EPA-660/2-74-069
June 1974
                         Environmental Protection  Technology Series
    Studies  of   Low Molecular

    Weight  Lignin  Sulfonates
                                   Office of Research and Development

                                   U.S. Environmental Protection Agency

                                   Washington, D.C. 20460

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            RESEARCH REPORTING SERIES
Research reports of the  Office  of  Research  and
Monitoring,  Environmental Protection Agency/ have
been grouped into five series.  These  five  broad
categories  were established to facilitate further
development  and  application   of   environmental
technology.   Elimination  of traditional grouping
was  consciously  planned  to  foster   technology
transfer   and  a  maximum  interface  in  related
fields.  The five series are;

   1.  Environmental Health Effects Research
   2.  Environmental Protection Technology
   3.  Ecological Research
   4.  Environmental Monitoring
   5.  Socioeconomic Environmental Studies

This report has been assigned to the ENVIRONMENTAL
PROTECTION   TECHNOLOGY   series.    This   series
describes   research   performed  to  develop  and
demonstrate   instrumentation,    equipment    and
methodology  to  repair  or  prevent environmental
degradation from point and  non-point  sources  of
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                                                EPA-660/2-74-069
                                                June 1974
                         STUDIES OF

           LOW  MOLECULAR WEIGHT LIGNIN  SULFONATES
                             by

   Wolfgang  G.  Glasser               Bjorn F.  Hrutfiord
     Josef S.  Gratzl                 Lennart N. Johanson
         Kaj  Forss                    Joseph L. McCarthy
                     Juanita J. Collins
                     Roap/Task 21 AZX 60
                      Project  12040 DEH
                   Program  Element 1BB037


                       Project Officer
                     Dr. H. Kirk Willard
     Pacific Northwest Environmental  Research Laboratory
            National Environmental  Research Center
                  Corvallis, Oregon  97330
                           for the

            OFFICE OF RESEARCH AND DEVELOPMENT
           U.S. ENVIRONMENTAL PROTECTION AGENCY
                 WASHINGTON,  D.C.  20460
For sale by the Superintendent of Documents, U.S. Government Printing Office, Washington, D.C. 20402 - Price $1.55

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              EPA Review Notice


This report has  been reviewed  by  the  Environmental
Protection Agency and approved for publication.
Approval  does not signify that the contents
necessarily reflect the views  and policies of
the Environmental Protection Agency,  nor  does
mention of trade names or commercial  products
constitute endorsement or recommendation  for use.
                       ii

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                             ABSTRACT





     Low molecular weight lignin sulfonates have been separated in



purified form and characterized by physicochemical  and chemical methods.



Their structures and reactions have been evaluated.   Preliminary studies



on the feasibility of industrial scale separations  have been performed.



     Lignin sulfonates from the spent sulfite liquor of a mild acid



bisulfite cook of Western Hemlock (Tsuga heterophylla) were purified and



fractionated in Sephadex G-25 column chromatography.   Samples with varying



molecular weights were analyzed using a new method  which aided the elim-



ination of the polydisperse nature of the material  under investigation.



This method which involved acetylation of hydroxyI-groups and ester ificat ion



of sulfonate-groups was widely developed in the course of this study using



model compounds.



     Complete elemental  and functional  group compositions were established



for  lignin sulfonates from a spent sulfite Iiquor and compared to  those



from milled wood  lignin preparation,  allowed  an  estimate of the



degree of sulfonation, condensation and demethylation as welI.



     Extended separation studies indicated the low  molecular weight lignin



sulfonates to be the reaction product of a difunctional vinyl-type poly-



merization, thus accounting for the widely different properties as compared



to their higher molecular weight counterparts (two- versus three-




dimensional network).



     The feasibility of large scale separations was piloted employing two




different separation principles:  one was the extraction and/or precipi-



tation of the dry matter in a spent sulfite liquor with alcohol, the
                                  iii

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second was the fractionation of the material by Ion exclusion in a



column arrangement.  Both methods seem to allow the separation of



basically three different classes of substances, namely, high molecular



weight LS, low molecular weight LS, and carbohydrate degradation



products.

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                             CONTENTS

Section                                                             Page
I         Conclusions                                                  I
11        Recommendations                                              3
11 I       Introduction                                                 5
IV       Objectives and Plans                                         9
V        Preparation, Fractlonation and Preliminary Characteriza-    II
           tion of Gymnosperm Lignin Sulfonates
VI        Preparation of Certain LOMOLS-like Monomers and Dimers and  19
           Characterization by NMR and Mass Spectroscopy
VII       Preparation of Acetyl Lignin Sulfonate Methyl Ester (ALSME)  29
           and their Spectroscopic Characterizations
VIII     Structural Studies of Acetyl Lignin Sulfonate Methyl Esters 39
           Derived from Milled Wood Lignin
IX       Structure and Reactivity of LOMOLS                          53
X        Preliminary Studies on Industrial Scale Separation of SSL   63
           Components
XI        Concluding Comments                                         73
X11       AcknowIedgements                                            75
XIII     References                                                  77
XIV      Publications and Patents                                    81
XV       Glossary                                                    83

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                                FIGURES

                                                              Page

 1      PREPARATION OF SPENT SULFITE LIQUOR                     12

 2      FRACTIONALON OF SULFONATES IN SPENT SULFITE LIQUOR     14
         BY GEL CHROMATOGRAPHY ON SEPHADEX G-25

 3      SHIFT OF THE WAVELENGTH OF THE ABSORPTION MAXIMUM       17
         NEAR 280 nm ON ALKALIZING FRACTIONS OF THE SPENT
         SULFITE LIQUOR

 k      REACTION SCHEME FOR THE TRANSFORMATION PROCEDURE        21

 5      THE FOUR TYPES OF LOMOLS-LIKE MONOMERS AND DIMERS       23
         SYNTHESIZED

 6      NMR-SPECTRUM OF A TYPICAL LOMOLS-LIKE DIMER             26

 7      MASS-SPECTRUM AND FRAGMENTATION PATTERN OF A TYPICAL    27
         LOMOLS-LIKE DIMER

 8      NMR SPECTRA OF ALSME DERIVATIVES,  PREPARED FROM VAR-    30
         IOUS FRACTIONS FROM SEPHADEX G-25 SEPARATIONS

 9      SEPHADEX LH-20 SEPARATIONS OF SOME ALSME FRACTIONS      32
         IN METHANOL

10      CORRELATION BETWEEN PHENOLIC HYDROXYL GROUPS AND ARO-   34
         MAT 1C PROTONS IN FRACTIONS FROM  SEPHADEX SEPARATIONS

11      THE CARBONYL REGION IN IR-SPECTRA  OF FRACTIONS FROM     36
         SEPHADEX SEPARATIONS

12      HYPOTHETICAL DIMER FORMATION MECHANISM                  38

13      ELUTION DIAGRAMS OF CALCIUM LIGNIN SULFONATES           42

14      ELEMENTAL AND FUNCTIONAL GROUP COMPOSITION OF MWL-      45
         ALSME

15      SCHEME 3                                                46

16      SCHEME 6                                                48

17      OXYGEN FUNCTION IN ALSME DERIVATIVES OF MWL             49

18      ELUTION DIAGRAM OF ES ALSME DERIVATIVES AND THE         56
         REFRACTIONATION PATTERNS OF SOME MER CLASSES
                                   vi

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                                                              Page

19     THE "REGENERATION PATHWAY" IN TERMS OF PEAKS, AS         59
         VISUALIZED FROM THE SEPHADEX LH-20 FRACTIONATIONS

20     ELUTION DIAGRAM OF BROMINATED ES'ALSME DERIVATIVES'  ?£ - 60
         AND THE REFRACTIONAT ION PATTERNS OF SOME MER CLASSES
                                         f
21     ACID HYDROLYSIS OF THE VERATRYL-GLYCERYL-6-ARYLETHER,    61
         ITS SULFONATION AND POLYMERIZATION PRODUCTS
                                                          ,.!."*
22     DISSOLUTION OF SSL SOLIDS AS A FUNCTION OF THE WATER     66
         CONTENT OF ETHANOL                   -••  ,         >   *

23     ELUTION DIAGRAM OF A SSL IN ION EXCLUSION CHROMA-        69
         TOGRAPHY
                                    vli

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                               TABLES

No.                                                            Page

1     Characteristics of Ultraviolet Absorption                 16

2     Chemical Shifts for Acetylated and Esterfied Lignin       25
        Sulfonates In NMR Spectroscopy

3     Empirical Formulae of ALSEME Derivatives of MWL           43

4     Extraction Conditions                                     65
                               viii

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                             SECTION I
                            CONCLUSIONS

Low molecular weight lignin sulfonates can be separated in purified form
from most other materials in spent sulfite liquors of the acid bisulfite
pulping process by use of ion exclusion processes functioning in packed
column equipment.  Selective extraction or precipitation with alcohol  of
lignin sulfonates In aqueous solution does not yield particularly useful
results.
Separation of purified lignin sulfonates into fractions of differing
average molecular weights can be conducted effectively on a laboratory
basis in aqueous solution by use of gel permeation with molecular sieve
materials such as Sephadex 25 contained in a column.
The separated lignin sulfonates from two separate sources (one from a
commercial spent sulfite liquor, and the other from a sulfonated milled
wood lignin) showed gel chromatography elution patterns, ultra violet
absorptions and certain other characteristics which were quite similar
to each other in view of the differences in the two preparation procedures.
It was concluded that further useful characterization of the lignin
sulfonate fraction might be accomplished by using a derivative soluble In
organic solvents and therefore a procedure was developed for preparation
of acetylated lignin sulfonate methyl esters (ALSME).
To provide experience toward synthesizing the ALSME preparations, acety-
lated methyl sulfonate ester derivatives were prepared for some eighteen
different lignin su I f onate*-1 i ke monomers and dimers.  These were
characterized by chemical analyses, NMR spectroscopy and mass spectroscopy.
                                 I

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Preparation of the ALSME fractions succeeded.  These materials gave rise
to NMR spectra which yielded further information concerning the structure
of the lignin sulfonate molecules of differing molecular weights.
Especially significant is the finding of an orderly change in phenolic
hydroxyl  content as a function of the molecular weight of lignin sulfonates.
Generally, the low molecular weight lignin sulfonates appear to arise
perhaps mainly as hydrolysis products of high molecular weight lignin
sulfonates, although some condensation or repolymerization of the low
molecular weight entities seems to occur simultaneously.

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                            SECTION II

                          RECOMMENDATIONS
 *         •             »

The Ion exclusion process for at  least partial separation of llgnln

sulfonates from sugars and other^materials in sulfite spent liquors should

be developed further toward application on at least a small pilot plant

industrial scale.  The process desirably will be multi-stage and may be

conducted intermittently or batchwise using a column packed with an

appropriate ion exchange resin.  Preferably the process should be carried

out using continuous Ion exclusion resion handling equipment as soon as

such equipment becomes available.

Further  laboratory studies should be carried out using the now-reported

separation procedure for ALSME derivatives dissolved in organic solvents

based upon use of an appropriate molecular sieve material such as

Sephadex LH?0» and directed toward securing highly effective laboratory

separations of lignin sulfonates of differing molecular weights.

Simultaneously, further searches should be made to find organic

solvents which dissolve lignin sulfonates and permit direct gel

permeation chromatorgraphy separation.  It seems possible that such

procedures may permit the isolation in approximately pure form of

lignin sulfonates with degree of polymerization up to five or

possibly even up to ten.

Practially oriented research and development work should be carried out

to learn how to make best economic use of the phenolic hydroxyl groupings

indicated to be present rather extensively in low molecular weight

lignin sulfonates.  For example, a variety of ethers and esters could

be produced which may have industrial uses.

                                 3

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The apparent capability of of the ALSME to polymerize under certain



conditions suggests that further studies on the polymerlzability of



lignin sulfonates should be conducted, and upon the nature and possible



commercial use of the resultant polymers.

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                           SECTION III



                          INTRODUCTION






     Lignln is a polymeric substance or class of substances, composed of



phenol propane type units, which makes up about 20% to 30% of wood tissue.



Throughout the world, wood cellulose or wood pulp is produced on a very



large scale from woody tissue, leaving the lignins and lignin derivatives



in spent pulping liquor which is usually evaporated and burned to recover



heat and chemicals.



     In one type of wood pulping process, the "sulfite" or "bisulfite



process," delignification is accomplished by the use of aqueous solutions



of metal bisulfites, either calcium, magnesium, sodium or ammonium bisul-



fite.  Extensive investigations have been conducted and are continuing to



be directed to the development of effective and economically competitive



sulfite process recovery processes based on the recovery of effluent



liquors, and then evaporating and burning to recover useful process chemi-



cals and heat.



     An alternative path is to develop methods for production of marketable



by-products from the lignin.  From the sulfite process, lignin sulfonates



may be produced.  Many studies have been conducted toward the objective



of producing useful products from these materials and success in applica-



tion and sales has been achieved in a few instances.



     For further progress toward the aim of developing useful products,



two main advances seem to be necessary, i.e., firstly, to secure more



information concerning the physical nature and chemical structure and




reactions of the lignin sulfonates and the 30$ of substances which coexist

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in the sulfite process effluent liquors, and secondly, to secure more



information concerning how effectively and economically to separate these



components one from another.



     Toward these general objectives, research has been continuing in this



laboratory over many years, and the studies now to be reported comprise a



continuation of this effort.



Earlier Studies



     Since about 1945, research on spent sulfite liquor and lignin sulfon-



ates has been carried out at the University of Washington.  During recent



years this research has been concentrated on lignin sulfonates and the



following specific work has been performed:  Very low molecular weight



lignin sulfonates, previously shown to comprise a few percent of the total



lignin sulfonates of gymnosperms,  have been fractionated using the tech-



niques of column chromatography and multistage partition between butanol



and water.  Two monomeric lignin sulfonates and a dimeric lignin sulfonate



have been isolated, crystallized,  and shown to be the major components



of the lowest molecular weight fractions.  Evidence has been obtained



for the presence of many other individual lignin sulfonates.



     Dioxane lignin was prepared from carefully extracted wood and sul-



fonated.  The resulting  lignin sulfonates were separated into a high and



low molecular weight fraction, using a new.and fast method based on the



solubility of low molecular weight sulfonates in n-butanol saturated with



water.  Upon chromatographic separation of the low molecular weight



material  and purification of the appropriate fractions, crystalline



material  was isolated and found to be identical with  low molecular weight



lignin sulfonates previously isolated from spent sulfite  liquor.

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     The two monomeric'lignin sulfonates were isolated, crystallized and



identified as (3-methoxy-4-hydroxyphenyI)-2-propene-l-sulfonate and I-



(3-methoxy-4-hydroxyphenyl)-l-propene-3-suIfonate.  The identity has been



verified by synthesis (I, 2).



Recent Studies



     In more recent work, sodium Iignin sulfonates from gymnosperm woods



were fractionated using Sephadex G-50 gel  columns and eluting with distilled


                -1       -4
water or with 10   to 10   M NaCI solutions.  Molecular weights of certain



Iignin sulfonate fractions were estimated by ultracentrifuge sedimentation



equilibrium and were found to range in an orderly manner from about 70,000



in the mostly excluded  initial eluates down to several hundred in the final



eluates.  The sizes of the Iignin sulfonate polymer molecules in terms of



equivalent Einstein spheres,  r , were estimated from the measured molecular



weights and from intrinsic viscosities calculated using relationships



reported by Goring and coworkers.  These ranged from about 7 to 70 A (3, 4).



     For a Iignin sulfonate of a particular molecular weight, r  was



estimated to be up to two times greater in water than in O.I M NaCI solu-



tion, behavior expected for an elastic network containing negative charge



sites in an environment of varying ionic strength.



     We have shown that the concentration of sodium chloride in the aqueous



eluant exerts a significant  influence upon the degree of success attained



in the fractionation of  Iignin sulfonates.  To secure satisfactory repro-



ducibility in fractionation,  the concentration of electrolyte must be held



constant.  To secure optimum fractionation of Iignin sulfonates, a par-



ticular level of eluant electrolyte concentration should be maintained



which is appropriate in relation to the pore size of the molecular sieve



material which is to be,used.

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     These relationships are of particular significance because our



research confirms the concept that the effective size of a lignin sulfon-



ate molecule may be changed substantially by change in the concentration



of electrolyte solution in which the molecule is dissolved.



     When the size of the lignin sulfonate molecules falls approximately



within the range of the sizes of the pores in the particular Sephadex



molecular sieve, effective fractionation may occur.  In further gel



chromatography fractionations, gymnosperm lignin sulfonates in aqueous



NaCI at 0.001 M and other molarities have been separated into ten sub-



stances or mixtures of substances amounting to about eighteen percent of



the weight of total lignin sulfonates.  The ultraviolet spectra of these



was about the same as that of the unfractionated sample.  Sedimentation



equilibrium molecular weights of the entities ranged from several hundred



up to about three thousand.  The entities appear to be the lower molecular



weight members of the polymer series of lignin sulfonates.



     Based on the molecular weights measured for these "peak" substances,



we have speculated that the peaks represent lignin sulfonate mers extending



up to the 10-mer or 12-mer, and possibly the 14-mer (4).
                                8

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                            SECTION IV
                       OBJECTIVES AND PLANS

Our general objective was to find new information concerning lignin
sulfonates, and especially those of low molecular weight, which would
provide a better foundation for development of profitable utilization
or the innocuous and economic disposal of these materials, and of the
spent sulfite liquors in which they are contained.

The specific aims of the research program were:
(a)  To secure further knowledge of how to purify low molecular weight
lignin sulfonates by separating them from other classes of materials, •
such as higher molecular weight lignin sulfonates, sugars and carbohydrates,
inroganic substances, etc.
(b)  To learn how to separate purified lignin sulfonates into fractions
of differing molecular weights with certain factions hopefully to consist
mainly of particular lignin sulfonate mers, such as monomers, dimers,
trimers, and higher mers.  It was anticipated that some crystalline monomers
might be obtained but mainly it was expected that a mixture of several
different mers would be found in each fraction;
(c)  To characterize each  lignin sulfonate fraction by a number of spectro-
scopic and other available procedures in order to secure additional
knowledge of the chemical structure and reactions of lignin sulfonates.
(d)  To prepare and characterize derivatives of low molecular weight
lignin sulfonates to augment the information gained by characterization
of the lignin sulfonates themselves;
(e)  To try to find new approaches to the economic utilization of  lignin
sulfonates.
                                 9

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                             SECTION V

            PREPARATION, FRACTIONAL ON, AND PRELIMINARY

         CHARACTERIZATION OF GYMNOSPERM LIGNIN SULFONATES



Introduction

     The first step taken to initiate the investigation was to proceed

with the preparation of the gymnosperms lignin sulfonates (for prior work,

see ref. 5,6,7). in view of the importance in the pulp and paper industry,

Western Hemlock wood was chosen as the basis for the investigation.

Purification and Separation

     By courtesy of the Weyerhaeuser Company in Everett, Washington,  spent
                t
sulfite liquor was prepared by pulping Western Hemlock in a laboratory

digester under mild conditions utilizing calcium base pulping liquor.

Mild conditions were used in order to secure a larger than usual  proportion

of  low molecular weight lignin sulfonates in the resultant calcium base

sulfite Iiquor.

     This calcium base  liquor was then treated in accordance with the

flow sheet given as Figure I; and then, more specifically, according to

the following procedure.  The liquor was degassed, passed through Dowex

50-8X to remove metal ions and yield free acids, then neutralized with

barium hydroxide.  The barium sulfate precipitate was removed by centri-

fuging and the final material concentrated by evaporation.

     A sample of this concentrated BaSSL was applied to a column contain-

ing Dowex 50W-X2 ion exchange resin to achieve separation of strong

electrolytes (ligpin sulfonates) from weak electrolytes Cacetic acid,

aldonic acids) and non-electrolytes especially including sugars.  The

effluent was collected  intermittently after having been examined by a

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                              FIGURE I


                 Preparation  of  Spent Sulfite Liquor
 Sulfite  Pulping
 Spent Sulfite  Liquor
  Dowex  50W-X8  De-ashing
  S0~  Stripping
  Ether  Extraction
  Ba(OH)2  Addition;  Centrifugation
                   T
I  Dowex  50W-X2:Ion  Exclusion  Separation
                   I
  Purified  Lignin  Sulfonates

                   Y
 Ca(OH)2  Neutralization
  Sephadex  G-25  Fractionation
                    I
  Low Molecular Weight  Lignin  Sulfonates
     Gel Iulose Pulps
     Ca
     SO
     Ether Solubles
    BaSCL,  etc.
-*.   Carbohydrates

    +  Aliphatic -  COOH
-*•   High  and  Medium
High and Med?

Mol. Wt. Lig.
                                                                 g.  SuIfonates
                                 12

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continuous UV recording apparatus, then neutralized with calcium hydroxide


and concentrated by evaporation.  This CaSSL was subjected to Sephadex G-25


gel chromatography and the absorbance at 280 nm of the resultant elution

liquid was recorded and is shown  in Figure 2.


     The relatively small size of the peak in the effluent volume range

2,200 - 2,600 ml in Figure 2 shows that the spent sulfite liquor contained

only a small proportion of Iignosulfonates excluded by Sephadex G-25, i.e.


Iignosulfonates with molecular weights larger than 10,000 (7).  This is
                      *
in all probability due to incomplete delignification during the cook that

was performed in order to produce a high proportion of low-molecular-weight


sulfonates.

     The eluted liquid was divided into a series of sixteen fractions

(A-PJ and  in each case, an overlapping peak was defined by thin layer

chromatography using isopropanol-water developer.   The mid-section of

corresponding peaks for a series of runs were combined and freeze dried.

The resultant material was subjected to analysis by ultraviolet and infra


red spectroscopy.


Characterization by UV-Spectroscopy

     Ultraviolet absorption spectra of a selection of fractions marked

A - P in Figure 2 were recorded on a Gary registering spectrophotometer


in neutral and alkaline solution.  The overall  shape of the spectra

obtained is well known to lignin chemists and therefore only the wave-


lengths of the absorption maxima and minima are shown in Table I.,


     As expected, all fractions A - P show in neutral solution an absorp-


tion maximum near 280 nm.  A closer examination reveals, however, that


fractions A - C exhibit the maximum at 281 nm whereas the maximum in
                                  13

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40-
            RELATIVE MIGRATION IN TLC
30-
20 -
10-
      COMPONENTS IMMOBILE ON TLC-PLATES
        	 I	   I
   2200
       A
       A
3000
 A
 B
A
c
     4000
A
D
A
E
 5000
A   A
F   6
A
H
 6000
A   A
I   J
A
K
A
L
 7000
A   A
M   N
A
0
A
P
                                                                   EFFLUENT VOLUME, ml
FIGURE 2.
Fractionatfon of  Sulfonates  In  Spent Sulfite  Liquor by Gel  Chromatography  on
Sephadex G-25 In  a  Column  10 feet by 2 Inches ID with Water as Eluant.

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fractions D - K is found at 280 nm and  in fractions L - P at 281-282 nm.


This very small difference in the  location of the absorption maximum can


also be seen in the spectra of the fractions of sulfonated milled-wood

Iignin.


     In neutral solution fractions A, B and C of both spent sulfite liquor

and milled wood Iignin show an absorption minimum at 260-261 nm whereas

fractions D, E and G show a minimum at 258 - 259 nm.  Fraction I  shows a

minimum at 256 -  257 nm.


     In alkaline  solution, fractions A, B and C show a maximum at 282 -

283 nm, fractions D, E and F at 285 - 286 nm.  Fractions G - K show maxima

in the region 287 - 293 nm with the maximum shifting towards longer wave-

lengths with increasing effluent volume (and probably decreasing molecular

weights).  Fractions L - P show the absorption maximum at 298 - 299 nm.
                        s
     A division of the fractions of Figure 2 into the four groups I  - IV

can be done on basis of the shift of the absorption maximum near 280 nm

on alkalizing the solution as Can be seen from Figure 3.

     Fi.gure 3 shows that fractions A - C of the spent sulfite liquor

showed a very small red-shift of only  I - 2 nm.  Fractions D - F showed a

red-shift of 5 -  6 nm, fractions G - K showed a red-shift of 8 - 13 nm and


fractions L - P a shift of 16 - 17 nm.


Characterization  by Thin Layer Chromatography

     About every  third 10 ml fraction of Figure 2 was further studied fay


means of thin  layer chromatography (TLC) on analytical silica gel G


("Merck") plates  using 4:1 isopropanol-water as eluent.  The spots were


visualized by  illuminating with ultraviolet  light.
                                  15

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                             TABLE I




           CHARACTERISTICS OF ULTRAVIOLET ABSORPTION

Fraction

A
B
C
D
E
F
G
H
1
J
K
L
M
N
0
P
SPECTRA OF FRACTI
Neutral
Maximum
281
281
281
280
280
280
280
280
280
280
280
281
282
282
282
282
ONS A - P IN
So 1 ut i on
Minimum
261
261
260
259
258
258
258
258
257
256
256
261
262
262
262
260
FIGURE 2
Alkal ine Solution
Maximum
282
282
282
286
286
286
288
290
291
293
293
298
299
299
299
298
     These studies showed that the fractions up to an effluent volume of



3,200 ml contained only solutes immobile on the TLC-plates.  The fractions



in the range 3,200 - 4,100 ml contained immobile as well as mobile compon-



ents.  In the fraction range 4,100 - 7,600 ml the fractions contained only



mobile components.



     Each fraction containing mobile components formed two or three spots



on the TLC-plates.  The location of these spots is indicated in Figure 2.



A comparison with Figure 3 shows that the immobile solutes are to be found



almost completely in fraction group I  that contains only small amounts of




                                16

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mobile solutes.  The mobile solutes are mainly to be found in fraction

groups II -  IV.
RED-SHIFT, nm
20
15


10
5
o
I





B C / j
f\ r^ ^^ i
m n* m m
i F4 ^^
I




G
0 E FJ
tf-Y
/
•MB
I
m

J K/
\/^
X^
^
	 SPENT SULFI'
	 SULFONATED
1 1
12
L M N 0
V




TE LIQUOR
MWL
1 1
2200 3000 4000 5000 6000 7000 8000
                                            EFFLUENT VOLUME, ml
    FIGURE  3.
    Shift of the Wavelength  of the  Absorption Maximum Near 280 nm
    on Alkalizing  Fractions  of the  Spent Sulfite  Liquor and of
    the Sulfonated Milled Wood Lignin  Shown  in  Fig. 2.
Conclusions

     From the presented  results,  it can be concluded that there are dis-

tinct differences between high- and  low-, as well as between  low- and low

molecular wight  lignin sulfonates.  These differences are revealed by

gel perme/atton as well as thin  layer chromatography and UV-spectroscopy.

Classification into four different groups (I-IV,) seemed to be approximate.


                                 17

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A substantial red-shift was evidenced upon alkallnation for the lowest



molecular weight lignin sulfonates, which indicates the presence of some



unique functional groups, probably in the side chains of the Cg-units of



the sulfonates.



     An examination of various fractions by TLC revealed that the sulfon-



ates could be divided into those immobile on TLC plates and those mobi[e.



The immobile sulfonic acids formed brown solutions.
                                18

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                             SECTION VI
           PREPARATION OF CERTAIN LOMOLS-LIKE MONOMERS  AND
      DIMERS  AND CHARACTERIZATION BY NMR AND MASS SPECTROGRAPHY

 Introduction
      Preliminary investigation of the fractions secured  from the Sephadex
 separations, as descrfbed in Section V  of this report,  indicated the need
 for application of the more refined analytical methods that are nowadays
 commonly used throughout organic chemistry.  Whereas,  NMR- and Mass-
 spectroscopy had been successfully applied to study  lignin and  Itgnin-
 like derivatives (8 - 12), these common methods could  not hitherto be
 used for Iignosulfonates.
      However, to apply these procedures, it was necessary to secure infor-
 mation concerning the spectra or patterns associated with particular
 groupings expected to be present in the LOMOL type materials.   It there-
 upon became  necessary to assemble and/or synthesize  certain LOMOLS like
 monomers and dimers in order to permit  the spectroscopy  to be carried out
 in consideration of the special chemical groupings of  interest.
      In contrast to other organic natural compounds, the analytical basis
 for the characterization of lignin sulfonates remained widely restricted
 because of the polyelectrolytic and polydisperse nature  of the material.
The  full elucidation of the  side chain  structures  and types of linkages
has  not been  achieved,  in  part  because  available analytical  methods have
not  provided  sufficient  information.  Due to the insolubility of lignin
sulfonates in organic solvents  and their thermal instability,  however,
methods such  as NMR- and  mass spectroscopy, extensively  used In structural
studies of organic natural compounds, could not be applied.  Our studies,

                                 19

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 therefore, were directed to establish modification procedures which



 allow the conversion of lignin sulfonate fractions into derivatives with



 the desired physical and structural properties by covering the polar



 groups such as hydroxyl- and sulfonic acid groups without evoking



 changes of the original side chain structures.



     Another requirement of the transformation procedures to be applied



 is their applicability to all the various  lignin structures over the



 entire range of molecular weights.  To cover both the phenolic- and the



 alcoholIc  hydroxyl groups as well, we applied the acetylation by pyridine/



 acetanhydride.



     To cover the sulfonic acid groups, the conversion to derivatives such



 as acid chlorides, acid amides and esters was considered (13).    Pre-



 vious attempts to characterize acetylated monomeric IignIn-type sulfochlor-



 ides by mass spectroscopy, however, gave unsatisfactory results (14).  As



 a consequence, we explored the possiblility of establishing a suitable



 method for esterifying the rather labile and reactive sulfonic acid groups



 dominant Iy located in the  a-posit ion (benzyl-sulfonic acids) of lignin



 side chains.



 Synthes i s



     A variety of lignin related model compounds featuring pertinent side



 chain structures and type of linkages were synthesized and sulfonated.



 By following the briefly outlined transformation procedure (Figure 4)  the



 corresponding acetylated methyl sulfonates were formed (15, 16).  The



obtained derivatives were soluble in organic solvents and purified fay



 recrystalIization and exhibited the physical properties required for NMR-



and mass spectroscopic analysis.




                                 20

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   I     6   ©

   CHS03Me
   OH
       OCH
        e  e
   CHS03Ag
   OCOCH
       OCH3
   CHS03CH3
        OCH3

   OCOCH3
*}    e  ©
CHS03Me
    OCH-

OCOCH-, '
                      R
   i
     ©. .e
CHSOgH
    OCH3

 OCOCH3
FIGURE 4.


REACTION SCHEME FOR THE TRANSFORMATION PROCEDURE.

-------
     As shown in Figure 4, sodium sulfonates were acetylated by pyridine/



acetanhydride.  The aqueous solution of the free acids prepared by cation



exchange was neutralized by silver oxide.  Reaction with methyl iodide



yielded the corresponding acetylated methyl sulfonates.



     The 18 model compounds that were synthesized in the course of this



study are represented by four types of monomeric and dimeric lignin build-



ing units, as shown in Figure 5.



     Type 2 represents monomers of the guaiacyl- and veratryl- series with



saturated and unsaturated sidechains.  It  includes all three possible reac-



tion products of the coniferylalcohol-type structure.  Among them is one



a - and one y~ sulfonic acid, each with a double bond, and one  a- y ~



disulfonic acid.  All of the three types of sulfonic acids have been iso-



lated earlier from sulfite liquors (I, 2),



     The second type of  linkage is expected to represent the major portion



of  linkages present in lignin.   The most  important one of them is the con-



figuration which carries an aryl-ether structure in  $-position and a



hydroxyl group in Y-position.  Other substituents to consider at the S-



carbon atom are a hydroxyIgroup or a carbon-to-carbon  linked second Cq



unit as it is formed from the coumaran structures in lignin in a neutral



sulfite cook.  A compound with  the latter configuration was supplied to us



by Dr. Josef Gierer from Sweden.  The fourth type of linkage represents the



d i phenyI structure.



NMR-Spectroscopy



     Extensive studies performed earlier  in this laboratory C8, 9)



revealed that NMR-spectroscopy  represents a valuable-method to study the



overall  structure of different lignin preparations.  However, the NMR





                                 22

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        TYPE  I
         CH2OR(
         irH
         CH
             OCH:
         OR2
        ir BE
      H or CH3
R,= H or  BENZOYL
                             HS03CH3     R=ALKYL
                                 OCH,
                     SULFONATION
                                            H
                                                 R- H
                                                    H   R -H
                                           CH2SO*
                                        
-------
spectra of sulfonated  lignin models and  lignin sulfonate fractions did not

yield satisfactory information mainly due to the  lack of solubility  in

organic solvents and due to the presence of strong .polar groups.  By pre-

paring the acetylated methyl sulfonates well resolved spectra could be

obtained.  Figure 6 shows a typical example of- the IMMR-spectrum of a sulfon-

ated dimer.  Following the  increasing magnetic field from the left to the

right side of the Figure, the aromatic protons are exhibited first, followed

by the protons of the benzyl ic carbon atoms which carry ace.toxy-groups.

Methine- and methylene-protons of the sidechains of Cg units generally

give rise to signals between the region of the aromatic protons and the

protons of the methoxy(groups, with which they interfere.

     Protons of acetyI groups are much less effected by other signals than

are methoxy-protons.  Aromatic acetoxy-protons usually appear at lower

field, well separated from their aliphatic counterparts; however, biphenyl

and phenyl-alkyl linkages ortho to acetoxy-groups cause a significant

shift of the acetyI-protons to higher field, where they interfere with the

aliphatic acetyI-groups.

     The average chemical shifts for acetylated and esterified lignin

sulfonates in NMR-spectroscopy are listed in Table 2.  This Table provides

the possibility of estimating rather precisely the relative distribution

of protons in LOMOLS-like materials and therefore, allows a nearly com-

plete functional group analysis of the acetylated methyl sulfonates.

Mass Spectroscopy

     Systematical mass spectroscopic studies of lignin related models had

not been reported before we started with our irwestigat ions. However,
                                                V
several  papers dealing with the mass spectroscopic fragmentations patterns
                                 24

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                               TABLE 2
            CHEMICAL SHIFTS FOR ACETYLATED AND ESTERIFIED
         LIGNIN SULFONATES IN NMR SPECTROSCOPY  ( T-VALUES)
Reg i on
Location of Signals
Type of Protons
2
3, 4
5
6
••" ." | 1 " IP"-"'- • 	 |n • !"— • •!-—-•
7
8
2.00 - 3.72
3.72 - 4.82
4,82 - 7.50
7,50 - 7.81
i
7.81 - 8.42
8.42 - 9.62
aromatic H, except in sulfo-
nated coumarans,
o-vinyl -protons
aromatic H in sulfonated
coumarans,
3-vinyl -protons
partial ly C.H
CaH-0-Ac ( fion-s u 1 f onated )
CciH-0-Ar (in coumarans)
Methoxy 1 -p rotons ,
sidechain protons other than
in 3, 4 and 8
Aromatic acetyl -protons,
except those ortho to bi-
phenyl-l inkages
..•I.... i...im.»—.T.i 	 — i,.— ..••^•..i. 	 .,n. 	 .in. 	 ,„..„..—,! 	 	 i i n, 	 .•.••^••Pllllili -i in niii ii •! 11..
A 1 i phat i c acety 1 -protons ,
aromatic acetyl -pro tons ortho
to biphenyl-l inkages
highly shielded, mostly side-
chain-protons
                                  25

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       CO
    0%0 CH-0
'H3<
OCH,
                           CMj|OCOCH3
                                                                                      IMS
2.0        3-0         4.Q        5.0
                                      PPM(r)  '
                                                        7.Q        8.0
                                                                 9-0
10
                 FIGURE  6,
                 PfR-SPECTRUM OF A  TYPICAL LOMOLS-LIKE DIMER.

-------
                                  313
   23 ft.
          252
           h...
                       282
                              3OO
 331


1
372
 ii
594
 i
426

 i
                                      MASS  UNITS
                                                                                 ;CH,
                                                                                   OCHj
                                                                                468 (43%)
FIGURE  7.

MASS-SPECTRUM AND FRAGMENTATION PATTERN OF A TYPICAL LOMOLS-LIKE DIMER..

-------
of rather simple models have been reported (II, 12).  Earlier attempts,



however, to obtain useful data from sulfonated lignin models failed



because of either the poor volatility or instabflfty at elevated tempera-



tures.



     The acetylated methyl sulfonates, however, were found to be volatile



and thermally stable enough to yield reasonable spectra.  Although the



base peaks were quite low Tn several cases, exact molecular weights could



be obtained.  In our studies we recorded the spectra of monomeric and



dimeric models.  A characteristic fragmentatton pattern is shown in Figure 7.



Conclusions



     Sulfonatton studies with Itgnin model  substances provided us with some



information about the principal  reaction pathway of the chemical  reaction



that occurs in the sulffte pulping of wood.



     The highly desirable use of modern analytical tools in organic chem-



istry was made possible through a new transformation procedure for sulfona-



ted lignin-Mke materials, which involved acetylation and esterif i cat ion.



This method allowed transformation of the  lignin sulfonates into deriva-



tives without electrolytic behavior.



     With the aid of such acetylated and esterified lignin sulfonate model



compounds the analytical basis for NMR and Mass spectroscopy studies with



lignin sulfonates from spent sulfite liquor was created.
                                 28

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                            SECTION VII
        PREPARATION OF ACETYL LIGNIN SULFONATE METHYLESTER
        (ALSME) AND THEIR SPECTROSCOPIC CHARACTERIZATIONS

Introduction
     The polyelectrolytic nature of lignin sulfonates has been the main
obstacle to their fracttonation and characterization in the past.  To
overcome the analytical difficulties which were caused by this property,
we investigated the transformation of these compounds into derivatives
with properties required for structural studies, especially for NMR- and
mass spectroscopy.  The synthetic basis for this transformation and the
analytical basts for the characterization of such derivatives had been
established before, using monomeric and dimeric lignin building units as
models.  (See Section VI for details.)  The transformation aimed at the
elimination of the polyelectric behavior by covering the polar groups:
hydroxyl groups by acetylation, and sulfonic acid groups by esterification.
Such acetylated JJgnin sulfonate methyl aster (hereafter called "ALSME")
would be sufficiently soluble in organic solvents to allow the applica-
tion of the more powerful analytical tools, such as NMR- and mass spec-
troscopy.
Transformedion Procedure
     The procedure used for the transformation of the LOMOLS-ltke monomers
and dimers was applied to lignin sulfonates with varying molecular weights
in a slightly modified form.  The so-obtained ALSME products were found
to be soluble in chloroform, the solvent commonly used for recording
NMR-spectra.
                                 29

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 2.0
3.0
4.0
5.0         6.0        7.0
       PPM (r)
8.0
9.0
FIGURE 8.
NMR SPECTRA OF  ALSME DERIVATIVES, PREPARED FROM  VARIOUS  FRACTIONS FROM SEPHADEX
G-25 SEPARATIONS.                    39

-------
     The transformation to ALSME  derivatives  resulted also  in a purifica-



tion of the original  lignin sulfonate  fractions obtained from the previ-



ously described Sephadex  fractionation (See Section V), which were contam-



inated with carbohydrate  degradation products to a certain degree.



     NMR Spectroscopy;  The spectra were  recorded using the same conditions



as descrtbed for the  LOMOLS-like  monomers and dimers (See Section VI).



The entire frequency  range of each spectrum was divided into several areas



that were classifted  on the basis of the model studies.  As shown in



Figure 8, the  LOMOLS  exhibited well resolved spectra in a wide range of



the investigated fractions.



     Chromatog raphy;  The separation of ALSME fractions using the cross-



linked Sephadex gel LH-20 and methanol  as eluant resulted in the fraction-



ation of low molecular weight mixtures into simple mixtures and into a



single, crystalline compound  (m.  p. 200-201 C).



     Analytical thin-layer chromatographic studies and fractionations by



Sephadex LH-20 gel chromatography in analytical scale indicate that the



fractions are composed of more or less complex mixtures of  low molecular



weight compounds ranging  from monomers to dimers and trimers and some




higher mers (See Figure 9).



Characterization by NMR Spectroscopy



     In general, the  spectra of all thirteen fractions studied allowed a



good correlation between  the protons of various functional groups.  Special



emphasis was placed upon  the content of aliphatic and phenolic hydroxyl



groups.  The correlation  between  these two hydroxyl fractions led finally



to a classification of the fractions in four different groups.  Constant



ratios—aliphatic to  phenolic hydroxyls—ranging from 0.5 Cfractlons  I to 7






                                  31

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ABSORBANCE
   A280nm
                                         PEAK A
                                EFFLUENT VOLUME

 FIGURE 9.
 SEPHADEX LH-20 SEPARATIONS OF SOME ALSME FRACTIONS IN METHANQL.
                          32

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CFractions  1-13 correspond with  fractions A-P  in Section V  in reverse
order]),  1.0 (fraction 8, 9), and  1.4  Cfractions 10,  II) were observed
(see Figure  10).   In the next higher fractions we found a continuous
increase of this ratio.
     A similar classification in a  somewhat  different fashion could be
made on the basis  of the UV-spectra (See Section V).  These findings were
finally supported  by the remaining  NMR signals which could be assigned
to protons of deffned side chain structures.  The main component in the
group consisting of the  lowest molecular fractions, fractions 1-5, (See
Section V and Figure 2) was  indicated  but not established to be a dimer
of a  lignan-type structure.
     The  next higher fractions  (6,  7)  represent mixtures of different
structural makeup.
     The  lignan-like compound was  finally isolated over Sephadex LH-20
and purified by recrystalIization.   Its melting point, its NMR-spectrum,
and its mass spectrum  indicate that it is of dimeric structure.  Its abso-
 lute configuration so  far  has not  yet  been established.
      In fractions  8, 9 a vinyl sulfonic acid type side chain structure
could be  detected.
     The  overlapping and broadening of the signals found in the spectra
of the  next  higher fractions does  not  allow  further studies on side chain
structures.  However, we did find  indications that condensation presumably
 in 5-position  increases with the molecular weight.  The first  indication
of condensation in this way  is observed in fraction 9 and seems to
 increase  steadily  in the higher  fractions.   It  remains unknown whether
this condensation  is induced secondarily by  the sulfonation reaction, or
whether it  is present  in the original  lignin in the plant.

                                 33

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CO
Q-
O
   0.5
§  °-
 o
\
              \
     \
                                                          OOL  A-	&	
                                             A	A	-A
                                                       — o
                                                                  ,o-~-o'
             •       I      »      i       I       •      |      %       T
            13     12     11      10      9      8      7      6      5
                                    Fraction Number

         FIGURE 10.
         CORRELATION  BETWEEN PHENOLIC HYDROXYL GROUPS AND AROMATIC PROTONS IN
         FRACTIONS FROM SEPHADEX SEPARATIONS.
                                      34

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Characterization by  IR Spectroscopy




     The  IR spectra of ALSME  derivatives are all very similar and without



characteristic features.  The sulfonate group exhibits a strong band



around  II and  12 , which  is "rather untypical.  The acetyl groups raise



strong ester bands in the neighborhood of  5.8 , thus covering eventually



present carbonyl groups.  These carbonyl groups, however, can be detected



in the  IR spectra of the  untransformed fractions.  It could be shown that



the carbonyl content of the LOMOLS is usually very low.  Some fractions,



however,  in the very  low  molecular weight  range exhibit a distinct con-



centration of CO-bands (See Figure  II).  No attempts were made to investi-



gate the nature of the carbonyl groups, which might also be due to incomplete



separation from carbohydrate  degradation products.



Conclusions



     The polyelectrolytic and polydisperse nature of the LOMOLS could be



eliminated by a relatively simple transformation procedure that covered



the highly polar groups.  We  assume  that this transformation did not induce



any particular changes in the original structures of the LOMOLS.  The so-



obtained ALSME derivatives were found to be soluble in organic solvents,



which aided considerably  their analysis.



     The most valuable analytical method proved to be NMR spectroscopy.  It



could be demonstrated that the NMR spectra of low molecular ALSME deriva-



tives provide  information on  structures which could not be obtained from



other analytical and spectroscopic methods so far.  Indications on typical



side chain structures and types of condensations can be as well derived



as an almost complete functional group analysis,   It could be demonstrated



that the content of aliphatic and phenolic hydroxyl groups can be estimated
                                  35

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                                                Fraction Number
1600   cm
     1800
FIGURE II.
THE CARBCNYL REGION IN IR - SPECTRA OF FRACTIONS FROM  SEPHADEX SEPARATIONS.

-------
in higher molecular  Ifgnin sulfonate  fractions with an accuracy never
accomplTshed before, even by applying rather elaborate analytical tech-
niques.  The NMR spectroscopic technique  represents the only method known
in llgnln chemistry  so  far which allows us to distinguish between these
two types of hydroxyl groups.
     The correlatton between these  two hydroxyl functions led to a classi-
fication of the fractions  in four different groups.  A similar classifica-
tion in a somewhat different fashion  could be made on the basis of the UV
spectra (see Section V).
     Significant changes  in the structural makeup of the low molecular
weight fractions of  the ALSME were  found.  The predominant component in
the first five  fractions exhibits features characteristic for Iignan-type
structures.  Since unextracted Western Hemlock was used for acid bisulfite
                i
pulping the presence of sulfonated  Iignans would not be surprising. Another
explanation, however, seems to be that this dimer  Is formed by a vinyl-
type condensation of two monomers with conjugated double bonds.  Based on
the assumption  that  coniferyl alcohol is  the only precursor, our findings
can be interpreted as depicted  in the reaction scheme in Figure 12,
     Homocondensation of coniferyl  alcohol forms a  lignan*-type dimer with
the structure that represents the main compound  in fractions  1-5.  Further
condensation between the dimer and  coniferyl alcohol and subsequent allyl
type rearrangement of the  coniferyl  alcohol side chain to a vinyl-type
structure  leads to a product with the spectral features observed in frac-
tions 8 and 9.
     Although there  Is  considerable doubt about the validity of the pro-
posed condensation mechanism, this  hypothesis could very^welI explain some
of the observed discrepancies of  LOMOLS.   Further experiments are  necess-
ary to support  this  hypothesis.
                                 37

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           DIMER EXPLANATION  I
                                                           GH.oH
        Fraction 1-5
               (6 7)

                  DIMER EXPLANATION  2
     OH-       DH
Fraction 8,9
FIGURE 12.

HYPOTHETICAL  DIMER FORMATION  MECHANISM.
                        38

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                            SECTION  VIM
           STRUCTURAL  STUDIES  OF  ACETYL  LIGNIN SULFONATE
       METHYL ESTERS  (ALSME) DERIVED  FROM  MILLED WOOD  LIGNIN

 Introduction
     The separation of lignin  sulfonates from spent  liquors of sulflte
 pulping processes  has  been  studied  extensively in this  laboratory during
 previous years  (3, 4,  17).  The major obstacle has been repeatedly shown
 to be a complete separation of aromatic  substances derived from sulfona-
 tion and dissolution of  Ifgnin in wood,  from the sugars which are formed
 at the same ttme by acid  hydrolysis of carbohydrates (.17).  Some sort of
 separation based on the  ionic  strength of  the compounds to be separated
 (ion exclusion  separation)  seems  to provide the best method so far (3, 17,
                                               ^
 18); however, neither  the lignin  nor  the carbohydrate part can be obtained
 absolutely pure and free  of contaminations by the ion exclusion method.
 Ten-20$ contaminations of the  respective counterpart seems to be a rea-
 sonable goal to be achieved by ion  exclusion chromatography.  Complete
 separation of aromatic- and sugar-components and complete recovery of both
 parts from spent sulfite  liquor (SSL), both of which are requirements for
 a scientific investigation  of  structural phenomena, had been out of reach
 with the methods available  so  far.
     To get a better founded and  more complete approach to our research
objectives, it  appeared necessary to  study the sulfonation reaction (as
 used in the acid sulfite  pulping  process of wood) with a variety of models
 for lignin in wood (See Section VI).
    - We started this approach  with  the preparation of various LOMOLS-like
monomers and dimers.   Their sulfonation  and transformation to acetylated

                                  39

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lignin sulfonate methyl ester (ALSME) derivatives taught us first the
principal sulfonation pathway of compounds with different functional
groups and active sites, and second, the potential use of highpowered
analytical tools such as NMR- and mass-spectroscopy.
      The application of these synthetic and analytical approaches to
various LOMOLS-fractions secured from SSL by Sephadex G-25 separations
has been discussed in Section VII in detail.
      Milled wood lignin (MWL) (19-21) is the genuine plant material,
isolated from wood by a special  mild procedure (ball milling and dioxane
extraction).   It is free of carbohydrates and extractives, yet widely
considered to be unchanged lignin.  It is a "model" by definition, since
it comprises only about 25-50$ of the total lignin-part in wood, and
since it has another physical form and environmeht than in wood.  The
lack of  incrustation in a cell wall  or between cell walls (middle
lamella) affects the melting and softening behavior of the material
and lets questions of accessibility appear irrelevant.  The different
solubility of the isolated lignin allows most reactions to proceed as
homdgeneous reactions (22).
      The advantage of working with MWL as a model for lignin (the DP of
MWL is reported to be around 60, molecular weight about 11,000 is based
on the fact that MWL is a homogeneous material, free of carbohydrates and
extractives.  An empirical formula,  based on the assumption of Cg- monomertc
units, can be designed for the material and a balance of certain functional
groups can be established.  That means that the starting material of the
reaction (e.g., sulfonation) can be well defined.  Changes that occur
during the reaction can be well  detected and controlled.

                                 40

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      In sulfonation  reaction  in  particular, the  sulfonates do not have to
be separated  from any  carbohydrates.   Control over all the organic material
is guaranteed.
Experimental
      Milled wood  Itgntn,  isolated  from Western Hemlock, was sulfonated
under mild conditions  CIOO°C, pH 1,5,  24  h).  The reaction product was
freed from excess S02  and  sulfate  ions.   The calcium salts of the lignin
sulfonates .-were fractionated over  Sephadex G-25  in water.  Twelve fractions
were  collected and separately transformed to ALSMES.
      These ALSMES were purified  and  investigated by NMR spectroscopy and
elemental analysts.  The empirical formulae were calculated for each of
the  12 fractions.
ResuIts and Discuss ion
      Representativeness of Mi I led  Wood Lignin;  The elution diagram of
Ca-LS from sulfonated  MWL  is compared  with that of Ca-LS from a spent
sulfite  liquor in Figure  13.
      Differences between both elution  diagrams can be visualized in the
very  high- and the very low molecular  weight region.  Both differences
signify the peculiarity of the MWL preparation.  The highest molecular
weight portion is absent since  it  cannot  be extracted with neutral  sol-
vents from the fiber.   The lowest  molecular weight material and the
extractives are missing as well, due to their removal prior to the isola-
tion  of the wood lignin.
Structu raI  Phenomena
      By Elemental Composition;   The empirical formulae for the Cg-basis
were  calculated for all of the twelve  fractions.  They are compiled in

                                 41

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            RELATIVE MIGRATION IN TLC
            1.0
       COMPONENTS IMMOBILE ON TLC*PLATES
   2200
  i
A280nm
3000
4000
5000
6000
7000
  2000
                                              6000   EFFLUENT VOLUME, ml
               FIGURE  13.

               ELUTION   DIAGRAMS  OF   CALCIUM  LIGNIN  SULFONATES
               Above:  Secured from Spent Sulfite  Liquor
               Below:  Prepared from  Milled Wood Lignin
               *TLC - Thin Layer Chromatography
                                     42

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                                                    TABLE 3

                                EMPIRICAL  FORMULAE OF ALSME DERIVATIVES OF MWL
Fraction
Number C
Original
Sample • 9.00
1 9.00
2 9.00
3 9.00
4 9.00
5 9.00
6 9.00
7 9.00
8 9.00
9 9.00
10 9.00
II 9.00
12 9.00
H
8.40
7.80
7.28
8.59
7.09
7.23
7.12
7.44
7.22
7.26
7.57
7.50
7.26
0*
2.98
3.09
2.73
3.15
2.77
2.77
2.60
2.73
2.71
2.56
2.61
2.73
2.89
OCH7;
0.94
0.45
0.58
0.1-5**
0.65
0.68
0.67
0.73
0.66
0.76
0.69
0.71
0.70
S07OCH,
—
0.35
0.39
0.40
0.46
0.46
0.51
0.49
0.48
0.48
0.45
0.36
0.33
CH3-CO
phenol ic
—
0.81
0.63
0.50
0.49
0.42
0.45
0.44
0.41
0.37-
0.33
0.29
0.34
CH3-CO
al iphat.
—
0.75
0.73
0.80
0.80
0.70
0.78
0.81
0.82
0.76
0.80
0.60
0.81
Mol. W._
Ave.for C^ Z H
193.4
279.5
272.9
265.9
279.5
272.5
279.2
282.4
278.0
274.2
270.9
254.3
264.4
11.2
14.9
14.3
14.1
14.3
14.0
14.3
14.9
14.3
14.4
14.4
13.4
13.8
Oxyg.
Bal .
3.919
3.889
3.696
3.703
3.889
3.906
3.779
3.950
3.854
3.798
3.750
3.802
3.920
 * Oxygen-determination by difference.
** After repeating the analysis for F_,  the OCHL-content  is about 0.60 per Cg.

-------
Table 3.  The phenolic- and aliphatic- acetyl groups were determined by



NMR spectroscopy.  The most essential functional groups were plotted in



diagrams CFigure 14).  It is demonstrated that the content of phenolic



hydroxyl groups increases from high to low mol. w. material.  The increase



seems to be steady in the high molecular weight range, exponential in the



low molecular weight range.  The content of phenolic OH groups in MWL has



been reported to be about 0.3 per Cg unit.  Apparently phenolic hydroxyls



are generated by the splitting of mainly a-arylether bonds CFigure 15);



however, the sharp increase of phenolic OH-groups in the LMWLS region



(fraction 6-1) cannot be explained only by this type of ether splitting,



but must involve some other reactions.



     The diagram of ether-OCH,-groups per C_ unit signifies this other



mode of phenolic OH group formation.  The content of methoxyl groups remains



constant in the high molecular weight LS region, but drops off drastically



in the LMWLS region.  This means that methoxyl  groups are cleaved by the



sulfonation reaction under the formation of phenolic hydroxyl groups in



3-position (23).  Sulfonate groups hav§ been reported to increase steadily



for high molecular weight LS (24).  This could  not be verified.  In con-



trast, the S-content of the various fractions as well as the content of



S03-groups per Cg unit exhibits a be I I-shaped curve with the culmination



point in fraction 6.  Forss derived a lignin formulation from the fact



that the S-content for high molecular weight lignin sulfonates is steadily



increasing (25).  He calculated that units of 10-18 Cg units share each



eight S03 groups.  A similar calculation resulted in 15-20 CQ units for




every eight sulfonate groups in the same region of the elution diagram of



MWL.




                                  44

-------
                  FIGURE  14.      ELEMENTAL AND FUNCTIONAL GROUP COMPOSITION OF MWL - ALSME.
    t.o  ,
  cr>
   0.8
 _ 0.6  •
 K
 O
PHENOLIC  OH
   (NMR)
 §
   0.4
   0.2
            10    8     6   4     2
                         Fraction Number
                                                       OS
1.0. -


0.8 •

0.6
                                          sf
                                             o.2
            so
                                                      10   8    64    2
                                                                   Fraction Number
                                                                                                              in
    0.8
    0.6
I   0.44
   0.2
                      >tarting Material
                                                         1.0
  OCH
            10    8    6    42
                         Fraction Number
                                                       CO
                       By Theory
                       Of Forss
                                                                  8 SO,
                                                      10   8
                   642
                     Fraction Number

-------
H2CY
H2C3
H Ca-0
                           Scheme 1
                           H2C-
                           H2f
                           H C®
                                                   0—
                                 OCH3
                                                                HO
                                                                    OCH3
        6
        5
CHOH
     CH3
        >,HS03-
-CH2OH?

Scheme 2
                                   OH
                                                    0-
OCH3
                  0
                  Scheme 3
                                             Major
                                               Minor
                                                   CH30
                                                          0<
                                        OCH3
                                                           CHS03-
                                 FIGURE 15
                                  46
                                                               OCH3

-------
     By Oxygen Function;   It  is well known that condensation reactions


compete with sulfonation reactions  (Scheme 3, Figure  15) C26).  In the


sulfonation reaction, a hydroxyl group  is substituted by a sulfonate group


whereas condensation means elimination  of a molecule of water.


     A balance of oxygen atoms per  CQ unit for all fractions is able to
                 i

give hints for the  location of condensed LS in the Sephadex diagram.  For


this reason all oxygen atoms  per Cg unit are added up (Scheme 4, Figure 16).
                   ' \j

If a sulfonate group has substituted an OH-group, it  is counted as I oxygen,
                      : O
The oxygens attached to the sulfur  atom are not counted.
     The MWL starting material had 3.92 0/Cg  (see Table 3).  The deviation

from this value for each of the  12 fractions  has been calculated and plot-

ted in Figure  17.  All oxygen values  lower than 3.92 0/Cq  indicate

condensation (or other  loss of water).

     The shape of the curve in Figure  17  indicates that condensed LS are

"located" in the high- as well as the  low molecular weight material, whereas

the material right between both  areas  (fraction 6) indicates no condensation

at all.  Interestingly, this fraction  is also the fraction with the highest

SO, content of all.  Condensed LS are  found mainly in fractions 2 and 3 and

9-11.  The degree of deviation of oxygens from the starting material

(0 - 0.25 0/Cg) can be considered to be an expression of the degree of con-


densation.  Thus, fractions 2 and 3 contain LS, where every 4. or 5. aromatic


ring is condensed onto the side  chain  of another unit (probably mainly in

6-position).  Both fractions comprise  about 10$ of the total lignin sul-


fonates.

     By NMR-Spectroscopy;  This  method has been shown to be a powerful


instrument in the analysis of lignin model compounds as we I I as  lignins
                                  47

-------
 H2COH
 H C-
 H COH
         OCHa
   0—
4 0/C9
               Scheme 4
H2C OH
                                      CH=CH2
                                      CHS03
                                               OCH3
                                        OH
                                        CH=CH-CH2S03-
                                               OCH3
                 Scheme 5
   OH
                 Scheme 6

                FIGURE 16

                      48

-------
           OXYGEN DEVIATION FROM 0.56 PER C
             (theoretically sulfonatable
              groups)
                                                —-  0.56  =
                      65432
                       Fraction Number
FIGURE  11

OXYGEN FUNCTION IN ALSJ4E; DERIVATIVES CF MWL.
                     49

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Csee Section VI  and VII).  Side chain configurations as wall as ring



substituents can be es-tfmated or determined with high accuracy.



     The application of NMR spectroscopy to the 12 fractions of the MWL



fractionation revealed some more specific features of the structure of LS.



Fractions 2 and 3 proved to contain some sulfonation products of coniferyl-




alcohol (Scheme 5, Figure 16).



     These compounds, however, were very probably not present as monomers



but rather attached to oligomeric fragments as indicated by thin layer and



Sephadex LH-20 chromatography.  The C-6 atom of the aromatic ring is the



position of intermolecular linkage.  Since both vinyl-compounds have only



three oxygen functions per Cg, not all  oxygen deviation shown in Figure 17



can be due to condensation;  some of it must be due to these unique side



chain configurations.



     The NMR spectra of fractions 8 upward show signs of increasing inten-



sity of carbon-carbon condensation in position 5 of the aromatic ring.



Condensation has been indicated also by the oxygen deviation of these



fractions, shown in Figure 17.



Cone I us ions




     Sephadex chromatography, elemental analysis and NMR spectroscopy



helped to elucidate some of  the structure of LS.



     It was shown that phenolic hydroxyI-groups are formed through demeth-



ylation of aromatic methoxyI-groups (Scheme 2, Figure 15).  In the lowest



molecular fraction of the lignin sulfonates from MWL, about every second



Cg unit was demethylated. The para positions of these newly formed



phenolic hydroxyI groups (position 6 of the Cg unit) are the most activated



nucleophilfc sites of the entire lignin (Scheme 6, Figure 16).





                                 50

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     These nucleophiles are, therefore, the most probable ones to undergo



condensation with carbon turn  ions  (Scheme 3, Figure  15), thus contributing



to the  lowering of the methoxyl content of the  llgnin sulfonates.  The



sulfur content of IS- is represented by a bell-shaped curve, wtth the cul-



mination point at the border between high- and  low molecular weight LS.



In LMWLS the sulfonation products of coniferyl  alcohol have been found,



probably attached to ollgomeric fragments of  lignin through the 6-posltion



of the aromatic ring.



Summary



     Milled wood lignin CMWL) of Western Hemlock has been mildly sulfonated



and analyzed by Sephadex G-25 chromatography, NMR spectroscopy and elemental



analysis.  A comparison of SSL from pulping of  wood chips was found to be



In good agreement with the sulfonated MWL in all essential parts, except



for the very low- and very high molecular weight range.  Results from the



MWL are, therefore, believed to be representative also for the lignin from



wood.



     An exact division between low- and high molecular weight LS Is pro-



posed by employing Sephadex chromatography, solubility in ether and ele-



mental analysis.  According to this division, MWL is composed of 30% LMWLS



and 1Q% high molecular weight particles.



     Structural studies revealed the-content of phenolic hydroxyl-,



methoxyl- and sulfonate-groups.  The degree of  condensation was estimated.



Certain unique structural  configurations could  be assigned to some of the



LMWLS.  An explanation for the demethylation observed was proposed,
                                 51

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                            SECTION  IX




                STRUCTURE AND REACTIVITY OF  LOMOLS




Introduction




     The structure of  LS has been elucidated so far nearly exclusively



on the basis of either chemical  reactions of lignin models, or physico-



chemical characterizations of LS by  gel permeation chromatography Csee



Section V, VI).   It has been our objective in this research enterprise



to separate these  isolated LS into a series of fractions each of which



consist mainly of particular mers, such as monomers, dinners, trimers, and



then mixtures of higher mers, and to characterize each mer class by several



methods Csee Section  tV).



     We approached these objectives  by purifying and fractionating LS



from a SSL over Sephadex G-25 Csee Section V).  Characterizations by UV



and I:R preceded the transformation  of the various LS fractions to ALSME



derivatives CSection VII).  The analytical basis for the characterization



of such ALSME derivatives had been created using LOMOLS-like monomers and



dimers as models  CSection VI).  The  use of Milled Wood Ligntn as an "ad-



vanced model" for wood allowed us to make concise statements about the



elemental composition  of lignin before and after sulfonation, and the fate



of most functional groups during this reaction CSection VIII).



     From the literature and from our earlier studies, we knew that LOMOLS



appeared different from the rest of  the LS by a number of characteristics,



as reflected in various chemical and physicochemical methods.  The most



important ones of them shall be  listed in the following.
                                 53

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      Forss and coworkers found that the UV absorption of the LOMOLS suf-
fered a severe red-shift when the solution was alkalized (7).  The UV
spectrum of HIMOLS appeared unaffected by the pH.  This Finnish group
also reported findings which demonstrated a significant difference in
solubility in sodium bisulfite solution of pH 5.5 - 6 between LO and HIMOLS
(6).  Fractionation of LS over ion exchange resin (DQWEX 50W-X2) separates
the LOMOLS from the HIMOLS (see Section V).  This separation can be visu-
alized also by the color:  LOMOLS are yellow, whereas HIMOLS are brown.
Fraetionation on Sephadex G-25 yields an elution diagram similar to that
from Dowex.  Very significant differences bewteen low and high molecular
weight parts of LS can be observed in the elemental  and functional  group
composition, as discussed in earlier sections of this report (Section V,
VI I, and VI I I).
      As to the origin of these differences that are in apparent disagree-
ment with the conventional understanding of lignin,  (particularly concerning
its homogeneity) (see ref. 27-29), Forss and coworkers believe that lignin
is as heterogeneous as the carbohydrate portion in wood (cf. hemi- and
holo-celIulose).  Other theories explain these differences with secondary
condensation of lignin material evoked by acid hydrolysis.
      To find a better understanding of the structure, origin, and reactivity
of LOMOLS we undertook two-fold studies:
      a.  We isolated lignin sulfonates into a series of fractions each of
          which consisted of particular mers, and we characterized each mer
          class by several methods;  and
      b.  We sulfonated the hydrolysis products of the most representative
          dimeric lignin model compound and investigated the reaction
          products.
                                 54

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Exper i mentaI SectIon




     Lfgnin sulfonates  from  a  spent  sulflte  liquor were purified as usual



(cf, Section V) and fractionated  by  ion  exclusion chroma tog raphy.  The LOMOLS



comprising  part was  neutralized, concentrated and freeze dried..  The total



portion was trans-formed to ALSME  derivatives  in accordance with the proced-



ure described  in Section VI.



     About  half of the  ALSME were fractionated over Sephadex LH-20 using



methanol as mobile phase.  The elution diagram exhibited a number of well



separated Individual  peaks,  the corresponding material of which were col-



lected and  recovered  by evaporation  and  drying under vacuum.  The separation



had a very  high degree  of reproducibiIity,  The substances from each indi-



vidual peak area were refractionated under the same conditions as used



before (see Figure 18).  Whereas  some peaks proved the high separation



potential of this method (peak d) other  peaks exhibited elution diagrams



very similar to the total ALSME fraction  (peak c).  Material  from corres-



ponding mer classes (peak areas)  was re-collected and recovered by evapora-



tion and drying.  The oily residues  were  dissolved in a little methanol  and



precipitated from ether 10:1.  The ether  solubles (ES) and the ether insolu-



bles (EIS) were recovered separately.  The samples were analyzed by NMR



spectroscopy and elemental composition.



     The other half of  the ALSME  derivatives was dissolved in chloroform,



and brominated under  very mild conditions (temp, below 5-10 C) until there



was no more discoloration of the  bromine.  Then the material  was recovered



and treated the same  way as  outlined above for unbrominated ALSME,



     Veratryl^-glyceryl-3-arylether was submitted to a mild acid hydrolysis



(ACIDOLYSIS) following  the procedure of Adler et. al. (30, 31) (0.2 N HCI in



dioxane:water 9:1;  reflux for  four hours).  At that time, no more unreacted




                                  55

-------
                                   A 280
ui
o\
                     E. VOL.                     E.VOL.                    E. VOL                        E.VOL.

      FIGURE  18.


      ELUTION DIAGRAM  OF ES  ALSME DERIVATIVES AND THE REFRACT IONAT ION PATTERS OF SOME MER CLASSES.

-------
3-ether was  left,  as  indicated  by  TLC.  Without cooling, excess sodium



bisulfite  in  little water  was added  to  the  solution and reflux continued



for two days.  Afterwards  the solution  was  concentrated under vacuum and



redfssolved  in water.   The aqueous solution was extracted several times



with plenty of chloroform  to remove  the chloroform solubles (unsulfonated



organics).  About  2/3  of the starting material was recovered in the organic



phase.  The  rest  (aqueous  solution)  was concentrated and run over an ion



exchange column  in H-form  to liberate the anions.  The free acids were



freed  from S02,  neutralized, concentrated and  freeze dried to yield mainly



the sodium salts of the sulfonated hydrolysis  products of the B-ether.



The usual  transformation  (cf. Section VI) yielded the ALSME derivative



which  was  divided  into an  ether soluble and an ether insoluble part by



precipitation from ether.   AlI  steps were control led by TLC, Sephadex G-25



and LH-20  chromatography,  IR- and  NMR-spectroscopy, as far as possible.



The elemental composition  of the EIS ALSME  derivative was determined and



its empirical formula  calculated.



Results and Discussion



     The refractionations  were  undertaken with the idea in mind to prove



the potential of  isolating individual compounds from LH-20 separations.



This potential seemed  to be very high,  since the  peaks exhibited were tall



and slender,  indicating excellent  separations  (see Figure 18, 20).  Also



NMR spectroscopy  indicated good separation  of  the  individual fractions.



     However, upon refractionation most mers or mer classes did not exhibit



elution diagrams with  single peaks,  but demonstrated a rather peculiar



instability,  indicated in  the "regeneration" of certain other peaks; as  if



there was  an .equilibrium of the compounds represented by these peaks.  By
                                  57

-------
naming all  peaks according to their retention volume, certain "regenera-



tion pathways" could be established Csee Figure 19).



     The isolation of compound c seemed to be most  likely for several



reasons:  The NMR-spectrum indicated the predominant presence of a compound



with a typical vinyl side chain.  This compound had earlier been found to



comprise the major portion of the LOMOLS.  TLC demonstrated that thts com-



pound was present as monomer (comparison with an authentic sample with this



structure).  However, the refractionation of peak c yielded the desired



material only in minor amounts, and the fractionation pattern exhibited



resembles strikingly much the original elution pattern of the ES ALSME



derivatives.



     These results allowed the conclusion that some compound, possibly the



one with the/5-vinyl structure, rearranges and/or isomerfzes extremely



readily to nearly everything we call LOMOLS.  Since the isomertzation



behavior of compound I  had been studied before, a reaction pathway Involv-



ing a double bond was suspected; therefore, the second half of the ES ALSME



was brominated prior to its fractionation.



     After bromination, the only obviously altered peak appears to be d.



It  is interesting to note that this peak was found to be the direct pre-



cursor of the polymerization (vinyl-plym.), as stated from the previous



experiment (see Figure 19).




     Refractionation of the mer class representing compound d, resulted



indeed  in the isolation of a single, stabilized peak d.  The refractionation



of the other mer classes showed again the known instability (see Figure 21).



No satisfactory explanation was found for the observation that the vinyl



compound I  was again present in the brominated ES ALSME.  There Is no reason





                                 58

-------
     (b)
                                          (d)
                                                                   (e)
                                                                  (a)
                                                                  (POLYMER)
 OAC
(b)
 CH=CH2
 CH-S03CH3
                                                 (a)   (POLYMER)
             (c)
(d)
           FIGURE  19.

           THE  "REGENERATION PATHWAY"  IN TERMS OF PEAKS, AS
           VISUALIZED FROM THE SEPHADEX LH-20 FRACTIONATIONS.
                        59

-------
                     Effluent Volume
                    Effluent Volume
FIGURE 20.
Elution Diagram of Bromlnated ES ALSME Derivatives and the
Refractionation Patterns of Some Her Classes.
                       60

-------
                                  -ArOH
                                               POLYMER
      POLYMER
FIGURE  21.

ACID HYDROLYSIS OF THE VERATRYL^GLYCERYL-^
-ARYLETHER, ITS SULFONATION- AND POLYMERI-
ZATION PRODUCTS.
                    61

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why its double bond should survive bromination,   It seems as  If this double

bond is generated not only by coniferyl alcohol endgroups as was assumed

hftherto.

     The questTon as to the origin of th.e vinyl-groups is belteved to be

answered only unsatisfactorily wtth contferyl alcohol end-groups,  tt could

be demonstrated that the most abundant intermediate of the acido lysis reaction

pathway of the 3-ether, as described by Adler, et.al., was able to form a

sulfonate with bisulfite ions (see Figure 21).  Thfs compound formed two

spots on TLC after acetylation with acetic anhydride and pyridine.  Since

it also contained a carbonyl-group, its structure is expected to match com-

pound II and acetylation forms the enoI acetate III and the ketoh II.

     After transformation to ALSME-derivatives, 85% of the sulfonate appeared

as polymeric ether insoluble amorphous powder.  The residual  \5% ether-

solubles, showing efght distinct spots on TLC, exhibit an abnormal amount of

vinyl-groups in their NMR-spectrum (most of them conjugated to the aromatic

ring) and an acetyl-peak, the location of which matches an enoI acetate.

Conclusions

     LOMOLS seem to be a mixture of several particular mers and mer classes

that are in an equilibrium with each other and that rearrange and/or isomer-

ize easily to "regenerate" this mixture.   The main reaction apparently involves

a double bond, which indicates vinyl  polymerization as the mode of formation

of higher mers.  Guaiacyl-propene-2-sulfonic-acid-l  seems to play a key role

in this reaction.  Its double bond stems obviously not only from coniferyl

alcohol  endgroups.

     It was found that hydrolysis products of 3-ethers undergo sulfonation,

and that these sulfonates are capable of forming vinyl groups via keto-enol

tautomerism, where the enol form polymerizes readily, probably in a vfnyl-

type polymerization.
                                  62

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                             SECTION X




                 PRELIMINARY STUDIES ON  INDUSTRIAL




                SCALE SEPARATION OF SSL COMPONENTS
 ntreduction
       In the  light of the  investigations reported in the earlier sections



of this report and prior work  in this  laboratory, preliminary experiments



were carried  out directed  toward investigation of feasibility of industrial



scale separation of SSL components.



      Two techniques were  given preliminary study.  One was solvent extrac-



tion of spent sulfite  liquor solids by butanol-water and ethanol-water



mixtures.  The other technique was a further study of the use of ion-



exchange resins on a column arrangement.  LOMOLS are separated from HIMOLS



presumably through some molecular sieve mechanism and from sugars in recog-



nition of the fact that the non-ionic sugars would not be excluded from the



pores  in an ion-exchange resin, whereas the  lignin sulfonates would be so



excluded.



      Earlier work in this  laboratory showed that high molecular weights



lignins can be separated from the rest of the substances in SSL, perhaps



technically although not necessarily economically by dialysis (31) and



by the formation of amine  salts of  lignin sulfonates.  Quantitative



separation from sugars was achieved by precipitation or solvent extraction



of the amine salts of  lignin sulfonates.  This salt formation was reversed



by use of sodium hydroxide or another strong base to give rise to freeing



the amine and formation of the metal salts of the lignin sulfonates which



is perfectly soluble in water.





                                 63

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Separation by Alcohol Extraction


      In this  laboratory, a considerable effort has  been made toward


separating lignin sulfonates of various molecular weight  (32-36).  One


of the approaches has been the fractionation by ethanol-water mixtures  (37).
                      ''i.                     '•••

It could be demonstrated that the MW of the dissolved  fractions  increased
                                       r ,

with  the water content of the eluant.  Preliminary  tests  have shown that
                                        i   • • j, '•

SSL solids can only be extracted with ethanol-water mixtures with water
                     /vi" "~ i                • .3."; ,"'*
contents up to \5%.  At higher water contents, the  solids yielded a sticky


unextractable tar.


Experimental


      Steam-stripped fermented spent sulfite liquor  from gymnosperms was


provided by the Georgia-Pacific Corp., in Bellingham, Washington.  The


liquor was neutralized with sodium hydroxide, freeze dried, and then extrac-


ted with ethanol-water mixtures beginning with 95%  ethanol and followed by


exhaustive extraction with ethanol containing increasing proportions of


water.  The extracts and extracted solids were analyzed by Sephadex gel


chromatography applying controlled ionic strength and the results are shown


in Table 4.


      In a second similar experiment spent sulfite liquor solids CCalcium


base) were extracted with ethanol  and ethanol-water mixtures and the weight


of the dissolved solids and the absorbance of solutions of the same was


determined.  A material balance by weight and absorption at 280 nm was


established.


Results and Discussion


     Treatment with 95% ethanol  resulted in the extraction of about 2% of


the organic matter which contained only 255? UV absorbing material (see


                                 64

-------
                                                TABLE 4
Extraction Conditions:  lOg CaSSL extracted with 500 ml. ethanol  and ethanol:water mixtures for twelve
                        hours at room temperature.


Starting Material
Ex 100
Ex 95
Ex 90
Ex 85
Ex 80
* Tarry residue
Precipitation (dissolved
Starting Material
95-S
90-S
80-S
a
(g)
10.0
0.6
0.9
1.50
2.20
3.20*

matter)
20.00
4.48
6.00
8.20
a weight (g) recovered.
b % weight based on starting material
c average absorbance of samples.
d % of total absorbance at 280 nm.
e theoretical weight of
f % weight of absorbing
b
%
100.0
6.0
9.0
15.0
22.0
32.0*

100.0
22,5
30.0
41.0
Column Expl
•
absorbing material where a,~a
material (LS) based on start i
c
Aa
9.100
0.022
0.184
0.980
1.430
1.430

18.2
2.40
3.65
6.40
anation

Q assumed
ng materi
d
*A280
100.0
0.24
2.0
10.8
15.8
15.8

100.0
13.3
20.0
35.0

constant at
al. l/b X(e
e f
(g) %s
7.6 76.
0.018 0.12
0.15 1.5
0.82 8.2
1.19 1 1.9
1.19 11.9

15.20 76.0
2.02 10.2
3.05 15.2
5.30 26.5

12.0.
X 100)
g
%r
76.
3.0
16.7
54.5
54.5
37.2*

76.
45.
50.
64.


g  % weight of absorbing material (LS) based on recovered  fraction.

-------
Starting
    Materia
    Dissolved
                                                              x
                                                           x-  LS
                                                               So IubIes
                                                               (Precip.)
                                      Total
                                  Solubles
                               (Precip.)
                                                      Tota
                                                   SoIubIes
                                                  (Extr.)
                                                            LS Solubles
                                                            (Extr.)
                                                  -
                                                 >S             20
                                                 % Water in Ethanol

                     FIGURE 22.
                     DISSOLUTION OF SSL SOLIDS AS A FUNCTION OF
                     THE WATER CONTENT OF ETHANOL.
                                    66

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Figure 22).  Two-thirds of the material  represented carbohydrate degrada-



tion products.  The extracted  Iignin sulfonate fraction gave a well resolved



elution pattern on gel chroma tog ra ph. i.c separation using SepKadex G-15.  It



could be  demonstrated that the so-extracted LOMOLS fraction consists



mainly of very  low molecular weight material.



     Subsequent extraction with 88% ethanol, carried out in three stages,



resulted in the dissolution of 22$ of the organic matter consist-ing of



about 50% of the  I ignin sulfonates..  The ratio between absorbing (lignin-



like) and non-absorbing (carbohydrate-like) material in all three stages



was practically the same.  The elution 'diagrams obtained from analytical



Sephadex separations  indicate that these fractions consist also of very



low molecular weight  materials.



     In another set of experiments we studied the precipitation of Iignin



sulfonates from aqueous solutions by ethanol.  We established the material



balance and found that the ratio between carbohydrate degradation products



and  Iignin sulfonates over the  investigated range of ethanoI-water mixtures



(up to 2Q% water)  remained constant.  Comparative gel-chromatographic LOMOLS



obtained by the two different techniques (extraction and precipitation)



have a very similar composition.



Conclusions



     These preliminary studies allow the conclusion that a certain amount



of carbohydrate degradation products (e.g., monosaccharides) can be extracted



with absolute ethanol, or generally, high percentage ethanol (.beyond 95%)',



however, a satisfactory separation of  lignin sulfonates and carbohydrate



reaction products by  more extraction with, or precipitation from, ethanol



water mixtures does not seem to be feasible.
                                  67

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Separation by Ion Exclusion                        ,.



     Several years ago In this  laboratory, pioneering research had been



conducted on sugar llgnin sulfonate separations using ion exchange resins



(17).  A fractfonation of SSL components  into sugar-rich and  llgnin sulfonr



ate-rich portions was achieved.   Iri recent years, this technique has been
                                 <,."


studied and improved in several academic and industrial   laboratories C7, 38)	
                             -5*


To evaluate the separation under optimal conditions, we carried out some



studies applying extremely low  loadfngs and very slow flow rates and



established material  balances.



Experimental



     Freeze dried spent sulfite liquor was dissolved in distilled water,



loaded onto a column filled with Dowex 50W-X2, samples eluted with water,

                                                                           _/

and fractions collected with an automatic fraction collector.  These were



examined using UV absorption at 280 nm and the elution diagram was plotted



(see Figure 23).  Each fraction was quantitatively neutralized with sodium



hydroxide, thus determining the acid number.  The neutralized sodium spent

                                   -.j -,j .
sulfite liquor was then concentrated, freeze dried, and the dry matter



content of each sample was determined.   The elution diagrams from analyti-



cal gel chromatography using Sephadex G-25 and G-50 were also determined.



Results and Discussions



     By using the ion-exchange resin in H-form we expected a better separa-



tion of charged molecules, such as lignin sulfonates, aldonic acids and



sugar sulfonic acids, from non-charged molecules such as mono-, dt- and



poly saccharides.  Due to the low loading and slow flow rate, we observed



complete exchange of ions within the first 5 to 10  inches of the total



column length (7 feet).  The remaining separation was exclusively governed



by the principle of  ion-exclusion.
                                68

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WEIGHT
     RECOVERED
     C9J
                                       P-.
UNIDENTIFIED
                                          \/  MATTER
                                                           ^REDUCING
  so        7o        fo         no        >bo
                                                         ELUTION VOLUME
   FIGURE 23.
   ELUTION DIAGRAM OF A SSL  IN  ION EXCLUSION CHROMATOGRAPHY.
                             69

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     Although no complete categorical separation of the SSL components



could be achieved, the accomplished separation into three main fractions



with distinct different composition  is of enormous technical and scientific



interest.



     The main fraction comprises about 55% of the total material and con-



tains high and middle molecular weight Itgni'n sulfonates, contaminated



with carbohydrate degradation products to an extent of about 10$ or less.



     The second fraction consists of low and middle molecular weight Iig-



nin sulfonates and carbohydrate degradation products in about equal  pro-



portions (1:1).  Since the content of reducing groups is moderate, we



assume that the non UV absorbing material consists mainly of aldonic acids.



The fraction amounts to about \5% of the total  material.



     The remaining 30% contains only traces of lignin sulfonates and com-



prises carbohydrate degradation products with the bulk, of mono- and  dl-



saccharides.



Conclus ions



     The reported pre Iimi nary study demonstrated that a crude separation



of spent sulfite  liquor components into three major fractions by ion



exchange exclusion chromatography can be achieved.



     From an industrial  point of view, all  of the three fractions have a



utilization potential.   The last two fractions contain practically all  of



the carbohydrate degradation products which may represent a valuable source



for a number of salable products.



     Both experiments gave rise to preferential separation of low molecular



weight ligntn sulfonates.  This is indicated in the graphs of Figure 22



and Figure 23.   In the separation with alcohol, 10$ of the lignin sulfonates
                                 70

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were separated and proved to be of  low molecular weight and relatively


low content of sugar components.   In the  unique  ion exclusion separation


similar results were obtained  as shown  in Figure 23.
      *

     Of special interest  in most cases are the  results obtained on separa-


tion of the resultant  low molecular weight Iignin sulfonate fraction when


subjected to gel  chromatography using Sephadex G-25 or Sephadex G-50.


     The  results  from  the  ton  exclusion experiment demonstrated that three


different types of  fractions could  be obtained:


      Fraction  I represented about  55% of  the total material containing


high  and medium  low  molecular  weight  LS contaminated with carbohydrate


degradation products  up  to  15$.


      Fraction  II  consisted  of  low  to  middle molecular weight LS and about


50% carbohydrate  degradation  products,  most of which were non-reducing and


of unknown  structure (possibly aldonic  acids).


      Fraction  Ml contained mainly sugars.
                                  71

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                            SECTION XI




                        CONCLUDING COMMENTS





     Lignin sulfonates from the spent sulfite pulping  liquor of Western



Hemlock have been separated in purified form using an alcohol extraction



and precipitation method as well as  ion exclusion chromatography.  Both



methods resulted  in the isolation of mainly three fractions:  high and



medium molecular weight lignin sulfonates,  low mol. v. LS, and carbohy-



drate degradation products.   In the alcohol extraction and/or precipita-



tion method, the separation was of  lower quality than  in the separation by



ion exclusion.  Neither separation method, however, was capable of isola-



ting pure LOMOLS.



     The characterization of  lignin sulfonates worked best after covering



the highly polar hydroxyl- and sulfonate-groups by acetylation and



esterification.  NMR spectroscopy allowed a complete functional group



analysis and overall, appeared to be the most useful analytical method.



     Summarizing the structural evaluation of low and high molecular



weight LS, it appears that LOMOLS are different from HI.MOLS by configura-



tions that affect the color as well as surface tension properties.  LOMOLS



were found to contain more phenolic hydroxyl-groups, more double bonds,



and probably more carbony I-groups.  The major type of  linkage seems to be



one similar to a vinyl-polymer (two dimensional).  This appears to be the



result of the sulfonation of acid hydrolysis products of alky I-aryI-ethers,



Most properties of LOMOLS can be discussed  in terms of this formation




hypothesis.
                                 73

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                            SECTION XI I




                          ACKNOWLEDGEMENTS






Dean R.W. Moulton, Chairman of the Department of Chemical Engineering,



University of Washington, provided helpful administrative assistance



for the project.  Ms. June Demont did the secretarial work.






Professors K.V. Sarkanen and G.G. Allan made valuable suggestions



and their cooperation on several occasions is appreciated.






The support of the project by the Office of Research and Monitoring,



Environmental Protection Agency, and the help provided by Mr. George R.



Webster and Dr. H. Kirk Willard, the Grant Project Officer, is



acknowledged with sincere thanks.
                                  75

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                              SECTION XI I I

                              REFERENCES

 1.  Schubert, S. W. , Audrus, M.  G.,  Ludwig,  C.,  Glenn ie, D., and
      nn£y;   --'CcrySt?n!ne Low Mol*cular  Weight Llgnin-Type
     Sulphonates.   II.  Synthesis  and  Establishment of Structure "
     TAPPI. 50,,  186-193 (1967).

 2.  Glennie, D. W. , "Chemical Structure of Lignin Sulphonates. III.
     Some Reactions of  Monomeric  Lignin Sulphonates." TAPPI, 49, 237-
     Z4Z  (1966).                                      "" ~— ~" """"

 3.  Gupta, P. R., and  McCarthy,  J. L., " Lignin XIV.  Gel Chromato-
     graphy and  the Distribution  in Molecular Size of Lignin Sulphonates
     at Several  Electrolyte Concentrations," Macromolecules. 1, 236-244
     (1968).                                            "~— * "~

 4.  Gupta, P. R., and  J. L. McCarthy, "Lignin XV.  Preliminary Char-
     acterization of Several Low  Molecular Weight Ligninsulfonate
     Mers," Macromolecules. \_, 495-498 (1968).

 5.  Forss, K. ,  "The Composition  of a  Spent Spruce Sulfite Liquor,"
     Dissertation, Abo  Akademi, 1961.

 6.  Forss, K. and Fremer, K. E. , "The Dissolution of Wood Components
     Under Different Conditions of Sulfite Pulping," TAPPI, 47(8),
     485-493  (1964).                                 - L  ~

 7.  Jenson, W. , Fremer, K. E. and Forss, K. , "The Separation of the
     Components  in Spent Sulfite  Liquor," TAPPI, 4_5_(2) ,  122-127 (1962).

 8.  Ludwig, C.  H., Mist, B. J.,  and McCarthy, J. L., "Lignin XII.  The
     High Resolution Nuclear Magnetic Resonance Spectroscopy of Protass
     in Compounds Related to Lignin," J.  Amer. Chem.  Soc.,  86,  1186-1196
     (1964).                          -   — '

 9.  Ludwig, C. H., Nist, B. J.,  and McCarthy, J. L., "Lignin XIV.  The
     High Resolution Nuclear Magnetic Resonance Spectroscopy of Protass
     in Acetylated Lignlns," J. Amer. Chem.  Soc., 8£, 1196-1202 (1964).

10.  Lenz, B.  L., "Application of Nuclear Magnetic Resonance Spectro-
     scopy to Characterization of Lignin," TAPPI, 5J_, 511-519 (1968).

11.  Kovacik,  V., "Massenspectrometric Einiger Model 1 subs tanzer des
     Llgnins,  I," Chem.  Ber. ,  102, IS13-I522 (1969).

12.  Kovacik,  V., "Massenspectrometric Einiger Modellsubstanzer des
     Llgnins,  II," Chem. Ber., 102, 3623-3631 (1969).
                                  77

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13.   King, E. G., Brauns, F., and Hibbert, H.,  "Studies on Lignln and
     Related Compounds XVIII. Lignin Sulpharlc  Acid - A .Preliminary
     Investigation on Its Isolation and Structure," Can. J. Research,
     J3.B, 88-92  (1935).                                            "

14.   Parrish, J. R.t "Monomeric Lignin Sulphonie Acids. Part II,"
     J. Chem. Soc. (C), 1145-I'50 (1967).

15.   Gellerstedt, G., and Gierer, J., "The Reactions of Lignin During
     Neutral Sulphite Cooking.  Part I. The Behavior of (3-Arylether
     Structures," Acta. Chem. Scand., 22_,  2510-2518 (1968).

16.   Gellerstedt, G., and Gierer, J., "The Reactions of Lignin During
     Neutral Sulphite Cooking.  Part II. The Behavior of Phenyleoumaran
     Structures," Ibid., 22_, 2029-2031(1968).

17.   Felicetta, V, F., Lung, M.  and McCarthy, J. L., "Spent Sulphite
     Liquor VII. Sugar-Lignin Sulphonate Separations Using Ion Ex-
     change Resins," TAPP'I,  42_,  496-501 (1959).

18.   Benko, J., "Separation  of Solutions of Spent Sulphite or Kraft
     Liquors and Bark Extracts," U.  S. Patent No. 3.509.121, April 28,
     1970.

19.   Bjorkman, A., "Studies  on  Finely Divided Wood, Part I." Svensk
     Papperstidning, 59, 477-485 (1956).

20.   Bjorkman, A., and Person,  B., "Studies on  Finely Divided Wood,
     Part II." Ibid, 60, 158-169 (1957).

21.   Bjorkman, A., "Studies  on Finely Divided Wood. Part III. (i) Extrac-
     tion of Lignin Carbohydrate Complexes with Neutral Solvent,"
     Ibid, 60, 243-251, 285-292, 329-335 (1957).

     (ii) Studies,,on Finely  Divided Wood.  Part  IV. Some Reactions
     of the Lignin Extracted by Neutral Solvents from Picea abies.
     1 us.

     (iii) Studies on Finely Divided Wood, Part V. The Effect of
     Milling.

22.   Bjorkman, A., Grenoble  - Symposium.

23.   Lundquist, K. and Ericsson, L., "Acid Degradation of Lignin VI.
     Formation of Methanol," Acta Chem. Scand., 2_5_ 756-758 (1971).

24.   Forss, K. and Fremer, K. E., " The Repeating Unit in Spruce
     Lignin," Paper? ja Puu, 47., 443-454 (1965).

25.   Forss, K., Fremer, K. E.,  and Stenlund, B., " Spruce Lignin and
     Its Reactions in Sulfite Cooking - II. The Reactions in Sulfite
     Cooking," Paper? ja Puu, 4j[, 669-676 (1966).
                                  78

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26.  Gierer, J., "The Reactions of Llgnln During Pulping.  A Des-
     cription and Comparison of Conventional Pulping Processes,"
     Svensk Papperstidning. 73., 571-596  (1970).

27.  Freudenberg, K., "Uber einen Foromelvarschlag fur das
     Fichtenlignin," Holzf.. 22. 65-66   (1968).

28.  Forss, K., "Das Fichtenlignin." Holzf.. 22_, 66-68  (1968).

29.  Freudenberg, K., "Antwort," Holzf.. 22_, 68-69   (L968).

30.  Adler, E., "Guaicylglyceral and its B-Guaicyl Ethyl." Acta
     Chem. Scand.. 9_, 341-342   (1955).

31.  (i) Lundquist,  K.,  "On the Separation of Lignin Degradation
     Products," Acta Chem. Scand.. J8, 1316  (1964).

     (ii) Lundquist, K.,  "Isolation of 3-Hydroxy-1-(4-hydroxy-3-
     methoxy pheny1)-2-propanone from Lignin," Acta Chem. Scand..
     J6_, 2303-2304   (1962).

32.  Peniston, Q. P. and McCarthy, J. L., "Lignin  I. Purification
     of Lignin Sulphonic Acids by Continuous Dialysis," J. Amer.
     Chem. Soc..  70.  1324-1328    (1948).

33.  Moscanin, J., Felicetta, V. P., Mailer, W. and McCarthy, J. L.,
     "Lignin VI.  Molecular Weights of Lignin Sulphonates by Light
     Scatterings," J. Amer. Soc., 77, 3470-3474 (1955).

34.  Felicetta, V. P., Ahola, A., and McCarthy, J. L., "Lignin VII.
     Distribution in Molecular Weight of Certain Lignin Sulphonates,"
     J. Amer.  Chem.  Soc.. 78_, 1899-1904  (1956).

35.  Mokihara, E., Tuttle, M. J., Felicetta, V. P., and McCarthy, J. L.,
     "Lignin VIII. Molecular Weights of  Lignin Sulphonates during
     Delignification by  Bisulfite-Sulfurans Acid Solutions," J. Amer.
     Chem. Soc..  79, 4495-4499  (1957).

36.  Felicetta, V. P., and McCarthy, J.  L., "Lignin  IX. Molecular
     Weights of Lignin Sulfonates as  Influenced by Certain Acidic
     Conditions," J. Amer. Chem.  Soc.. 79_, 4499-4502 (1957).

37.  Moscanin, J., Halson, H.,  Felicetta, V. P., and McCarthy, J. L.,
     "Lignin XI.  Estimation of Polymolecularity in Lignin Sulfonate
     Polymers  from Diffusion Measurements," J. Amer. Chem. Soc., 81,
      2054-2056 (1959).

38.  Markham, A.  E., Feniston, Q. P. and McCarthy, J.  L., "Lignin  III.
     Fractional Precipitation of  Barium  Lignin Sulfonates from Water
     vs. Ethanol," J. Amer. Chem. Soc.,  T\_,  3599-3607   (1949).

39.  Benko, J.. U. S. Patent No.  3.509.121. April  28,  1970,  Dryden
     Chemicals Ltd., Oakville, Ontario,  Canada.
                                   79

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                            SECTION XIV

                     PUBLICATIONS AND PATENTS


The following publications have been produced or are anticipated to be

produced as a result of this  project:

      SPENT SULFITE      Preparation, Fractionation, and Preliminary
      LIQUOR XIV.        Characterization of Cymnosperm Lignin
                         Sulfonates from Spent Sulfite Liquor and
                         Milled Wood Lignin.  Forss, K., Collins, J.J.,
                         Glasser, W.G., Gratzl, J.S., and McCarthy,
                         J.L., Tappi, 55_,  1329-1333 (1972).

      LIGNIN XVI.        Synthesis, Nuclear Magnetic Resonance, and
                         Mass Spectroscopy of Several Monomeric and
                         Dimeric  Lignin-like Sulfonates.  Glasser,
                         W.G., Gratzl, J.S., Collins, J.J., Forss, K.,
                         and  McCarthy, J.L., Macromolecules, 6,
                          114  (1973)

      LIGNIN XVII.       Preparation and Characterization of Acetyl
                          Lignin Sulfonate Methyl Esters.  Glasser,
                         W.G., Gratzl, J.S., Collins, J.J., Forss, K.,
                         and  McCarthy, J.L.  To be submitted for
                         publication  in Macromolecules.

 It appears that  no  patentable developments have arisen from the

present study.

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                             SECTION  XV




                              GLOSSARY



ALSME - Acetylated llgnin sulfonate methyl ester.



Ca/Na-SSL - Calcium or sodium base spent sulfite liquor.



DP_- Degree of polymerization.



EIS - Ether insoluble.




GPC - Gel permeation chromatography.



HI MOIS - High molecular weight  lignin sulfonates.



LOMOLS - Low Molecular Weight Lignin  Sulfonates.



LS - Lignin Sulfonates.



MW - Molecular Weight



NMR - Nuclear magnetic  resonance.



SSL - Spent sulfite  liquor.



TLC - Thin  layer chromatography



UV - Ultra  violet spectroscopy.
                                   83

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SELECTED WATER
RESOURCES ABSTRACTS

INPUT TRANSACTION FORM
•"l.ariceport'rfo.-

  is

l:
                                                        '2,' •- , !*
                                                                   3. Accession No.
                            w
 4. Title

  Studies of Low Molecular Weight Lignin Sulfonates
 7. Autnorw  B. F. Hrutfiord, L. N. Johanson, J.  L. McCarthy,
  K.  Forss, W. Glasser, J. Gratzl, J. Collins
                            10. Project No.
     University of Washington
                            11. Contact/Grant No.

                              12040 DEH
              ization
« "•; =  '^ *,*'^'
._g.-'_i-_-   -... • Vg-
 15. Supplementary Notes

  Environmental Protection Agency Report No.  EPA-660/2-74-069, tfune
 16.-Abstract  LOW molecular weight lignin sulfonates  have been separated in purified form and
  characterized by physicochemical and chemical methods.   Their structure and reactions
  have been evaluated.
       Lignin sulfonates from the spent  sulfite liquor of a mild acid bisulfite cook of
  Western Hemlock (Tsaga heterophylla) were  purified and  fractionated in Sephadex 6-25
  column chromatography.  Samples were analyzed using acetylation of hydroxyl-groups and
  esterification of sulfonate-groups which aided  the elimination of the polydisperse
  nature of the material under investigation.
       Complete elemental and functional  group compositions were established for lignin
  sulfonates from a spent sulfite liquor and compared to  those from milled wood lignin
  preparation.  This allowed an estimate of  the degree of sulfonation, condensation and
  demethylation as well.
       Extended separation studies indicated the  low molecular weight lignin sulfonates t<
  be the reaction product of a difunctional  vinyl-type polymerization, thus accounting
  for the widely different properties as compared to their higher molecular wefght
  counterparts.  The feasibility of  large scale separations was determined using (1)
  the extraction and precipitation of the dry matter in a spent sulfite liquor with
  alcohol, and (2) the fractionation of  the  material by ion exclusion in a column
  arrangement.
 17a. Descriptors
  Sulfonates, lignin, pulp wastes,  chemical  analysis, by-products, molecular structure,
  organic wastes, separation  techniques, sulfite liquors, waste identification, Pacific
  Northwest U.S.


 17b. Identifiers

  Lignin sulfonate  separation,  chemical  composition, spent sulfite liquore
 17c. COWRR Field &. Group
18. Availability }- 19, Security 'Class. ?
, (Report) " •* '
1 ' * "',"%"'.*
20 •* Security Ctev
! 	 ,.(^ase) _ c
Abstractor H. Kirk Will ard
<• 21 No', of |
> fages -•!
"«. ' .. - f~ ]
22. PWMT 't.'"i
Send To:
WATER RESOURCES SCIENTIFIC INFORMATION CENTER
U.S. DEPARTMENT OP THE INTERIOR
WASHINGTON. OjC. 20240
institution EPA - Pacific NW Environmental Res. Lab.
WRSIC 102 (REV. JUNE 1971!
                                                                                 Q P O 488-935

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