR 162.1 He), and thereby determines whether a
product needs to be classified for "restricted use."  If the Standard does
classify a pesticide for "restricted use," this determination is stated in the
second chapter.

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Requirement _to Re-register Under the Standard

    FIFHA Section 3(g), as amended in  1978, directs EPA to re-register  all
currently registered products as expeditiously as possible.  Congress also
agreed that re-registration should be accomplished by the use of  Registration
Standards.
    Each registrant of a currently registered product to which this  Standard
applies, and who wishes to continue to sell or distribute his product in
commerce, must apply for re-regisration.  His application must contain  proposed
labeling that complies with this Standard.
    EPA will issue a notice of intent to cancel the registration  of  any
currently registered product to which this Standard applies if the registrant
fails to comply with the procedures for re-registration set forth in the
Guidance Package which accompanies this Standard.


"Product Specific" Data and "Generic" Data

    In the course of developing this Standard, EPA has determined the types of
data needed for evaluation of the properties and effects of products to which
the Standard applies, in the disciplinary areas of Product Chemistry,
Environmental Fate,  Toxicology, Residue Chemistry, and Ecological Effects.
These determinations are based primarily on the data Guidelines proposed in
1978 (43 FR 29686, July 10, 1978, and 43 FR 37336, August 2, 1978), as applied
to the use patterns of the products to which this Standard applies.  Where it
appeared that data from a normally applicable Guidelines requirement was
actually unnecessary to evaluate these products, the Standard indicates that
the requirement has been waived.  On the other hand, in some cases studies not
required by the Guidelines may be needed because of the particular composition
or use pattern of products the Standard covers;  if so, the Standard explains
the Agency's reasoning.  Data guidelines have not yet been proposed  for the
Residue Chemistry discipline, but the requirements for such data  have been in
effect for some time and are, the Agency believes, relatively familiar  to
registrants.  Data which we have found are needed to evaluate the
registrability of some products covered by the Standard may not be needed  for
the evaluation of other products, depending upon the composition,-formulation
type, and intended uses of the product in question.  The Standard states which
data requirements apply to which product categories.  (See the second chapter.)
    The various kinds of data normally required for registration  of a pesticide
product can be divided into two basic groups;

    (A)  data that is "product specific," i.e., data that relates only to
         the properties or effects of a product with a particular composition
         (or a group of products with closely similar composition); and
    (B)  "generic" data that pertains to the properties or effects of a
         particular ingredient, and thus is relevant to an evaluation of the
         risks and benefits of all products containing that ingredient  (or all
         such products having a certain use pattern), regardless  of any such
         product's unique composition.

    The Agency requires certain "product specific" data for each  product to
characterize the product's particular composition and physical/chemical
properties (Product Chemistry), and to characterize the product's acute
toxicity (which is a function of its total composition).  The applicant for
registration or re-registration of any product, whether it is a manufacturing-
use or end-use product, and without regard to its intended use pattern, must

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submit or  cite  enough of  this  kind  of data to allow EPA to evaluate the
product.   For such  purposes, "product specific"  data on any product other than
the applicant's is  irrelevant,  unless the  other  product is closely similar in
composition  to  the  applicant's.  (Where it has been found practicable to group
similar products  for purposes  of evaluating,  with a single set of tests,  all
products in  the group,  the  Standard so indicates.)  "Product specific" data on
the efficacy of particular  end-use  products is also required where the exact
formulation  may affect  efficacy and where  failure of efficacy could cause
public health problems.
    All other data  needed to evaluate pesticide  products concerns the
properties or effects of  a  particular ingredient of products (normally a
pesticidally active ingredient, but in some cases a pesticidally inactive,  or
"inert," ingredient).   Some data in this "generic" category are required to
evaluate the properties and effects of all products containing that ingredient
[e.g., the acute LD-50 of the  active ingredient  in its  technical or purer
grade; see proposed 40  CFR  163.81-1 (a), 43 FR 37355].
    Other  "generic" data  are required to evaluate all products which both
contain a  particular ingredient and are intended for certain uses (see,  e.g.,
proposed 40  CFR 163.82-1, 43 FR 37363,  which  requires subchronic oral testing
of the active ingredient  with  respect to certain use patterns only).  Where a
particular data requirement is use-pattern dependent, it will apply to each
end-use product which is  to be labeled for that  use pattern (except where such
end-use product is  formulated  from  a registered  manufacturing-use product
permitting such formulations)  and to each  manufacturing-use product with
labeling that allows it to  be  used  to make end-use products with that use
pattern.   Thus, for example, a subchronic  oral dosing study is needed to
evaluate the safety of any  manufacturing-use  product that legally could  be  used
to make an end-use, food-crop  pesticide.   But if an end-use product's label
specified  it was  for use  only  in ways that involved no  food/feed exposure and
no repeated  human exposure, the subchronic oral  dosing  study would not be
required to  evaluate the  product's  safety; and  if a manufacturing-use
product's  label states that the product is for use only in making end-use
products not involving food/feed use or repeated human  exposure,  that
subchronic oral study would not be  relevant to the evaluation of the
manufacturing-use product either.
    If a registrant of a  currently  registered manufacturing-use or end-use
product wishes  to avoid the costs of data  compensation  [under FIFRA  Section
3(c)(1)(D)]  or  data generation  [under Section 3(c)(2)(B)] for "generic" data
that is required  only with  respect  to some use patterns,  he may elect to  delete
those use  patterns  from his labeling at the time he re-registers his product.
An applicant for  registration of a  new  product under this Standard may
similarly  request approval  for  only certain use  patterns.


Data Compensation Requirements  under FIFRA 3(c)(1)(D)

    Under  FIFRA Section 3(c)(1)(D),  an  applicant for registration,  re-
registration, or  amended  registration must offer to pay compensation for
certain existing  data the Agency has  used  in  developing  the Registration
Standard.  The  data for which compensation must  be offered is all data which is
described by all  the following  criteria:

    (1)  the data were first submitted  to  EPA (or to its  predecessor agencies,
         USDA or  FDA),  on or after  January 1,  1970;
    (2)  the data were submitted to  EPA  (or USDA or FDA)  by some other
         applicant or registrant in support of an  application  for an

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         experimental use permit, an amendment adding a  new  use  to a
         registration, or for re-registration, or  to support or  maintain in
         effect an existing registration;
    (3)  the data are relevant to the Agency's decision  to register or re-
         register the applicant's product under th,e Registration Standard,
         taking into account the applicant's product's composition and intended
         use pattern(s);
    (4)  the data are determined by EPA to be valid and  usable in reaching
         regulatory conclusions; and
    (5)  the data are not those for which the applicant  has  been exempted by
         FIFRA Section 3(c)(2)(D) from the duty to offer to  pay  compensation.
         (This exemption applies to the "generic" data concerning the  safety of
         an active ingredient of the applicant's product, not to "product
         specific" data.  The exemption is available only to applicants  whose
         product is labeled for end-uses for which the active ingredient in
         question is present in the applicant's product  because  of his use of
         another registered product containing that active ingredient  which  he
         purchases from another producer.)

    An applicant for re-registration of an already registered product  under
this Standard, or for registration of a new product under this Standard,
accordingly must determine which of the data used by EPA in  developing the
Standard must be the subject of an offer to pay compensation, and oiust submit
with his application the appropriate statements evidencing his compliance with
FIFRA Section 3(c)(1)(D).
    An applicant would never be required to offer to pay for "product  specific"
data submitted by another firm.  In many, if not in most cases,  data which are
specific to another firm's product will not suffice to allow EPA to evaluate
the applicant's product, that is, will not be useful to  the  Agency in  determin-
ing whether the applicant's product is registrable.  There may be cases,  how-
ever,  where because of close similarities between the composition of two or
more products, another firm's data may suffice to allow  EPA  to evaluate  some or
all of the "product specific" aspects of the applicant's product.   In  such a
case,  the applicant may choose to cite that data instead of  submitting data
from tests on his own product,  and if he chooses that option, he  would have  to
comply with the offer-to-pay requirements of Section 3(C)(1)(D)  for that data.
    Each applicant for registration or re-registration of a  manufacturing-use
product, and each applicant for registration or re-registration  of an  end-use
product, who is not exempted by FIFRA Section 3(c)(2)(D), must comply  with the
Section 3(c)(1)(D) requirements with respect to each item of "generic" data
that relates to his product's intended uses.
    A detailed description of the procedures an applicant must follow  in
applying for re-registration (or new registration) under this Standard is found
in the Guidance Package for this Standard.


Obtaining Data to Fill "Data Gaps"; FIFRA 3(c)(2)(B)

    Some of the kinds of data EPA needs for its evaluation of the properties
and effects of products to which this Standard applies have  never been
submitted to the Agency (or, if submitted, have been found to have deficiencies
rendering them inadequate for making registrability decisions) and 'nave  not
been located in the published literature search that EPA conducted as  part of
preparing this'Standard.  Such instances of missing but  required data  are
referred to in the Standard as "data gaps".

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    FIFRA  Section  3(c)(2)(B),  added  to  FIFRA by  the  Congress  in 1978,
autnorizes EPA  to  require  registrants to whom a  data requirement applies to
generate (or otherwise  produce)  data to fill such  "gaps"  and  submit  those data
to  EPA.  EPA must  allow a  reasonably sufficient  period for this to be
accomplished.   If  a  registrant fails to take appropriate  and  timely  steps to
fill  the data gaps identified  by a section 3(c)(2)(B)  order,  his product's
registration may be  suspended  until  the data are submitted.   A mechanism is
provided whereby two or more registrants may agree to share  in the costs of
producing  data  for which they  are both  responsible.
    The Standard lists, in its summary  second chapter, the "generic" data gaps
and notes  the classes of products to which these data gaps pertain.  The
Standard also points out that  to be  registrable  under the Standard,  a  product
must  be supported  by certain required "product spe::fic"  data.  In some cases,
the Agency may  possess  sufficient "product specific" data on  one currently
registered product,  but may lack such data on another. Only  those Standards
which apply to  a very small number of currently  registered products  will
attempt to state definitively  the "product specific" data gaps on a 'product by
product' basis.  (Although the Standard will in  some cases note which  data that
EPA does possess would  suffice to satisfy certain  "product specific" data
requirements for a category of products with closely similar  composition
characteristics.)
    As part of  the process of  re-registering currently registered products, EPA
will  issue Section 3(c)(2)(B)  directives requiring the registrants to  take
appropriate steps  to fill  all  identified data gaps — whether that data in
question is "product specific" or "generic" — in  accordance  with a  schedule.
    Persons who wish to obtain registrations for new products under  this
Standard will be required  to submit  (or cite) sufficient  "product specific"
data  before their  applications are approved.  Upon registration, they  will be
required under  Section  3(c)(2)(B) to take appropriate steps to submit  data
needed to  fill  "generic" data  gaps.  (We expect  they will respond to this
requirement by entering into cost-sharing agreements with other registrants who
previously have been told  they must  furnish the  data.) The Guidance Package
for this Standard  details  the  steps  that must be taken by registrants  to comply
with  .Section 3(c)(2)(B).
Amendments to the Standard

    Applications for registration which  propose  uses or  formulations  that  are
not presently covered by the Standard, or which  present  product compositions,
product chemistry data, hazard data,  toxicity  levels, or labeling  that  do  not
meet the requirements of the Standard, will automatically be considered by the
Agency to be requests for amendments  to  the Standard.  In response to such
applications, the Agency may request additional  data to  support the proposed
amendment to the Standard, or may deny the application for  registration on the
grounds that the proposed product would  cause  unreasonable  adverse effects to
the environment.  In the former case, when additional data  have been
satisfactorily supplied, and providing that the  data do  not indicate  the
potential for unreasonable adverse effects, the  Agency will then amend  the
Standard to cover the new registration.
    Each Registration Standard is based  upon all data and information available
to the Agency's reviewers on a particular date prior to  the publication date.
Tnis "cut-off" date is stated at the beginning of the second chapter.   Any
subsequent data submissions and any approved amendments  will be incorporated
into the Registration Standard by means  of addenda, which are available for
inspection at SPA in Washington, D.C., or copies of which may be requested from

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the Agency.  When all the present "data gaps" have been filled and the
submitted data have been reviewed, the Agency will revise the Registration
Standard.  Thereafter, when the Agency determines that the internally
maintained addenda have significantly altered the conditions for registration
under the Standard, the document will be updated and re-issued for publication.
    While the Registration Standard discusses only the uses and hazards of
products containing the designated active ingredient(s), the Agency is also
concerned with the potential hazards of some inert ingredients and impurities.
Independent of the development of any one Standard,  the Agency has initiated
the evaluation of some inert pesticide ingredients.   Where the Agency has
identified inert ingredients of concern in a specific product to which the
Standard applies, these ingredients will be pointed  out in the Guidance Package.
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                REGULATORY POSITION

    This chapter presents the Agency's decision on what

Standards of product composition, toxicity, use, labeling,

and packaging are required for the pesticide active ingredient

in question.  The decision complies with the rules and

regulations (40 CFR 162) used to implement the Federal

Insecticide, Fungicide, and Rodenticide Act, as amended

(FIFRA), and with the Agency's present regulatory policies.

There are different requirements for manufacturing-use

chemicals and for each type of end-use formulation which

present a significantly different set of hazards.   This

Registration Standard is based upon all data and information

on Aspon^* available to the Agency's reviewers as  of February 27,

1979.

    Companies which have submitted data in support of

their registrations of Aspon® products are Chevron Chemical

Company and Stauffer Chemical Company, both of Richmond,

Calif., and O.M. Scott & Sons of Marysville, Ohio.  These

data may be cited by other registrants or applicants for

registration,  when appropriate,  to support the registration(s)

of their own product(s), provided they have offered and
*  Aspon^ is a registered trade name of Stauffer Chemical
Company.  Its use in this document does not constitute
endorsement or recommendation for use by this Agency.  Since
there is no acceptable common name for this compound, the
trade name will be used in this document for convenience.
                       -Q-

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agreed  to pay compensation,  as  required by FIFRA Sections



3(c) (1) (d). and  3(c) (2) (d) .



Manufacturing-Use Aspon™



     The Agency  has  reviewed  all data available to



it.  Although incomplete,  these  data indicate that



manufacturing-use Aspon™ (which includes both the



technical material  and  the granular formulation interme-



diate)  is suitable  for  registration because  it does



not  meet or exceed  the  risk  criteria leading to a



Rebuttable Presumption  Against Registration  [Chapter 40,



Section 162.11(a) of  the  Code of Federal Regulations],



Data gaps have  been identified; when these data are



supplied, the Agency  will again review the registration



status  of this  compound.



     In  order to be  covered under this Standard, a manufactur-



ing-use Aspon® product  must  comply with the  following



standards. A manufacturing-use Aspon™ product must contain



Aspon™  (0,0,0,0-Tetrapropyl  dithiopyrophosphate)  as an



active  ingredient.  Given current manufacturing-use product



grades and formulation  methods, the Agency expects that most



technical material  will  range above 90% a.i. and that most



granular formulation  intermediates will range above 25% a.i.



Should an applicant desire to register a manufacturing-use



product that departs greatly from those currently registered,



that applicant should contact the Agency for specific



directions on how to accomplish registration. Because



Aspon^ is corrosive to  steel, manufacturers of the technical



material may not ship it  in  unlined steel containers.  The



                        -10-

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acute toxicology testing on a manufacturing-use Aspon0'



product must demonstrate into which Toxicity Category (I



through IV) the product falls for the following acute



effects:



         Acute Oral Toxicity;



         Acute Dermal Toxicity;



         Acute Inhalation Toxicity;



         Primary Eye Irritation; and



         Primary Dermal Irritation.



    Labels for currently registered manufacturing-use


     (ft
Asporf£y products must include the following:



    1.  The intended end-use of products formulated from



manufacturing-use products determines which data applicants



for (re)registration of the manufacturing-use product are


                                                        (ft
required to submit or cite.  All manufacturing-use Aspon**



products must therefore carry one of the following statements



on the label:



    a.  For Formulation Into End-Use Insecticide Products



    Intended Only for Domestic, Non-Food, Outdoor Use;



    b.  For Formulation Into End-Use Insecticide Products



    Intended Only for Non-Domestic, Non-Food, Outdoor Use;



    or



    c.  For Formulation Into End-Use Insecticide Products



    Intended Only for Domestic or Non-Domestic, Non-Food,



    Outdoor Use.




                       -11-

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    2.  All manufacturing-use Aspon° products must carry



the following warning on the label, under the "Hazards



to Wildlife" section:



    This pesticide is toxic to fish.  Do not discharge



    into lakes, streams, ponds, or public water unless



    in accordance with NPDES permit.  For guidance, contact



    your Regional Office of the EPA.



    3.  All technical Aspon™ products must carry the



following warning on the label:



    This product is corrosive to steel.  Do not transport



    or store in unlined steel containers.



    4.  Manufacturing-use product labels must comply with



the requirements of 40 CFR 162.10 regarding label format,



including placement of hazard warnings on the label, type



size and color, etc.



    To be covered under this Standard, all applicants for



registration or re-registration of technical and formulation



intermediate products must agree to cite or submit the



following information on the composition and toxicity of



each proposed product.  After each data gap is listed the



section in the Proposed Guidelines which describes that type



of data and when it is required [43 FR, No. 132, 29696 of



July 10, 1978;  and 43 FR, No. 163, 37336 of August 22,



1978].  While the Agency does have some limited data on the



product chemistry of Aspon^, possible changes in the



manufacturing processes or product formulation methods may






                       -12-

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affect the product's physical/ chemical characteristics.

All normally required data on physical/chemical  characteristics

are therefore being listed as data gaps, so  that the Agency

can obtain the most current data.
                                          Guidelines  Section
  Product Chemistry
    For Both Technical and Formulation
    Intermediate
    1)  Product Identity	 163.61-3(a)
    2)  Disclosure of Ingredients	 163.61-3(c)
    3)  Description of Manufacturing
       Process	 163.61-4
    4)  Formation of Unintentional
       Ingredients	 163.61-5
    5)  Declaration of Limits.	 163.61-6(a)
    6)  Certification of Limits	 163.61-6(b)
    7)  Analytical Methods	 163.61-7(a)
    8)  Analytical Results	 163.61-7 (b) (1)
    For Technical
    9)  Color	 163.61-8(c) (1)
    10) Odor	 163.61-8(c) (2)
    11) Melting Point	 163.61-8 (c) (3)
    12) Solubility (in quantitative
        terms)	 163. 61-8 (c) (4)
    13) Stability	 163.61-8 (c) (5)
    14) Octanol/Water Partition
        Coefficient	 163.61-8 (c) (6)
    15) Physical State	 163.61-8 (c) (7)
    16) Density or Specific Gravity	163.61-8(c) (8)
    17) Boiling Point	 163.61-8 (c) (9)
    18) Vapor Pressure	 163.61-8 (c) (10)
    19) pH	 163.61-8(c) (11)
    For Formulation Intermediate
    20) Density or Specific Gravity	163.61-8 (c) (8)
    21) Storage Stability	 163.61-8 (c) (12)
    22) Flammability	 163.61-8 (c) (13)
    23) Oxidizing or Reducing Action	163.61-8 (c) (14)
    24) Explosiveness	 163.61-8 (c) (15)
    25) Corrosion Characteristics	 163.61-8 (c) (18)
                       -13-

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                                          Guidelines Section
 *Toxicology
    1) Acute Oral Toxicity Study	 163.81-1
    2) Acute Dermal Toxicity Study	 163.81-2
    3) Acute Inhalation Toxicity Study... 163.81-3
    4) Primary Eye Irritation Study	 163.81-4(c)
       OR
       Data on pH of the Product	 163.81-4 (b)
    5) Primary Dermal Irritation Study... 163.81-5
    6) Dermal Sensitization Study	 163.81-6

    To be covered under this Standard, applicants  for

registration or re-registration of technical and formulation

intermediate products which are labeled for formulation into

products intended for non-domestic or domestic, outdoor,

non-food, use must agree to submit or cite all of  the

information required above, as well as the following informa-

tion:

Non-Domestic or Domestic Use
                                          Guidelines Section
  Environmental Fate
    1) Hydrolysis	 163.62-7(b)
    2) Photolysis (in water)	 163.62-7(c)
    3) Aerobic Soil Metabolism	 163.62-8(b)
    4) Microbial Metabolism	 163.62-8 ( f) (2)
    5) Activated Sludge Metabolism	 163.62-8 (g)
    6) Leaching	 163.62-9(b)
    7) Adsorption/Desorption	 163.62-9(d)
    8) Field Dissipation study on
       representative emulsifiable con-
       centrate and granular formula-
       tions	 163.62-10'
    9) Fish Accumulation	 163.62-ll(d)
  Toxicology
    1) Teratogenicity Study	 163.83-3
    2) Acute Delayed Neurotoxicity	 163.81-7
"*A demonstration that a manufacturing-use
product has a composition substantially similar to a
manufacturing-use product for which the Agency already
has acceptable acute toxicity data will satisfy acute
toxicity data requirements for the former product.  Both
active and inert ingredients will be considered in making
determinations of similarity.
                       -14-

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                                          Guidelines  Section
   Ecological  Effects
     1) Microbial  Metabolism	 163. 62-8 ( f) (3)
     2) The  avian  acute  oral  LD-50  for
       one  species  of waterfowl  (pref-
       erably  the mallard) ££  one  species
       of upland  game bird  (preferably
       the  bobwhite, other native  quail,
       or the  ring-necked pheasant)	 163.71-1
     3) A 48-hour  LC-50  (or EC-50)  for
       one  species  of aquatic  inverte-
       brate  (preferably Daphnia magna).. 163.72-2
Rmulsif iable Concentrate
     In order  to be covered under  this Standard, an  end-use

emulsif iable  concentrate  (EC) Aspon™ product must contain

     (ft
Aspon0* (0,0,0, 0-Tetrapropyl dithiopyrophosphate) as an

active ingredient.  FIFRA Section 162.11(c) lists the

criteria for  classifying pesticides for restricted, non-

domestic, or  domestic use.
            (»
     EC Aspon0* products which are shown to have a Toxicity

Category I rating for any of the following acute effects

must be classified for restricted use (i.e., for retail sale

to and application only by certified applicators or persons

under their direct supervision) :

         Acute Oral Toxicity;

         Acute Dermal Toxicity; or

         Acute Inhalation Toxicity.

    EC Aspon^ products which are shown to have a Toxicity

Category II rating for any of the following acute effects

must be classified for non-domestic use:

         Acute Oral Toxicity;
                       -15-

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         Acute Dermal Toxicity; or

         Acute Inhalation Toxicity.
            (6)
    EC Aspon"^ products which are shown to have any of the

following Toxicity Category ratings may be classified for

domestic use:

         Acute Oral Toxicity:  Category III or IV

         Acute Dermal Toxicity:  Category III or IV

         Acute Inhalation Toxicity: Category III or IV

         Primary Eye Irritation:  Category I through IV

         Primary Dermal Irritation:  Category I through IV

EC products  intended for domestic use with Toxicity Category

I or II ratings for primary eye or dermal irritation must

meet the criteria for child-resistant packaging [see FR

44(48):13019-13024, March 9, 1979].

    Labels for currently registered EC Aspon^ products

must include the following:

    1.  If EC Aspon® products contain petroleum distillates,

the statement "Contains petroleum distillates" must appear

on the label in close proximity to the ingredient statement.

Active ingredient:
    0,0,0,0-Tetrapropyl dithiopyrophosphate	     %
Inert Ingredients*	     %
Total	  100%
*Contains Petroleum Distillates
    2.  If the EC Aspon0' product has an Acute Oral Toxicity

Category IV and contains greater than 10% by weig-ht petroleum

distillates, the following first aid statement must appear

on the label (see also Table 2, Appendix A):

                       -16-

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    If_ swallowed;   If the patient  is unconscious, main-



    tain breathing  and heart rate  (CPRrcardiopulmonary



    resuscitation).  Contact your  local Poison Control



    Center, physician, or hospital  immediately-  Do Not



    Induce Vomiting!



    If the EC Aspon® product has an Acute Oral Toxicity



Category I and contains greater than 10% by weight petroleum



distillates, the following first aid statement must appear



on the label (see also Table 2, Appendix A):



    ^_f swallowed;   If the patient  is unconscious, main-



    tain breathing  and heart rate  (CPR:cardiopulmonary



    resuscitation).  Contact your  local Poison Control



    Center, physician, or hospital  immediately.  If the



    patient is conscious, induce vomiting (syrup of ipecac;



    if not available, stimulate the back of the throat



    with finger).  Never give anything by mouth to an



    unconscious person!



    If the EC Aspon™ product has an Acute Oral Toxicity



Category II or III  and contains greater than 10% by weight



petroleum distillates, the following first aid statement



must appear on the label (see also Table 2, Appendix A):



    If swallowed;  If the patient  is unconscious, main-



    tain breathing  and heart rate  (CPR:cardiopulmonary



    resuscitation).  Contact your local Poison Control



    Center, physician, or hospital immediately.





                       -17

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    The question of whether vomiting should or should



not be induced will be determined on a case-by-case basis



based on a review of the toxicity of active ingredients,



inert ingredients, and impurities.



    3.  All EC Aspon® products must carry the following



warning on the label:



    Keep children and pets off treated areas for 48 hours



    after application and until the grass has completely



    d r i ed.



    4.  All EC Aspon^ products must carry the following



warning on the label, under the "Hazards to Wildlife"



section:



    This pesticide is toxic .to fish.  Do not contaminate



    water by cleaning of equipment or disposal of wastes.



    5.  All currently registered EC Aspon™ products



between 12% and 28% a.i. must carry on the label the acute



toxicity hazard warnings and first aid statements required



for the following Toxicity Categories (see Appendix A):



    Acute Dermal Toxicity - III



    Primary Eye Irritation - I



    Primary Dermal irritation - II



    6.  EC product labels must comply with the requirements



of 40 CFR 162.10 regarding label format, including placement



of hazard warnings on the label, type size and color,  etc.



In addition, all labels and labeling intended for agricultural



uses must bear the statement, "This product must be applied



in accordance with 40 CFR 170."  (Registrants may amplify





                       -18-

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 this  statement  on  labels  or  labeling  by  stating the require-

 ments  of  40 CFR Part  170  or  additions thereto  if they

 choose.)

    To be  covered  under  this  Standard, all  applicants for

 registration or  reregistration  of  EC  Aspon™ products  must

 agree  to  submit or  cite  the  following information  on  the

 composition of  each proposed  product.  After each  data gap

 is listed  the section  in  the  proposed Guidelines which

 describes  that  type of data  and when  it  is  required [43 FR,

 No. 132,  29696  of July 10, 1978; and  43  FR,  No.  163,  37336

 of August  22, 1978].

                                          Guidelines  Section
  Product Chemistry
    1)  Product  Identity	 163.61-3(a)
    2)  Disclosure of Ingredients	 163.61-3(c)
    3)  Description of Manufacturing
        Process.	 163.61-4
    4)  Formation of Unintentional
        Ingredients	 163.61-5
    5)  Declaration of Limits	 163.61-6(a)
    6)  Certification of Limits	 163.61-6(b)
    7)  Analytical Methods	 163.61-7(a)
    8)  Analytical Results	 163.61-7 (b) (1)
    9)  Color	 163.61-8(c) (1)
    10) Odor	 163.61-8(c) (2)
    11) Density or Specific Gravity	163.61-8(c) (8)
    12) Storage Stability	 163.61-8 (c) (12)
    13) Flammability	 163.61-8 (c) (13)
    14) Oxidizing or Reducing Action	 163.61-8(c)(14)
    15) Explosiveness	 163.61-8 (c) (15)
    16) Miscibility	 163.61-8 (c) (16)
    17) Viscosity	 163.61-8 (c) (17)
    18) Corrosion Characteristics	 163.61-8 (c) (18)
    19) Dielectric Breakdown Voltage	163.61-8 (c) (19)

    Listed below are the Toxicology data which must be

 submitted or cited to obtain  registration or re-registration

 for EC Aspon™ products.  After each data gap is  listed  the

Section in the Proposed Guidelines of August 22, 1978  (43

 FR, No. 163, 37336) which describes that type  of data  and

when it is required.  The Agency has  determined  that  currently
                       -19-

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registered EC products between 12% and 28% a.i. are substan-

tially similar in composition, and that EC products between

65% and 68% a.i. are substantially similar in composition.

Acute toxicity data available on any one product  in either

group may be cited in support of the registration of any

other product in that group, provided compensation has been

offered for use of these data.  Currently registered EC

Aspon^ products which contain other active ingredients

must be tested individually for each acute effect.

                                          Guidelines Section
ECs Between 12% and 28% a.i.*
         1) Acute oral toxicity (rat)
            on product in upper range
            (i.e., @ 25% a.i.)	 163.81-1
         2) Acute inhalation  (rat)
            on product in upper range
            (i.e., 0 25% a.i.)	 163.81-3

ECs Between 65% and 68% a.i.*
         1) Acute oral toxicity (rat)	 163.81-1
         2) Acute dermal toxicity
            (rabbit)	 163.81-2
         3) Acute inhalation  (rat)	 163.81-3
         4) Primary eye irritation
            (rabbit)	 163.81-4 (c)
            OR
            Data on pH of the Product.... 163.81-4(b)
         5) Primary skin irritation
            (rabbit)	 163.81-5
              (ft
ECs With Asjponv and Other Active Ingredients
         1) Acute oral toxicity (rat).... 163.81-1
         2) Acute dermal toxicity
            (rabbit)	 163.81-2
         3) Acute inhalation  (rat)	 163.81-3
*  A demonstration that an EC Aspon0' product has a composi-
tion substantially similar to an EC product for which the
Agency already has acceptable acute toxicity data will
satisfy acute toxicity data requirements for the former
product.  Both active and inert ingredients will be considered
in making determinations of similarity.
                       -20-

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                                          Guidelines Section
         4) Primary eye  irritation
            (rabbit)	 163.81-4 (c)
            OR
            Data on pH of the Product.... 163.81-4 (b)
         5) Primary skin irritation
            (rabbit)	 163.81-5
Granular Aspon^

    In order to be covered under this Standard, an end-use

granular Aspon® product must contain Aspon®  (0,0,0,0-

Tetrapropyl dithiopyrophosphate) as an active ingredient.

FIFRA Section 162.11 (c) lists the criteria for classifying

pesticides for restricted, non-domestic, or domestic use.

    Granular Aspon™ products which are shown to have a

Toxicity Category I rating for any of the following acute

effects must be classified for restricted use (i.e., for

retail sale to and application only by certified applicators

or persons under their direct supervision):

         Acute Oral Toxicity;

         Acute Dermal Toxicity; or

         Acute Inhalation Toxicity.

    Granular Aspon® products which are shown to have a

Toxicity Category II rating for any of the following acute

effects must be classified for non-domestic use:

         Acute Oral Toxicity;

         Acute Dermal Toxicity; or

         Acute Inhalation Toxicity.

    Granular Aspon® products which are shown to have any

of the following toxicity Category ratings may be classified


                       -21-

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for domestic use:



         Acute Oral Toxicity:  Category III or IV



         Acute Dermal Toxicity:  Category III or IV



         Acute Inhalation Toxicity: Category III or IV



         Primary Eye Irritation:  Category I through IV



         Primary Dermal Irritation:  Category I through IV



Granular products intended for domestic use with Toxicity



Category I or II ratings for primary eye or dermal irritation



must meet the criteria for child-resistant packaging [see PR



44(48):13019-13024, March 9, 1979].



    Labels for currently registered granular Aspon^



products must include the following:



    1.   All granular Aspon^ products must carry the



following warning on the label:



    Keep children and pets off treated areas for 48 hours



    after application and until the grass has completely



    d r i ed .


                          (8)
    2.   All granular Aspon** products must carry the



following warning on the label, under the "Hazards to



Wildlife" section:



    This pesticide is toxic to fish.  Do not contaminate



    water by cleaning of equipment or disposal of wastes.


                                               (ft
    3.   All currently registered granular Aspon0^ products



between 1% and fi% a.i. must carry on the label the acute



toxicity hazard warnings and first aid statements required



for the following Toxicity Categories (see Appendix A).





                       -22-

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Without Fertilizer
1) Acute Oral Toxicity - III
2) Acute Dermal Toxicity - III
3) Primary Eye Irritation - III
4) Primary Dermal Irritation - III

With Fertilizer
1) Acute Oral Toxicity - III
2) Acute Dermal Toxicity - III
3) Primary Eye Irritation - II
4) Primary Dermal Irritation - III

    4.  Granular product labels must comply with the require-

ments of 40 CFR 162.10 regarding label format, including

placement of hazard warnings on the label, type size and

color, etc.  In addition, all labels and labeling intended

for agricultural use must bear the following statement,

"This product must be applied in accordance with 40 CFR

170."  (Registrants may amplify this statement on labels or

labeling by stating the requirements or 40 CFR Part 170 or

additions thereto if they choose.)

    To be covered under this Standard, all applicants

for registration or reregistration of granular Aspon®

products must agree to submit or cite the following informa-

tion on the composition of each proposed product.   After

each data gap is listed the section in the Proposed Guidelines

which describes that type of data and when it is required

[43 FR, No. 132,  29696 of July 10,  1978;  and 43 FR, No. 163,

37336 of August 22, 1978].

                                          Guidelines Section
  Product Chemistry
    1)  Product Identity	  163.61-3(a)
    2)  Disclosure of Ingredients	  163.61-3(c)
    3)  Description of Manufacturing
       Process	  163.61-4
    4)  Formation of Unintentional
       Ingredients	  163.61-5
    5)  Declaration of Limits	  163.61-6(a)
                       -23-

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[Footnote concluded from previous page.]
**  An acute inhalation toxicity study  is required for
granular products if "20 percent or more of the aerodynamic
equivalent of the formulated product (as registered or under
conditions of use) is composed of particulates not larger
than 10 microns in diameter" [Guidelines Section
1*3.81-3(a) (2)(ii)] .  An acute inhalation test on any
currently registered granular product between 1% and 6% a.i.
may be submitted or cited in support of the registrations of
all currently registered granular products.  A request for
a waiver of this requirement based on percent of particulates
not larger than 10 microns must be made individually
for each product.
                       -24-

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             ASPON®
                 MANUFACTURING-USE 	
          (TECHNICAL AND  FORMULATION  INTERMEDIATE)


I.  Regulatory Position


  A.  Regulatory Decision


    The Agency has reviewed all data available  to  it.


Although  incomplete, these data indicate that manufacturing-


use Aspon® is suitable for registration  because  it does


not meet  or exceed the risk criteria leading to  a Rebuttable


Presumption Against Registration  [Chapter 40, Section


152.11(a) of the Code of Federal Regulations],   Data gaps


have been identified; when these data are supplied, the


Agency will again review the registration status of this


compound.

                                                          (ft
    The Agency has determined that manufacturing-use Aspon**


does not appear to cause an unreasonable adverse effect


with proper label directions and precautions.  Those manufac-


turing-use products currently registered may be  reregistered


subject to the conditions imposed for data requirements, and


new products may also be registered under the terms of this


Standard.


  B.  Criteria for Registration Under the Standard


    To be registered under this Standard, manufacturing-use


       products must meet the following  conditions:


    1.   The manufacturing-use product contains  Aspon® as


    an active  ingredient;


    2.   The manufacturing-use product bears  required labeling;
-25-

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    3.   The manufacturing-use product must list on the label
    the intended end-use(s)  of formulated products produced
    from the manufacturing-use product; and
    4.   The applicant for registration of manufacturing-
    use products complies with all other terms and conditions
    specified in this Standard and hereby offers and agrees
    to  pay compensation to other persons, with regard to the
    approval of this application, to the extent required by
    3(c)(l)(d)  and 3(c)(2)(d) of the Federal Insecticide,
    Fungicide,  and Rodenticide Act [FIFRA], as amended, 7
    U.S.C. 136(c) (1) (d)  and 136 (c) (2) (d) .
  C.  Acceptable Ranges and Limits
    1.   Product Composition Standards
    To  be covered under this Standard, all technical and
formulation intermediate products must contain Aspon^
ro,0,0,0-Tetrapropyl dithiopyrophosphate]  as an active
ingredient.  The Agency will consider for registration
manufacturing-use products which contain any percentage of
active  ingredient.  In addition, currently registered and
proposed manufacturing-use products must agree to submit or
cite the information on product composition identified as
data gaps in Section I.D of this document.
    Standards have not yet been set for contaminants and
inerts  in manufacturing-use Aspon® products.  When standards
are set for any contaminants or inerts in manufacturing-use
Aspon^ products, manufacturing-use products must comply
with those standards.
                       -26-

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     2.   Acute  Toxicity  Limits



     The  Agency will  grant  registration  to  manufacturing-use



 Aspon® products which have Toxicity  Category  I  through  IV



 ratings  for  any of the  following  acute  effects:



   1)  Acute  Oral Toxicity;



   2)  Acute  Dermal Toxicity;



   3)  Acute  Inhalation  Toxicity;



   4)  Primary  Eye Irritation; and



   5)  Primary  Dermal Irritation.



     3.   Use  Patterns



     To be covered under this Standard, manufacturing-use



 (i.e., technical and formulation  intermediate) products must



 carry label  directions  permitting further  formulation into



 end-use  pesticides which are intended only for outdoor,



 non-food, domestic or non-domestic use.  Directions for



 formulation  into products intended for other  end-uses must



 be supported by appropriate data and a petition to amend  the



 Standard to  permit the  extended uses.



  D.  Data Gaps



     To be covered under this Standard, applicants for



 registration or re-registration of technical  and formulation



 intermediate products must agree to cite or submit the



 following information on the composition and  toxicity of



 each proposed product.   After each data gap is listed the



 section  in the Proposed Guidelines which describes that type



 of data  and when it is  required [43 FR,  No. 132, 29696 of



July 10,  1978;  and 43 FR,  No. 163, 37336 of August 22,



 1978].






                       -27-

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                                          Guidelines Section
  Product Chemistry
    For Both Technical and Formulation
    Intermediate
    1)  Product Identity	 163.61-3(a)
    2)  Disclosure of Ingredients	 163.61-3(c)
    3)  Description of Manufacturing
       Process	 163.61-4
    4)  Formation of Unintentional
       Ingredients	 163.61-5
    5)  Declaration of Limits	 163.61-6(a)
    6)  Certification of Limits	 163.61-6(b)
    7)  Analytical Methods	 163.61-7(a)
    8)  Analytical Results	 163.61-7(b) (1)
    For Technical
    9)  Color	 163.61-8(c) (1)
    10) Odor	 163.61-8(c) (2)
    11) Melting Point	 163.61-8 (c) (3)
    12) Solubility (in quantitative
        terms)	 163. 61-8 (c) (4)
    13) Stability	 163.61-8 (c) (5)
    14) Octanol/Water Partition
        Coefficient	 163.61-8 (c) (6)
    15) Physical State	 163.61-8 (c) (7)
    16) Density or Specific Gravity	163.61-8(c) (8)
    17) Boiling Point	 163.61-8 (c) (9)
    18) Vapor Pressure	 163.61-8 (c) (10)
    19) pH	 163.61-8(c) (11)
    For Formulation Intermediate
    20) Density or Specific Gravity	163.61-8 (c) (8)
    21) Storage Stability	 163.61-8 (c) (12)
    22) Flammability	 163.61-8 (c) (13)
    23) Oxidizing or Reducing Action	163.61-8 (c) (14)
    24) Explosiveness	 163.61-8 (c) (15)
    25) Corrosion Characteristics	 L63.61-8(c)(18)
 *Toxicology
    1)  Acute Oral Toxicity Study	 163.81-1
    2)  Acute Dermal Toxicity Study	 163.81-2
    3)  Acute Inhalation Toxicity Study... 163.81-3
    4)  Primary Eye Irritation Study	 163.81-4(c)
       OR
       Data on pH of the Product	 163.81-4(b)
    5)  Primary Dermal Irritation Study... 163.81-5
    6)  Dermal Sensitization Study	 163.81-6
*  A demonstration that a manufacturing-use Aspon**
product has a composition substantially similar to a
manufacturing-use product for which the Agency already
has acceptable acute toxicity data will satisfy acute
toxicity data requirements for the former product.  Both
active and inert ingredients will be considered in making
determinations of similarity.
                       -28-

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    To be covered under this Standard, applicants  for

registration or re-registration of technical and formulation

intermediate products which are labeled for formulation  into

products intended for outdoor, non-food, non-domestic or

domestic uses must agree to submit or cite all of  the

information required above, as well as the following informa-

tion:

Non-Domestic or Domestic Use
                                          Guidelines Section
  Environmental Fate
    1) Hydrolysis	 163.62-7(b)
    ?.) Photolysis (in water)	 163.62-7(c)
    3) Aerobic Soil Metabolism	 163.62-8(b)
    4) Microbial Metabolism	 163.62-8( f) (2)
    5) Activated Sludge Metabolism	 163.62-8(g)
    6) Leaching	 163.62-9(b)
    7) Adsorption/Desorption	 163.62-9(d)
    8) Field Dissipation study on
       representative emulsifiable con-
       centrate and granular formula-
       tions	 163.62-10
    9) Fish Accumulation	 163.62-ll(d)
  Toxicology
    1) Teratogenicity Study	 163.83-3
    2) Acute Delayed Neurotoxicity	 163.81-7
  Ecological Effects
    1) Microbial Metabolism	 163.62-8 (f) (3)
    2) The avian acute oral LD-50 for
       one species of waterfowl (pref-
       erably the mallard)  o_r one species
       of upland game bird (preferably
       the bobwhite, other native quail,
       or the ring-necked pheasant)	 163.71-1
    3) A 48-hour LC-50 (or EC-50)  for
       one species of aquatic inverte-
       brate (preferably Daphnia magna).. 163.72-2

  R.  Required Labeling

    1.  Product Chemistry

    The ingredient statement will list the active  ingredient

as:   0,0,0,0-Tetrapropyl dithiopyrophosphate.   In all cases,
                       -29-

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the percentage by weight of active ingredient and inerts

must equal 100%.

Active Ingredient:
    0,0,0,0,-Tetrapropyl dithiopyrophosphate	     %
Inert Ingredients		%
Total	  100%

    ?.  Human Hazard - Precautionary Labeling

    The hazard warnings and first aid statements on all

manufacturing-use product labels must correspond to the

^oxidty Category assigned to that product for each acute

effect.  Tables 1 and 2 in Appendix A list the required

labeling for each acute Toxicity Category (for more detailed

information, see 40 CFR 162.10 on labeling requirements).

    3.  Environmental Hazards

    All manufacturing-use product labels must include the

following warning:

    "This pesticide is toxic to fish.  Do not discharge

    into lakes, streams, ponds, or public water unless

    in accordance with NPDES permit.  For guidance, contact

    your Regional Office of the EPA."

    4.  Physical or Chemical Hazards

    Manufacturers of the technical chemical may not ship it

to formulators in unlined steel containers.  In addition,

the technical label should include the following warning,

for the information of formulators who use the technical

product to manufacture end-use products:

    "This product is corrosive to steel.  Do not transport

    or store in unlined steel containers."


                       -30-

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    5.  Use Patterns



    All manufacturing-use Aspon™ products must list on the



label the intended end-use(s)  of formulated products produced



from the manufacturing-use products.   All manufacturing-use



Aspon^ product labels must contain one of the following



statements:



    1.  "For Formulation Into  End-use Insecticide Products,



    Intended Only For Domestic, Non-food, Outdoor Use";



    or



    2.  "For Formulation Into  End-use Insecticide Products,



    Intended Only For Non-domestic, Non-food, Outdoor Use";



    or



    3.  "For Formulation Into  End-use Insecticide Products,



    Intended Only For Domestic or  Non-domestic,  Non-food,



    Outdoor Use."
                       -31-

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 II.  Regulatory Rationale



  A.  Regulatory Decision



    The Agency has determined that the technical and  formula-


                       (R>
 tion intermediate Aspoa0^ products described  in  this



 Standard can be registered as manufacturing-use pesticides



 for sale, distribution, and reformulation in the United



 States.  There are no data currently available which  suggest

          (Ok

 that Asporf0' meets any of the risk criteria for unreasonable



 adverse effects, as listed in 40 CFR 162.11(a).  In addition,



 to be covered under this Standard, applicants must agree to



 submit or cite the data listed in Section I.D of this



 document.



  R.  Acceptable Ranges and Limits



    1.   Product Composition Standards



    The Agency will consider for registration manufacturing-



 use products which contain any percentage of Aspon™ as



 an active ingredient.  Nevertheless,  given current manufac-



 turing-use product grades and formulation methods,  the



Agency expects that most technical material will range



above 90% a.i.  and that granular formulation intermediates



will range above 25% a.i.   Should an  applicant desire to



 register a manufacturing-use product  that departs greatly



from those currently registered, that applicant should



contact the Agency for specific directions on how to



accomplish regi-stration.
                       -33-

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    2.  Acute Toxicity Limits
    The Agency will register manufacturing-use Aspon®
products which have Toxicity Category I through IV ratings
because the use pattern does not result in possible exposure
to the general public, and because the pesticide industry
can be required to provide safe working conditions (i.e.,
specialized protective clothing such as respirators)  which
will mitigate possible hazards from products with high
toxicity ratings.
    3.  Use Patterns
    Manufacturing-use pesticides may be used only in the
formulation of specific end-use products, because [under
the Proposed Guidelines, 163.40-2(c)  and (d)]  manufactur-
ing-use pesticides are not intended for pesticidal applica-
tion as registered.
  C.  Data Gaps
    The data which applicants are required to submit or
cite in order to obtain (re)registration for manufacturing-use
Aspon^ are listed in Section I.D of this document.
    A field dissipation study on representative emulsifiable
concentrate and granular products is required for all
manufacturing-use products because they are labeled for
formulation into end-use Aspon® products intended for
terrestrial use.  A teratology study is required for
manufacturing-use products labeled for formulation into
domestic or non-domestic end-use products because the use
                       -34-

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pattern could result in exposure to pregnant women.  Other



chronic studies, such as oncogenicity, are not currently



required because the use pattern is not expected to  result



in repeated exposure to humans over a significant portion of



the human life-span.



  D.   Required Labeling



    Acute toxicity hazard warnings must accurately reflect



the product's level of toxicity (products may not be labeled



to show either greater or lesser hazard from the product



than  in fact exists).  Because the currently registered 90%



a.i.  technical product has been determined to be corrosive



to steel, technical manufacturers may not ship the technical



to formulators in unlined steel containers; in addition, the



current label must be modified to include a warning against



transportation or storage in unlined steel containers (see



Section I.E).
                       -35-

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III.  Product Chemistry



    FIFRA 3(c)(2)(A)  requires  the Agency  to  establish



guidelines for  registering pesticides  in  the United  States.



The Agency requires  registrants  to  provide quantitative  data



on all added ingredients, active and inert,  which  are



equal to or greater  than 0.1%  of the product by weight.



    To establish the  composition of products proposed



for registration, the Agency requires  data and informa-'



tion not only on the  manufacturing  and formulation pro-



cesses, but also a discussion  on the formation of manu-



facturing impurities  and other product ingredients,  inten-



tional and unintentional.  Further, to assure that the



composition of  the product as marketed will  not vary



from the composition  evaluated at the  time of registra-



tion, applicants are  required  to submit a statement certify-



ing the upper and lower composition limits for the added



ingredients,  or upper limits only for  some unintentional



ingredients.   Subpart D suggests specific precision limits



for ingredients based on the percentage of ingredient



and the standard deviation of the analytic method.



    In addition to the data on product composition, the



Agency also requires data to establish the physical and



chemical properties of both the pesticide active ingredient



and its formulations.  For example,  data are needed concerning



the identity and physical state of the active ingredient



(e.g., melting'and boiling point data,  vapor pressure






                       -37-

-------
and solubility).  Data are also required on the properties

of the formulated product to establish labeling cautions

(e.g., flammability, corrosivity or storage stability).  The

Agency use.s these data to characterize each pesticide and to

determine its environmental and health hazards.


DISCIPLINARY REVIEW

Chemistry Profile
Data Gaps
Required Labeling

Chemistry.Profile

    "Aspon^" is a trade name for Of0,0,0-Tetrapropyl

dithiopyrophosphate.  The technical material  is a straw-to-

dark amber liquid with a moderately aromatic  odor.  It  is

stable at room temperature, miscible with most organic

solvents, and compatible with commonly-used pest control

materials.  It is corrosive to steel.

Data Gaps

    Listed below are Product Chemistry data needed  to

obtain registration or reregistration for all manufacturing-

use Aspon® products.  After each data gap is  listed the

section  in the Proposed Guidelines (July 10,  1978,  43 FR,

No. 132, 2969*5) which describes that type of  data and when

it is required.

                                          Guidelines Section
    For  Both Technical and Formulation
    Intermediate
    1) Product Identity	 163.61-3 (a)
    2) Disclosure of Ingredients	 163.61-3(c)
    3) Description of Manufacturing
       Process	 163.61-4
    4) Formation of Unintentional
       Ingredients	 163.61-5
    5) Declaration of Limits	 163.61-6(a)
    6) Certification of Limits	 163.61-6(b)
    7) Analytical Methods	 163.61-7(a)
    8) Analytical Results	 163.61-7 (b) (1)
                        -38-

-------
     For Technical
     9T~Color	  163. 61-8 (c) (1)
     10) Odor	  163.61-8(c) (2)
     11) Melting  Point	  163.61-8 (c) (3)
     12) Solubility  (in  quantitative
        terms)	  163. 61-8 (c) (4)
     13) Stability	  163. 61-8 (c) (5)
     14) Octanol/Water Partition
        Coefficient	  163. 61-8 (c) (6)
     15) Physical State	  163.61-8 (c) (7)
     16) Density  or  Specific  Gravity	  163.61-8 (c) (8)
     17) Boiling  Point	  163. 61-8 (c) (9)
     18) Vapor  Pressure	  163. 61-8 (c) (10)
     19) pH	•	  163.61-8(c) (11)
     20) Flammability	  163. 61-8 (c) (13)
     21) Explosiveness	  163. 61-8 (c) (15)
     22) Viscosity	  163. 61-8 (c) (17)
     23) Corrosion Characteristics	  163.61-8(c) (18)
     For Formulation Intermediate
     24) Density  or  Specific  Gravity	  163.61-8 (c) (8)
     25) Storage  Stability	  163. 61-8 (c) (12)
     26) Flammability	  163. 61-8 (c) (13)
     27) Oxidizing or Reducing  Action	  163.61-8 (c) (14)
     28) Explosiveness	  163. 61-8 (c) (15)
     29) Corrosion Characteristics	  163.61-8 (c) (18)

Required Labeling

     Ingredient Statement:  The ingredient  statement  will

list the active  ingredient as  0,0,0,0-Tetrapropyl  dithiopyro-

phosphate.

     Physical Hazard Precautionary  Labeling;   Since the

technical product is corrosive to  steel, technical manufac-

turers may not ship it  to formulators  in unlined  steel

containers, and  the technical  label must carry the following

warning:

     "This product is corrosive to  steel.   Do  not  transport

     or store  in steel  containers."
                       -39-

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TOPICAL DISCUSSIONS

    Corresponding to each of the Topical Discussions

listed below is the number of the section in the 'Pro-

posed Guidelines for Registering Pesticides' of July

10, 1978 (43 FR, No. 132, 29696), which explains the minimum

Product Chemistry data needed in order to obtain registration

or reregistration for manufacturing-use Aspon^ products.

                                          Guidelines Section
Chemical Identity ........................ 163.61-3
Manufacturing Processes .................. 163.61-4
Formation of Unintentional Ingredients... 163.61-5
Ingredients in Pesticide Products ........ 163.61-6
Product Analytical Methods and Data ...... 163.61-7
Physical/Chemical Properties ............. 163.61-8

Chemical Identity

    At present, there is no acceptable common name for

the insecticide, 0,0,0,0-Tetrapropyl dithiopyrophosphate.

         C.H-0.    5   S
          •5 '  ^   n   n
                   ?P-0-
                             OC3H7
Other names, as listed on Chemline (March 1980) are as

follow:

         Thiopyrophosphoric acid [ ( (HO) 2PS) 20] , tetra-

propyl ester (SCI)

         Thiodiphosphoric acid [ ( (HO) 2P (S) ) 20] , tetra-

propyl ester (9CI)

         NPD

         Tetra-n-propyl dithionopyrophosphate

         Tetra-n-propyl dithiopyrophosphate

         Propyl thiopyrophosphate [ ( (PrO) 2P (S) )20]


                       -40-

-------
  Other structural identifiers are:

           CAS Registry No. 3244-90-4


           MF C12H28°5P2S2

           Mol. Wt. 378.43

  Manufacturing Process

      Although details of the present manufacturing process


  are not available,  the published literature  (Sittig, 1971,


  MRDI GS0019-002; Sittig, 1977, MRID GS0019-003) , as well as

  the applicable U.S. patent No. 2,663,722 (1953, MRID GS0019-


  006)  indicate the following reactions occur:



(1)  1        S   I                          S   S
     1C H 0^^ "   f                  c-Pi°\ "   " J^-pi
   21 J   ^>P-C1| + H,0 + 2CcH,.N - >  J   ">P-0-P 2C5H5N + H2° "*" C°2 + 2NaC1

  The  manufacturing processes are not sufficiently detailed

  to satisfy Proposed Guidelines requirements and may not even


  be relevant unless the manufacturer actually uses them.


  Formation of Unintentional Ingredients

      There is no information available to the Agency on the

  formation of unintentional ingredients during the manufacture


  of Aspon"' products.
                         -41-

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Ingredients in Pesticide Products



    For all Aspon^ products, the Agency requires a



listing of the upper and lower limits established  (by



the producer or formulator) for each active ingredient,



and the upper limit for each impurity, reaction product,



and degradation product which is known to be present or



which might reasonably be  identified.



          (a)  manufacturing-use preparation:  the only



    currently registered technical product contains a



    minimum of 90.00% active ingredient (a.i.).



          (b)  formulation  intermediate:  the only currently



    registered formulation  intermediate (25-G) contains



    25.00% a.i.



Product Analytical Methods and Data



    Stauffer (1970, MRDI GS0019-005) and Ja et al.  (1966,



MRID GS0019-001) identify  two methods, infrared (IR) and



thin-layer chromatographic  (TLC)-colorimetric, for  the



analysis  of technical Aspon™.  The IR method is included



in the EPA manual of chemical methods for pesticides (EPA,



1976, MRID GS0019-015).  (The high-resolution nuclear



magnetic  resonance (NMR) spectra of analytical-grade



Aspon®, as a structural identification aid and reference



source, is available from  the literature [Keith et  al.,



1968, MRID 005004395]).



Physical/Chemical Properties



    Color;  The technical  material is a straw-to-dark amber



color  (Stauffer, 1968, MRID GS0019-004).





                       -42-

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    Odor;  The  technical material has  a moderately  aromatic



odor  (Stauffer, 1968, MRID GS0019-004).



    Melting Point;  The melting point  of the  technical



material  is below -40°F  (given as the  freezing point)



[Stauffer, 1968, MRID GS0019-004].



    Solubility;  The solubility of the technical material  is



0.16%  in water  at room temperature (Stauffer, 1968, MRID



GS0019-004) and soluble with difficulty in light petroleum



(Martin and Worthing, 1977, MRID GS0019-017).  It is completely



miscible with all common organic solvents (Stauffer, 1968,



MRID GS0019-004).



    Stability;  The technical material is stable with



insignificant hydrolysis in water at room temperature and



stable for at least 24 hours at 100°C  (Stauffer,  1968,



MRID GS0019-004); it is compatible with commonly-used pest



control materials (Spencer, 1973, MRID GS0019-018).



    Octanol/Water Partition Coefficient;   No data are



available on the technical material.



    Physical State;  The technical material is in liquid



form.  The formulation intermediate is in granular form.



    Density or Specific Gravity;   The technical  material's



specific gravity is 1.119 to 1.123 at 68/68°F [Stauffer,



1968, MRin GS0019-004].   No data are  available on the



formulation intermediate.



    Boiling Point;   The boiling point for the technical



material is 104 C at 0.01 mm Hg (Martin and Worthing,
                       -43-

-------
197*7, MRID GS0019-017)  and 148°C at 2 mm Hg (Spencer, 1973,



MRID GS0019-018).



    Vapor Pressure;  No data are available on the technical



product.



    pH;  No data are available on the technical product.



    Storage Stability;   No data are available on the formula-



tion intermediate.



    Flammability;   The technical material's flash point



[open cup]  is 300°F [Stauffer, 1968, MRID GS0019-004] .  No



data are available on the formulation intermediate.



    Oxidizing or Reducing Action;  No data are avail-



able on the formulation intermediate.



    Explosiveness;  The technical material decomposes



[without explosive hazard] at 300°F [Stauffer, 1968, MRID



GS0019-004].  No data are available on the formulation



intermediate.



    Viscosity;  The technical material's viscosity is 12.5



cp at 70°F [Stauffer, 1968, MRID GS0019-004].



    Corrosion Characteristics;  The technical material may



cause discoloration and physical changes on prolonged



contact with metal; it is corrosive to steel  (Martin and



Worthing, 1977, MRID GS0019-017).  No data are available on



the formulation intermediate.
                       -44-

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                      BIBLIOGRAPHY
 MRID
 GS0019-015
GS0019-001
 005004395
rs0019-017
005001354
005002074
GS 0019-002


GS0019-003


GS0019-018



GS 0019-004


GS0019-005



005004479



GS0019-006
 CITATION
 Chemline,  Chemical Information on Line [Data base].
     Bethesda,  Md:  National  Library of Medicine.
     March  1980.

 EPA.   1976.   EPA manual  of  chemical methods  for
     pesticides and devices.   AOAC,  Arlington,  Virginia.

 Ja, W.;  Smith  W.J.;  Below, J.F.   1966.   The  analysis
     of technical Aspon,  Richmond  Report No.  RR-66-35.
     Stauffer Chemical  Co., New York,  N.Y.

 Keith,  L.H.; Garrison, A.W.;  Alford,  A.L.  1968.  The
     high resolution NMR  spectra of  pesticides.   I.
    organophosphorus pesticides.  J.  Assoc.  Off. Anal.
    Chem.  51(5):1063-1094.

 Martin,  H.; Worthing,  C.R., eds.  1977.  Pesticide
     index: basic information  on the chemicals  used
    as  active  components of pesticides.  5th ed.
    British Crop Protection Council,  Worcestershire,
    England.

 McMahon, B.; Burke, J.A.  1978.  Analytical  behavior data
    for  chemicals  determined  using AOAC multiresidue
    methodology  for pesticide residues  in foods.  J. Assoc.
    Off. Anal. Chem.  61:640-652.

 Ruzicka, J.H.; Thomson, J.; Wheals, B.B.; Wood, N.F.
    1968.  The application of gel chromatography to the
    separation of  pesticides.  Part I.  Organophosphorus
    pesticides.  J. Chromatog.  34(l):14-20.

 Sittig, M.  1971.  Agricultural chemicals manufacture.
    Noyes Data Corp., Park Ridge, N.J.

 Sittig, M.  1977.  Pesticides process encyclopedia.
    Noyes Data Corp., Park Ridge, N.J.

 Spencer, E.Y.  1973.  Guide to the chemicals used in
    crop protection.  6th ed. Canada Dept. of Agri-
    culture, Ontario, Canada.

 Stauffer Chemical Co.  1968.  Aspon insecticide,
    technical information bulletin.  New York, N.Y.

 Stauffer Chemical Co.  1970.  Infrared procedure to
    determine the assay of Aspon, method no. MPO 25-3.
    (Unpublished).  New York, N.Y.

Toy, A.D.F.  1951.   Tetraethyl dithionopyrophosphate
    and related tetraalkyl dithionopyrophosphates.
    J. Am. Chem.  Soc.  73:4670-4674.

 U.S. Patent No. 2,663,722.  1953.  Method of preparing
    tetraalkyl dithionopyrophosphates.
                              -45-

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IV.  Environmental Fate

DISCIPLINARY REVIEW

Environmental Fate Profile
Data Gaps

Environmental Fate Profile

    There are no data currently available on the environ-
                    (R>
mental fate of Aspoa0'.

Data Gaps

    Listed below are the Environmental Fate data needed to

obtain registration or re-registration for manufacturing-use

Aspon® products.  After each data gap is listed the

section in the Proposed Guidelines of July 10, 1978  (43 FR,

Mo. 132 29696) which describes that type of data and when it

is required.

                                          Guidelines Section
    1) Hydrolysis	 163.62-7(b)
    2) Photolysis (in water)	 163.62-7(c)
    3) Aerobic Soil Metabolism	 163.62-8(b)
    4) Microbial Metabolism	 163.62-8 ( f) (2)
    5) Activated Sludge Metabolism	 163.62-8(g)
    6) Leaching	 163.62-9(b)
    7) Adsorption/Desorption	 163.62-9(d)
    8) Field Dissipation study on
       representative emulsifiable con-
       centrate and granular formula-
       tions	 163.62-10
    9) Fish Accumulation	 163.62-ll(d)
                       -47-

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v.   Toxicology

DISCIPLINARY  REVIEW

Toxicology  Profile
Data Gaps
Required Labeling

Toxicology  Profile

     No data are  available  on  technical  or  formulation

                  
-------
    Applicants for registration or re-registration of

technical and formulation intermediate products which are

formulated into products intended for outdoor, non-food,

non-domestic or domestic use must also agree to submit or

cite the following information:

Non-Domestic ££ Domestic Use
                                          Guidelines Section
    1) Teratogenicity Study	 163.83-3
    2) Acute Delayed Neurotoxicity	 163.81-7

Required Labeling

    Product-specific acute toxicity precautionary labeling

is required.  Acceptable categories of acute toxicity,

and the corresponding required precautionary labeling

statements, appear in Appendix A to this document.


TOPICAL DISCUSSIONS

    Corresponding to each of the Topical Discussions

listed below is the number of the section in the 'Proposed

Guidelines' of August 22, 1978 (43 FR, No. 163, 37336) which

explains the minimum Toxicology data needed in order to

obtain registration or reregistration for manufacturing-use

Aspon^ products.

                                          Guidelines Sections
Acute Effects	 163.81-1, -2, -3, and -7
Local irritation	 163.81-4 and -5
Sens itizat ion	 163.81-6
Subchronic 21-Day Dermal	 163.82-2
Subchronic Neurotoxicity	 163.82-5
Teratology	 163.83-3
Mutagenicity	 163.84-1 thru -4
                       -50-

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Acute Effects



    Acute Oral Toxicity



         The minimum data requirement for testing acute oral



    toxicity (LD-50) is one test on each technical and



    formulation intermediate product, preferably using the



    laboratory rat.   No data are available for assessing the



    acute oral LD-50 toxicity of either the technical or the



    formulation intermediate chemicals.



    Acute Dermal Toxicity



         The minimum data requirement for testing acute



    dermal toxicity  (LD-50)  is one test, preferably using



    the albino rabbit,  for each technical and formulation



    intermediate product.  This test should be conducted on



    both intact and  abraded skin.   No data are available for



    assessing the acute dermal LD-50 of  either the technical



    or the formulation  intermediate chemicals.



    Acute Inhalation Toxicity



         The minimum data requirement for testing acute



    inhalation toxicity (LC-50)  is one test for each technical



    and  formulation  intermediate product,  preferably using



    the  laboratory rat.   No  data are available for assessing



    the  acute inhalation LC-50 of  either the  technical  or



    the  formulation  intermediate chemicals.



    Acute Delayed  Neurotoxicity



         Data are  required on the  technical material  if the



    active ingredient,  or any of its metabolites,  degradation
                      -51-

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    products,  or impurities, cause esterase depression or



    are structurally related to a substance that induces



    delayed neurotoxicity-



         Aspon^ is an organophosphate.  Organophosphorus



    pesticides must be tested for acute delayed neurotoxicity.



    The preferred species for testing is the female domestic



    chicken (hen).



         No data are available for assessing the acute



    delayed neurotoxicity of the technical chemical.



Local Irritation



    Primary Eye Irritation



         The minimum data requirement for testing primary



    eye irritation is one test for each technical and



    formulation intermediate product, conducted on a mammal,



    preferably the albino rabbit.  Data which demonstrate



    that the test substance has a pH of 1-3 or 12-14 should



    be submitted instead of data from a primary eye irritation



    test.  For all regulatory purposes, the Agency will



    assume that substances with the above pH values or which



    cause Category I skin effects are corrosive (i.e., have



    a Toxicity Category I rating).  No data are available



    for assessing the primary eye irritation potential of



    either the technical or formulation intermediate chemicals,



    Primary Dermal Irritation



         The minimum data requirement for testing primary



    dermal irritation is one test for each technical and
                       -52-

-------
     formulation  intermediate  product, conducted  on  a  mammal,


     preferably the albino  rabbit.  No data  are available  for


     assessing the primary  dermal  irritation  potential  of


     either the technical or the formulation  intermediate


     chemicals.


Dermal Sensitization


     The minimum  data requirement  for dermal  sensitization


is an intradermal test on  all manufacturing-use  products,


preferably using the albino guinea pig.  These data are


required if repeated human skin contact, under the conditions


of use, is expected.  No data are available  for  assessing


the  dermal sensitization of the technical or formulation


intermediate chemicals.


Subchronic 21-Day Dermal


     This testing may be required on the technical material,


depending on data to be submitted on the persistence of

     /C7\                                                  ft<\
Aspon" as applied under use directions for end-use Aspon0'


products.


Subchronic Neurotoxicity


     This testing may be required on the technical material,


depending on results of the acute delayed neurotoxicity


studies required in this chapter.


Teratology


     The minimum data requirement for teratology  is a test on


the  technical material in two mammalian species.   This test


is required to support the registration of manufacturing-use
                       -53-

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products when their pesticidal end-use may reasonably be


expected to result in significant exposure to human females.


No data are available for assessing the teratology of the


technical product.


Mutagenicity


    The following studies represent only  the minimum require-

                                                          (ft
ments for data on the potential heritable effects of Aspon**:


1.  A mammalian in vitro point mutation test;


2.  A sensitive sub-mammalian point mutation test (bacteria,


    fungi, insect);


3.  A primary DNA damage test (i.e., sister chromatid


    exchange or unscheduled DNA synthesis);


4.  A mammalian in vitro cytogenetics test.  If this test


    suggests a positive result, a dominant lethal or


    heritable translocation test may be required.


    After results from these test systems and other toxicology


disciplines have been considered, additional testing may be


required to further characterize or quantify the potential


genetic risks.


    Although the Agency's mutagenic testing requirements


are not final, the standards for these tests should be


based on the principles set forth therein (FR 43, No.


163, Tuesday, August 22, 1978).  Protocols and choices of


test systems should be accompanied by a scientific rationale.


Substitutions of test systems for those listed above will


be considered after discussion with the Agency.
                       -54-

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    These requirements should be considered an interim



guide and not final Agency policy.  However, the Agency



does consider the above testing scheme to be a reasonable



minimum requirement.



    No data are available for assessing the mutagenicity of



the technical product, but testing may be required when the



Agency's Guidelines on mutagenicity testing are completed.
                       -55-

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VI.  Residue Chemistry

                (6)
    Use of Asporr* is not likely to  result  directly


in residues in human food and animal  feed  items  because


it has not been registered for use  on  food or  feed  crops,


There are no residue data requirements for non-food uses


of Aspon®.
                      -57-

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 VT I.   Ecological  Effects

 DISCIPLINARY  REVIEW

 Ecological  Effects  Profile
 Data  Gaps
 Required Labeling

 Ecological  Effects  Profile

    From the  available  studies,  it  is  apparent  that the

 technical material  is very highly toxic  to  aquatic  organisms,

 particularly  fish.  The technical was  shown  to  be practically

 non-toxic to  birds  in dietary  tests.

 Data  Gaps

    Listed  below are the Ecological Effects  data which must

 be submitted  or cited to obtain  registration or re-registra-
                                a\
 tion  for manufacturing-use  Aspon" products.  After  each

 data  gap is listed  the  section in the  Proposed Guidelines  of

 July  10, 1978  (43 FR, No.  132, 29696)  which  describes that

 type  of data  and when it is required.

                                          Guidelines Section
    1) Microbial Metabolism	 163.62-8 (f) (3)
    2) The avian acute  oral LD-50 for
       one species  of waterfowl  (pref-
       erably  the mallard)  p_r one species
       of upland game bird  (preferably
       the bobwhite, other  native quail,
       or the  ring-necked pheasant)	 163.71-1
    3) A 48-hour LC-50  (or EC-50) for
       one species  of aquatic inverte-
       brate  (preferably Daphnia magna).. 163.72-2

Required Labeling

    All technical and formulation intermediate products intended

 for shipment must bear  the warning:   "This pesticide is

toxic to fish.  Do  not discharge into  lakes, streams, ponds,

or public water unless  in accordance with NPDES permit.  For

guidance, contact your Regional Office of the EPA."


                       -59-

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TOPICAL DISCUSSIONS

    Corresponding to each of the Topical Discussions

listed below is the number of the section in the 'Pro-

posed Guidelines for Registering Pesticides' of July

10, 1978 (43 PR, No. 132, 29696), which explains the minimum

Ecological Effects data needed  in order to obtain registration

                                             (ft
or reregistration for manufacturing-use Aspon^ products.

                                          Guidelines Sections
Microbes	 163.62-8 (f) (3)
Birds	 163.71-1 and  .71-2
Aquatic Invertebrates	 163.72-2
Fish	 163.72-1

Microbes

    Data on the effects of pesticides on microbes are

required to support the registration of manufacturing-

use products labeled for formulation into end-use products

intended for terrestrial, noncrop uses.  There are no

microbial data available on Aspon^.

Birds

    A determination of the single-dose, oral LD50 for

one bird species is required to support the registration

of every manufacturing-use product.  There are no avian

LD_  data available on Aspon^.

    A determination of the avian subacute dietary LC 0

(5-day dietary exposure) is required to support the  registra-

tion of all manufacturing-use products. Acceptable data are

                                 (ft
available on the effects of Aspon0^ in the diet of several

species [see Table 3].  These data indicate that Aspon® is
                       -60-

-------
 practically  non-toxic,  subacutely, to upland game birds and



 wild waterfowl.




                                             (ft
 Table  3.   Subacute  Dietary Toxicity of Aspon^ to Birds
Species
Mallard
duck
Bobwhite
quail
Ring-necked
pheasant
Mallard
duck
Japanese
quail
Formulation
93%
Technical
93%
Technical
95%
Technical
95%
Technical
95%
Technical
LC-50
(ppm)
4353
8414
>5000
>5000

>5000
Reference
Joiner, 1975,
MRID 000004830
Fink and Reno,
1976, MRID
000004831
Hill et al. ,
1975, MRID
GS0019-010
MRID GS0019-01

MRID GS0019-01




0

0
    A decision to require chronic  toxicity data  (reproductive



or simulated and actual field tests), however, will  depend



upon the results of studies on persistence, degradation



rates, and accumulation.



Aquatic Invertebrates



    A determination of the 48-hour EC.... or LC.-,,
                                     50      50


for an aquatic invertebrate species  is required  to support



the registration of all manufacturing-use products.  There



-^_ ..~ ~w._~ v,v.*J.-^J.». „„ „-£-"" .



    The decision to require life-cycle or other  tests on



aquatic invertebrates will depend upon the results of



studies on persistence, degradation  rates, and accumulation.
                       -61-

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Freshwater Fish

    The minimum data required for establishing the acute

toxicity of Aspon*^ in fish is a determination of the

96-hour LC p both for one coldwater fish species (preferably

rainbow trout) and for one warmwater fish species  (preferably

bluegill).  Acceptable data are available on the acute

toxicity of Aspon™ to fish in several EPA tests which

studied its effects on coldwater as well as warmwater fish.

Based on these findings, which are summarized in Table 4,

Aspon^ can be considered to be very highly toxic to

coldwater and warmwater fish species.


Table 4.  Acute Toxicity of Technical Aspon® to Fresh-
          water Fish
 Species
Formulation
LC-50
(ppm)
Reference
 Rainbow Trout
 Rainbow Trout
 Bluegill
90% (Tech.)    0.07
93% (Tech.)    0.1
90% (Tech.)    0.1
        EPAf 1975,
        MRID GS0019-
        007

        EPA, 1976,
        MRID GS0019-
        008

        EPA, 1976,
        MRID GS0019-
        009
    Due to the highly toxic nature of Aspon^ with respect

to coldwater and warmwater fish, further testing  (i.e.,

embryo-larvae and life-cycle tests [Proposed Guidelines

Section 163.72-4]) will depend upon the results of studies

on persistence, degradation rates, and accumulation.
                       -62-

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                    BIBLIOGRAPHY

MRID          CITATION!
GS0019-007    EPA.  1975.  Report on  the  toxicity of  technical
                  Aspon  to rainbow trout.   (U.S. EPA, Chemical  and
                  Biological  Investigations Branch, Beltsville,
                  Maryland, Static jar  test No. 913,  unpublished  report.)

GS0019-008    EPA.  1976.  Report on  the  toxicity of Aspon technical
                  to rainbow  trout.   (U.S.  EPA, Chemical and Biological
                  Investigations Branch,  Beltsville, Maryland, Static
                  jar test No. 932, unpublished.)

GS0019-009    EPA.  1976.  Report on  the  toxicity of Aspon Technical
                  to bluegill sunfish.  (U.S. EPA, Chemical and Biologi-
                  cal Investigations  Branch, Beltsville, Maryland, Static
                  jar test No. 998, 7/14/76, unpublished report.)

000004831     Fink, R.; Reno, F.E.  1976.   Final report:  eight-day
                  dietary LC-50 — bobwhite quail:  project no. 132-129.
                  (Unpublished study  received March 8, 1976 under 476-
                  2163; prepared by Hazleton Laboratories America, Inc.
                  in cooperation with Maryland Dept. of Agriculture, Div.
                  of Inspection and Regulation, submitted by Stauffer
                  Chemical Co., Richmond, Calif.; CDL:225231-A).

GS0019-010    Hill, E.F.; Heath, R.G.; Spann, J.W.; Williams, J.D.
                  1975.  Lethal dietary toxicities of environmental
                  pollutants to birds.  Special Scientific Report—
                  Wildlife No. 191. U.S. Fish and Wildlife Service,
                  Washington, D.C.

000004830     Joiner,  R.L.  1975.  Safety evaluation of Aspon Technical
                  by a five-day feeding test in mallard ducks:  T-5397.
                  (Unpublished study received June 26, 1975 under 476-
                  2163; submitted by Stauffer Chemical Co., Richmond,
                  Calif.; CDL: 223289-A) .
                              -63-

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             EMULSIFIABLE CONCENTRATE ASPON®



I.  Regulatory Position



  A.  Regulatory Decision



    The Agency has reviewed all data available to  it.



Although incomplete, these data indicate that emulsifiable



concentrate (EC)  Aspon® is suitable for registration



because it does not meet or exceed the risk criteria leading



to a Rebuttable Presumption Against Registration [Chapter



40, Section Ifi2.11(a) of the Code of Federal Regulations].



Data gaps have been identified; when these data are supplied,



the Agency will again review the registration status of this



compound.


                                           (R)
    The Agency has determined that EC Aspon0^ does not



appear to cause an unreasonable adverse effect with proper



label directions  and  precautions.   Those EC products currently



registered may be reregistered subject to  the conditions



imposed for data  requirements, and new products may also be



registered under  the  terms of this Standard.



  B.   Criteria for Registration Under the  Standard



    To be registered  under this Standard,  EC  formulations  of



       must meet  the  following conditions:



    1.  The EC product contains Aspon® as  an  active



    ingredient  [if an unregistered source  of Aspon® is



    used in formulating,  then  the  data outlined  under



    Section 162.18-2(c) (d) (1) (iii)  will  be  required];
                       -65-

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    2.   The EC Aspon^ product is within the acute toxicity



    limits  for restricted or general use and bears the



    required labeling;



    3.   The EC Aspon® product is within acceptable



    ranges  for use patterns and application methods;



    and



    4.   The applicant for registration of EC products



    complies with all other terms and conditions specified



    in  this Standard and hereby offers and agrees to pay



    compensation to other persons, with regard to the



    approval of this application, to the extent required by



    3(c)(l)(d) and 3(c)(2)(d) of the Federal Insecticide,



    Fungicide, and Rodenticide Act [FIFRA], as amended, 7



    (I.S.C.  13fi(c)(l)(d)  and 136(c) (2) (d) .



  C.  Acceptable Ranges and Limits



    1.   Product Composition Standards



    To be covered under this Standard, all EC products must



contain Aspon^ [0,0,0,0-Tetrapropyl dithiopyrophosphate]



as an active  ingredient.  The Agency will consider for



registration EC products which contain any percentage of



active ingredient.  In addition, currently registered and



proposed EC products must agree to submit or cite the



information on product composition identified as data



gaps in Section I.D of this document.



    Standards have not yet been set for contaminants and


                  (ft
inerts in EC Aspon** products.  When standards are set for
                       -66-

-------
 any contaminants  or  inerts  in  EC  Aspon° products,  EC



 end-use  products  must  comply with those standards.



    2.   Acute Toxicity Limits



    a.   Restricted Use



    The  Agency will  grant registration  to EC Aspon^



 products as  restricted pesticides  (i.e., for retail sale  to



 and application only by Certified Applicators or persons



 under their  direct supervision) for non-food, outdoor use



 which have a Toxicity  Category I  rating  for any of  the



 following acute effects:



    1) Acute Oral Toxicity;



    2) Acute Dermal Toxicity;



    3) Acute Inhalation Toxicity;



    4) Primary Eye Irritation;  and



    5) Primary Dermal  Irritation.



    b.   Non-Domestic Use



    The  Agency will grant registration  to EC Aspon™



products intended for  non-domestic, non-food,  outdoor use



which have a Toxicity  Category II rating for any of the



following acute effects:



    1) Acute Oral Toxicity;



    2) Acute Dermal Toxicity; or



    3) Acute Inhalation Toxicity;


                                             (ft
The Agency will grant  registration to EC Asponcy products



intended for non-domestic,  non-food, outdoor use which



have a Toxicity Category I  or II rating for  either  of





                       -67-

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the following acute effects:



    1)  Primary Eye Irritation; and



    2)  Primary Dermal Irritation.



    c.   Domestic Use



    The Agency will grant registration to EC Aspon®



products intended for domestic, non-foodf outdoor use which



have a Toxicity Category III or IV rating for any of the



following acute effects:



    1)  Acute Oral Toxicity;



    2)  Acute Dermal Toxicity;



    3)  Acute Inhalation Toxicity;



The Agency will grant registration to EC Aspon^ products



intended for domestic, non-food, outdoor use which have



a Toxicity Category I through IV rating for either of



the following acute effects:



    1)  Primary Eye Irritation; and



    2)  Primary Dermal Irritation.



    3.   Use Patterns and Application Methods



    To be covered this Standard, EC products may be used



only as an insecticide on home lawns or ornamental turf.



Application may not be made aerially or by air blast methods,



Currently registered EC products must retain present



recommendations for dosage rates on the labels.  Applicants



who wish to increase the dosage recommendations on currently



registered products, or who wish to register new products



with higher dosage recommendations than those currently






                       -68-

-------
registered, may be  required to  submit  additional  supporting

data.

    D.  Data Gaps

    To be covered under this Standard, applicants  for

registration or reregistration  of EC Aspon® products must

agree to submit or  cite the following  information  on the

composition and toxicity of each proposed product.  After

each data gap is listed the section in the Proposed Guidelines

which describes that type of data and when it  is  required

[43 PR, No. 132, 29696 of July  10, 1978; and 43 FR, No. 163,

37336 of August 22, 1978].

                                          Guidelines Section
  Product Chemistry
    1) Product Identity	 163.61-3(a)
    2) Disclosure of Ingredients	 163.61-3(c)
    3) Description of Manufacturing
       Process	 163.61-4
    4) Formation of Unintentional
       Ingredients	 163.61-5
    5) Declaration of Limits	 163.61-6(a)
    6) Certification of Limits	 163.61-6(b)
    7) Analytical Methods	 163.61-7(a)
    8) Analytical Results	 163.61-7 (b) (1)
    9) Color	 163.61-8(c) (1)
    10)  Odor	 163.61-8(c) (2)
    11)  Density or Specific Gravity	163 .61-8(c) (8)
    12)  Storage Stability	 163.61-8 (c) (12)
    13)  Flammability	 163.61-8 (c) (13)
    14)  Oxidizing or Reducing Action	163.61-8 (c) (14)
    15)  Explosiveness	 163.61-8 (c) (15)
    16)  Miscibility	 163.61-8 (c) (16)
    17)  Viscosity	 163.61-8 (c) (17)
    18)  Corrosion Characteristics	 163.61-8 (c) (18)
    19)  Dielectric Breakdown Voltage	163.61-8(c) (19)
                       -69-

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                                          Guidelines Section
 *Toxicology
ECs Between 12% and 2ft% a. i.
         1) Acute oral toxicity  (rat)
            on product in upper  range
            (i.e., P 25% a.i.)	 163.81-1
         2) Acute inhalation  (rat)
            on product in upper  range
            (i.e., P 25% a.i.)	 153.81-3

ECs Between 65% and 68% a.i.
         1) Acute oral toxicity  (rat).... 163.81-1
         2) Acute dermal toxicity
            (rabbit)	 163.81-2
         3) Acute inhalation  (rat)	 163.81-3
         4) Primary eye irritation
            (rabbit)	 163.81-4 (c)
            OR
            Data on pH of the Product.... 163.81-4 (b)
         5) Primary skin irritation
            (rabbit)	 163.81-5

ECs With Aspon^ and Other Active Ingredients
         1) Acute oral toxicity  (rat).... 163.81-1
         2) Acute dermal toxicity
            (rabbit)	 163.81-2
         3) Acute inhalation  (rat)	 163.81-3
         4) Primary eye irritation
            (rabbit)	 163.81-4 (c)
            OR
            Data on pH of the Product.... 163.81-4(b)
         5) Primary skin irritation
            (rabbit)	 163.81-5

  E.  Required Labeling

    1.  Product Chemistry

    The ingredient statement will list the active  ingredient

as:  0,0,0,0-Tetrapropyl dithiopyrophosphate.  In  all cases,

the percentages by weight of active  ingredient and inerts

must equal 100%.
*  A demonstration that an EC Asponty product has a composi-
tion substantially similar to an EC product for which the
Agency already has acceptable acute toxicity data will
satisfy acute toxicity data requirements for the former
product.  Both active and inert ingredients will be considered
in making determinations of similarity.
                       -70-

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Active Ingredient:
  0,0,Of0-Tetrapropyl dithiopyrophosphate	      %
Inert Ingredients		%
Total	  100%

If EC products contain petroleum distillates, the statement

"Contains petroleum distillates" must appear on the label  in

close proximity to the ingredient statement.

Active Ingredient:
  0,0,0,0-Tetrapropyl dithiopyrophosphate	      %
Inert Ingredients*		%
Total	  100%
* Contains Petroleum Distillates

    2.  Human Hazard - Precautionary Labeling

    The hazard warnings and first aid statements on all

EC product labels must correspond to the Toxicity Category

assigned to that product for each acute effect (see Appendix

A). Specifically, all currently registered ECs between  12%

and 28% a.i. must carry on the label the acute tbxicity

hazard warnings and first aid statements required for the

following Toxicity Categories:

    1) Acute Dermal Toxicity - III

    2) Primary Eye Irritation - I

    3) Primary Dermal Irritation - II
                   /R\
    If the EC Aspon^ product has an Acute Oral Toxicity

Category IV and contains greater than 10% petroleum distillates,

the following first aid statement must appear on the label

(see also Table 2, Appendix A):

    If swallowed;  If the patient is unconscious,  main-

    tain breathing and heart rate (CPR:cardiopulmonary

                       -71-

-------
    resuscitation).  Contact your local Poison Control

    Center, physician, or hospital immediately.  Do Not

    Induce Vomiting!

                   (O\
    If the EC Aspon4* product has an Acute Oral Toxicity


Category I and contains greater than 10% petroleum distillates,


the following first aid statement must appear on the label


(see also Table 2, Appendix A):

    If swallowed;  If the patient is unconscious, main-


    tain breathing and heart rate (CPRrcardiopulmonary


    resuscitation).  Contact your local Poison Control

    Center, physician, or hospital immediately.  If the


    patient is conscious, induce vomiting (syrup of ipecac;

    if not available, stimulate the back of the throat


    with finger).  Never give anything by mouth to an

    unconscious person!


    If the EC Aspon*^ product has an Acute Oral Toxicity

Category II or III and contains greater than 10% petroleum

distillates, the following first aid statement must appear


on the label (see also Table 2, Appendix A):

    I_f swallowed;  If the patient is unconscious, main-

    tain breathing and heart rate (CPRrcardiopulmonary

    resuscitation).  Contact your local Poison Control

    Center, physician, or hospital immediately.

    The question of whether vomiting should or should

not be induced will be determined on a case-by-case basis

based on a review of the toxicity of active ingredients,

inert ingredients, and impurities.


                       -72-

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    3.  Environmental Fate



    Because the use pattern clearly indicates the possibility



of post-application exposure to children and pets, the



following warning must appear on all EC labels:  "Keep



children and pets off treated areas for 48 hours after



application and until the grass has completely dried."



Other environmental precautions not in conflict with specific



parts of this Standard should be retained.



    4.  Environmental Hazards



    All EC products must bear the label warning:  "This



pesticide is toxic to fish.   Do not contaminate water



by cleaning of equipment or  disposal of wastes*"
                      -73-

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II.  Regulatory Rationale



    A.  Regulatory Decision

                                               /«

    The Agency has determined that the EC Aspon4* products



described in this Standard can be registered for sale,



distribution, and use in the United States.  There are no



data currently available to the Agency which suggest that



Aspon^ meets any of the risk criteria for unreasonable



adverse effects, as listed in 40 CFR 162.11(a).  In addition,



to be covered under this Standard, applicants must agree to



submit or cite the data listed in Section I.D of this



document, and must also meet the standards for use as listed



in Section I.e.2 of this document.



    B.  Acceptable Ranges and Limits



    1.  Product Composition Standards



    The Agency will consider for registration EC products



which contain any percentage of Aspon® as an active



ingredient as long as the products meet the acute  toxicity



standards listed in Section I.e.2 for domestic, non-domestic,



or restricted use.  The Agency considers that the  use



restrictions and required protective clothing for  the



several acute toxicity levels will adequately protect humans



and the environment from unreasonable adverse effects.



    2.  Acute Toxicity Limits



    a.  Restricted Use


                                     (ft
    The Agency will register EC Asponcy products for



restricted,  non-food,  outdoor use which have a Toxicity





                       -75-

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Category I rating because certified applicators can legiti-


mately be expected to provide the specialized protective


clothing  (for themselves or those under their supervision)


which are required for products with a Toxicity Category I
                                               «
rating.


    b.  Non-Domestic Use


    The Agency will register EC Aspon® products for


non-domestic, non-food, outdoor use which have a Toxicity


Category II rating for acute oral, dermal, or inhalation


toxicity, or which have a Toxicity Category I or II rating


for primary eye or dermal irritation because non-domestic


users can legitimately be expected to provide the specialized


protective clothing (for themselves or their employees)


which are required for products with these Toxicity Category


ratings.  The Agency considers that these restrictions,


together with use of the required protective clothing, will


adequately protect humans from unreasonable adverse effects.


    c.  Domestic Use

                                     /a
    The Agency will register EC Aspori0' products for


domestic, non-food, outdoor use which have a Toxicity


Category III or IV rating for acute oral, dermal, or inhala-


tion toxicity, or which have a Toxicity Category I through


IV rating for primary eye or dermal irritation.  EC products


intended for domestic use with Toxicity Category I or II


ratings for primary eye or dermal irritation must meet the


criteria for child resistant packaging [see FR 44 (48) :13019-



                       -76-

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13024, March 9, 1979].  The Agency considers  that  the



economic and aesthetic benefits  from Aspon® use outweigh



the risks from products with acute Toxicity Category ratings



of III or IVf and that the use of child-resistant  packaging



for products with Toxicity Category I or II ratings for



primary eye or dermal irritation will adequately protect



humans from unreasonable adverse effects.



    3.  Use Patterns and Application Methods


            (ft
    EC Aspon0' products may be registered for  use as an



insecticide only on lawns and ornamental turf.  EC products



may not be used on food crops because the hazard of such



uses and of residue ingestion has not been evaluated nor has



such an evaluation been requested. Application may not be



made aerially or by air blast methods because these two



methods can reasonably be expected to result  in high exposures



to applicators, other persons,  or wildlife close to the



application site.   Currently registered EC products must



retain the dosage recommendations on the labels, in the



absence of data to support higher rates.



    C.  Data Gaps



    The data on the physical/chemical composition and acute



toxicity which applicants are required to submit or cite for



EC Aspon^ products are listed in Section I.D of this



document.  These data are required in order to obtain



registration for any proposed end-use product.
                       -77-

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    D.  Required Labeling



    Acute toxicity hazard warnings must accurately reflect



the product's level of toxicity (products may not be labeled



to show either greater or lesser hazard from the product



than in fact exists).  Proper emergency medical treatment of



patients who have ingested petroleum distillates is a



controversial subject. Two significant risks must be weighted



in reaching a decision on whether or not to induce emesis



[vomiting]  or perform gastric lavage.  If vomiting is



induced, or gastric lavage is performed, petroleum distillates



may be aspirated, possibly resulting in a fatal chemical



pneumonitis.  However, retaining a highly toxic pesticide in



the stomach even for a short period of time may also prove



fatal. In reaching a decision on appropriate labeling policy



for products, the Agency considers the toxic properties of



active ingredients, inerts, and impurities; the Agency also



considers that emergency treatment may not be readily



available and that first aid will usually be administered by



a member of the family or general public who has little or



no medical training.  In general, therefore, the Agency



believes that the best advice is to seek medical help



immediately and to keep the patient breathing until medical



help is available.  The following first aid statement must



therefore appear on all labels of EC Aspon^ products which



contain greater than 10% by weight petroleum distillates:





                       -78-

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    1.  If patient  is  unconscious, maintain  breathing  and



hearbeat  (CPR:cardiopulmonary  resuscitation).   Contact your



local Poison Control Center, hospital, or physician  immediately,



In addition to Statement #1, all products which contain



greater than 10% by weight petroleum distillates and are in



Oral Toxicity Category I must  carry the following statement



on the label:



     2.   If patient is conscious, induce vomiting (syrup



of ipecac; if not available, stimulate back  of  throat  with



finger). Never give anything by mouth to an  unconscious



personl



In addition to Statement #1, all products which contain



greater than 10% by weight petroleum distillates and are in



Oral Toxicity Category IV must carry the following statement



on the label:



   3.  Do not induce vomiting!



Products in Oral Toxicity Categories II and  III will be



dealt with on a product-by-product basis at  the time of



registration; labeling cautions will be based on a review of



active ingredient toxicity, inert ingredients, and impurities.



    Because the use pattern indicates the possibility of


                                           
exposure to children and pets, all EC Aspon"' products must



carry the following warning:   "Keep children and pets off



treated areas for 48 hours and until grass has completely



dried."





                       -79-

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 III.  Product Chemistry

 DISCIPLINARY REVIEW

 Chemistry Profile
 Data Gaps
 Required Labeling

 Chemistry Profile

    "Aspon®" is a  trade name  for  0,0,0,0-tetrapropyl

 dithiopyrophosphate.  No change was  reported  in  the  composi-

 tion of a 15% EC formulation  after 13 months  at  68 and

 100°F.  No other data are available  on  the  physical/chemical

 characteristics of any EC formulation.

Data Gaps

    Listed below are the Product  Chemistry  data  needed  to

obtain registration or re-registration  for  EC Aspon"^

products.  After each data gap is listed  the  section  in  the

Proposed Guidelines (July 10, 1978,  43  FR,  No. 132, 29696)

which describes that type of data and when  it is  required.

                                          Guidelines  Section
    1) Product Identity	 163.61-3(a)
    2) Disclosure of Ingredients	 163.61-3(c)
    3) Description of Manufacturing
       Process	 163.61-4
    4) Formation of Unintentional
       Ingredients	 163.61-5
    5) Declaration of Limits	 163.61-6(a)
    6) Certification of Limits	 163.61-6(b)
    7) Analytical Methods	 163.61-7(a)
    8) Analytical Results	 163.61-7 (b) (1)
    9) Color	 163.61-8(c) (1)
    10)  Odor	 163.61-8 (c) (2)
    11)  Density or Specific Gravity	 163.61-8 (c) (8)
    12)  Storage Stability	 163.61-8 (c) (12)
    13)  Flammability	 163. 61-8 (c) (13)
    14)  Oxidizing or Reducing Action	163.61-8(c) (14)
    15)  Explosiveness	 163.61-8 (c) (15)
    16)  Miscibility	 163. 61-8 (c) (16)
    17)  Viscosity	 163.61-8 (c) (17)
    18)  Corrosion Characteristics	163.61-8(c) (18)
    19)  Dielectric Breakdown Voltage	 163.61-8 (c) (19)
                       -81-

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Required Labeling

    Ingredient Statement;  The ingredient statement will

list the active ingredient as 0,0,0,0-Tetrapropyl dithiopyro-

phosphate.  If EC products contain petroleum distillates,

the statement "Contains petroleum distillates" must appear

on the label in close proximity to the ingredient statement.


TOPICAL DISCUSSIONS

    Corresponding to each of the Topical Discussions

listed below is the number of the section in the 'Pro-

posed Guidelines for Registering Pesticides' of July

10, 1978 (43 FR, No. 132, 29696), which explains the minimum

product Chemistry data needed in order to obtain registration

or reregistration for EC Aspon  products.

                                          Guidelines Section
Chemical Identity	 163.61-3
Manufacturing Processes	 163.61-4
Formation of Unintentional Ingredients... 163.61-5
Ingredients in Pesticide Products	 163.61-6
Product Analytical Methods and Data	 163.61-7
Physical/Chemical Properties	 163.61-8


Chemical Identity

    At present, there is no acceptable common name for

the insecticide, 0,0,0,0-Tetrapropyl dithiopyrophosphate.

For a discussion of other identifiers of this active ingredient,

see the Product Chemistry chapter in the section of this

document on manufacturing-use products.

Manufacturing Process

    The Agency has no information on present-day manufacturing

processes for any EC product.

                       -82-

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Formation of Unintentional Ingredients



    The Agency has no  information on  the possible  formation



of unintentional  ingredients  in any EC product.



Ingredients in Pesticide Products



    For all pesticide  products, the Agency requires a



listing of the upper and lower limits established  (by



the producer or formulator) for each active ingredient,



and the upper limit for each  impurity, reaction product,



and degradation product which is known to be present or



which might reasonably be identified.  Currently registered



EC products range from 12.10  to 67.64% a.i.



Product Analytical Methods and Data



    No methods for analysis of EC products have been



submitted or reported.



Physical/Chemical Properties



    Color;  There are no data available on any EC formulation.



    Odor;  There are no data  available on any EC formulation.



    Physical State;  EC products are in liquid form.



    Density o_r Specific Gravity;   There are  no data available



on any EC or granular formulation.



    Storage Stability;   Chevron (1975, MRID  000004843}



reports no change in the composition of a 15%  EC formulation



after 13 months at 68 and 100°F.



    Flammability;   No data are available on  any EC formulation.



    Oxidizing ££ Reducing Action;   No data are avail-



able on any EC formulation.






                       -83-

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      Explosiveness;  No data are available  on any EC formula-

  tion.

      Miscibility;   No data  are available  on any EC formu-

  lation.

      Viscosity;   No data  are available  on any EC formulation.

      Corrosion Characteristics;  No data  are available on  any

  EC formulation.

      Dielectric Breakdown Voltage;  No  data are available  on

  any EC  formulation.


                  BIBLIOGRAPHY

MRID        CITATION
000004843    Chevron Chemical  Co.  1975.  Product research and
                services; shelf-life test; Ortho Chinch Bug
                Lawn  Spray.   (Unpublished study  received Dec. 3,
                1975  under 239-2445; CDL;228761-A.)
                           -84-

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IV.  Environmental Fate

DISCIPLINARY REVIEW

Environmental Fate Profile
Exposure Profile
Required Labeling

Environmental Fate Profile

    There are no data currently available on the environ-

mental fate of Aspon .

Exposure Profile

    Because of the lack of environmental fate data for

Aspon^, the Agency can make only brief generalizations about

the possibility and extent of exposure.

    For persons involved in the dilution, mixing, and

application of EC products, there is little chance of oral

                                                    
-------
Required Labeling



    Although there are no data available on the environmental


             (R)
fate of Aspon" from which to determine label precautions,



the use pattern (on home lawns) clearly indicates the



possibility of post-application exposure to children and



pets. The following warning must therefore appear on all EC



labels:



     "Keep children and pets off treated areas for 48 hours



     after application and until the grass has completely



     dried."
                       -86-

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V.  Toxicology

DISCIPLINARY REVIEW

Toxicology Profile
Toxicology Hazard Assessment
Data Gaps
Required Labeling

Toxicology Profile

    The acute dermal toxicity in rabbits (2.0 g/kg) indicates

a potentially low acute dermal toxicity in humans  for

the 13% a.i. EC product tested.  No data were available to

assess the acute oral or acute inhalation toxicity of

any EC product.  Data are insufficient to assess the full

range of acute toxicity of all EC formulations.

    Several eye irritation studies conducted on rabbits

showed a wide variety of results (persistent eye irritation

and corneal opacity at day 14 to slight eye irritation at 1

hour and no corneal opacity)  which indicate a possibly

severe eye irritant to humans from the 13-14.2% EC product

tested.  A study conducted with a 13-14.2% EC on rabbits to

assess primary dermal irritation resulted in severe irritation

at 72 hours which indicates a potentially severe skin

irritant to humans.  Sufficient data were not available to

totally assess the primary eye irritation or primary dermal

irritation of all EC formulations.

Toxicology Hazard Assessment

    The 'Exposure Profile1  which appears in the Environmental

Fate chapter lists the chance of oral exposure to EC products
                       -87-

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as small with some (unknown) possibility of dietary exposure



from residues on home garden crops.  No oral toxicology



hazard assessment can be made for any EC product, however,



because of the lack of data.



    Similarly, although some chance of inhalation exposure



to EC products exists, dependant on the vapor pressures and



viscosities of the various products, no inhalation toxicology



hazard assessment can be made for any EC product because of



the lack of data.



    Application of EC products can result in dermal exposure



to applicators and homeowners, including ocular exposure.



In addition, for home uses, children and pets may be exposed



to treated lawns.  The amount of exposure cannot be determined


                                                       (ft
because of data gaps on the environmental fate of Aspon .



Eye exposure to a 13% a.i. EC product can result in



irreversible corneal opacity and severe eye irritation.



Although the acute dermal toxicity of the 13% EC tested is



low to moderate, dermal exposure can result in primary



dermal irritation, including severe irritation or moderate



erythema and edema.  No toxicology hazard assessment can be



made for EC products with a percent a.i. higher than 13%



because of the lack of data.



Data Gaps



    Listed below are the Toxicology data which must be



submitted or cited to obtain registration or re-registration
                       -88-

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 for  EC  Aspon** products.*   After  each data gap is listed

 the  Section  in the  Proposed  Guidelines  of August 22, 1978

 (43  PR, No.  163,  37336) which describes that type of data

 and  when  it  is required.   The Agency has determined that

 currently registered  EC products between 12% and 28% a.i.

 are  substantially similar  in  composition,  and that EC

 products  between  65%  and 68%  a.i.  are substantially similar

 in composition.   Acute toxicity  data  available  on any one

 product in either group may  be cited  in  support of the

 registration  of any other  product  in  that  group,  provided

 compnesation  has  been offered  for  use of these  data.

 Currently  registered EC Aspon™ products  which contain

 other active  ingredients must  be  tested  individually  for

 each acute effect.

                                          Guidelines  Section
 ECs Between 12% and 28% a.i.
          1) Acute oral toxicity  (rat)
            on product in  upper  range
             (i.e., @ 25% a.i.)	  163.81-1
          2) Acute inhalation  (rat)
            on product in  upper  range
             (i.e., @ 25% a.i.)	 163.81-3

 ECs Between 65% and 68% a.i.
          1) Acute oral toxicity  (rat).... 163.81-1
          2) Acute dermal toxicity
             (rabbit)	 163.81-2
          3) Acute inhalation  (rat)	 163.81-3
         4) Primary eye irritation
             (rabbit)	 163.81-4 (c)
            OR
            Data on pH of  the Product.... 163.81-4(b)
         5) Primary skin irritation
            (rabbit)	 163.81-5
*  A demonstration that an EC Aspori"' product has a composi-
tion substantially similar to an EC product for which the
Agency already has' acceptable acute toxicity data will
satisfy acute toxicity data requirements for the former
product.  Both active and inert ingredients will be considered
in making determinations of similarity.
                       -89-

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ECs With Asponv and Other Active Ingredients
         1) Acute oral toxicity  (rat)	 163.81-1
         2) Acute dermal toxicity
            (rabbit)	 163.81-2
         3) Acute inhalation  (rat)	 163.81-3
         4) Primary eye irritation
            (rabbit)	 163.81-4 (c)
            OR
            Data on pH of the Product.... 163.81-4(b)
         5) Primary skin irritation
            (rabbit)	 163.81-5

Required Labeling

    Product-specific acute toxicity precautionary labeling

is required.  Acceptable categories of acute  toxicity,

and the corresponding required precautionary  labeling

statements, appear  in Appendix A to this document.

    If the EC Aspon® product  has an Acute Oral Toxicity

Category IV and contains greater than 10% by  weight  petroleum

distillates, the following first aid statement must  appear

on the label (see also Table  2,  Appendix A):

    I_f swallowed;   If the patient  is unconscious, main-

    tain breathing  and heart  rate  (CPRrcardiopulmonary

    resuscitation).  Contact  your  local Poison Control

    Center, physician, or hospital  immediately.  Do  Not

    Induce Vomiting!
                   (ft
    If the EC Aspon'"' product  has an Acute Oral Toxicity

Category I and contains greater  than 10% by weight petroleum

distillates, the following first aid statement must  appear

on the label (see also Table  2,  Appendix A):

    If^ swallowed:   If the patient  is unconscious, main-

    tain breathing  and heart  rate  (CPRicardiopulmonary

                       -90-

-------
     resuscitation).   Contact  your  local  Poison Control

     Center,  physician,  or  hospital  immediately.   If  the

     patient  is  conscious,  induce vomiting  (syrup of  ipecac;

     if  not available, stimulate the  back of  the  throat

     with  finger).  Never give  anything by mouth  to an

     unconscious  person!

     If  the EC Asppn® product has an Acute Oral Toxicity

Category  II  or  III and  contains greater than  10%  by  weight

petroleum distillates,  the  following first aid statement

must appear  on  the label (see  also Table 2, Appendix A):

     I_f  swallowed;  If the patient 'is unconscious, main-

     tain  breathing and  heart rate (CPR:cardiopulmonary

     resuscitation)!   Contact your local Poison Control

     Center,  physician,  or hospital immediately.

    The question of whether vomiting should or should

not be  induced for products with Acute Oral Toxicity Categories
     *
of II and III will be determined on a case-by-case basis

based on  a review of  the toxicity of active ingredients,

inert ingredients, and  impurities.



TOPICAL DISCUSSIONS

    Corresponding to each of the Topical Discussions

listed below is the number of the  section in the  'Proposed

Guidelines'  of August 22, 1978 (43  FR,  No.  163, 37336)  which

explains the minimum Toxicology data needed in order to

obtain registration or  reregistration for EC Aspon®

products.

                       -91-

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                                          Guidelines Sections
Acute Effects	 163.81-1, -2, and -3
Local Irritation..	 163.81-4 and -5

Acute Effects

    Acute Oral Toxicity

         The minimum data requirement for testing acute oral

    toxicity (LD-50) is one test on a registered product

    from each group of substantially similar products (see

    the Data Gaps section in this chapter) , preferably using

    the laboratory rat.  No data are available for assessing

    the acute oral LD-50 of any EG product.

    Acute Dermal Toxicity

         The minimum data requirement for testing acute

    dermal toxicity (LD-50) is one test, preferably using

    the albino rabbit, for a registered product from each

    group of substantially similar products (see the Data

    Gaps section in this chapter).  The acute dermal LD-50

    for a 13-14.2% EC in male rabbits is greater than 2.0

    g/kg (Rittenhouse and Narcisse, 1972, MRID 000004838).

    Moderate skin irritation was noted but was not persistent

    at 72 hours.  The data are adequate to assign the

    13-14.2% EC product tested to Toxicity Category III for

    acute dermal toxicity.  Currently registered products

    between 12% and 28% should also be assigned to Category

    III for acute dermal toxicity.  No data are available

    for assessing the acute dermal toxicity of any EC

    product between 65% and 68% a.i., or any EC product

    which contains Aspon® plus other active ingredients.


                       -92-

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    Acute Inhalation Toxicity
         The minimum data  requirement  for  testing  acute
    inhalation toxicity  (LC-50) is one  test  for a  regis-
    tered product from each group of substantially similar
    products (see the Data Gaps section in this chapter),
    preferably using the laboratory rat. No  data are available
    for assessing the acute inhalation  LC-50 of any EC
    product.
-Local Irritation
    Primary Eye Irritation
         The minimum data requirement for testing primary
    eye irritation is one test for a registered product from
    each group of substantially similar products (see the
    Data Gaps section in this chapter), conducted on a
    mammal, preferably the albino rabbit.  Data which demons-
    trate that the test substance has a pH of 1-3 or 12-14
    should be submitted instead of data from a primary eye
    irritation test.  For all regulatory purposes,  the
    Agency will assume that substances with the above pH
    values or which cause Category I skin effects ar-e
    corrosive (i.e., have a Toxicity Category I rating).
         Disparate test results were obtained in three
    adequate tests conducted on rabbits using a 13% EC
    product.  In one study (Narcisse,1972, MRID 000004836),
    male rabbits were observed for 7 days  after applcation
    of a 13% EC to the eye.  Persistent eye irritation was

                       -93-

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noted at day 7, the last day of observation.  Another



study was conducted (Bullock and Narcisse, 1974, MRID



000004835).  Male and female rabbits were observed for



14 days after application of a 13% EC product to the



eye.  Persistent iritis, conjuctival redness, and



discharge were noted until day 7; corneal opacity was



reported in half the test animals at day 14.



     In yet another study (Gregory and Narcisse, 1974,



MRID 000004833), female rabbits were observed for 14



days after application of a 13% EC product to the eye.



Slight eye irritation was noted at 1 hour.  No corneal



opacity was noted in any test animal.



     The existing data are sufficient to assess the



primary eye irritation potential of the 13% EC product



tested and to place it in Toxicity Category I, indicating



severe eye irritation hazard.  Currently registered



products between 12% and 28% a.i. should also be assigned



to Category I for primary eye irritation.  No data are



available for assessing the primary eye irritation of



any EC product between 65% and 68% a.i., or any EC



product which contains Aspon™ plus other active



ingredients.



Primary Dermal Irritation



     The minimum data requirement for testing primary



dermal irritation is one test for a registered product



from each group of substantially similar products (see





                   -94-

-------
the Data Gaps section in this chapter) , conducted on a
mammal, preferably the albino rabbit.  Narcisse (1972,
MRID 000004837)  observed rabbits after application of a
13% EC product to the skin.  The dermal exposure resulted
in mild to severe erythema with no edema.  The existing
data are adequate to assign the 13% EC product tested to
Toxicity Category II for primary dermal irritation.
Currently registered products between 12% and 28% a.i.
should also be assigned to Category II for primary
dermal irritation.  No data are available for assessing
the primary dermal irritation of any EC product between
    and 68% a.i., or any EC product which contains
       plus other active ingredients.
                   -95-

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                    BIBLIOGRAPHY

MRID          CITATION
000004835     Bullock, C.H.; Narcisse, J.K.  1974.  The eye irri-
                  tation potential of Ortho Chinch Bug Spray (CC
                  5109): S-668: SOCAL 588/XX:24.  (Unpublished study
                  received Aug. 5, 1974 under 239-765; submitted by
                  Chevron Cehmical Co., Richmond, Calif.; CDL:022718-A).

000004833     Gregory, L.K.; Narcisse, J.K.  1974.  The eye irrtiation
                  potential of CC-5495: S-745: SOCAL 674/XX:117.  (Un-
                  published study received June 25, 1975 under 239-765;
                  submitted by Chevron Chemical Co., Richmond, Calif.;
                  CDL:220001-C).

000004836     Narcisse, J.K.  1972.  Eye irritation potential of Ortho
                  Bug Spray: S-362: SOCAL 283/71:114.  (Unpublished
                  study received Nov. 14, 1974 under 239-765; submitted
                  by Chevron Chemical Co., Richmond, Calif.; CDL:051023-A)

000004837     Narcisse, J.K.  1972.  Skin irritation potential of
                  Ortho Chinch Bug Spray: S-363: SOCAL 284B/VI:114.
                  (Unpublished study received Nov. 14, 1974 under 239-765;
                  submitted by Chevron Chemical Co., Richmond, Calif.;
                  CDL:051023-B).

000004838     Rittenhouse, J.R.; Narcisse, J.K.  1972.  The acute dermal
                  toxicity of Ortho Chinch Bug Spray: S-363: SOCAL
                  284A/VI:117. (Unpublished study received Nov. 14, 1974
                  under 239-765; submitted by Chevron Chemical Co.,
                  Richmond, Calif.; CDL:051023-C).
                              -96-

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 VI.   Ecological  Effects

 DISCIPLINARY  REVIEW

 Ecological  Effects  Profile
 Required  Labeling

 Ecological  Effects  Profile

    The available data show  that  a  13%  EC  is  highly

 toxic  to  fish and freshwater  aquatic  invertebrates,  the

 invertebrates being more sensitive  than fish.

    Tests on  a 13%  EC indicate  that there  is  no  phytotoxicity

 to turf grass if used at recommended  rates  (3.7  pounds a.i.

 per acre)  ,  and that it is only  slightly phytotoxic to

 certain varieties of turf at  2  to 4 times  recommended

 rates.

 Required Labeling

    Based on data discussed  in  the Manufacturing-Use section

 of this document, all EC products must  bear the  label

 warning: "This pesticide is toxic to  fish.  Do not contaminate

 water by cleaning of equipment  or disposal of wastes."


 TOPICAL DISCUSSIONS

    Applicants for registration of end-use EC products are

 not required to submit information on ecological effects.

 The following discussions present supplemental information

 available to the Agency on EC formulations.

Terrestrial Plants

    Tests  on a 13% EC (Chevron, 1971,  MRID 000004849)

 indicate that there is no phytotoxic  response by turfgrasses


                       -97-

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when used at the recommended rate of 3.7 pounds a.i. per

acre.  The response to the EC varies from no reaction to

moderate phytotoxic symptoms when used at 2 to 4 times the

recommended rate, depending on the variety of turfgrass

tested (Lindemann 1974).  This type of data is not, at

present, required for registration.

Aquatic Invertebrates

    A 48-hour toxicity test (EPA, 1975, MRID GS0019-011)

using a 13% EC formulation was performed on the water flea,

Daphnia magna.  The 48-hour LC-50 = 0.625 ppm (0.5 to 0.77

ppm, 95% c.i.).  These data are sufficient to characterize a

13% EC formulation as highly toxic to aquatic invertebrates.

Freshwater Fish

    Data discussed in the section on Manufacturing-use

products indicate that Aspon*^ can be considered very

highly toxic to coldwater and warmwater fish species.

    Addtional data, which are summarized in Table 7,

are also available on the 96-hour LC-50 of a 13% EC formula-

tion.  These data indicate that the 13% EC formulation

tested is highly toxic to rainbow trout.
Table 7.  Acute Toxicity of Formulated Aspon*
          Products to Freshwater Fish
Species
Rainbow Trout
Formulation
13%
EC
LC-50
(ppm)
1.0
Reference
EPA, 1975,
MRID GS0019-
011
1
1
1
1
1
1
                        -98-

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                    BIBLIOGRAPHY

MRID          CITATION
000004849     Chevron Chemical Co.  1971.  Summary: Ortho Sod
                  Webworm Control.  (Unpublished study including
                  OR 513 report  nos. 387-1, 387-41, 621-37, 621-36,
                  623-07, 623-06, 504-23, received Dec. 20, 1971
                  under 239-2389; CDL:001557-A).

GS0019-011    EPA.  1975.  Report on the toxicity of Ortho Sod
                  Webworm (13% active ingredient) to Daphnia magna.
                  (U.S. EPA, Chemical and Biological Investigations
                  Branch, Beltsville, Maryland, Static jar test No.
                  865, 8/21/75, unpublished.)

GS0019-012    EPA.  1975.  Report on the toxicity of Ortho Sod-Webworm
                  13% active ingredient to rainbow trout.   (U.S. EPA,
                  Chemical and Biological Investigations Branch, Belts-
                  ville, Maryland, Static jar test No.  848, 7/8/75,
                  unpublished report.)

000005003     Lindemann, R.H.; Massey,  V.C.;  Coltharp,  J.L.;  Bryant,
                  W.F. 1974.  Product performance report:  OR report no.
                  657-10.  (Unpublsihed study including OR-513 report
                  nos. 705-41, 748-21,  748-22,  705-25,  705-23 and 705-42,
                  received June 25,  1975 under  239-2389;  submitted by
                  Chevron Chemical Co., Richmond, Calif.;  CDL:133068-C).
                              -99-

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                  GRANULAR ASPO



I.  Regulatory Position



  A.  Regulatory Decision



    The Agency has reviewed all data available to  it.



Although incomplete, these data indicate that granular



Aspon® is suitable for registration because it does not



meet or exceed the risk criteria leading to a Rebuttable



Presumption Against Registration [Chapter 40, Section



162.11(a) of the Code of Federal Regulations],  Data gaps



have been identified; when these data are supplied/ the



Agency will again review the registration status of this



compound.



    The Agency has determined that granular Aspon^ does



not appear to cause an unreasonable adverse effect with



proper label directions and precautions.  Those granular



products currently registered may be reregistered subject to



the conditions imposed for data requirements, and new



products may also be registered under the terms of this



Standard.



  B.  Criteria for Registration under the Standard



    To be registered under this Standard, granular Aspon®



products must meet the following conditions:



    1.  The granular product contains Aspon®



as an active ingredient [if an unregistered source of



Aspon™ is used in formulating, then the data  outlined



under Section 162.18-2(c) (d) (1) (ill)  will be  required];





                       -101-

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    2.  The granular Aspon™ product is within the acute



toxicity limits for restricted or general use and bears the



required labeling;



    3.  The granular Aspon® product is within acceptable



ranges for use patterns and application methods; and



    4.  The applicant for registration of granular products



complies with all other terms and conditions specified in



this Standard and hereby offers to pay compensation to other



persons, with regard to approval of this application, to the



extent required by 3(c)(l)(d)  and 3(c)(2)(d) of the Federal



Insecticide, Fungicide, and Rodenticide Act [FIFRA], as



amended, 7 U.S.C. 136(c)(l)(d) and 136 (c) (2) (D) .



  C.  Acceptable Ranges and Limits



    1.  Product Composition Standards



    To be covered under this Standard, all granular products



must contain Aspon® [0,0,0,0-Tetrapropyl dithiopyrophosphate]



as an active ingredient.  The Agency will consider for



registration granular products which contain any percentage



of active ingredient.  In addition, currently registered and



proposed granular products must agree to submit or cite the



information on product composition identified as data



gaps in Section I.D of this document



    Standards have not yet been set for contaminants and



inerts in granular Aspon" products.  When standards are



set for any contaminants or inerts in granular Aspon®



products, granular end-use products must comply with those



standards.
                       -102-

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     2.  Acute Toxicity Limits



     a.  Restricted Use



     The Agency will grant registration to granular



products as restricted pesticides  (i.e., for retail sale  to



and  application only by Certified  Applicators or persons



under their direct supervision) for non-food, outdoor use



which have a Toxicity Category I rating for any of the



following acute effects:



     1) Acute Oral Toxicity;



     2) Acute Dermal Toxicity;



     3) Acute Inhalation Toxicity;



     4) Primary Eye Irritation; or



     5) Primary Dermal Irritation.



     b.  Non-Domestic Use



     The Agency will grant registration to granular Aspon®



products intended for non-domestic, non-food, outdoor use



which have a Toxicity Category II rating for any of the



following acute effects:



     1) Acute Oral Toxicity;



     2) Acute Dermal Toxicity; or



     3) Acute Inhalation Toxicity;



The Agency will grant registration to  granular Aspon®



products intended for non-domestic, non-food,  outdoor



use which have a Toxicity Category I or II  rating for



either of the following acute effects:



     1) Primary Eye Irritation;  and



    2) Primary Dermal Irritation.
                       -103-

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    c.  Domestic Use
    The Agency will grant registration to granular
products intended for domestic, non-food, outdoor use which
have a Toxicity Category III or IV rating for any of the
following acute effects:
    1) Acute Oral Toxicity;
    2) Acute Dermal Toxicity; or
    3) Acute Inhalation Toxicity;
The Agency will grant registration to granular Aspon®
products intended for domestic, non-food, outdoor use which
have a Toxicity Category I through IV rating for either of
the following acute effects:
    1) Primary Eye Irritation; and
    2) Primary Dermal Irritation.
    3.  Use Patterns and Application Methods
    To be covered under this Standard, granular products may
be used only as an insecticide on home lawns or ornamental
turf.  Application may not be made aerially.  Currently
registered granular products must retain present recommen-
dations for dosage rates on the labels.  Applicants who wish
to increase the dosage recommendations on currently registered
products, or who wish to register new products with higher
dosage recommendations than those currently registered may
be required to submit additional supporting data.
  D.  Data Gaps
    To be covered under this Standard, applicants for
registration or reregistration of granular Aspon® products
                       -104-

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 must agree  to submit or cite the following information on

 the  physical/chemical composition and toxicity of each

 proposed  product.   After each data gap is listed the

 section in  the Proposed Guidelines which describes that type

 of data and when  it is  required [43 FRf  No.  132, 29696 of

 July 10,  1978;  and  43 FR,  No.  163, 37336 of  August 22,

 1978] .

                                           Guidelines Section
  Product Chemistry
     1)  Product Identity	  163.61-3(a)
     2)  Disclosure of Ingredients	  163.61-3(c)
     3)  Description  of Manufacturing
        Process	  163.61-4
     4)  Formation of Unintentional
        Ingredients	  163.61-5
     5)  Declaration  of Limits	  163.61-6(a)
     6)  Certification of Limits	  163.61-6(b)
     7)  Analytical Methods	  163.61-7(a)
     8)  Analytical Results	  163.61(b)(l)
     9)  Color	  163.61-8(0(1}
     10) Odor	  163.61-8(c) (2)
     11) Density or  Specific Gravity	163.61-8(c) (8)
     12) Storage Stability	  163.61-8 (c) (12)
     13) Oxidizing or Reducing Action	  163.61-8(c)(14)
     14) Explosiveness	  163.61-8 (c) (15)
     15) Corrosion Characteristics	163.61-8(c) (18)
 *Toxicology
Granulars Between 1%  and 6%
          1)  Acute inhalation  (rat)**	  163.81-3
*A demonstration that a granular Aspon^ product has
a composition substantially similar to a granular product
for which the Agency already has acceptable acute toxicity
data will satisfy acute toxicity data requirements for
the former product.  Both active and inert ingredients will
be considered in making determinations of similarity.
**  An acute inhalation toxicity study is required for
granular products if "20 percent or more of the aerodynamic
equivalent of the formulated product (as registered or under
conditions of use) is composed of particulates not larger
than 10 microns in diameter" [Guidelines Section
163.81-3(a) (2) (ii)].  An acute inhalation test on any
currently registered granular product between 1% and 6% a.i.
may be submitted or cited in support of the registrations of
all currently registered granular products.  A request for
a waiver of this requirement based on percent of particulates
not larger than 10 microns must be made individually
for each product.

                       -105-

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  E.  Required Labeling

    1.  Product Chemistry

    The ingredient statement will list the active ingredient

as:  0,0,0,0-Tetrapropyl dithiopyrophosphate.  In all cases,

the percentages by weight of active ingredient and inerts

must equal 100%.

Active Ingredient:
  0,0,0,0-Tetrapropyl dithiopyrophosphate	     %
Inert Ingredients		%_
Total	  100%

    2.  Human Hazard - Precautionary Labeling

    The hazard warnings and first aid statements on all

granular product labels must correspond to the Toxicity

Category assigned to that product for each acute effect

(see Appendix A).  Specifically, all currently registered

granulars between 1% and 6% a.i. must carry on the label

the acute toxicity hazard warnings and first aid state-

ments required for the following Toxicity Categories:

Granulars Without Fertilizer
1) Acute Oral Toxicity - III
2) Acute Dermal Toxicity - III
3) Primary Eye Irritation - III
4) Primary Dermal Irritation - III

Granulars With Fertilizer
1) Acute Oral Toxicity - III
2) Acute Dermal Toxicity - III
3) Primary Eye Irritation - II
4) Primary Dermal Irritation - III

    3.  Environmental Fate

    Because the use pattern clearly indicates the possibility

of post-application exposure to children and pets, the
                        -106-

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following warning must appear on all granular labels:  "Keep



children and pets off treated areas for 48 hours after



application and until the grass has completely dried."



Other environmental precautions not in conflict with specific



parts of this Standard should be retained.



    4.  Environmental Hazards



    All granular products must bear the label warning:



"This pesticide is toxic to fish.   Do  not contaminate water



by cleaning of equipment or disposal of wastes."
                      -107-

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 II.  Regulatory Rationale
    A.  Regulatory Decision
                                                 
-------
Category I rating because certified applicators can legiti-



mately be expected to provide the specialized protective



clothing (for themselves or those under their supervision)



which are required for products with Toxicity Category I



rating.



    b.  Non-Domestic Use



    The Agency will register granular Aspon® products



for non-domestic, non-food, outdoor use which have a Toxicity



Category II rating for acute oral, dermal, or inhalation



toxicity, or which have a.Toxicity Category I or II rating



for primary eye or dermal irritation, because non-domestic



users can legitimately be expected to provide the specialized



protective clothing (for themselves or their employees)



which are required for products with these Toxicity Category



ratings. The Agency considers that these restrictions,



together with use of the required protective clothing, will



adequately protect humans from unreasonable adverse effects.



    c.  Domestic Use



    The Agency will register granular Aspon^ products for



domestic, non-food, outdoor use which have a Toxicity



Category III or IV rating for acute oral, dermal, or inhala-



tion  toxicity, or which have a Toxicity Category I through



IV rating for primary eye or dermal irritation.  Granular



products intended for domestic use with Toxicity Category I



or II ratings for primary eye or dermal irritation must meet



the criteria for child-resistant packaging [see PR 44(48):
                       -110-

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 13019-13024,  March  9,  1979].   The Agency  considers  that the
 economic  and  aesthetic  benefits  from  Aspon^ use  outweigh
 the  risks  from products with  acute Toxicity Category  ratings
 of III or  IV, and that  the  use of child-resistant packaging
 for  products  with Toxicity  I  or  II ratings  for primary  eye
 or dermal  irritation will adequately  protect humans from
 unreasonable  adverse effects.
     3.  Use Patterns and Application  Methods
     Granular  Aspon® products  may be registered for use  as
 an insecticide only on lawns  and ornamental  turf.  Granular
 products may  not be used on food crops because the hazard of
 such uses  and of residue ingestion has not  been evaluated
 nor  has such  an evaluation been requested.   Application  may
 not  be made aerially because  this method can reasonably  be
 expected to result  in high exposures  to applicators, other
 persons, or wildlife close to the application site.   Currently
 registered granular products must retain the dosage  recommen-
 dations on the labels, in the absence of data to support
 higher rates.
    C.  Data Gaps
    The data on the physical/chemical composition and acute
 toxicity which applicants are required to submit or  cite for
granular Aspon*^ products are listed in Section I.D of this
document.   These data are required in order  to obtain
 registration for any proposed end-use product.
                       -Ill-

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    D.   Required Labeling



    Acute toxicity hazard warnings must accurately reflect



the product's level of toxicity (products may not be labeled



to show either greater or lesser hazard from the product



than in fact exists).  Because the use pattern indicates the



possibility of exposure to children and pets,  all granular


     (R)
Aspon** products must carry the following warning:  "Keep



children and pets off treated areas for 48 hours and until



grass has completely dried."
                       -112-

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 TTT.   Product  Chemistry

 DISCIPLINARY REVIEW

 Chemistry  Profile
 Data Gaps
 Required Labeling

 Chemistry  Profile

     "Aspon®" is  a  trade name  for  0,0,0,0-tetrapropyl

 dithiopyrophosphate.  No data  are  available  on  the  physical/-

 chemical characteristics of any granular  formulation.

 Data Gaps

     Listed below are the Product Chemistry data which must

 be submitted or cited to obtain registration or re-registra-
                       (ft
 tion for granular Aspon^ products.  After each data gap  is

 listed the section in the Proposed Guidelines (July 10,

 1978,  43 PR, No. 132, 29696) which describes that type of

 data and when  it is required.

                                          Guidelines Section
     1) Product Identity	 163.61-3(a)
     2) Disclosure of Ingredients	 163.61-3(c)
     3) Description of Manufacturing
       Process	 163.61-4
     4) Formation of Unintentional
       Ingredients	 163.61-5
     5) Declaration of Limits	 163.61-6(a)
    6) Certification of Limits	 163.61-6(b)
    7) Analytical Methods	 163.61-7(a)
    8) Analytical Results	 163.61(b)(l)
    9) Color	 163.61-8(c) (1)
    10) Odor	 163.61-8(c) (2)
    11) Density or Specific Gravity	163.61-8 (c) (8)
    12) Storage Stability	 163.61-8 (c) (12)
    13) Oxidizing or Reducing Action	163.61-8 (c) (14)
    14) Explosiveness	 163.61-8 (c) (15)
    15) Corrosion Characteristics	 163.61-8 (c) (18)

Required Labeling

    Ingredient Statement;   The ingredient statement will

 list the active ingredient as 0,0,0,0-Tetrapropyl dithiopyro-

phosphate.
                       -113-

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TOPICAL DISCUSSIONS

    Corresponding to each of the Topical Discussions

listed below is the number of the section in the 'Pro-

posed Guidelines for Registering Pesticides' of July

10, 1978 (43 FR, No. 132, 29696), which explains the minimum

Product Chemistry data needed in order to obtain registration

or reregistration for granular Aspon™ products.

                                          Guidelines Section
Chemical Identity	 163.61-3
Manufacturing Processes	 163.61-4
Formation of Unintentional Ingredients... 163.61-5
Ingredients in Pesticide Products	 163.61-6
Product Analytical Methods and Data	 163.61-7
Physical/Chemical Properties	 163.61-8


Chemical Identity

    At present, there is no acceptable common name for

the insecticide, 0,0,0,0-Tetrapropyl dithiopyrophosphate.

For a discussion of other identifiers of this active ingredient,

see the Product Chemistry chapter in the section of this

document on manufacturing-use products.

Manufacturing Process

    The Agency has no information on present-day manufacturing

processes for any granular product.

Formation of Unintentional Ingredients

    The Agency has no information on the possible formation

of unintentional ingredients in any granular product.

Ingredients in Pesticide Products

    For all pesticide products, the Agency requires a

listing of the upper and lower limits established (by the
                       -114-

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producer or  formulator) for each active  ingredient,  and
the  upper  limit  for each  impurity, reaction product,  and
degradation  product which  is known to be present or  which
might  reasonably be identified.  Currently registered
granular products range from 1.32% to 5% a.i.
Product Analytical Methods and Data
    No methods for analysis of granular products have been
submitted  or reported.
Physical/Chemical Properties
    Color;  There are no data available on any granular
formulation.
    Odor;  There are no data available on any granular
formulation.
    Physical State;  Granular products are in solid form.
    Density ojr Specific Gravity;  There are no data available
on any granular formulation.
    Storage Stability;  There are no data available on any
granular formulation.
    Oxidizing ££ Reducing Action;  No data are avail-
able on any granular formulation.
    Explosiveness;   No data are available on any granular
formulation.
    Corrosion Characteristics;   No data are available on any
granular formulation.
                       -115-

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 IV.  Environmental  Fate

 DISCIPLINARY  REVIEW

 Environmental Fate  Profile
 Exposure  Profile
 Required  Labeling

 Environmental Fate  Profile

    There are no data  currently  available  on  the  environ-
                    (ft
 mental fate of Aspon**.

 Exposure  Profile

    Because of the  lack of environmental fate data  for

     (ft
 Aspon", the Agency  can make only brief generalizations

 about the possibility  and extent of exposure.

     For  persons involved in the application of granular

 products, there is  little chance of oral exposure except

 through accidental  ingest ion.  Aspon® is not registered

 for use on food or  feed crops, so there is very little

 possibility of dietary exposure to the general public.

 (Depending on the leaching and mobility characteristics of

 the granular  products, home use may result in contamination

 of home garden vegetables.)   Dermal and eye exposure to

granular formulations  (and to dust particles of the formula-

 tions)  can occur.  Inhalation exposure to granular formulations

can also occur through inhalation of dust-sized particles by

applicators and homeowners.

Required Labeling

    Although  there are no data available on the environmental

fate of Aspon^ from which to determine label precautions,
                       -117-

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the use pattern (on home lawns) clearly indicates the



possibility of post-application exposure to children and



pets. The following warning must therefore appear on all



granular labels:



     "Keep children and pets off treated areas for 48 hours



     after application and until the grass has completely



     dried."
                       -118-

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V.  Toxicology

DISCIPLINARY REVIEW

Toxicology Profile
Toxicology Hazard Assessment
Data Gaps
Required Labeling

Toxicology Profile

    The acute oral toxicity in rats (males, >6.0 g/kg;

females = 3.4 g/kg) indicates a potentially low acute oral

toxicity in humans for the 3.2-3.9% granular product tested.

The acute dermal toxicity in rabbits (4.65 g/kg)  indicates a

potentially low acute dermal toxicity in humans for the 5%

granular tested.  No data were available to assess the acute

inhalation toxicity of any granular product.  Data are

insufficient to assess the full range of acute toxicity of

all granular formulations.

    An eye irritation study conducted on rabbits indicates a

mild, transitory eye irritation potential for humans from

the 3.2% granular (without fertilizer)  tested.  A study

conducted on rabbits to assess primary dermal irritation

indicates a slight, transitory dermal irritation potential

for humans from the 3.2% granular tested.  Data on other

active ingredient products which contain fertilizer indicate

a possible increase in the primary eye irritation potential

of such products from the fertilizer component.

Toxicology Hazard Assessment

    The 'Exposure Profile1 which appears in the Environmental

Fate chapter lists the chance of exposure to granular


                       -119-

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products as small with some (unknown) possibility of dietary



exposure from residues on home garden crops.  The acute oral



toxicity of a 3.9% granular product  is low.  Whether possible



oral exposure to granular products would occur at levels



high enough to be of concern cannot  be determined, because



of the lack of data.



    Similarly, although some chance  of inhalation exposure



to granular products exists, dependant on the size of the



dust particles of the formulations, no inhalation toxicology



hazard assessment can be made for any granular product



because of the lack of data.



    Application of granular products can result in dermal



exposure to applicators and homeowners, including ocular



exposure from dust particles of the product.  In addition,



for home uses, children and pets may be exposed to treated



lawns.  The amount of exposure cannot be determined because



of data gaps on the environmental fate of Aspon^.  Data



indicate that a 3.2% a.i. granular product has low acute



dermal toxicity and low primary dermal irriation.  The



primary eye irriation potential of a 5% a.i. granular



product is also low. Whether possible dermal and eye exposure



to granular products would occur at levels high enough to be



of concern cannot be determined because of the lack of



data.



Data Gaps



    Listed below are the Toxicology data which must be



submitted or cited to obtain registration or re-registration





                       -120-

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 for granular Asporv^ products.*  After  each  data  gap is

 listed  the Section  in  the  Proposed Guidelines  of August  22,

 1978  (43 FR, No. 163,  37336) which describes that type of

 data  and when  it is required.  The Agency has  determined

 that  currently  registered  granular products between  1% and

 6% a.i. are substantially  similar in composition,   except

 that  currently  registered  granular Aspon™ products  between

 1% and  6% a.i.  which contain fertilizer will be  considered

 substantially similar  in composition for determining primary

 eye irritation.  Acute toxicity data available on any one

 product in either group may be cited in support  of the

 registration of any other  product in that group,  provided

 compensation has been offered for use of these data.

                                          Guidelines Section
Granulars Between 1% and 6%
         1) Acute TrThanTtTon (rat)**	 163.81-3
*A demonstration that a granular Aspon0' product has
a composition substantially similar to a granular product
for which the Agency already has acceptable acute toxicity
data will satsify acute toxicity data requirements for
the former product.  Both active and inert ingredients will
be considered in making determinations of similarity.
**  An acute inhalation toxicity study is required for
granular products if "20 percent or more of the aerodynamic
equivalent of the formulated product (as registered or under
conditions of use)  is composed of particulates not larger
than 10 microns in diameter" [Guidelines Section
163.81-3(a) (2) (ii)].  An acute inhalation test on any
currently registered granular product between 1% and 6% a.i.
may be submitted or cited in support of the registrations of
all currently registered granular products.  A request for
a waiver of this requirement based on percent of particulates
not larger than 10 microns must be made individually
for each product.
                       -121-

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Required Labeling


    Product-specific acute toxicity precautionary labeling


is required.  Acceptable categories of acute toxicity,


and the corresponding required precautionary statements,


appear in Appendix A to this document.



TOPICAL DISCUSSIONS


    Corresponding to each of the Topical Discussions


listed below is the number of the section in the 'Proposed


Guidelines' of August 22, 1978 (43 FR, No. 163, 37336)


which explains the minimum Toxicology data needed in order


to obtain registration or reregistration for granular

     (Ok
Aspon0' products.


                                          Guidelines Sections
Acute Effects	 163.81-1, -2, and -3
Local Irritation	 163.81-4 and -5


Acute Effects


    Acute Oral Toxicity


         The minimum data requirement for testing acute


    oral toxicity (LD-50) is one test on any registered


    product between 1% and 6% a.i., preferably using the


    laboratory rat.  The acute oral LD-50 for a 3.2-3.9%


    a.i. granular is 6.0 g/kg for male rats and 3.4 g/kg for


    female  rats (Eisenlord, 1978, MRID 000004857). The data


    indicate that the 3.2-3.9% granular tested should be


    assigned Toxicity Category III for acute oral toxicity.


    Currently registered products between 1% and 6% a.i.  -


    should  also be assigned to Category III for acute oral


    toxicity.
                       -122-

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Acute Dermal Toxicity



     The minimum  data  requirement  for  testing  acute



dermal  toxicity  (LD-50)  is  one  test, preferably  using



the albino  rabbit,  for  any  registered  product  between  1%



and <5%  a.i.  The  acute  dermal LD-50 for  a  5% granular  in



rabbits is  4.65 g/kg  (Bullock,  1970, MRID  000004858).



No skin irritation  or signs of  toxicity  were noted  at



this dose level.  The data  indicate that the 5% granular



tested  should be  assigned Toxicity Category III for



acute dermal toxicity.   Currently  registered products



between 1%  and 6% a.i.  should also be  assigned to



Category III for  acute  dermal toxicity.



Acute Inhalation Toxicity



     The minimum data requirement  for  testing acute



inhalation  toxicity (LC-50)  is one test  for any regis-



tered product between 1% and 6% a.i.,  preferably using



the laboratory rat.  An  acute inhalation toxicity study



is required for granular products  if "20 percent or more



of the aerodynamic equivalent of the formulated product



(as registered or under  conditions of  use)  is composed



of particulates not larger than 10 microns in diameter"



[Guidelines Section 163 .81-3 (a)  (2)  (ii)  ] .  An acute



inhalation  test on any currently registered granular



product between 1% and 6% a.i.  may be  submitted or cited



in support of the registrations  of all currently registered



granular products.  A request for a waiver of this
                   -123-

-------
    requirement based on percent of participates not larger
    than 10 microns must be made individually for each
    product.  No data are available for assessing the acute
    inhalation LC-50 of any granular product.
Local Irritation
    Primary Eye Irritation
         The minimum data requirement for testing primary
    eye irritation is one test for a registered product from
    each group of substantially similar products, conducted
    on a mammal, preferably the albino rabbit (unless the
    pesticide product has a pH of 1-3 or 12-14 or demonstrates
    severe skin corrosivity).  Data which demonstrate that
    the test substance has a pH of 1-3 or 12-14 will be
    submitted instead of data from a primary eye irritation
    test.  For all regulatory purposes, the Agency will
    assume that substances with the above pH values or Which
    cause Category I skin effects are corrosive (i.e.,
    have a Toxicity Category I rating).  [For purposes
    of determining primary eye irritation potential, the
    Agency has determined that there are two groups of
    substantially similar granular Aspon^ products: 1)
    those between 1% and 6% a.i. which do not contain
    fertilizer, and 2) those between 1% and 6% a.i. which jJo
    contain fertilizer.]
         A primary eye irritation study was conducted on
    rabbits using a 3.2% granular without fertilizer  (Bullock,

                       -124-

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1976, MRID 000004861).  The  application  (0.1  ml)  of  the



3.2% granular  in the  eye  resulted  in moderate,  transient



conjunctival redness  and  a slight  discharge of  the



conjunctivae at 1 hour; all  eyes were normal  at  24



hours.  In addition,  no corneal opacity was observed.



The data are adequate to  assign the 3.2% granular tested



to Toxicity Category  III  for primary eye irritation.



Currently registered  products between 1% and  6%  a.i.



which do not contain  fertilizer should also be assigned



to Category III for primary eye irritation.


                                (R)
     Data available on non-Aspon'0' products with



fertilizer indicate that  such products should be



assigned to Toxicity Category II for primary  eye irrita-



tion (The Andersons [sic], 1980, GS0019-019; Biesemeior,



1978, GS0019-020;  O.M. Scott & Sons, Co., 1979, GS0019-021;



O.M. Scott & Sons,  Co., 1979, GS0019-022; Raltech



Scientific Services, Inc., 1980, GS0019-023; Thompson,



1980, GS0019-024;  Thompson,  1979, GS0019-025;  Thompson,



1980, GS0019-026).   In the absence of specific data, the

                        /p|

Agency assumes that Asponv°' products with fertilizer



should also be assigned to Toxicity Category II for



primary eye irritation.  When the data requested on



product chemistry  of granular products have been submitted,



the Agency will review those data to determine substantial



similarity of composition, in which case Category II



will be assigned.   If similarity cannot be established,





                   -125-

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additional testing will be required of the applicant to



establish an appropriate eye irritation toxicity category



Registrants also have the option of submitting data on



the pH of their product (if appropriate) or submitting



data from a primary eye irritation test on their specific



product.
                   -126-

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       Primary Dermal  Irritation

             The minimum data  requirement  for testing primary

       dermal  irritation is one  test for  any registered product

       between 1% and  6% a.i., conducted  on a mammal, preferably

       the  albino rabbit.   Eisenlord (1978,  MRID 000004859)

       observed rabbits after application of a 3.2%  granular

       product to the  skin.  Transient, slight erythema with

       and without edema was observed at  24  and 48 hours;

       however all animals were  normal at  72 hours.   The

       data  are adequate to assign  the 3.2%  granular  tested

       to Toxicity Category III  for primary  dermal irritation.

       Currently registered products between 1% and  6%  a.i.

       should  also be  assigned to Category  III  for primary

       dermal  irritation.


                   BIBLIOGRAPHY

MRID         CITATION
000004858     Bullock, C.H.  1970.  Toxicology lab report—T 1520;
                 T 1549.  (Unpublished study received Apr. 18, 1978
                 under 239-2032; prepared by Stauffer Chemical Co.,
                 submitted by Chevron Chemical Co., Richmond, Calif.;
                 CDL:234497-C).

000004861     Bullock, C.H.  1976.  The eye irritation potential of
                 CC 7187: S-972; SOCAL 937/27:76.  (Unpublished
                 study received Apr.  18, 1978 under 239-2032; sub-
                 mitted by Chevron Chemical Co., Richmond, Calif.;
                 CDL:234497-F).

000004857     Eisenlord, G.H.   1978.  The acute oral toxicity of
                 Ortho Chinch Bug and Sod Webworm Control: S-1178;
                 SOCAL 1179/31: 116.   (Unpublished study received
                 Apr. 18, 1978 under 239-2032; submitted by Chevron
                 Chemical Co., Richmond, Calif.; CDL:234497-B).

000004859     Eisenlord, G.H.   1978.  The skin irritation potential
                 of .Ortho Chinch Bug  and Sod Webworm Control: S-1179;
                 SOCAL 1180/30:132.  (Unpublished study received Apr.
                 18, 1978 under 239-2032;  submitted by Chevron Chemical
                 Co., Richmond, Calif.;  CDL:234497-D).
                           -127-

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Addenda
MRID

GS0019-019
GS0019-020
GS0019-021
GS0019-022
GS0019-023
GS0019-024
GS0019-025
GS0019-026
CITATION

The Andersons [sic],  1979.  Primary eye irritation
study in .the albino rabbit, primary skin irritation
study in the albino rabbit, acute dermal toxicity
study in the albino rabbit, acute oral toxicity study
in rats - Turf Care 20-4-10 with Benefin and chlor-
pyrifos.  (Unpublished studies, received May 30,
1979, under 9198-37).

Biesemeior, J.  1978.  Toxicology lab report [acute
oral LD-50, acute dermal LD-50, skin irritation, eye
irritation] reference no. F-8649.  (Unpublished study
received Apr. 24, 1979, under 538-156; prepared by
Raltech Scientific Services, Inc. [Warf Institute,
Madison, Wis.]; submitted by O.M. Scott & Sons, Marys-
ville, Ohio).

O.M. Scott & Sons, Co.  1979.  Acute oral toxicity,
acute dermal toxicity, primary eye irritation, primary
dermal irritation - Kwit and Western Lawn Insect
Control.  (Unpublished studies received May 5, 1980,
under 538-69.)

O.M. Scott & Sons, Co.  1979.  Acute oral toxicity,
acute dermal toxicity, primary eye irritation, primary
dermal irritation - Western Lawn Insect Control Plus
Fertilizer.  (Unpublished study received May 5, 1980,
under 538-94.)

Raltech Scientific Services, Inc.  1980.  Eye irrita-
tion, Lab report 760871.  (Unpublshed study received
May 1, 1980 under 538-137; submitted by O.M. Scott &
Sons Co., Marysville, Ohio.)

Thompson, G.W.  1980.  The primary eye irritation study
of F6713.   (Unpublished study received June 12, 1980,
under 538-72; prepared by Raltech Scientific Services,
Inc.; submitted by O.M. Scott & Sons, Marysville, Ohio.
Accession # 243155.)

Thompson, G.W.  1979.  Toxicology lab report - F9348.
 (Unpublished study received Nov. 6, 1979, under 538-160;
prepared by Raltech Scientific Services, Inc.; submitted
by O.M. Scott & Sons, Marysville, Ohio.  Accession #
241350.)

Thompson, G.W.  1980.  Toxicology lab report (acute
oral LD-50, acute dermal LD-50, skin irritation and eye
irritation), lab report 765242.  (Unpublished study
received March 24, 1980, under 538-163; prepared by
Raltech Scientific Services, Inc.; submitted by O.M.
Scott & Sons, Marysville, Ohio.)
                               -128-

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VI.   Ecological  Effects

DISCIPLINARY  REVIEW

Ecological  Effects Profile
Required  Labeling

Ecological  Effects Profile

    Information  on the acute  toxicity of a granular  form  to

laboratory  mammals is supplied  in the Toxicology chapter.

The toxicity  of  a 3.2% formulation ranges from  "slightly" to

"practically  non-toxic" to rats.  A 3.2% granular  is moderately

toxic to warmwater fish. Tests  on a 3.2% granular  formulation

indicate no phytotoxic response by turf when the product  is

applied at  14.6  pounds a.i. per acre, which is  4 times the

recommended rate.

Required Labeling

    Based on  data discussed in the Manufacturing-Use section

of this document, all granular products must bear  the label

warning: "This pesticide is toxic to fish.   Do  not contaminate

water by cleaning of equipment or disposal  of wastes."


TOPICAL DISCUSSIONS

    Applicants for registration of end-use  granular products

are not required to submit information on ecological effects.

The following discussions present supplemental  information

available to  the Agency on granular  formulations.

Terrestrial Plants

    Tests on  a 3.2% granular product (Chevron, 1974, MRID

000004854) indicate no phytotoxic response  by turf when
                      -129-

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exposed to 14.6 pounds a.i. per acre, which is 4 times the

recommended rate.  This type of data is not, at present,

required for registration.

Freshwater Fish

    Data discussed in the section on Manufacturing-use

products indicate that Aspon® can be considered very

highly toxic to coldwater and warmwater fish species.

    Additional data, which are summarized in Table 3,

are also available on the 96-hour LC-50 of a 3.2% granular

formulation.  The data indicate that the 3.2% granular is

moderately toxic to bluegills.
Table 3.  Acute Toxicity of Formulated Aspon*
          Products to Freshwater Fish
Species
Bluegill
Bluegill
Formulation
3.2% Gran.
3.2% Gran.
LC-50
(ppm)
5.6
3.8
Reference
EPA, 1975,
MRID GS0019-
013
EPA, 1975,
MRID GS0019-
014
                        -130-

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                    BIBLIOGRAPHY

MRID          CITATION
000004854     Chevron Chemical Co.  1974.  Aspon, Dursban  (Unpublished
                  study including report nos. 627.02, 627.27, 623.09-
                  623.12, 504.23, 504.26, 366.10, 658.29, 657.35, 519.23,
                  748.20, 727.23, 519.30, 727.24, 727.30, 627.23, 627.24,
                  received May 6, 1975 under 239-2032; CDL:222347-C).

GS0019-013    EPA.  1975.  Report on the toxicity of Ortho Chinch Bug
                  Control, 3.2% a.i., to bluegills.  (U.S. EPA, Belts-
                  ville, Maryland, Static jar test No. 876, 9/22/75,
                  unpublished report.)

GS0019-014    EPA.  1975.  Report on the toxicity of Ortho Chinch Bug
                  Control on bluegills.  (U.S. EPA, Chemical and Bio-
                  logical Investigations Branch, Beltsville, Maryland,
                  Static jar test No. 866, 8/21/75, unpublished.)
                              -131-

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     Guide  to Use  of This Bibliography

Content of  Bibliography.  This  bibliography  contains
citations of all the studies  reviewed by EPA in  arriving
at the positions and conclusions  stated elsewhere  in
this Standard.  The bibliography  is divided  into 3
sections: (1) citations  that  contributed information
useful to the review of  the chemical and considered to
be part of  the data base supporting registrations under
the Standard, (2)  citations examined and judged  to be
inappropriate for  use  in developing the Standard, and
(3) standard reference material.  Primary sources for
studies in  this bibliography  been the body of data
submitted to EPA and its predecessor agencies in support
of past regulatory decisions, and the published  technical
literature.

Units of Entry.  The unit of  entry in this bibliography
is called a "study."  In the  case of published materials,
this corresponds closely to an article.  In  the case
of unpublished materials submitted to EPA, the Agency
has sought  tof identify documents at a level parallel to
a published article from within the typically larger
volumes in which they were submitted.  The resulting
"studies" generally have a distinct title (or at least a
single subject), can stand alone  for purposes of review,
and can be described with a conventional bibliographic
citation.  The Agency has attempted also to  unite basic
documents and commentaries upon them, treating them as a
single study.

Identification of  Entries.   The entries in this bibliog-
raphy are sorted by author,  date of the document, and
title.  Each entry bears, to  the left of the citation
proper, an eight-digit numeric identifier.   This number
is unique to the citations,  and should be used at any
time specific reference is required.  This number is
called the "Master Record Identifier",  or "MRID".  It is
not related to the six-digit  "Accession Number"  which
has been used to identify volumes of submitted data;  see
paragraph 4(d)(4)  below for a further explanation.   In a
few cases, entries added to  the bibliography late in the
review may be preceded by a nine-character temporary
identifier.   This  is also to be used whenever a specific
reference is needed.

Form of the  Entry.   In addition to the Master Record
Identifier (MRID),  each entry consists of a bibliographic
citation containing standard elements followed,  in
the case of  materials  submitted to EPA,  by a description
of the earliest known  submission.   The bibliographic
                   -133-

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conventions used reflect the standards of the American
National Standards Institute (ANSI), expanded to provide
for certain special needs.  Some explanatory notes of
specific elements follow:

a.  Author.  Whenever an author could confidently be
    identified, the Agency has chosen to show a personal
    author.  When no individual was  identified, the
    Agency has shown an  identifiable laboratory or
    testing facility as  author.  As  a last resort,
    the Agency has shown the first  known submitter as
    author.

b.  Document Date.  When the date appears as four
    digits with no question marks,  the Agency took it
    directly from the document.  When a four digit date
    is followed by a question mark,  the bibliographer
    deduced the date from evidence  in the document.
    When the date appears as (19??), the Agency was
    unable to determine  or estimate  the date of the
    document.

c.  Title.  This is the  third element in the citation.
    In some cases it has been necessary for Agency
    bibliographers to create or enhance a document
    title. Any such editorial insertions are contained
    between square brackets.

d.  Trailing Parentheses.  For studies submitted to the
    Agency in the past,  the trailing parentheses include
    (in addition to any  self-explanatory test) the
    following elements describing the earliest known
    submission:

    (1)  Submission Date.  Immediately following the
         word 'received* appears the date of the earliest
         known submission.

    (2)  Administrative  Number.  The next element,
         immediately following the  word 'under1, is the
         registration number, experimental permit
         number, petition number, or other administrative
         number associated with the  earliest known
         submission.

    (3)  Submitter.  The third element is the submitter,
         following the phrase 'submitted by'.  When
         authorship is defaulted to  the submitter,
         this element is omitted.
                   -134-

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(4)   Volume Identification.   The final element in
     the trailing parenthesis identifies the EPA
     accession number of the volume in which the
     original  submission of  the study appears.  The
     six-digit accession number follows the symbol
     'CDL1, standing  for "Company Data Library".
     This accession number  is in turn followed by an
     alphabetic suffix which shows the relative
     position  of the  study within the volume.   For
     example,  within  accession number 123456,  the
     first study would be 123456-A;  the second,
     123456-B;  the 26th,  123456-Z;  and the 27th,
     123456-AA.
              -135-

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                 OFFICE OF PESTICIDE PROGRAMS
              REGISTRATION STANDARD BIBLIOGRAPHY
       Citations Considered to be Part of the Data Base
        Supporting Registrations Under the Standard

Product Chemistry
MRID          CITATION

000004843     Chevron Chemical Company.  1975.  Product research
                  and services:  shelf-life test - Ortho Chinch
                  Bug Lawn Spray. (Unpublished study received Dec.
                  3f 1975 under 239-2445; CDL:228761-A)

GS0019-001    Ja, W., W.J. Smith, and J.F. Below.  1966.  The
                  analysis of technical Aspon, Richmond report
                  no. RR-66-35. Stauffer Chemical Co., New York, N.Y.

005004395     Keith, L.H.; Garrison, A.W.; Alford, A.L.  1968.
                  The high resolution NMR spectra of pesticides.
                  I. organophosphorus pesticides.  J. Assoc.  Off.
                  Anal. Chem. 51(5):1063-1094.

005001354     McMahon, B.; Bourke, J.A.  1978.  Analytical behavior
                  data for chemicals determined using AOAC multi-
                  residue methodology for pesticide residues  in
                  foods.  J. Assoc. Off. Anal. Chem.  61:640-652.

005002074     Ruzicka, J.H.; Thomson, J.; Wheals, B.B.; Moods, N.F.
                  1968.  The application of gel chromatography to
                  the separation of pesticides. Part I. organophos-
                  phorus pesticides.  J. Chromatog.  34(1):14-20.

GS0019-002    Sittig, M.  1971.  Agricultural chemicals manufacture.
                  Noyes Data Corp., Park Ridge, N.J.

GS0019-003    Sittig, M.  1977.  Pesticides process encyclopedia.
                  Noyes Data Corp., Park Ridge, N.J.

GS0019-004    Stauffer Chemical Company.  1968.  Aspon insecticide,
                  technical information bulletin.  New York,  N.Y.

GS0019-005    Stauffer Chemical Company.  1970.  Infrared procedure
                  to determine the assay of Aspon, method no. MPO 25-3,
                  New York, N.Y.  (Unpublished).
                                 -136-

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                 OFFICE OF PESTICIDE PROGRAMS
               REGISTRATION STANDARD BIBLIOGRAPHY
       Citations Considered to be Part of the Data Base
        Supporting Registrations Under the Standard

Product Chemistry
MRID           CITATION

005004479      Toy, A.D.F.  1951.  Tetraethyl dithionopyrophosphate
                  and related tetraaalkyl dithionopyrophosphates.
                  J. Amer. Che. Soc.  73:4670-4674.

GS0019-006     U.S. Patent No. 2,663,722.  1953.  Method of preparing
                  tetraalkyl dithionopyrophosphate.

Toxicology

000004858      Bullock, C.H.  1970.  Toxicology lab report—T 1520;
                  T 1549.  (Unpublished study received Apr. 18,
                  1978 under 239-2032; prepared by Stauffer Chem-
                  ical Co., submitted by Chevron Chemical Co.,
                  Richmond, Calif.; CDL:234497-C).

000004861      Bullock, C.H.  1976.  The eye irritation potential
                  of CC 7187: S-972; SOCAL 937/27:76.  (Unpublished
                  study received Apr. 18, 1978 under 239-2032; sub-
                  mitted by Chevron Chemical Co., Richmond, Calif.;
                  CDL:234497-F).

000004835      Bullock, C.H.; Narcisse, J.K.   1974.  The eye irri-
                  tation potential of Ortho Chinch Bug Spray (CC
                  5109): S-668: SOCAL 588/XX:24.  (Unpublished
                  study received Aug. 5,  1974 under 239-765; sub-
                  mitted by Chevron Chemical Co., Richmond, Calif.;
                  CDL:022718-A).

000004857     Eisenlord, G.H.  1978.  The acute oral toxicity of
                  Ortho Chinch Bug and Sod Webworm Control: S-1178;
                  SOCAL 1179/31:116.  (Unpublished study received
                  Apr. 18, 1978 under 239-2032;  submitted by Chevron
                  Chemical Co., Richmond, Calif.;  CDL:234497-B).

000004859     Eisenlord, G.H.  1978.  The skin irritation poten-
                  tial of Ortho Chinch Bug and Sod Webworm Control:
                  S-1179;  SOCAL 1180/30:132.   (Unpublished study
                  received Apr.  18,  1978  under 239-2032;  submitted
                  by Chevron Chemical Co., Richmond,  Calif.; CDL:234497-D)
                              -137-

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                 OFFICE OF PESTICIDE PROGRAMS
              REGISTRATION STANDARD BIBLIOGRAPHY
       Citations Considered to be Part of the Data Base
        Supporting Registrations Under the Standard
Toxicology
MRID
CITATION
000004833     Gregory/ L.K.; Narcisse, J.K.  1974.  The eye irri-
                  tation potential of CC-5495:  S-745; SOCAL
                  674/XX:117. (Unpublished study received June 25,
                  1975 under 239-765; submitted by Chevron Chemical
                  Co., Richmond, Calif.; CDL:220001-C).

000004836     Narcisse, J.K.  1972.  Eye irritation potential of
                  Ortho Bug Spray:  S-362; SOCAL 283/71:114.  (Un-
                  published study received Nov. 14, 1974 under
                  239-765; submitted by Chevron Chemical Co.,
                  Richmond, Calif.; CDL:051023-A).

000004837     Narcisse, J.K.  1972.  Skin irritation potential of
                  Ortho Chinch Bug Spray:  S-363; SOCAL 284B/VT:114.
                  (Unpublished study received Nov. 14, 1974 under
                  239-765; submitted by Chevron Chemical Co.,
                  Richmond, Calif.; CDL:051023-B).

000004838    Rittenhouse, J.R.; Narcisse, J.K.  1972.  The acute
                  dermal toxicity of Ortho Chinch Bug Spray: S-363;
                  SOCAL 284A/VT:117.  (Unpublished study received
                  Nov. 14, 1974 under 239-765; submitted by Chevron
                  Chemical Co., Richmond, Calif.; CDL:051023-C).

Ecological Effects
GS0019-007   EPA.  1975.  Report on the toxicity of technical
                  Aspon to rainbow trout.  (U.S. EPA, Chemical
                  and Biological Investigations Branch, Belts-
                  ville, Maryland, Static jar test No. 913,
                  unpublished report.)
GS0019-008   EPA.
     1976.  Report on the toxicity of Aspon tech-
    nical to rainbow trout.  (U.S. EPA, Chemical
    and Biological Investigations Branch, Belts-
    ville, Maryland, Static jar test No. 932,
    unpublished.)
                                 -138-

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                 OFFICE OF PESTICIDE PROGRAMS
              REGISTRATION STANDARD BIBLIOGRAPHY
       Citations Considered to be Part of the Data Base
        Supporting Registrations Under the Standard

Ecological Effects
MRID          CITATION

GS0019-009    EPA.  1976.  Report on the toxicity of Aspon
                  technical to bluegill sunfish.  (U.S. EPA,
                  Chemical and Biological Investigations Branch,
                  Beltsville, Maryland, Static jar test No. 998,
                  7/14/76, unpublished report.)

000004831     Fink, R.; Reno, F.E.  1976.  Final report:  eight-
                  day dietary LC-50—bobwhite quail:  project no.
                  132-129. (Unpublished study received March 8,
                  1976 under 476-2163;  prepared by Hazleton Labor-
                  atories America, Inc. in cooperation with Mary-
                  land Dept. of Agriculture, Div. of Inspection and
                  Regulation, submitted by Stauffer Chemical Co.,
                  Richmond, Calif.; CDL:225231-A).

GS0019-010    Hill, E.F.; Heath, R.G.;  Spann, J.W.; Williams, J.D.
                  1975.  Lethal dietary toxicities of environmental
                  pollutants to birds.   Special  Scientific Report—
                  Wildlife No. 191. U.S.  Fish and Wildlife Service,
                  Washington, D.C.

000004830     Joiner, R.L.  1975.   Safety evaluation of Aspon tech-
                  nical by a five-day feeding test in mallard ducks:
                  T-5397. (Unpublished  study received June 26, 1975
                  under 476-2163;  submitted by Stauffer Chemical Co.,
                  Richmond, Calif.; CDL:223289-A).
                                 -139-

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                 OFFICE OF PESTICIDE PROGRAMS
              REGISTRATION STANDARD BIBLIOGRAPHY
       Citations Considered to be Part of the Data Base
        Supporting Registrations Under the Standard

Toxicology - Addenda
MRID          CITATION

GS0019-019    The Andersons [sic].  1979.  Primary eye irritation
              study in the albino rabbit, primary skin irritation
              study in the albino rabbit, acute dermal toxicity
              study in the albino rabbit, acute oral toxicity study
              in rats - Turf Care 20-4-10 with Benefin and chlor-
              pyrifos.  (Unpublished studies, received May 30,
              1979, under 9198-37).

GS0019-020    Biesemeior, J.  1978.  Toxicology lab report [acute
              oral LD-50, acute dermal LD-50, skin irritation, eye
              irritation]  reference no. F-8649.  (Unpublished study
              received Apr. 24, 1979, under 538-156; prepared by
              Raltech Scientific Services, Inc. [Warf Institute,
              Madison, Wis.]; submitted by O.M. Scott & Sons, Marys-
              ville, Ohio).

GS0019-021    O.M. Scott & Sons, Co.  1979.  Acute oral toxicity,
              acute dermal toxicity, primary eye irritation, primary
              dermal irritation - Kwit and Western Lawn Insect
              Control.  (Unpublished studies received May 5, 1980,
              under 538-69.)

GS0019-022    O.M. Scott & Sons, Co.  1979.  Acute oral toxicity,
              acute dermal toxicity, primary eye irritation, primary
              dermal irritation - Western Lawn Insect Control Plus
              Fertilizer.  (Unpublished study received May 5, 1980,
              under 538-94.)

GS0019-023    Raltech Scientific Services, Inc.  1980.  Eye irrita-
              tion, Lab report 760871.  (Unpublshed study received
              May 1, 1980 under 538-137; submitted by O.M. Scott &
              Sons Co., Marysville, Ohio.)

GS0019-024    Thompson, G.W.  1980.  The primary eye irritation study
              of F6713.   (Unpublished study received June 12, 1980,
              under 538-72; prepared by Raltech Scientific Services,
              Inc.; submitted by O.M. Scott & Sons, Marysville, Ohio.
              Accession # 243155.)
                               -140-

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                 OFFICE OF PESTICIDE PROGRAMS
              REGISTRATION STANDARD BIBLIOGRAPHY
       Citations Considered to be Part of the Data Base
        Supporting Registrations Under the Standard

Toxicology - Addenda
MRID          CITATION

GS0019-025    Thompson, G.W.  1979.  Toxicology lab report - F9348.
              (Unpublished study received Nov. 6, 1979, under 538-160;
              prepared by Raltech Scientific Services, Inc.; submitted
              by O.M. Scott & Sons, Marysville, Ohio.  Accession #
              241350.)

GS0019-025    Thompson, G.W.  1980.  Toxicology lab report (acute
              oral LD-50, acute dermal LD-50, skin irritation and eye
              irritation), lab report 765242.  (Unpublished study
              received March 24, 1980, under 538-163; prepared by
              Raltech Scientific Services, Inc.;  submitted by O.M.
              Scott & Sons, Marysville,  Ohio.)
                             -141-

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                 OFFICE OF PESTICIDE PROGRAMS
              REGISTRATION STANDARD BIBLIOGRAPHY
       Citations Examined and Judged Inappropriate For
                Use in Developing the Standard

MRID          CITATION
005004090     Bagdon, R.E.; DuBois, K.P.  1955.  Pharmacologic
                  effects of chlorthion, malathion and tetra-
                  propyl dithionopyrophosphate in mammals.  Arch.
                  Inter. Phatmacod. Therap.  Cin (2/3): 192-199.

000004829     Bresolin, P.M.  1975.  Toxicology laboratory report
                  T-5284: Aspon technical.  (Unpublished study
                  received Dec'. 5, 1975 under 476-2163; submitted
                  by Stauffer Chemical Co., Richmond, Calif.;
                  CDL:223288-A).

000004853     Chevron Chemical Company.  19??.  Summary statement:
                  Ortho Chinch Bug and Sod Webworm Control.  Sum-
                  mary of studies 222347-B through 222347-C.  (Un-
                  published study received May 6f 1975 under
                  239-2032; CDL: 222347-A).

000004855     Chevron Chemical Company.  19??.  Summary statement:
                  Ortho Sod Webvrorm Control.  Summary of studies
                  222348-B through 222348-C.  (Unpublished study
                  received Apr. 18, 1975 under 239-2389; CDL:222348-A)

000004841     Chevron Chemical Company.  19??.  Summary table:
                  efficacy data at 3.7 Ib Ai/A (Aspon).  (Unpub-
                  lished study received March 31, 1960 under 239-765;
                  CDL:222167-B) .

000004849     Chevron Chemical Company.  1971.  Summary:  Ortho
                  Sod Webworm Control.  (Unpublished study includ-
                  ing OR 513 report nos. 378-1, 387-41, 621-37,
                  621-36, 623-07, 623-06, 504-23, received Dec. 20,
                  1971 under 239-2389; CDL:001557-A).

000004842     Chevron Chemical Company.  1974[?].  Sunmary state-
                  ment: Ortho Chinch Bug Spray.  Summary of studies
                  2222170-B through 222170-C.  (Unpublished study
                  received Apr. 24, 1975 under 239-765; CDL:222170-A).

000004854     Chevron Chemical Company.  1974.  Aspon, Dursban.
                  (Unpublished study including report nos. 627.02,
                  627.27, 623.09-623.12, 504.23, 504.26, 366.10,
                  658.29, 657.35, 519.23, 748.20, 727-23, 519.30,
                  727.24, 727.30, 627.23, 627.24, received May 6,
                  1975 under 239-2032; CDL: 222347-C).
                                 -142-

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                  OFFICE OF PESTICIDE PROGRAMS
               REGISTRATION STANDARD BIBLIOGRAPHY
        Citations Examined and Judged Inappropriate For
                 Use in Developing the Standard

 MRID          CITATION
 000004832     Chevron Chemical Company.   1975.   Summary statement.
                   Summary of study 220001-D.   (Unpublished study
                   received June 25,  1975  under  239-765;  CDL: 220001-A).

 000004847     Chevron Chemical Company.   1975.   Summary statement—
                   phytotoxicity:   Ortho Chinch  Bug  Lawn  Spray.
                   Summary of study 2288758-B.   (Unpublished study
                   received Dec.  3,  1975 under 239-2445;  CDL:228758-A).

 000004845     Chevron Chemical Company.   1975.   Summary  statement -
                   phytotoxicity:   Ortho Sod Webworm Lawn Spray.
                   Summary of study 228762-B.  (Unpublished  study
                   received Dec.  16,  1975  under  239-2446; CDL:228762-A)

 000004850     Chevron Chemical Company.   1975.   Summary  statement:
                   Aspon.   Summary of study 133068-C.   (Unpublished
                   study received  June 25, 1975  under 239-2389;
                   CDL:133068-A).

 GS0019-011     EPA.  1975.   Report on the  toxicity of Ortho  Sod
                   Webworm  (13% active ingredient) to Daphnia magna.
                   (U.S.  EPA,  Chemical  and Biological Investigations
                   Branch,  Beltsville,  Maryland, Static jar  test No.
                   865,  8/21/75, unpublished.)

GS0019-012     EPA.  1975.   Report on the toxicity of Ortho Sod-
                  Webworm  13%  active  ingredient to  rainbow trout.
                   (U.S.  EPA, Chemical  and Biological Investigations
                   Branch,  Beltsville, Maryland, Static jar test No.
                   848,  7/8/75, unpublished report.)

GS0019-013     EPA.  1975.  Report on  the toxicity of Ortho Chinch
                  Bug Control, 3.2% a.i., to bluegills.  (U.S. EPA,
                  Beltsville, Maryland, Static jar test No. 876,
                  9/22/75, unpublished report.)

GS0019-014    EPA.  1975.  Report on  the toxicity of Ortho Chinch
                  Bug Control on bluegills.   (U.S. EPA, Chemical
                  and Biological  Investigations Branch, Beltsville,
                  Maryland, Static jar test  No.  866, 8/21/75,
                  unpublished.)
                                 -143-

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                 OFFICE OF PESTICIDE PROGRAMS
              REGISTRATION STANDARD BIBLIOGRAPHY
       Citations Examined and Judged Inappropriate For
                Use in Developing the Standard

MRID          CITATION
000005003     Lindemann, R.H.; Massey, V.C.; Coltharp, J.L.;
                  Bryant, W.F.  1974.  Product performance report:
                  OR-513 report no. 657-10.  (Unpublished study
                  including OR report nos. 705-41, 748-21, 748-22,
                  705-25, 705-23 and 705-42, received June 25, 1975
                  under 239-2389; submitted by Chevron Chemical Co.,
                  Richmond, Calif.; CDL: 133068-C).

000004848     Pate, D.A.  1967.  Ortho Chinch Bug Control with
                  fertilizer. (Unpublished study including OR-513
                  report nos. 238-40, 238-41, 237-20, 230-47, 234-5,
                  234-2, 230-26, 230-49, received May 6, 1968 under
                  239-2265; submitted by Chevron Chemical Co.,
                  Richmond, Calif.; CDL:001512-A).

000005377     Radeleff, R.D.; Wbodard, G.T.  1957.  The toxicity
                  of organic phosphorus insecticides to livestock.
                  J. Amer. Vet. Med. Assoc.  130(5): 215-216.

000004860     Rittenhouse, J.R.  1978.  The acute inhalation
                  toxicity of Ortho Chinch Bug and Sod Webworm
                  Control: S-1180; SCCAL 1181/28:142.  (Unpub-
                  lished study received Apr. 18, 1978 under 239-
                  2032; submitted by Chevron Chemical Co., Richmond,
                  Calif.; CDL:234497-E).

000004834     Sherman, M.; Chang, M.T.Y.; Herrick, R.B.  1969.  Fly
                  control, chronic toxicity, and residues from feed-
                  ing propyl thiopyrophosphate to laying hens.  J.
                  Econ. Entonol.  62(6):1494-1499.

005004694     Sherman, M; Ross, E.; Chang, M.T.Y.  1964.  Acute and
                  subacute toxicity of several organophosphorus in-
                  secticides to chicks.  Toxicol. Appl. Pharmacol.
                  6(2):147-153.
                                 -144-

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MRID
GS0019-015



GS0019-016


GS0019-017
GS0019-018
   OFFICE OF PESTICIDE PROGRAMS
REGISTRATION STANDARD BIBLIOGRAPHY
   Standard Reference Material

CITATION
Chemline, Chemical Information on Line [Data base].
    Bethesda, Md:  National Library of Medicine.
    March 1980.

EPA.  1976.  EPA manual of chemical methods for
    pesticides and devices.  AOAC, Arlington,
    Virginia.

EPA.  1979.  Pesticide chemical use pattern profile
    for Aspon.  Washington, D.C.  (Unpublished).

Martin, H.; Worthing, C.R., eds.  1977.  Pesticide
    index: basic information on the chemicals used
    as active components of pesticides.  5th ed.
    British Crop Protection Council, Wbrcestershire,
    England.

Spencer, E.Y.   1973.   Guide to the chemicals used in
    crop protection.   6th ed.   Canada Dept.  of Agri-
    culture, Ontario, Canada.
                                -145-

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                                        Appendix A
             Table 1.   Required Toxlcity Category Warning Statements for Aspon^Products
(Exposure
I  Route
I
                  I
                 T
I
iToxiclty Category I      |Toxlcity Category II     iToxiclty Category III    iToxicity Category IV
ty Catego
If swallc
ty Categ
 fatal I
I Oral*
[Fatal If swallowed.  WashlMay be fatal  if swal-  -| Harmful ^fswallowed.
(throroughly with soap   (lowed. Nash thoroughly  (Mash thoroughly after
(and water after handling!with soap and water af- (handling.
(and before eating or    |ter handling  and before j
I smoking.	j eating or smoking.	|	
(No precautionary state-
jmerit required.
I Dermal*     (Fatal if absorbed       I May be fatal  if absorbed) Harmful  If abosrbed
             (through skin.  Do not get)through skin.  Do not  get)through  skin.  Avoid
             Jin eyes, on skin, or on j in eyes, on skin, or  on (contact  with skin,  eyes,
             (clothing. Wear protec-  (clothing. Wear protec-  (or clothing. Wash thor-
             (tive clothing  and rubberItlve clothing  and rubberjoughly after handling.
             (gloves. Wash thoroughly (gloves. Wash  thoroughly
             (after handling and be-  (with soap and  water af-
             jfore eating or smoking, jter handling  and before
             (Remove contaminated     (eating or smoking.  Re-
             jclothing and wash be fore (move contaminated cloth-
             jreuse.                  (ing and wash  before
             I	(reuse.	
                                                                           No precaautlonary state-
                                                                           ment  required.
(Inhalation* (Fatal If inhaled. Do notlMay be fatal  It Inhaled.(Harmful  If Inhaled.
             (breathe dust (vapor or  (Do not breathe dust (va-|Avoid  breathing  dust
             (spray mist). Wear a masMpor or spray  mist). Wear) (vapor or  spray  mist).
             (or pesticide respirator (a mask or pesticide res-(Remove contaminated
             .'jointly approved by the jpirator jointly approved)clothing and wash before
             (Mining Enforcement and  (by the Mining Enforce-  (reuse. Keep container
             (Safety Administration   |merit and Safety Admlni- (closed when not  in use.
             ((formerly the U.S. Bur- (stration (formerly the  (Use only with  adequate
             jeau of Mines) and the   (U.S. Bureau of Mines)    (ventilation.
             (National Institute for  (and the National Insti-
             lOccupational Safety and (tute for Occupational
             (Health. Remove contami- (Safety and Health. Re-
             (nated clothing and wash (move contaminated cloth-
             jbefore reuse.           (Ing and wash  before
             I	             (reuse.
                                                                           No precautionary  state-
                                                                           ment  required.
                              -147-

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                           Appendix A
Table 1.  Required Toxlcity Category Warning Statements  for AsporP'Products
(Exposure 1 1 1 1
Route 1 Toxlcity Category I iToxlclty Category II (Toxlclty Category III j Toxlcity Category IV
IRye effects (Corrosive. Causes eye (Causes eye Irritation. (Avoid contact with eyes
(damage. Harmful or fatallHarmful If swallowed. Dolor clothing. Wash thor-
jlf swallowed. Do not getfnot get In eyes or on joughly after handling.
jln eyes, or oh clothing. (clothing. Mash thorough- I
(Wear goggles, or face jly after handling. Re-
jshleld. Mash thoroughly (move contaminated cloth-l
(after handling. Remove (Ing and wash before re-
jcontamlnated clothing (use.
(and wash before reuse. I
Skin effectslCorroslve. Causes burns. (Causes skin Irritation. Avoid contact with skin
(Do not get on skin or on|Do not get on skin or on|or clothing. Hash thor-
jclothlng. Wear protec- (clothing. Wash tho rough- joughly after handling.
Itlve clothing and rubber |ly after handling. Re-
jgloves.l Wash thoroughly (move contamlned clothing)
(after handling. Remove .(and wash before reuse, j
(contaminated clothing I I
(and wash before reuse, j
(Signal Word 1 DANGER I WARNING CAUTION
INo precautionary
Intent required.
No precautionary
ment required.
state-
state-
CAUTION
* Any product which falls Into Toxlcity Category I for the oral, dermal, or Inhalation acute toxiclty categories
will be required to carry the word "Poison" on the label with a skull and crossbones.
1 The need for gloves must be determined on an Individual basis. Some products cause blistering If confined
under clothing.
                 -148-

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          Appendix A
                Table 2.  Required First Aid Statements
1 Exposure 1 I 1 I
1 Route (Toxlcity Category I JToxlcity Category II JToxicity Category III JToxicity Category IV
lOral |IC swallowed: Drink 1 or 2
|g lasses of water and induce vomit-
ling by touching back of throat
(with finger. Do not give anything
(by mouth to an unconscious person.
(Get medical attention.
(For ECs with >10% petroleum dis-
jtillates; If the patient is uicon-
jsclous, maintain breathing and
(heart beat (CPR:cardiopulmonary
(resuscitation). Contact your local
(Posion Control Center, hospital,
(or physician immediately. If the
(patient is conscious. Induce votni-
jting (syrup of Ipecac; if not
(available, stimulate the back of
(throat with finger). Never give
(anything by mouth to an uncon-
jscious person!
Dermal (If on skin: Wash with plenty of
(soap and water.
Inhalation (If inhaled: Remove victim to fresh
jaTr. If not breathing, give arti-
jficial respiration, preferably
jmouth-to-mouth. Get medical at ten-
It Ion.
Same as for Toxicity Category I. (Same as for Toxiclty Category I. 1
For ECs with >10% petroleum dls- (For ECs with >10% petroleum dis-
tillates: If the patient is uncon-
sclous, maintain breathing and
heart beat (CPR:cardiopulmonary
resuscitation). Contact your local
Poison Control Center, hospital,
or physician immediately. [The.
question whether to Induce vomit-
ing will be determined on a case-
by case basis.]
Same as for Toxiclty Category I.
Same as for Toxicity Category I.
tillates; If the patient is uncon-|
scious, maintain breathing and
heart beat (CPR:cardiopulmonary
resuscitation). Contact your local
Poison Control Center, hospital,
or physician Immediately. [The
question whether to induce vomit-
ing will be determined on a case-
by case basis.]
No first aid statement
required.
For ECs with >10» petro-
leum distillates: If the
patient is unconscious,
maintain breathing and
heart beat (CPR:cardio-
pulmonary resuscita-
tion) . Contact your lo-
cal Poison Control Cen-
ter, hospital, or physi-
cian immediately. Do not
induce vomiting!
Same as for Toxicity Category I. |No first aid statement
(required.
Same as for Toxicity Category I.
No first aid statement
required.
-149-

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                                         Appendix A
                                               Table 2.   Required First Aid Statements CONTINUED
(Exposure
I  Route
             iToxiclty Category I
                          fg°ry
                          Flush
I
iToxicity Category II
I
IToxicity Category III
Ity C.
 skin
r
IToxicity Category IV
(Eye effects lit in eyes;  Flush with water tor  (Sane  as  for Category I, except
             ITS minutes.  Get medical attention.jomit  Note  to  Physician.
             (If swallowed:  Drink  promptly a
             (Targe quantity of milk, egg
             (whites, gelatin solution, or;  If
             (these are  not  available, drink
             (large quantities of  water. Avoid
             (alcohol.   NOTE TO*PHYSICIAN: Prob-
             lable mucosal damage  may contrain-
  	jdicate the use of gastric lavage.
                                   |If on skin;  Wash with  plenty of   |No first aid statement
                                   jsoap and water.   Get medical at-   (required.
                                   |tent Ion if irritation  persists.
Skin effects|I£ on skin: Wash with  water. Get
             (medical  attention.
             (If swallowed:  Drink  promptly a
             (Targe quantity of milk, egg
             (whites,  gelatin solution, or, if
             (these are not  available, drink
             (large quantities of  water. Avoid
             (alcohol. NOTE TO PHYSICIAN: Prob-
             lable  mucosal damage  may contraIn-
  	Idicate the use of gastric lavage.
                                                Same as for Category I, except
                                                omit Note to Physician.
                                   (It on skin; Washwitn plenty of
                                   jsoap and water.  Get medical at-
                                   |tentIon  if  irritation persists.
                                   No  first aid  statement
                                   required.
                                                                                                      •U S GOVERNMENT PRINTING OFFICE:  1980 341-085/3045
                             -150-

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