United States                      EPA 600/6-84-010
                Environmental Protection
                Agency	FEBRUARY 1984
&EPA        Research and

                Development
                DATA ACQUISITION FOR ENVIRONMENTAL
                TRANSPORT AND FATE SCREENING FOR
                COMPOUNDS OF INTEREST TO THE OFFICE
                OF SOLID WASTE
                Prepared for
                OFFICE OF SOLID WASTE
                Prepared by

                Office of Health and
                Environmental Assessment
                Washington DC 20460

-------
                                           February 1984
DATA ACQUISITION FOR ENVIRONMENTAL TRANSPORT AND FATE SCREENING
     FOR COMPOUNDS OF INTEREST TO THE OFFICE OF SOLID WASTE
                               By

              H.  M. Jaber, W. R. Mabey, A. T.  Liu,
              T.  W. Chou, H. L. Johnson, T. Mill,
                R.  T.  Podoll, and J.  S. Winterle
                       SRI International
                     333 Ravenswood Avenue
                     Menlo Park,  CA   94025

                  EPA Contract No.  68-03-2981
                     Work Assignment No. 15
                        Project Officer
                         Lee A. Mulkey
               Environmental Research Laboratory
              U.S.  Environmental Protection Agency
                       Athens,  GA   30613
                   Technical Project Monitor
                          Gregory Kew
                   Exposure Assessment Group
         Office of Health and Environmental Assessment
               Office of Research and Development
              U.S. Environmental Protection Agency
                     Washington, DC   20460
         OFFICE OF HEALTH AND ENVIRONMENTAL ASSESSMENT
               OFFICE OF RESEARCH AND DEVELOPMENT
              U.S. ENVIRONMENTAL PROTECTION AGENCY
                     WASHINGTON, DC   20460

-------
                         DISCLAIMER

     This report has been reviewed in accordance with U.S.
Environmental Protection Agency policy and approved for
publication.  Mention of trade names or commercial products
does not constitute endorsement or recommendation for use.

-------
                                 FOREWORD
     The Exposure Assessment  Group  of  EPA's Office of Research and
Development has  three  main functions:   1)  to conduct exposure
assessments; 2)  to  review assessments  and  related documents;  and 3)  to
develop guidelines  for Agency exposure assessments.  The activities
under each of  these functions are  supported by and respond to the needs
of the various EPA  program offices.  In relation to the first function,
the Exposure Assessment Group sponsors projects for the purpose of
gathering data used in exposure assessments.  This study is one of those
projects and was done  for the Office of Solid Waste (OSW) .
     The Resource Conservation and  Recovery Act of 1976 (RCRA)
authorizes a. regulatory program to  identify those wastes which pose  a
substantial hazard  to  human health  or  the  environment and to establish
management standards sufficient to  prevent such harm.  A portion of  this
program focuses  on  individual chemicals and requires determining their
toxicity, capacity  to  be transported to susceptible populations, and
potential fate in the  environment.   The data compiled in this report are
intended to assist  OSW in predicting the probable fate and transport
properties of  compounds selected by OSW after study of various
industrial waste streams.
                                             James W. Falco, Director
                                             Exposure Assessment Group
                                 ii

-------
                                ABSTRACT
     Physical properties, equilibrium, and kinetic constants for
evaluating the transformation and transport in aquatic systems for
organic chemicals of interest to the Environmental Protection Agency
have been obtained from the literature and calculated from theoretical
or empirical relations.  Values for selected physical properties such as
melting point, boiling point, vapor pressure, water solubility, and
octanol/water partitioning, and for rate constants such as hydrolysis,
microbial degradation, photolysis, and oxidation are listed for each
chemical along with the source of the data.  Values are reported in
units suitable for use in a current aquatic fate model.  A discussion of
the empirical relationships between water solubility, octanol/water
partition coefficients, and partition coefficients for sediment and
biota is presented.
     This report was submitted in partial fulfillment of Contract No.
68-03-2981 by SRI International under the sponsorship of the U.S.
Environmental Protection Agency.  This report covers a period from 1 May
1983 to 30 September 1983 and work reported herein was completed as of
30 September 1983.
                                 iii

-------
                                CONTENTS

FOREWORD                                                            ii

ABSTRACT                                                           ill

    1.   Introduction	  1

           Purpose	  1
           Background	  2
           References	  8

    2.   Definition  of  Processes  and  Sources  of Data	  9

           Basis  for derivation of  data	  9
           Chemical  name,  Chemical  Abstracts  Service registry
             number, and molecular  weight	 10
           Water  solubility	 10
           Melting  and  boiling point	 11
           Vapor  pressure	 11
           Molecular weight to oxygen ratio	 12
           Octanol/water partition  coefficient	 12
           Hydrolysis rate constants	 13
           Mlcrobial degradation  rate constant	 14
           Photolysis rate constant	 16
           Oxidation rate  constant	 16
           References	 20

    3.   Data  Sheets for Chemicals  of Interest	 22

           List of  data sheets	 23
           List of  source  codes	 26
           Data sheets	 28
           References	102

    4.   Calculation of Partition Coefficients  of  Organic
         Chemicals  in Aquatic Environments	104
                               iv

-------
                                SECTION 1
                              INTRODUCTION

PURPOSE

     Decisions on possible regulatory action  or  cost-effective  remedial
measures for toxic chemicals require an understanding of  environmental
and human risks associated with the manufacture, use, and disposal  of
chemicals.  Part of the risk assessment requires the best scientific
information about what the concentration  of a chemical  is in the
environment.  In the absence of reliable  and  extensive  monitoring data,
the concentration of a chemical can be estimated using  one of several
fate models and data for the individual processes  that  may be dominant
for that chemical.  These data may be measured in  the laboratory,
obtained from literature sources, or estimated using appropriate
structure-activity relationships  (SARs) or correlation  methods.  These
data used with environmental parameters in a  mathematical model
constitute the process modeling approach  (Baughman and  Burns, 1980;
Baughman and Lassiter, 1978; Smith et al., 1977; Mill,  1978).
     The compounds listed in this report  were of concern  to the Office
of Solid Waste after study of waste streams from certain  industrial
processes.  Others are recognized by-products or potential trace  by-
products which might have substantial health  impacts if appropriate
waste disposal practices are not  followed.  The  Office  of Solid Waste
has requested that chemical-specific Health and Environmental Effects
Profiles, or preliminary risk assessments, be prepared  from existing
literature sources to assist in deciding  whether the chemical should  be
listed as hazardous wastes under  provisions of the Resource Conservation
Act and Recovery Act of 1976, Section 3001.   The Office of Health and
Environmental Assessment, consequently is examining the toxicological,

-------
 environmental and chemical literature as background for this work.  This
 report  compiles literature data or estimates for 10 fundamental physical
 and  chemical parameters for 74 chemicals which subsequently will be
 analyzed to predict their potential environmental transport, fate and
 persistence.
     These data are to be used to decide what chemicals clearly would
 not  persist in aquatic environments because of exceptional reactivity
 and  what environments may be of particular concern because of dominant
-volatilization or sorption processes.  This information will also be
 used to decide what data gaps exist and what particular process data
 need to be obtained for subsequent and more detailed assessments.
     The data are made available in this report with the expectation
 that they may be of interest in other assessment-efforts.  Use of the
 data in the context of other assessments requires that each user
 understand the sources and limitations of the data.  Each user must
 decide  what additional data are required for the particular
 assessment.  Any user of these data must particularly recognize that
 some values were estimated by SRI staff with expertise in the process of
 Interest, and that considerable subjective judgment was applied for some
 of  the  estimates.  Such judgments based on even crude analogies are
 indeed  valuable and acceptable in screening level evaluations.  In cases
 where  even expert judgment cannot be used to provide a value, no value
 was  entered.  Users of these data are encouraged to conduct more
 intensive literature searches or to consult other knowledgeable
 scientists to augment or supplant data in this report.
      In this report, "process data" are defined as data relating to rate
 constants, equilibrium constants, or physical properties that describe
 the  intrinsic processes the chemicals may undergo independent of
 environmental influences.  "Environmental parameter" in this report
 refers  to properties or data that describe (or are a function of) the
 environment.

-------
BACKGROUND
     The processes  that can be important for  transforming or transport-
ing a chemical  in an aquatic environment are  shown in  Figure 1.1.  The
following discussion summarizes the mathematical  basis for the process
modeling approach applied to aquatic systems:   (1)  the evaluation of
rates of loss of chemical due to transformations  and volatilization
processes,  (2)  the  influence of sorption processes on  the rates of loss
of chemical, and (3)  the prediction of concentration and half-life of
chemical in the aquatic environment, including  terms for input of
chemical, dilution,  and flow out of the environment.   This discussion
assumes that sorption to particulates in the  environment is not
kinetically controlled (i.e., sorption equilibrium is  attained
instantaneously).
          Inflow of
          Chemical
         Outflow of
           Chemical
                            Volatilization
                          Organic Chemical
                             in Aquatic
                            Environment
                         Sorption/Desorption
                            to Particulates,
Chemical Transformations
    Photochemistry
    Hydrolysis
    Oxidation
B iotransf ormations
    Hydrolysis
    Oxidation
    Reduction, etc.
                               II
                            Sedimentation
             FIGURE 1.1   TRANSPORT AND TRANSFORMATION PROCESSES IN
                         AQUATIC ENVIRONMENTS

-------
EVALUATION OF  CHEMICAL LOSS  RATES
     The rate  of  loss  of a chemical due to the above transformation
processes and  volatilization,  Rj,  is given by the sum of the rates of
the individual processes,  R^,  according to the equation
                                                                  (i.i)
where k^' is  the  rate  constant  for  the i-th process, [Ej]  is an
environmental parameter that is kinetically important for  the i-th
process, and  [C]  is  the concentration of the chemical.  The calculations
of R^ for individual processes  from environmental parameter and process
data are discussed  in  subsequent sections.  The important  environmental
parameters  for  each  process have been reviewed, and the use of the
parameters  in the calculations  of environmental transformation rates has
been discussed  in detail by Baughman and Burns (1980) , Mill (1978) , and
Smith et al.  (1977).
     The above  expression for R« assumes that the loss of  chemical is
first order in  the  chemical concentration, as certainly must be the case
at the highly dilute concentrations expected in the environment.
Equation (1.1)  also  requires that the rate of loss of chemical due to
any one process KJ  is  first order in the environmental parameter term
E*; RJ is then  considered as following overall second-order kinetic
behavior .   If it  is  assumed that the low concentration of  chemical in
the environment has  no significant  effect on the environment (for
example, does not change pH, biomass, dissolved oxygen, etc.) and that
the environmental parameter, E^, is constant over a specific region and
time period,  the  term k^' [E^]  can be expressed as a simple pseudo-
first-order rate  constant, k^,  and  then
or
                                 \ = ^±                         (1.3)
where kq.  is  the  overall pseudo-first-order rate constant for loss of
chemical  due to  transformation and volatilization.  The half-life for

-------
loss of chemical due  to  these  processes  is then given by


                              t1/2 - InZ/k^,                       (1.4)
INFLUENCE OF SORPTION
     In addition  to  losses  of  chemicals due to these transformation and
volatilization processes, sorption  to  particulates can also reduce the
concentrations of chemicals in aquatic systems.  These particulates may
be either suspended  sediments  or  biotic in origin and the particulates
may eventually be deposited into  benthic sediments.  The suspended or
benthic sediment may  later  serve  as a  source of chemical from sorption-
desorption equilibrium  as the  chemical in solution volatilizes or
undergoes transformation in the water  column.  If biotransformation does
not occur in biota (such as bacteria,  algae, and fish), the chemical may
be released back  into solution when the organism dies and decomposes.
The understanding of  chemical  transformation when the chemical is sorbed
onto particulates is  inadequate to  predict or measure the rates of such
reactions for use in  modeling. Therefore, the following discussion
assumes that no transformations occur  on particulates and that sorption
is completely reversible and rapid  in  comparison with transformations
that occur in solution.
     The partitioning of a  chemical between particulates (sediment or
biota) and water at  the low concentrations of chemicals usually found in
the environment can  be  expressed  as a  partition coefficient K_:

                                VCs/Cw                        (1'5)
where C_ and Cu are  the equilibrium concentrations of chemical on
       3      W
sediment and in water,  respectively (Baughman and Lassiter, 1978; Smith
and Bomberger, 1982).
     By convention, IL,  is unitless  when Cg is in units that are
equivalent to GW  (i.e., Cg  is  in  g  chemical/g particulate and GW is in g
chemical/g water).   In  this discussion, [Cw] will be defined in  these
weight units and  [C]  will be defined in molecular units (moles L  );

-------
because 1 g water  is  approximately 1 mL,  it follows that [C]  = 103[CW][MW]"1
where MW is the molecular  weight  of chemical.   Note that [C]  and [Cw]
can be used interchangeably in expressions such as equation (1.2)
because first-order rate  constants are concentration independent, but
the rate of loss  term,  R,  is of course defined in units corresponding to
[Cw] or [C].
     For a chemical in  aqueous solution containing particulates, the
chemical is equilibrated  between  the water and particulate P  according
to the relation
                                            C-P                   (1.6)
and the partition  coefficient can be rewritten as
                               K  »  [C-P1                         ri „
                                P   [Cw][P]                        (1'7)
where  [C-P]  is  the mass  of  sorbed chemical  per unit solution volume and
[P] is the mass  of sorbing  particulate per  unit solution volume.  The
mass balance of  chemical in the solution-sediment system is given by
                            [Cj.]  =  [C-P] + [Cw]
                                                                  (1.8)
where  [C_] is  the  total  mass of chemical in a unit solution volume of
water  containing [P]  grams  of particulate.   Combining equations (1.7)
and (1.8) then  gives  the fraction of the total chemical dissolved in
solution:
                                        i
                                    Kp[P]
Baughman and  Lassiter (1978)  have pointed out that,  given the relation-
ship  shown  in equation (1.9), the fraction of chemical in solution may
be quite high in spite of a large Kp value because the sediment or biota
loading,  [P] , is often low in aquatic systems (i.e., K_[P] < 1).
     The concentration of chemical in solution [C ]  in the presence of a
particulate-water system is then given by

-------
                                      [CT]
                                    [P]Kp
Substituting equation  (1.10)  into  equation (1.2)  for  the rate of loss of
chemical then gives
                                   [P]K  + 1
This relationship  shows  that unless  transformation on particulate is as
fast as or faster  than  that  in  solution,  the  net effect of sorption will
be to reduce the overall rate of  loss  of  chemical from the aquatic
system.  From equation  (1.11),  it also follows that the half-life of the
chemical is given  by

                                 ([P]K  + I)ln2
     The process modeling  approach  is  then a valuable tool in risk
assessments.  Although  values  of  t\/2  or  Cw can be manually calculated,
the calculations are more  easily  done  using computer  programs.  One such
computer model is EXAMS, which allows  the user  to choose environmental
parameters and is able  to  accommodate  chemicals when  several processes
compete to be the important  fate  pathway.   Computer models also allow
for sophisticated and environmentally  realistic dynamic models to be
used rather than assuming  steady-state conditions.

-------
                               REFERENCES

Baughman, G. L., and L. A. Burns.  1980.  Transport and Transformation of
     Chemicals: A Perspective.  In:  The Handbook of Environmental Chemistry,
     Vol. 2, Part A.  0. Hutzinger, Ed.  Springer-Verlag, New York.

Baughman, G. L., and R. R. Lassiter.  1978.  Prediction of Environmental
     Pollutant Concentration.  In:  Estimating the Hazard of Chemical
     Substances to Aquatic Life.  ASTM STP 657.  J. Cairns, Jr., K. L.
     Dickson, and A. W. Maki, Eds. American Society for Testing and
     Materials, Philadelphia, PA.

Mill, T. 1978.  Data Needed  to Predict Environmental Fate of Organic
     .Compounds.  Symposium on Environmental Fate held at American
     Chemical Society Meeting, Miami, FL, September 1978.

Smith, J. H. , and D. C. Bomberger.  1982.  Volatilization from Water.
     In:  Laboratory Protocols for Evaluating the Fate of Organic Chem-
     icals in Air and Water.  EPA-600/3-82-022.  U.S. EPA, Washington, DC.

Smith, J. H. , W. R. Mabey, N. Bohonos, B. R. Holt, S. S. Lee, T.-W. Chou,
     D. C. Bomberger, and T. Mill.  1977.  Environmental Pathways of
     Selected Chemicals in Freshwater Systems.  Part I.  Background and
     Experimental Procedures.  EPA-600/7-77-113.  U.S. EPA, Washington, DC.

-------
                                SECTION  2
              DEFINITIONS OF PROCESSES AND SOURCES OF DATA
BASIS FOR DERIVATION OF DATA
     The data on chemicals given in this report were obtained from the
literature and from calculations based on theory, SARs, or empirical
calculations.  In general, the physical properties of a chemical are
functions of the molecular structure as an entity; that is, the
elemental composition, spatial relationships and size, molecular weight,
and functional groups of the molecule all may contribute to the property
of the chemical.  In contrast, the chemical or biological reactivity of
a.molecule is usually caused by selected functional groups in the
molecular structure, and the functional group may undergo transformation
with sometimes only minor changes in the total structure of the
molecule.
     The individual processes that chemicals may undergo can then be
classified and evaluated according to specific physical properties or
the reactive functional groups that these chemicals may have in
common.  The basis for the empirical correlations between KQW and Sw is
discussed in Section 4.  These constants describe equilibrium processes
for the chemical between water and a second (organic) phase.  Similarly,
the volatilization of a chemical can be evaluated in terms of Henry's
constants, which are functions of vapor pressure and water solubility.
     The reactivity of a chemical can be classified according to select
functional groups in the molecular structure.  For evaluations of
hydrolysis reactions, chemicals are classified as carboxylic acid esters
(-C02R), carboxylic acid amides (-CONH2), alkyl halides (R-X), and
phosphoric acid esters ((RO^PO), to name only a few.  Data for
hydrolysis of a chamical can often be estimated by analogy to another
chemical with a similar functional group or calculated by more formal

-------
procedures using linear  free-energy relationships such as the Taft
equation, the Hammett equation, or other such correlations (Mill, 1979;
Wolfe et al., 1978 and 1980).
     Chemical oxidation  rate constants can be calculated by evaluating
the reaction of an oxidant at a particular type of carbon-hydrogen bond
(i.e., hydrogen abstraction process) or at an olefinic bond.  No SAR or
correlation method is available for predicting a direct photolysis rate
constant except by analogy to other chemicals, which is often unreliable
because of the complex chemistry of photoexcited states.
     For this report, data obtained from calculations involving theory,
SARs, or empirical correlations have been clearly identified so that the
user can recognize the source of such data and can recalculate data
using current or improved procedures.
     The following briefly describes the environmental processes and the
process data important in aquatic fate assessments.  The process data
are discussed in the order that they appear on the data sheets.  The
sources of the process data are also discussed.
CHEMICAL NAME, CHEMICAL  ABSTRACTS SERVICE REGISTRY NUMBER, AND MOLECULAR
WEIGHT
     The names of the chemicals used on the data sheets are those as
given on the original EPA list.  The Chemical Abstracts Service (CAS)
number has been obtained mainly from the original EPA list.  Handbooks,
catalogs, or the CAS were used when necessary.  The molecular weight
(MW) has been calculated from the molecular formula.  Although the MW is
not used for environmental assessments, it is required for conversion of
units from ppm to molar  units (M).  The MW has also been used to
calculate the molecular  weight/oxygen ratio.
WATER SOLUBILITY
     Water solubility (Sw) data are required for calculating Henry's
constant and for calculating other partition coefficients using the
correlation equations discussed in Section 4.  Values of Sw (ppm or
mg L-1) were calculated from KQW using a correlation equation developed
by Yalkowsky and Valvani (1980).

                                  10

-------
     For organic pollutants that are liquid in their pure state at 25°C

                 log Sw - -1.08 log Kow + 3.70 + log MW          (2.1)

where MW is the molecular weight of the pollutant (g mole"1).  For
organic pollutants that are solid in their pure state at 25°C

                                                  ASF
        log Sw = -1.08 log Kow + 3.70 + log MW - (13^)(mp - 25) (2.2)

where mp is the melting point of the pollutant (°C) and ASp is the
entropy of fusion of the pollutat
known, it may be approximated by
entropy of fusion of the pollutant (cal mol'^deg"1).  If ASj. is not
                        ASF ~ 13.6 + 2.5  (n - 5)                  (2.3)
where n is the number of flexible atoms (i.e., atoms not involved in
double bonds, triple bonds, or part of a ring structure) in the
pollutant molecule, other than hydrogen.   If n is less than 5, n - 5 is
set equal to zero.
     For solids that had no literature melting points available, Sw was
calculated using the equation for liquids.  This results in a maximum Sw
and should be used only for a screening risk assessment.
MELTING AND BOILING POINT
     These data are not used directly in aquatic fate assessments, but
they show in which phase (gas, liquid, solid) the pure chemical is found
under environmental conditions.  Boiling point data are cited for 760
torr (1 atmosphere) unless otherwise noted.  The melting point should be
used in the calculation of water solubility from octanol/water partition
coefficient (KQW) data for compounds that are solids above 25°C.
VAPOR PRESSURE
     The vapor pressure Py (torr) of an organic chemical is, in itself,
a qualitative or relative measure of the volatility of the chemical in
                                   11

-------
its pure state and  can  be used to calculate the Henry's constant used in
volatilization rate constant calculations.  Unless otherwise specified,
the PV values listed are at 25°C.
     Vapor pressure data not found in the literature were calculated
using procedures described by Grain (1982).  The method uses a
modification of the Watson correlation to express the temperature
dependence of AH  such  that

                       AHv "   AHvb [3  "  2
-------
coefficients (see Section 4).  The calculation of KQW from structural
features of the molecule is also discussed in Section 4.
HYDROLYSIS RATE CONSTANTS
     Hydrolysis refers to reaction of a. chemical with water, usually
resulting in the introduction of a hydroxyl function into a molecule and
loss of a leaving group -X:
                      R-X + H20         '  ROH + HX               (2.5)
The hydrolyses of some classes of compounds are catalyzed by acid or
base, and therefore the hydrolysis rates of these chemicals in the
environment can be pH dependent.   The subject of hydrolysis in aquatic
systems has been reviewed in detail by Mill et al. (1982), and an
extensive compilation of hydrolysis data was published in a review by
Mabey and Mill (1978).
     The rate of hydrolysis of a compound at a specific pH value is
given by the equation
                 RH " khtC]  -  (kA[H] + kN + kB[OH-])[C]          (2.6)
where k^ is the first-order rate constant for hydrolysis at the pH, kA
and kg are second-order rate constants for acid- and base-promoted
hydrolyses respectively, and kN is the first-order rate constant for the
pH-independent , neutral hydrolysis process.  Using the autoprotolysis
equilibrium expression
                             [H+][OH-] - K,,                      (2.7)
equation (2.6) can be rewritten as
                        kL  = k [H+] + k^ + -2J1                 (2.8)
                          HA       M   [Jf]
Equation (2.8) shows that kh will depend on the pH of the aquatic system
and on the relative values of k^, kg, and kN.  At present, no reliable
information shows that hydrolysis rates in aquatic environments will be
catalyzed by species other than [H+] or  [OH~] .
                                   13

-------
     The  hydrolysis rate constants  kA,  kg,  and kN used to calculate kh
as a function  of  pH are described below along with the source codes for
calculating  or estimating the values  of the rate constants.
ACID-PROMOTED  HYDROLYSIS RATE CONSTANT
     The acid-promoted hydrolysis  rate  constant kA  (M"!*") is for the
acid-promoted hydrolysis of  a chemical.   In  regions where only kA
contributes  to  hydrolysis (i.e., kA[H+]  » kN =» kB[OH~]), kh will
decrease by  a factor of 10 for each  1-unit increase in pH.
BASE-PROMOTED HYDROLYSIS RATE CONSTANT.
     The base-?promoted hydrolysis  rate  constant kg  (M"1!!"1) is for the
base-promoted (OH~)  hydrolysis of  a  chemical.  In regions where only kg
contributes  to  hydrolysis, k^ will increase  by a factor of 10 for each
1-unit  increase in pH.
NEUTRAL-HYDROLYSIS RATE CONSTANT.
     The neutral-hydrolysis  rate constant kN (h'1)  is for the pH-
independent  hydrolysis of a  chemical.   Data  or sources pertaining to the
hydrolysis of the organic chemicals  have been entered in the data sheets
in several ways.   When a chemical  structure  had op jiydrolyzable
^functional groups, NHFG was  entered. When chemical hydrolysis occurs
only at extreme pH values or temperatures or with catalysts not
available in aquatic environments, HNES was  entered (hydrolysis opt
^nvironmentally jignificant) .  Other data for hydrolysis are referenced
or are  based on analogy to similar chemicals.
MICROBIAL DEGRADATION RATE CONSTANT
     Biotransformations  are  undoubtedly  important processes for
degradation of  chemicals in  aquatic  environments, resulting in
hydrolysis,  oxidation, and reduction of  the chemical structure to
ultimately  produce carbon dioxide  and water.  The complex factors
influencing the biotransformation  of a chemical  include pH, temperature,
dissolved oxygen,  available  nutrients, other organic chemicals
(synthetic  or naturally  occurring) that  may serve as cometabolites or
                                   14

-------
alternative energy sources, and the populations and types of organisms
capable of transforming the chemical.  For most assessments, the initial
biotransformation step is of prime importance (i.e., removal of the
specific chemical from the environment).  However, the biotransformation
process is still too complex to be used to reliably predict a
biotransformation rate constant using theoretical approaches such as
those available for chemical and physical processes.
     Maki et al. (1980) recently reviewed some of the aspects of the
measurement of biotransformation rates and the use of such data.  The
rates of biotransformation are complex functions of chemical concen-
tration and microbial biomass.  However, at the typical concentrations
of a chemical in the environment (< 1 ppm), the rates may be expected to
follow second-order kinetics because they are first order in chemical
kinetics and first order in biomass kinetics.  Furthermore, the
microorganism growth due to consumption of the chemical may not be
significant; therefore, the rates of biotransformation are pseudo-first-
order as a function of the chemical concentration.
     The biotransformation data given in this report were estimated for
the approach described by Baughman et al. (1980), in which the rate of
biotransformation of a chemical, RB, is given by the expression
where kj, is a second-order rate constant for biotransformation of a
chemical by bacteria of population [B] in the solution phase of the
water column.  When kb is given in mL cell"1 h"1, the units of [B] are
in cell mL  •  Because data for k^ were not available for most chemicals
covered by this report, the rate constants were estimated solely for use
in aquatic fate modeling by EPA.  These data were estimated using on
relative rates of biodegradation of the chemicals as reported in
literature, structural analogies, and judgment of SRI staff with
expertise in biotransformation studies.  These data have been estimated
and appropriate caution should be exercised in the use of the data.
                                  15

-------
PHOTOLYSIS RATE CONSTANT
     The direct photolysis rate constants kp (h~^) for most of the
chemicals cannot be estimated because of insufficient spectral and
quantum yield data.  For chemicals where no light absorption occurs
above the solar cutoff  (300 nm), the rate constant can be considered as
zero, and therefore photolysis is not environmentally ^relevant (NER).
     In cases where the chemical is expected to photolyze in the
environment but no data are available, no value is entered. Similarly,
no value is entered if nothing is known about a chemical's photolytic
reactivity.  No data for indirect photolysis of chemicals is provided in
this report except that which results from oxidation processes (see next
section).
OXIDATION RATE CONSTANTS
     Chemical oxidation of organic chemicals in aquatic environments may
be caused by several different oxidants, among which are singlet oxygen
(102), alkyl peroxyl radical (R02«), alkoxy radical (R0»), or hydroxyl
radical («OH).  The source of these oxidants is primarily photochemical,
but because the oxidants react with chemicals in their ground state, and
oxidation therefore does not involve the photochemistry of the chemical
itself, oxidations are reasonably considered as discrete processes apart
from photochemistry.  Each oxidant has a unique reactivity toward
organic moieties, and the relative and absolute concentrations of these
oxidants will vary with environmental parameters, such as concentration
and origin of humic-fulvic materials and sunlight intensity.
     Literature information classifies reported data on oxidation of
organic chemicals by oxy radicals such as RO-* and ^02.  The laboratory
study conducted by Mill et al. (1982) using natural waters indicates
                                            -9
that R02* radical concentrations of ~ 1 x 10   M may be present in the
surface waters of sunlit water bodies.  Oxidation reactions initiated
by RO-» include the following:
                                   16

-------
                     R02«  + -C-H 	- R02H H- -O              (2.10)

                     R02»  +  C=C 	•- R02-C-O                (2.11)

                     R02»  + ArOH 	»• R02H + ArO«             (2.12)

                     R02- + ArNH2	 R02H + ArNH            (2.13)

Of these reactions, the last two are quite rapid in aquatic environments

(cl/2 < several days), whereas the others are slower and usually will
not be important for most chemicals.

     Zepp et al. (1978) have shown that  ^02 can be formed at
        —1 7
" 1 x 10 *•*• M concentrations in sunlit natural waters.  The most

important reactions for ^2 with organic chemicals are those involving
reaction with olefinic moieties (Ranby and Rabek, 1978).
G-C=CH

OOH
I  I/CH2-
C-C               » products
I  I
0-0
                                                                 (2.14)
Some rate constants for  Q£ and R0»» are listed in a review by Mill
(1980).

     The rate of loss of organic chemicals RQX by oxidation is
      ROX ~ kRO .fR02*][C] + kl  1()2
               2               02
where k/jy and [OX] are the rate constants and concentration values for
other unspecified oxidants.  Only data for the second-order rate

constants k__   and k.   have been estimated for this report.  When two
           ™2*      102
rate constants are given on the data sheets, the second-order rate

constants should be multiplied by their respective oxidant concentra-
tions to determine which of the first-order rate constant values is

larger, and that rate constant should be used for an assessment.
                                   17

-------
     Apart from a direct measurement of a rate constant at a specific
temperature (which is rare), most rate constants in this report were
obtained either from extrapolation of a rate constant for the organic
chemical measured at another temperature or from a correlation of
structure with reactivity as discussed below.
RATE CONSTANT FOR OXIDATION BY ALKYL PEROXYL RADICAL
     Because many chemicals on the list of chemicals of concern have
several kinds of reactive centers for oxidation by R02«, the overall
rate constant k_Q   (M~^h~^)was obtained by first calculating the
individual rate constants for each reactive site and then summing these
rate constants.  For example, acrolein has two reactive sites:  (1)
addition to the double bond and (2) H-atom transfer from the carbonyl
k
"RO. = ki +


(2.17)
(2.18)
When one oxidation process was found to be fast, the important oxidant
was listed and the other reactions were ignored.  When there were more
than one -CH bond of a given kind, the rate constant was multiplied by
the number of similar -CH bonds to give the correct total rate constant
for oxidation of that CH-bond.
     Two procedures were used to calculate individual k0X values
for RO • reactions.  In the first, when a structure was analogous to
another chemical structure with a measured rate constant at a similar
temperature, the measured rate constant was used directly (Hendry et
al., 1974).  (The -CHO bond in acrolein is an example.)  The second
procedure, used most often, is based on SARS established by Howard and
coworkers for H-atom transfer (Korcek et al., 1972) and addition to
double bonds (Howard, 1972), as shown below.
     For the H-atom transfer reaction
                     log k_n  - 18.96 - 0.2[D(R-H)]              (2.19)
                          R0
                                  18

-------
where D(R-H) is the bond dissociation energy of the CH-bond.
     For the R02 addition to double bonds
                  log kRQ  =  [16.54 - 0.2D(XCR2-H)]/0.75          (2.20)
where D(XCR2~H) is the bond dissociation energy of a species that gives
the radical formed by R02 addition and where R02 is assumed to have the
same effect as methyl (Me) on D(C-H).   Thus for oxidation of vinyl
chloride
             \
      R°2* + /C=C\   	-R02C-C»                           (2.21)
the closest analog would be MeCH2CHCl, and the value of D(MeCH2CHCl-H)
would be used in equation (2.20).  Bond dissociation energies were taken
from Furuyama et al. (1969).
RATE CONSTANT FOR OXIDATION BY SINGLET OXYGEN
     Only a few of the chemicals tabulated in this report are reactive
toward  02; these include some polycyclic aromatic and a few olefinic
double bond or diene systems.  All reactive chemicals were assigned rate
constants by analogy with similar structures that have shown rate
constants for reaction with singlet oxygen.  For cyclic olefins, the
values of Matsuura et al. (1973) were used.  For alicyclic olefins and
other structures, the rate data summarized by Gollnick (1978) were used.
                                 19

-------
                               REFERENCES

Baughman, G. L. , D. L. Paris,  and W. C.  Steen.  1980.  Quantitative
     Expression of Biotransformation Rate.   In:  Biotransformation and
     Fate of Chemicals in Aquatic Environments.  A. W. Maki, K. L. Dickson,
     and J. Cairns, Jr., Eds.  American  Society for Microbiology, Washing-
     ton, DC.
Furuyama, S. , D. M. Golden, and  S. W. Benson.  1969.  J. Am. Chem. Soc.
     JJ1, 7564-7569.

GSllnick, K.  1978.   In: Singlet Oxygen.  B. Ranby and J. F. Rabek, Eds.
     John Wiley and Sons, New  York.

Grain, C.  1982.  Vapor Pressure.  In: Handbook of Chemical Property
     Estimation Methods.  W. J.  Lyman, W. F. Reehl, D. H. Rosenblatt,
     Eds.  McGraw-Hill Book Company, New York.

Hansch, C., and A. Leo.  1979.   Substituent  Constants for Correlation
     Analysis in Chemistry and Biology.  Wiley-Interscience. New York.

Hendry, D. G. , T. Mill, L. Piszkiewicz,  J. A. Howard, and H. K. Eigenmann.
     1974.  J. Phys.  Chem. Ref.  Data.  3_, 937-978.

Howard, J. A.  1972.  Adv. Free  Radical  Chem. b_, 49-174.

Kenaga, E. E., and C. A. I. Goring.  1978.   Relationship Between Water
     Solubility, Soil-Sorption,  Octanol/Water Partitioning, and Bio-
     concenttation of Chemicals  in Biota.  In: Aquatic Toxicology, ASTM
     STP 707, J. G. Eaton, P.  R. Parrish, and A. C. Hendricks, Eds.
     American Society for Testing and Materials, Philadelphia, PA.'

Korcek, S., J. H. B.  Chenier,  J. A. Howard,  and K. U. Ingold.  1972.
     Can. J. Chem. 50, 2285-2297.

Matey, W. R. , and T.  Mill.  1978.  J. Phys.  Chem. Ref. Data. _7, No. 2,
     383-415.

Mabey, W. R. , T. Mill, and R.  T. Podoll.  1983.  Estimation Methods for
     Process Constants and Properties Used in Fate Assessments.  Final
     Report for Work  Assignment  No. 5 in partial fulfillment of EPA
     Contract No. 68-03-2981,  U.S. EPA,  Athens, GA.

Maki, A. W. , K. L. Diickson, and  J. Cairns, Jr., Eds.  1980.  Bio trans-
     formation and Fate of Chemicals in  Aquatic Environments.  American
     Society for Microbiology, Washington, DC.

Matsuura, T., A. Horinaka, and R. Nakashima.  1973.  Chem. Lett. 887-890.

Mill, T.  1979.  Structure Reactivity Correlations for Environmental
     Reactions.  EPA-560/11-79-012.  U'.S;' EPA, Washington, DC.
                                    20

-------
                               REFERENCES

Mill, T.  1980.  Photooxidation in the Environment.  In:  The Handbook
     of Environmental Chemistry, Vol. 2, Part A.  0. Hutzinger,  Ed.
     Springer-Verlag, New York.

Mill, T., W. R. Mabey, and D. G. Hendry.  1982.  Hydrolysis  in Water.
     In:  Laboratory Protocols for Evaluating the Fate of Organic
     Chemicals in Air and Water.  EPA-600/3-82-022.  U.S. EPA, Washington.

Ranby, B., and J. F. Rabek, Eds.  1978.  Singlet Oxygen.  John Wiley and
     Sons, New York.

Wolfe, N. L., L. A. Burns, and W. C. Steen.  1980.  Chemosphere. 9_,
     393-402.

Wolfe, N. L., R. G. Zepp, and D. F. Paris.   1978.  Water Res. 1.2,  561-563.

Yalkowsky, S. H., and S. C. Valvani.  1980.  J. Pharm. Sci.  69,  No.  8,
     912-922.

Zepp, R. G., N. L. Wolfe, G. L. Baughman, and R. C. Hollis.  1978.   Nature.
     267, 421-423.
                                   21

-------
                               SECTION 3
                 DATA SHEETS FOR CHEMICALS OF INTEREST
This section contains a list of data sheets showing the Chemical Abstract
Services registry number and compound name, a list of source codes for the
data sheets, and the data sheets and references for this work assignment.
                                   22

-------
                          LIST OF DATA  SHEETS
              CAS
Number   Registry Number

   1        102-36-6
   2        102-82-9
   3        314-40-9
   4        330-55-2
   5        624-92-0
                     Compound Name
6
7
8
9
10
11
12
13
14
15
16
17
18
19
110-81-6
30453-31-7
68-85-0
93-58-3
99-04-7
99-94-3
619-21-6
619-66-9
88-99-3
100-21-0
120-61-6
1679-64-7
121-91-5
528-44-9
  20
2303-16-4
3,4-Dichlorophenylisocyanate
Tributylamine
Bromacil
Linuron
Dimethyldisulfide
(2,3-Dithiabutane)

Diethyldlsulfi.de
(3,4-Dlthlahexane)
Ethylpropyldlsulfide
(3,4-Dithiaheptane)
Benzole acid
Methylbenzoate
3-Methylbenzoic acid

4-Methylbenzoate
3-Formylbenzoic acid
4-Formylbenzoic acid
Phthalic acid
Terephthalic acid

Dimethylterephthalate
Methylterephthalate
Isophthalic acid
Trimellitic acid
(1,2,4-Bemzenetricarboxylic acid)
Diallate
  21
  22
  23
  24
  25
2303-17-5
12427-38-2
1134-23-2
1929-77-7
1114-71-2
Triallate
Maneb
Cycloate
Vernolate
Pebulate
  26
  27
  28
  29
  30
2212-67-1      Molinate
2008-41-5      Butylate
1563-66-2      Carbofuran
63-25-2        Carbaryl
39076-02-3     sec-Butylcarbamic acid, methyl ester
                                   23

-------
                     LIST OF DATA SHEETS (continued)
              CAS
Number   Registry Number

  31        148-18-5
  32        8018-01-7
  33        12122-67-7
  34        759-94-4
  35        623-80-3

  36        529-34-0

  37        447-53-0
  38        447-53-0
  39        119-64-2

  40        825-51-4

  41        90-15-3
  42        135-19-3
  43        104-90-5
  44        1696-17-9
  45        96-45-7
                            Compound Name
46
47
48
49
50
51
52
1563-38-8
289-16-7
57-14-7
540-73-8
593-60-2
106-93-4
30496-13-0
  53
  54
  55

  56
  57
  58
  59
  60

  61
  62
  63
  64
  65
108-86-1
583-53-9
106-37-6

608-21-9
626-39-1
22311-25-7
634-89-9
608-90-2

87-82-1
608-33-3
615-56-5
615-58-7
626-41-5
Dithiocarbamate
Mancozeb
Zineb
EPTC
Carbamodithioic acid, S,S-diethyl ester

3,4-Dihydro-l(2H)-naphthalenone
(cr-Tetralone)
3,4-Dihydronaphthalene
1,2-Dihydronaphthalene
1,2,3,4-Tetrahydronaphthalene
(Tetralin)
Decahydronaphthol-2

1-Naphthol
2-Naphthol
2-Methyl-5-ethylpyridine
N,N-Diethylbenzamide
2-Imidazolidinethione
(Ethylenethiourea)

2,3-Dihydro-2,2-dimethyl-7-benzofuranol
1,2,4-Trithiolane
1,1-Dimethylhydrazine
1,2-Dimethylhydrazine
Bromoethene

1,2-dibromoethane
Tetrabromobisphenol A
(1,1,3,3-Tetrabromo-2,2-bis(4-
 phenolyl)propane)
Bromobenzene
1,2-Dibromobenzene
1,4-Dibromobenzene

1,2,3-Tribromobenzene
1,3,5-Tribromobenzene
1,2,3,4-Tetrabromobenzene
1,2,3,5-Tetrabromobenzene
Pentabromobenzene

Hexabromobenzene
2,6-Dibromophenol
3,4-Dibromophenol
2,4-Dibromophenol
3,5-Dibromophenol
                                   24

-------
                    LIST  OF  DATA  SHEETS  (continued)

              CAS
Number   Registry Number   	Compound Name	

  66        28165-52-8     2,5-Dibromophenol
  67        28514-45-6     Dibromophenol
  68        57383-80-9     2,3-Dlbromophenol
  69        1163-19-5      Decabromobiphenyl ether
  70        32536-52-0     Octabromobiphenyl ether

  71        598-94-7       N,N-Dimethylurea
  72        689-11-2       sec-Butylurea
  73        869-79-4       Di-sec-butylurea
  74        4128-34-7      Di-isopropylurea
                                  25

-------
                              LIST OF SOURCE CODES

Calc               Molecular weight/oxygen ratio was calculated directly.

CC-Kow             Value of the octanol/water partition coefficient  (K)  was
                   obtained by computer calculation using FRAGMENT calculation
                   procedure (see Section 4.4).

C-OX               Oxidation rate constants were calculated,  using functional
                   group reactivity toward alkyl peroxyl radical (R02) and
                   singlet  oxygen (SO).

C-Sw f Kow         The  water solubility (Sw) was calculated from the
                   octanol/water partition coefficient (Kpw)  usin8 tne
                   equation of Yalkowsky and Valvani (1980);  the calculation
                   of Sw values is discussed in  Section 2.

C-vp f bp          Vapor pressure (vp)  was calculated from the boiling point
                   (bp) using the method discussed by Grain (1982);  the method
                   is discussed in Section 2.

E-A-Carbaryl       Estimated by analogy to Carbaryl; hydrolysis data for
                   Carbaryl from Mabey  and Mill  (1978).

E-A-Dibromopropane Estimate by analogy  to dibromopropane; hydrolysis data  for
                   dibromopropane from  Vogel (1983).

E-A-MeBz           Estimate by analogy  to methyl benzoate; hydrolysis data for
                   methyl benzoate from Mabey and  Mill (1978).

E-A-TDI            Estimated by analogy to toluene diisocyanate; hydrolysis
                   data for toluene diisocyanate from Sopach and Boltromeyuk
                   (1974).

E-KB               Estimate of biotransformation rate constant (k^)  is based
                   on relative rates of transformation reported in literature
                   or on structure-reactivity analogies.

HNES               Hydrolysis is not environmentally significant. Chemical
                   hydrolysis occurs only at extreme pHs or temperatures or
                   with catalysts not available  in aquatic environments.

INERT              Oxidation reactions  at ambient  oxygen levels have half-life
                   greater  than 2 years and are  therefore considered
                   unimportant fate processes.
                                      26

-------
M-OX



NHFG

partial
PNER

R02

SO

VF-NBD
Oxidation rate constants were modelled using functional
group reactivity toward alkyl peroxyl radical (R02) and
singlet oxygen (SO).

No hydrolyzable functional groups in molecule.

Partial notation indicates that the computer calculated
octanol/water partition coefficient has not accounted for
each functional moiety of the molecule.  This occurs when  a
substituent fragment is not represented in the data base or
when there are possible hydrogen bonding interactions.

Photolysis is not environmentally relevant.

Alkyl peroxyl radical, R02.

Singlet oxygen,  02

Volatilization is too fast for biotransformatlon  studies to
be conducted.  No biotransformation data are therefore
available.
                                     27

-------
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                                   N=C=0
Compound Name:    3.4-dichlorophenylisocyanate
CAS Registry Number;  102-36-6
.Molecular Weight(g):
188
Parameters:
Water Solubility  (ppm)
Boiling Point  (°C)
Vapor Pressure  (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (MT^hr""1)
                  Reference
Acid Hydrolysis Rate
Constant  (M  hr""1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml  cell  hr~  )
Photolysis Rate  Constant (hr~l)
Oxidation Rate  Constant (M  hr~  )
260
161.9/100 torr
2.82 x 10"1
5.88
3.30 (partial)


3 x 10~5
1 x 10-10

INERT
C-Sw f Kow
Boublik. et al. (1973)
Dean (1979)
Calc
CC-Kow


E-A-TDI
E-KB

M-OX R02, ..SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                    28

-------
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                         CH2CH2CH2CH3
                          I
                         N
                                                    CH3CH2CH2CH2
Compound Name:   tributylamine
CAS Registry Number; 102-82-9
.Molecular Weight(g):
185.4
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant
Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant (ml cell  hr~ )
Photolysis Rate Constant (hr"1)
Oxidation Rate Constant '(M  hr~ )
                  Reference
31
71 fi-717
0.29
5.79
4.15
NHFG
NHFG
NHFG
3 x ID'12
PNER
INERT
C-Sw f Row
Merck (1976)
C-vp f bp
Calc
CC-Kow



E-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA,  and should not be used in more detailed assessments.
                                   29

-------
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
Compound Name:    Bromacil
CAS Registry Number;  314-40-9
                                                                CH,
.Molecular Weight(g):
261.11
Parameters;

Water Solubility  (ppm)
Melting Point  (°C)

Boiling Point  (°C)


Vapor Pressure  (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)


Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant  (hr~ )
Microbial Degradation
Rate Constant  (ml  cell  hr~  )
Photolysis Rate Constant  (hr~l)
Oxidation Rate  Constant  (M-1hr~  )
                  Reference
815
157.5-160
sublimes

8.16
1.32 (partial)



3 x lO'12

INERT
Spencer (1973)
Merck (1976)
Spencer (1973)

Calc
CC-Kow



E-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment to  be
 conducted by the EPA, and should not be used in more detailed assessments.
                                   30

-------
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                             CH3

                       N-C-N-OCH,
                       H  II        3
                          O
Compound Name:   Linuron
CAS Registry Number; 330-55-2
.Molecular Weight(g):
249.11
Parameters;

Water Solubility (ppm)

Melting Point  (°C)
Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
Acid Hydrolysis Rate
Constant (M'-Tir"1)
Neutral Hydrolysis Rate
Constant (hr  )
Microbial Degradation      -
Rate Constant (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M~1hr~ )
                  Reference
75
93-94

1.1 x 10~2/24°C
7.78
1.17 (partial)
HNES
HNES
HNES
1 x lO'10

INERT
Spencer (1973)
Merck (1976)

Spencer (1973)..
Calc
CC-Kow
Aly (1976)
Aly (1976)
Aly (1976)
E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                 31

-------
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
CH,-S-S-CH3
Compound Name:    dimethyldisulfide
CAS Reeistrv Number: 624-92-0 Molecular Weight(g): 94 2Q
Parameters: Reference ,
Water Solubilitv (Dt>m) 5.2 x 10
Soiling Point (°C) 112-118
Vapor Pressure (torr) 28,69
Molecular Weight/Oxygen 2.94
Log (Octanol/Water Partition
Coefficient) -0.04
Alkaline Hydrolysis Rate
Constant (M^hr'1) NHFG
Acid Hydrolysis Rate
rn.,L., t-a.n- CM"-"-!,^-!^ 	 ^\*f_y
Neutral Hydrolysis Rate
Constant (hr~ ) NHFG
Microbial Degradation - _g
RatP Hnnstant (ml cell~1hr~i>) 3 X 10
PNFTR
Oxidation Rate Constant (M'^r"1) INERT
C-Sw f Row
Verschueren (1977)
Osborn and Douslin (1966)
Calc
CC-Kow



E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  32

-------
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                       C2H5-S-S- C2H5
Compound Name:   diethyldisulfide   (.3,4-dithiahexanel

CAS Registry Number; HO-81-6	Molecular WeightCg):
                                                                  122.25
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M^hr"1)
Acid Hydrolysis Rate
Constant (M~ hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant (ml
                                                       Reference
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant
&_fi v irr
154
4.28
3.82
1.04
NHFG
NHFG
NHFG
3 x 10~9
PNER
INERT
C-Sw f Kow
Weast (1973)
Dreisbach (1961)
Calc
CC-Kow


•
E-KB

M-OX R02, SO
 These .data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                 33

-------
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
C2H5-S -S-C3H7
Compound Name:    ethylpropyldisulfide  (3,4-dithiaheptane)
CAS Registry Number: 30453-31-7 Molecular WeiehtCe): 136.27
Parameters;
Water Solubility (ppm) 1,3 x 104
Boiline Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen 4. 26
Log (Octanol/Water Partition
Coefficient) 1.58
Alkaline Hydrolysis Rate
Constant (M^hr"1) NHFG
Acid Hydrolysis Rate
rj_ ,,,.,.,,,.,. fM"~li1T--l\ 	 	 NHiG
Constant {M. nr J~)
Neutral Hydrolysis Rate
Constant (hr ) NHFG
Microbial Degradation _9
Rat-* Honstant (ml cell~1hr~-L) , 3 x 10
p-i. — 4.-T .-_ j r. Rife- rnTTSf-nnf ThT"^-^ rlNJiK
Oxidation Rate 'Constant (M^hr" ) INERT
Reference
C-Sw f Kow


Calc
CC-Kow



E-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                   34

-------
                                                           COOH
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
Compound Name:   benzole acid
CAS Registry Number; 68-85-0
.Molecular Weight(g):
JL22.12
Parameters;

Water Solubility (ppm)
Melting Point C"C)

Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M^hr'1)
                  Reference
Acid Hydrolysis Rate
Constant (M  hr""1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation _    .
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M~ hr~ )
T/inn
12? A
?£Q 9
i _?fi v in"3
3.82
1.87
NHFG
NHFG
NHFG
1 x 10~7
PNER
INERT
Merck riQ7fi>
Mo-rnV fTQ7^
Merck fl976")
Wiedemann fl Q7?"i
Calc
CC-Kow



E-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  35

-------
                                                          COOCH,
                      EPA CONTRACT 68-03-2981
                      WORK ASSIGNMENT NO. 15
CAS Registry Number: 93-58-3 Molecular Weight(g): 135 16
Parameters: Reference
Water Solubility (onm) 2600
Boiling Point (°C) 199.6
Vapor Pressure (torr) 0.3944
Molecular Weight/Oxygen 4.26
Log (Octanol/Water Partition
Coefficient) 2.24
Alkaline Hydrolysis Rate
Constant (M~1hr~1) 7
Acid Hydrolysis Rate , „ -Ln-3
,-,.,_,,.,.,.. rM~lii-r-l''i 	 .
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation _ _j
Rat-* flnnstant (ml cell~1hr~i) . 1 X 10
PVirt^rt 1 ire"i c Paf"a P^rnctrmt" TViT*" ^-^ rNKR
Oxidation Rate Constant (M~ hr" ) INERT
C-Sw f Kow
Weast (1973)
Dreisbach (1955)
Calc
CC-Kow
Mabey and Mill (1978)
Mabey and Mill (1978)
•
E-KB

M-OX R02, SO
These data were estimated for use in a preliminary assessment to be
conducted by the EPA, and should not be used in more detailed assessments.
                                 36

-------
                                                                             10
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                          COOH
                                                             CH,
Compound Name:   3-methylbenzoic acid
CAS Registry Number: 99-04-7
.Molecular Weight(g):
136.16
Parameters;

Water Solubility (ppm)

Melting Point (°C).
Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant
Oxidation Rate Constant  (M  hr~ )
                  Reference
180
ina_7s
263
9.6 x 10~4
4.26
2.54
NHFG
NHFG
NHFG
1 x 10~?
PNER
TNF.T3T
C-Sw f Kow
Verschueren (197.7)
Vo-ron'hiieT-on f!Q77^
C-vp f bo
Calc
CC-Kow



E-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  37

-------
                                                                            11
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                         COOCH,
Compound Name:   4-methylbenzoate
CAS Registry Number:  99-94-3
.Molecular Weight(g):
150
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M^hr"1)
                  Reference
Acid Hydrolysis Rate
Constant  (M  hr""1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation       .
Rate Constant  (ml cell  hr~  )
Photolysis Rate Constant  (hr'1)
Oxidation Rate Constant  (M  hr~  )
550

4.56 -x 10"1
4.69
2.90
1 x 10~3
7

1 x 10~7
PNER
INERT
C-Sw f Kow

Weast (1973)
Calc
CC-Kow
E-A-MeBz
E-A-MeBz

E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to  be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  38

-------
                                                                           12
COOH
EPA CONTRACT 68-03-2981 f()l
WORK ASSIGNMENT NO. 15 X^-k
CHO
Compound Name: 3-formylbenzoic acid
CAS Resistry Number: 619-21-6 Molecular Weight(g): ISO. 14
Parameters;
Water Solubilitv (ppm) 1100
Meltine Point (°C) 175
Boiline Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen 4.69
Log (Octanol/Water Partition
Coefficient) 1.23
Alkaline Hydrolysis Rate
Constant (M^hr'1) NHFG
Acid Hydrolysis Rate NHFG
Constant ^M nr •*)
Neutral Hydrolysis Rate
Constant (hr~X) . NHFG
Microbial Degradation -7
Ral-o rrmsfant Cml eell"1hr~1') 1 X 10

Oxidation Rate Constant (M^hr"1) INERT
Reference
C-Sw f Kow
Weast (1973)


Calc
CC-Kow



E-KB
-
M-OX R02, SO
These data were estimated for use in a preliminary assessment to be
conducted by the EPA, and should not be used in more detailed assessments.
                                 39

-------
                                                                            13
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
Compound Name:   4-formylbenzoic acid
CAS Registry Number;  619-66-9
                                                          COOH
                                                          CHO
.Molecular Weight (g):
150.14
Parameters;

Water Solubility (ppm)

Melting Point  C°C)
Boiling Point  (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M-1hr~ )
                  Reference
170
256
sublimes
-
4.69
1.23
NHFG
NHFG
NHFG
1 x 10~7

INERT
C-Sw f Kow
Weast (1973)
Weast (1973)

Calc
CC-Kow



E-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more  detailed assessments.
                                  40

-------
                                                                            14
                                                         COOH
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                              OOH
Compound Name:    phthalic acid
CAS Registry Number;  88-99-3
.Molecular Weight(g):
166.13
Parameters;

Water Solubility (ppm)

Melting Point C°C)
Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M"1^"1)
                  Reference
Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant (M-1hr~ )
320
191 (decomposes)


5.19
1.62
NHFG
NHFG
NHFG
1 x 10~7
PNER
INERT
C-Sw f Row
Hawley (19J7)


Calc
CC-Kow



E-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA,  and should not be used in more detailed assessments.
                                  41

-------
                                                                            15
                                                         COOH
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO.  15
                                                         COOH
Compound Name:    terephthalic acid
CAS Registry Number;  100-21-0
.Molecular Weight(g):
166.13
Parameters:
Water Solubility  (ppm)
Boiling Point  (°C)
Vapor Pressure  (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
Acid Hydrolysis Rate
Constant  (M"1^'1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation       .
Rate Constant  (ml  cell  hr~  )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M  hr~ )
                  Reference
26
300 (sublimes)
n.l5/20°C
S.1Q
1.62
NHFG
NHFG
NHFG
1 x 10~?
PNER
INERT
C-Sw f Kow
Mprck (1976")
Weber et al . (1981}
C.a 1 r-
CC-Kow


-
E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment  to be
 conducted by the EPA, and should not be used in more detailed  assessments.
                                  42

-------
                                                                             16
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                          COOCH3
                                                          COOCHj
Compound Name:   dimethylterephthalate
CAS Registry Number; 120-61-6
jiolecular Weight(g):
194,19
Parameters;

Water Solubility (ppm)

Melting Point C°C)
Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant (ml cell  hr  )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M-1hr~ )
                  Reference
200
140
300 (sublimes)
7.0 x 10~5
6.07
2.34
7
1 x 10~3

1 x 10~?
PNER
INERT
C-Sw f Kow
Verschueren (1977).
Verschueren (197J1
C-VTJ f bp
Calc
CC-Kbw
E-A-MeBz
E-A-MeBz

E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA,  and should not be used in more detailed assessments.
                                  43

-------
                                                                            17
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
Compound Name:    methylterephthalate
CAS Registry Number;  1679-64-7	Molecular Weight(g):
           180.19
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation _
Rate Constant  (ml cell  hr~  )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M-1hr~ )
Reference
6600


5.63
1.98
7
1 x 10~3

1 x 10~7
PNER
INERT
C-Sw f Row


Calc
CC-Kow
E-A-MeBz
E-A-MeBz

E-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment  to  be
 conducted by the EPA, and should not be used in more detailed  assessments.
                                  44

-------
                                                                             18
                                                        COOH
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                            COOH
Compound Name:   isophthalic acid
CAS Registry Number; 121-91-5
.Molecular Weight(g):
166.13
Parameters;

Water Solubility (ppm)
Melting Point (°C)

Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M-1hr~ )
                  Reference
130
345-348
sublimes

5.19
1.62
NHFG
NHFG
NHFG
1 x 10~7
PNTTR
INERT
Verschueren (1977)
Merck (1976)
Merck (1976)..

Calc
CC-Kow



E-KB

M-OX, R02. SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  45

-------
                                                                            19
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
Compound Name:    trimellitic acid  (1,2,4-benzenetricarboxylic  acid)

CAS Registry Number;  528-44-9	Molecular Weight(g):  	210.14
Parameters;

Water Solubility  (ppm)
Melting  Point (°C)

Melting Point (°C)


Vapor Pressure  (torr)


Molecular Weight/Oxygen
Log  (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
Acid Hydrolysis Rate
Constant  (M   hr"1)
Neutral Hydrolysis  Rate
Constant  (hr~  )
Microbial  Degradation      .
Rate Constant (ml cell  hr~ )
Photolysis  Rate Constant (hr"1)
 Oxidation Rate Constant (M-1hr~  )
Reference
400
218-220
238 (decomposes)

6.57
1.37
NHFG
NHFG
NHFG
3 x 10~9

INERT
C-Sw f Kow
Merck (19.76)
Weast (1973)

Calc
CC-Kow



E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                   46

-------
                                                                            20
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
,  ,  ^
(CHlCH
                              H
                              C
                              H
                                                                          Cl
Compound Name:   pjallate
CAS Registry Number; 2303-16-4
.Molecular Weight(g):
             .'273. S
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M~ hr  )
                  Reference
14
150/9 torr
6.8 x 10"3
8.55
0.73 (partial)



3 x 10~9

INERT
Snencer (1973)
Merck (1976)
C-vp f bp
Calc
CC-Kow


•
E-KB

M-OX RO7, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  47

-------
                                                                            21
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
               r   , -
               (CHJCH
                                                                   H

Compound Name:   Triallate
CAS Registry Number;  2303-17-5
.Molecular Weight(g):
305
Parameters;

Water Solubility  (ppm)

Melting Point  (°C)

Boiling Point  (°C)


Vapor Pressure  (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       ""
Acid Hydrolysis Rate
Constant  (M  hr""1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml  cell"  hr~  )
Photolysis Rate  Constant  (hr'1)
                  Reference
Oxidation Rate  Constant
                              "
4
29-in
148-149/9 torr
2.07 x 10~4
9.53
1.33 (partial)



3 x 10~9

INERT
Spencer (1973)

Spencer (1973) .
Grover et al. (1978)
Calc
CC-Kow



E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  48

-------
                                                                             22
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                      H2C-N-C-S
                                                                  X
H2C-N~C-S/
•     H  I
                                                                   Mn
Compound Name:   Maneb
CAS Registry Number; 12427-38-2	Molecular Weight(g):
            265.29
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
Acid Hydrolysis Rate
Constant  (M  hr""1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)


Oxidation Rate Constant  (M  hr~  )
 Reference

decomposes before
melting

8.29




3 x 10~9

INERT

Spencer (1973 X

Calc



•
E-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  49

-------
                                                                           23
                       EPA CONTRACT  68-03-2981
                       WORK ASSIGNMENT  NO.  15
/~\  >''
(    V-N-C-S-C2H5
Compound Name:	Cycloate	

CAS Registry Number; 1134-23-2	Molecular WeightCg):
              215.4
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant (hr~l)
Oxidation Rate Constant (M  hr  )
   Reference
75/20°C
146/10 torr
6.2 x 10~3
6.72
1.85



3 x 10~9

INERT
Snencer (1973)
Soencer (19.73)
Scencer (1973)
Calc
CC-Kow


-
E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  50

-------
                                                                             24
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15    CH3CH2CH2—S—C—
Compound Name:    Vernolate
CAS Registry Number; 1929-77-7	Molecular Weight(g):
           203.1
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (to'rr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr~l)
Oxidation Rate Constant  (M  hr~  )
Reference
90/20°C
140/20 torr
1.04 x 10~2
6.16
1.84



3 x 10~9

INERT
Spencer (1973)
Spencer (1973).
Spencer (1973)
Calc
CC-Kow


•
E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  51

-------
                                                                            25
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                            CH3CH2CH2-S-C-I<
                                                              >CH2CH2CH2CH3
Compound Name:   Pebulate
CAS Registry Number;  HI A-71-2
                                .Molecular Weight(g):
                                                203.36
Parameters:
Water Solubility  (ppm)
Boiling Point (°C)
Vapor Pressure  (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
                                                  Reference
Acid
Constant
Hydrolysis Ra
ant (M'-hir-1)
Rate
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml  cell   hr~  )
Photolysis Rate Constant  (hr"1)
Oxidation Rate  Constant

92/21°C
142/20. torr
3.5 x 10~2
3.3 x 10~2
6.36
1.84



3 x 10~9

INERT
Spencer (1973)
Merck (1976)
Ouellette and King (1977)
C-vp f bp
Calc
CC-Kow


•
E-KB

M-OX R02r SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  52

-------
                                                                             26
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                            C—SCHZCH3
Compound Name:    Molinate
CAS Registry Number; 2212-67-1
.Molecular WeightCg):
187.1
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant
Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M-1hr~ )
                  Reference
912/21°C
137/10 torr
5.6 x 10~3
1.9 x 10~2
5.84
0.90



3 x 10~9

INERT
Spencer (1973)
Spencer (1973)
Ouellette and King (1977)
C-vp f bp
Calc
CC-Kow



E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  53

-------
                                                                            27
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
              CH3CH2-S-C-NN
Compound Name:   Butvlate
CAS Registry Number: 2008-41-5
    CH3

 CH2CHCHj

 CHjCHCHj

    CH3
.Molecular WeightCg):
217.4
Parameters:

Water Solubility


Boiling Point  (°C)


Vapor Pressure  (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation       1
Rate Constant  (ml  cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M  hr~  )
                  Reference
36/20°C
138/21.5 torr
1.3 x 10~2
6.79
2.12



1 x ID'10

INERT
Snencer (1973)
Soencer (1973)
Spencer (19.73)
Calc
CC-Kow



E-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment to  be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  54

-------
                                                                             28
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
Compound Name:   Carbofuran
CAS Registry Number; 1563-66-2
.Molecular Weight(g):
221.3
Parameters;

Water Solubility (ppm)

Melting Point (°C)
Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr  )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M  hr~ )
                  Reference
7nn
150-153
-
<1.4 x 10~5
6.91
2.55
1638
5.04 x 10~4
2.5 x 10~3
3 x 10~9

INERT
Stjencer (1973 t
Merck (19761

Jaber et al. (1983)
Calc
CC-Kow
E-A-Carbaryl
E-A-Carbaryl
E-A-Carbaryl
E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                   55

-------
                                                                            29
                                                           II  H
                                                        0-C-N-CH
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
Compound Name:    Carbaryl
CAS Registry Number;  63-25-2
                                .Molecular Weight(g):
                                                201.2
Parameters;

Water Solubility  (ppm)
Melting Point  (°C).

Boiling Point  (°C)


Vapor Pressure  (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
                                                  Reference
Acid
Constant
Hydrolysis Ra
ant (M'-'-hr'1)
Rate
Neutral Hydrolysis Rate
Constant  (hr~ )
Microbial Degradation
Rate Constant  (ml  cell  hr~  )
Photolysis Rate  Constant  (hr~l)
Oxidation Rate  Constant (M  hr~  )
40/30°C
145

<6 x 10~6
6.28
2.50
1638
5 x 10~4
2.5 x 10~3
3 x 10~9

INERT
Spencer (1973)
Merck (19J6)

Jaber et al. C1983)
Calc
CC-Kow
Mabey and Mill (1978)
Mabey and Mill (1978)
Mabey and Mill (1978)
E-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  56

-------
                                                                            30
H
EPA CONTRACT 68-03-2981 CH3-C-NH-COOCH3
WORK ASSIGNMENT NO. 15 '
CH2CH3
Compound Name: sec-butylcarbamic acid, methyl ester
CAS Reeistrv Number: 39076-02-3 Molecular WeightCs): 131
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
2.1 x 104


4.09
Log (Octanol/Water Partition
Coefficient) 1.39
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
Acid Hydrolysis Rate
Constant (M hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant (ml cell
Oxidation Rate Constant



hr-l<> 3 x 10~9
(hr'1) PNER
(M-1hr~ ) INERT
Reference
C-Sw f Kow


Calc
CC-Kow



E-KB

M-OX R02, SO
These data were estimated for use in a preliminary assessment to be
conducted by the EPA, and should not be used in more detailed assessments.
                                 57

-------
                                                                            31
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                      CHjCHj     /,
                  CHjCH/
                                                             N-C
                                   Na'
Compound Name:   DithiocarbaTnate
CAS Registry Number; 148-18-5
.Molecular Weight(g):
171.27
Parameters;

Water Solubility (ppm)
Melting Point  (8C)

Boiling Point  (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation       -
Rate Constant  (ml cell  hr~  )
Photolysis Rate Constant  (hr~l)
Oxidation Rate Constant  (M  hr~  )
                  Reference
1.2 x 105
94-96


5.35
0.04 (partial)



3 x 10~9
PNER
INERT
C-Sw f Kow
Merck (1976)


Calc
CC-Kow



E-KB

M-OX RO2. SO
 These data were estimated for use in a preliminary assessment  to  be
 conducted by the EPA, and should not be used in more detailed  assessments.
                                   58

-------
                                                                             32
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                      CH,-K-!-S.
                                                      CH2-N-C-S"
                                                          H  ||
   Mn
                                  Zn
Compound Name:   Mancozeb
CAS Registry Number: 8018-01-7
.Molecular Weight(g):
540
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation      ..
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M-1hr  )
                  Reference

decomposes
before melting

16.86




3 x 10"9

INERT

Spencer (1973)
•
Calc




E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                   59

-------
                                                                            33
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                      I!  H
                                                  -S-C-N-CH2
                                                           CH2—NH—C—S—Zn—
Compound Name:   Zineb
CAS Registry Number; 12122-67-7	Molecular Weight (g) :     (275.7).
Parameters;

Water Solubility  (ppm)


Boiling Point  (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
                                                  Reference
Acid
Constant
Hydrolysis Ra
ant (M^hr'1)
Rate
Neutral Hydrolysis, Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M  hr~ )
10
decomposes
before melting
negligible
8.62




3 x 10~9

INERT
Spencer (1973)
Spencer (1973)
Spencer (1973)
Calc




E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment  to  be
 conducted by the EPA, and should not be used in more detailed  assessments.
                                  60

-------
                                                                            34
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                 C2H5-S-C-N'
Compound Name:   EPTC
CAS Registry Number; 759-94-4
.Molecular Weight(g):
189.3
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant
Acid Hydrolysis Rate
Constant  (M  hr-1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation      .
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant
Oxidation Rate Constant  (M  hr~ )
                  Reference
375/20°C
137-138/30 torr
3.4 X 10"2
5.92
1.30



3 x 10" 9
PNER
INERT
Spencer (1973)
Spencer (1973)
Spencer (1973)
Calc
CC-Kow



E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  61

-------
                                                                            35
                      EPA CONTRACT 68-03-2981
                      WORK ASSIGNMENT NO. 15
C2H5-S-C-S-C?H,
CAS Registry Number: 623-80-3 Molecular Weight(g): 150
Parameters: Reference
Water Solubilitv (oom) 1<7 X 10
Boiline Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition .
Coefficient) ~U>J^
Alkaline Hydrolysis Rate
Constant (M^hr"1)
Acid Hydrolysis Rate
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation -9
**rp> Crmstant (ml cell~1hr~1') J X 10
PVint-nl v^ r- T?^^ff Pnn^f"nnf fhr~l^ "MbK
Oxidation Rate Constant (M"1^" ) INERT
C-Sw f Kow


Calc
CC-Kow



E-KB.

M-QX R02, SO
These data were estimated for use in a preliminary assessment to be
conducted by the EPA, and should not be used in more detailed assessments.
                                 62

-------
                                                                             36
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
Compound Name:   3,4-dihydro-l(2H)-naphthalenone  (a-tetralone)	

CAS Registry Number;  529-34-0	Molecular Weight(g):       146.19
Parameters;

Water Solubility (ppm)

Melting Point (°C)
Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant
Acid Hydrolysis Rate
Constant  (M^hr""1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M-1hr~ )
Reference
1.6 X 104
5.3-6
113-116/6 torr
3.0 x 10~2
4.57
1.53
NHFG
NHFG
NHFG
1 x 10~7

INERT
C-Sw f Row
Aldrich (1982)
Aldrich (1982)
C-vp f bp
Calc
CC-Kow



E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  63

-------
                                                                            .3Z
                                                                     same as  38
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
Compound Name:    3,4-dihydronaphthalene
CAS Registry Number;  447-53-0	Molecular Weight(g):    130.19
Parameters:
Water Solubility  (ppm)
Boiling Point  (°C)
Vapor Pressure  (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant
                                                       Reference
Acid
Constant
Hydrolysis Ra
ant  (M'-'-hr"1)
Rate
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml  cell  hr~  )
Photolysis Rate  Constant (hr"1)
Oxidation Rate  Constant (M
                              "
98
206-207
0.51
4.07
3.54
NHFG
NHFG
NHFG
1 x 10~7
-
INERT
C-Sw f Kow
Weast (1973)
C-vp f bp
Calc
CC-Kow


•
E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                   64

-------
                                                                            .38
                                                                     same as 37
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
Compound Name:   1,2-dihydronaphthalene
CAS Registry Number; 447-53-0
                                .Molecular Weight(g):    130.19
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (OctanoI/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
                                                  Reference
Acid
Constant
Hydrolysis Ra
ant (M~1hr~1)
Rate
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation       .
Rate Constant  (ml cell  hr~  )
Photolysis Rate Constant  (hr~l)
Oxidation Rate Constant  (M  hr~  )
98
206-207
0.51
4.07
3.54
NHFG
NHFG
NHFG
1 •* in"7

4 x 105
C-Sw f Row
Weast (1973)
C-vp f bp
Calc
CC-Kow


•
F.-UR

M-OX R02
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  65

-------
                                                                            39
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
Compound Name:    1,2,3,4-tetrahydronaphthalene   (Tetralin)	

CAS Registry Number;  119-64-2	Molecular Weight(g):    132.2
Parameters:
Water Solubility  (ppm)
Boiling Point (°C)
Vapor Pressure  (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell" hr~  )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M  hr~  )
Reference
35
207.6
0.3869
4.13
3.96
NHFG
NHFG
NHFG
3 x 10~9

INERT
C-Sw f Kow
Dreisbach (1955)
Dreisbach (1955)
Calc
CC-Kow



E-KB

M-OX R02
 These data were estimated for use in a preliminary assessment  to be
 conducted by the EPA, and should not be used in more detailed  assessments.
                                   66

-------
                                                                        40
                     EPA CONTRACT 68-03-2981
                     WORK ASSIGNMENT NO. 15
                                           CO""
Compound Name:   decahydronaphthol-2
CAS Registry Number;  825-51-4
                          .Molecular Weight(g):     154.25
Parameters:
Water Solubility (ppm)
Boiling  Point C°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
                                           Reference
Hydrolysi
(M-l-hr'1)
is Rate
Alkaline
Constant
Acid Hydrolysis Rate
Constant (M'-^hr'1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr   )
Photolysis  Rate Constant (hr-1)
Oxidation Rate Constant (M-1hr~ )
300
109/14 torr
1.18 x 10~2
4.82
3.15
NHFG
NHFG
NHFG
3 x 10~9
PNER
INERT
C-Sw f Row
Aldrich (1982)
Jaber et al. (1983)
Calc
CC-Kow



E-KB

M-OX R02, SO
 These data were estimated for use in a  preliminary assessment to be
 conducted by the EPA,  and should not be used in more detailed assessments.
                                67

-------
                                                                            41
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
Compound Name:    1-naphthol
CAS Registry Number:  90-15-3
.Molecular WeightCg):    144.16
Parameters;

Water Solubility  (ppm)

Melting Point C°C)
Boiling Point (°C)


Vapor Pressure  (torr)


Molecular Weight/Oxygen
Log  (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
Acid Hydrolysis Rate
Constant  (M^hr"1)
Neutral Hydrolysis  Rate
Constant  (hr~  )
Microbial Degradation
Rate Constant  (ml  cell  hr~  )
Photolysis  Rate  Constant (hr"1)
Oxidation Rate  Constant (M  hr~  )
                  Reference
210
96
288
1.07 X 10~4
4.51
2.62
NHFG
NHFG
NHFG
1 x 10~7

7 x 108
C-Sw f Row
: Merck (1976)
Merck (1976)
C-vp f bp
Calc
CC-Kow



E-KB

M-OX R02
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments,
                                  68

-------
                                                                             42
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO.  15
Compound Name:    2-naphthol
CAS Registry Number;  135-19-3
.Molecular Weight(g):
144.16
Parameters;

Water Solubility (ppm)

Melting Point (°C)
Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       ""
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~  )
Photolysis Rate Constant  (hr-1)
Oxidation Rate Constant  (M-1hr~  )
                  Reference
740
122
285-286
2.24 x 10~4
4.51
2.62
NHFG
NHFG
NHFG
1 x 10~7

1 x 108
Verschueren (1977)
Verschueren (1977)
Merck (1976)
Karyakin et al. (1968)
Calc
CC-Kow


•
E-KB

M-OX R02
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  69

-------
                                                                            43
EPA CONTRACT 68-03-2981 | 1
WORK ASSIGNMENT NO. 15 x\^
. C2H5
Compound Name: 2— methvl— 5— ethvlpvridine
CAS Registry Number: J04.-90-5 Molecular Weight Cg): 121.18
Parameters: Reference
Water Solubility (opm) 1100
Boiling Point (°C) 179.3
Vapor Pressure (torr) 1.13
Molecular Weight/Oxygen 3.78
Log (Octanol/Water Partition
Coefficient) 2.53
Alkaline Hydrolysis Rate
Constant (M^hr'1) NHFG
Acid Hydrolysis Rate
Neutral Hydrolysis Rate
Constant (hr ) NHFG
Microbial Degradation _-
RatP Constant (ml cell'-hir ) 3 x J,Q~

Oxidation Rate Constant (M hr~ ) INERT
C-Sw f Row
Boublik et al. (1973)
Van De Rostvne and Prausnitz
(1980)
Calc
CC-Kow


•
E-KB

M-OX R02, SO
These data were estimated for use in a preliminary assessment to be
conducted by the EPA, and should not be used in more detailed assessments.
                                  70

-------
                                                                            44
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO.  15
                 .O.
    XCH2CH3
   N^
O   CH2 CH3
Compound Name:    N.N-dlethylbenzamide
CAS Registry Number;  1696-17-9
.Molecular Weight(g):
     137
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant
Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation      -
Rate Constant (ml cell  hr~ )
Photolysis Rate Constant (hr"1)
Oxidation Rate Constant (M-1hr~ )
                  Reference
7inn


4.28
1.84
NHFG
NHFG
NHFG
3 x 10~9

INERT
C-Sw f ' Kow


("lair
CC-Kow


•
E-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment  to  be
 conducted by the EPA,  and should not be used in more detailed  assessments.
                                  71

-------
                                                                            45
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                        H
Compound Name:    2-imidazolidinethione   (ethvlenethiourea)

CAS Registry Number;  96-45-7	Molecular Weight(g):
102.16
Parameters:

Water Solubility  (ppm)

Melting Point (°C)
Boiling Point (°C)


Vapor Pressure  (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation _
Rate Constant  (ml  cell  hr   )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M-1hr~  )     4 x 10
                                                       Reference
1.1 x 105
203-204

•
3.19
-1.03 (partial)



i x m-10

4 x 1010
C-Sw f Row
Merck (1976).


Calc
CC-Kow



E-KR

M-OX SO
 These data were estimated for use in a preliminary assessment to  be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  72

-------
                                                                            46
                                                         04H
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
Compound Name:    2.3-dihydro-2,2-dimethyl-7-benzofuranol	

CAS Registry Number;     1563-38-8    Molecular WeightCg):  	220
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~  )
Photolysis Rate Constant
Oxidation Rate Constant  (M-1hr~  )      1 x 10
Reference
700


6.87
2.60
NHFG
NHFG
NHFG
1 x 10-10 '

1 x 107
Merck C19761)


Calc
CC-Kbw


•
K-TTR

M-OX R02
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                   73

-------
                                                                             47
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                         H2C
                           S
                           I
                           CH
Compound Name:    1,2,4-trithiolane
CAS Registry Number;  289-16-7
.Molecular Weight(g):
                           124
Parameters:
Water Solubility  (ppm)
Boiling Point (8C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M^hr -1)
Acid Hydrolysis Rate
Constant (M'-hir"1)
Neutral Hydrolysis Rate
Constant (hr  )
Microbial Degradation
Rate Constant  (ml cell  hr  )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant
                  Reference
1.7 x 106


3.87
-0.40



1 X ID"10
PNER
3 * 1010
C-Sw f Kow


Calc
CC-Kow



E-KB

ftf—nv sn
 These data were estimated for use in a preliminary assessment to  be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  74

-------
                                                                             48
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                     w
Compound Name:   1,1-dlmethylhydrazine
CAS Registry Number; 57-14-7
                            .Molecular  Weight(g):
                                                 60.10
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
                                              Reference
Alkaline
Constant
Hydrolysi
(M^hr'1)
is Rate
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell" hr" )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M-1hr   )
1.2 x 108
63.9
158
157
1.88
-2.42
NHFG
NHFG
NHFG
i x in'10
PNER
labile3
C-Sw f Kow
Merck (1976)
C-vp f bp
Verschueren (1977)
Calc
CC-Kow



F.-TCR

M-OX R02
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.

 GO Reacts  with oxygen directly.  Half-life estimated to be less than 10 days.
                                   75

-------
                                                                             49
                        EPA  CONTRACT  68-03-2981
                        WORK ASSIGNMENT NO.  15
                                        HN—NH

                                         C^CH,
Compound Name:    1.2—dimethvlhvdrazine
CAS Registry Number;   540-73-8
                     .Molecular Weight(g):
60.10
Parameters;

Water  Solubility  (ppm)


Boiling Point  (°C)


Vapor  Pressure (torr)


Molecular Weight/Oxygen
Log  (Octanol/Water  Partition
Coefficient)
                                       Reference
Alkaline
Constant
sis Rate
Acid Hydrolysis  Rate
Constant  (M'-Hir"1)
Neutral Hydrolysis Rate
Constant (hr~  )
Microbial  Degradation
Rate  Constant (ml cell  hr~  )
 Photolysis  Rate Constant (hr'1)
•Oxidation Rate Constant (M-1hr~ )
2.9 x 108
81/753 torr
75
fiQ.9
1.88
-2.76
NHFG
NHFG
NHFG
1 x 10-10
PNER
labile3
C-Sw f Kow
MprrV nPTfil
C-vp f bp
BotihUV, of al . (19731
Calc
CC-Kow



E-KB

M-OX
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
  Ca) Reacts with oxygen directly.  Half-life estimated to be less  than  10 days.
                                   76

-------
                                                                            50
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO.  15
                  H2C=CH
                        I
                        Br
Compound Name:
CAS Registry Number: S93-6Q-2
.Molecular Weight(g):      106.96
Parameters;

Water Solubility (ppm)


Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       '
                  Reference
Acid Hydrolysis Rate
Constant  (M~1hr~1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell" hr~ )
Photolysis Rate Constant  (hr~l)
Oxidation Rate Constant  (M  hr~  )
1.7 x 104
15.80
1033
3.34
1.38
HNES
HNES
HNES

PNER
INERT
C-Sw f Row
Dreishach fiqS9")
Dreisbach (1959)
Calc
CC-Kow


•
VT? - NRn

C-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  77

-------
                                                                            51
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                   Br  Br
                     —CH2
Compound Name:    1,2—dibromoethane
CAS Registry Number:  106-93-4
.Molecular Weight(g):
187.88
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation _
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr~l)
Oxidation Rate Constant  (M~1hr~ )
                  Reference
4300/30°C
131-132
11.70
5.88
1.76
HNES
HNES
3.7 x 10~5
1 x lO'10
PNER
INERT
Soencer (1973)
Merck (1976)
Dreisbach (1959)
Calc
CC-Kbw


E-A-Dibromopropane
E-KB

C-OX R02, SO
 These data were estimated for use in a preliminary assessment  to be
 conducted by the EPA, and should not be used in more detailed  assessments.
                                  78

-------
                                                                             52
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                    HO—
Compound Name: Tetrabromobisphenol A (1.1.3.3-tetrabromo-2.2-bis (4-phenolvl)propane)

CAS Registry Number; 3Q496-13-Q	Molecular Weight(g):  	543.8	
Parameters:

Water Solubility (ppm)

Melting Point (°C)
Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
Acid Hydrolysis Rate
Constant (M'nir"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant (ml cell  hr  )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant
Reference

180-184


17.0




3 x lO'12

2 x 107

Hawley (1977)


Calc



•
E-KB

M-OX R02
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA,  and should not be used in more detailed assessments.
                                   79

-------
                                                                            53
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                           Br
                    o
Compound Name:    bromobenzene
CAS Registry Number;  108-86-1
.Molecular Weight(g):
157.02
Parameters;

Water Solubility  (ppm)


Boiling Point (°C)


Vapor Pressure  (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M-1hr~ )
                  Reference.
450
156.2
4.18
4.91
3.00
NHFG
NHFG
NHFG
3 x 10~9
PNER
INERT
C-Sw f Kow
Dreisbach (1955)
Dreisbach (1955)
Calc
CC-Kow


•
E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment  to be
 conducted by the EPA, and should not be used in more  detailed  assessments.
                                80

-------
                                                                             54
                                                         Br
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                             Br
Compound Name:   1,2-dibromobenzene
CAS Registry Number; 583-53-9
.Molecular Weight(g):
235.9.2
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
Acid Hydrolysis Rate
Constant  (M'-hir"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation      .
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M-1hr~  )
                  Reference
80
224
0,193
7.37
3.86
NHFG
NHFG
NHFG
1 x 10-10

INERT
C-Sw f Kow
Aldrich (1982>>
Dreisbach f!955)
Calc
CC-Kow


•
K-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                   81

-------
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                        Br
                                                      6
                                                        Br
                                                                            55
Compound Name:   Ir4-
CAS Registry Number:  1Q6-37-6
.Molecular Weight(g):
                                                                 235.92
Parameters;

Water Solubility  (ppm)

Melting Point (°C)

Boiling Point (°C)


Vapor Pressure  (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M'-'-hr"1)
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation       .
Rate Constant  (ml cell  hr~  )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M~ hr~  )
                                                       Reference
19
87-89
220.4
0.025
7.37
3.86
NHFG
NHFG
NHFG
1 v in'10

INERT
C-Sw f Row
Aldrich (1982).
Merck C19761)
Jordan (195^
Calc
CC-Kow


•
E-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment to  be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  82

-------
                                                                             56
                                                             Br
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
Compound Name:   1.2.S-tribromobenzene
CAS Registry Number;   608-21-9
                            .Molecular  Weight(g):
                                              314.82
Parameters;

Water Solubility (ppm)

Melting Point (°C)
Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
                                              Reference
Hydrolysi
(M-ihr'1)
is Rate
Alkaline
Constant
Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant (ml cell  hr  )
Photolysis Rate Constant (hr"1)
Oxidation Rate Constant (M  hr~ )
12
87.8


9.84
4.73
NHFG
NHFG
NHFG
1 x ID'10

INERT
C-Sw f Kow
Weast (1973)


Calc
CC-Kow


•
E-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA,  and should not be used in more detailed assessments.
                                  83

-------
                                                                            57
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                          Br
Compound Name:    1,3,5-tribromobenzene
CAS Registry Number;  626-39-1
.Molecular Weight(g):
314.82
Parameters:

Water Solubility (ppm)

Melting Point (°C)

Boiling Point (°C)


Vapor Pressure  (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~  )
Photolysis Rate Constant
Oxidation Rate Constant  (M-1hr~  )
                  Reference
1.3
121-124
?71/7fiS 1-rvrr
6.4 x 10~4
9.84
4.73
NHFG
NHFG
NHFG
1 x lO'10

INERT
C-Sw £ Kow
Aldrich (1982)
Weast (1973)
C-vp f bp
Calc
CC-Kow



E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment  to be
 conducted by the EPA, and should not be used in more detailed  assessments,
                                  84

-------
                                                                            58
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
O
Compound Name:    1,2,3,4-tetrabromobenzene
CAS Registry Number;  22311-25-7      Molecular Weight(g):
          393.72
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log  (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant
Acid Hydrolysis Rate
Constant  (M  hr-1)
Neutral Hydrolysis Rate
Constant  (hr~ )
Microbial Degradation       .
Rate Constant  (ml  cell  hr~  )
Photolysis Rate  Constant  (hr-1)
Oxidation Rate  Constant  (M  hr~  )
 Reference
1.8


12.30
5.59
NHFG
NHFG
NHFG
3 x ID'12

INERT
C-Sw f Row


Calc
CC-Kow



E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                   85

-------
                                                                            59
                                                          Br
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                       Br
                                                         Br

                                                         Br
Compound Name:    1.2.3.5-tetrabromobenzene
CAS Registry Number;    634-89-9	Molecular Weight(g):
                                                             393.72
Parameters;

Water Solubility  (ppm)

Melting Point C°C)
Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M^hr"1)
Acid
Constant
                                                  Reference
Hydrolysis Rate
,ant (M'-Hir"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell" hr~  )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant

1.8
99-100
329
1.3 x 10~6
12.30
5.59
NHFG
NHFG
NHFG
i v in'12

INERT
C-Sw f Row
Weast (1973)
Weast (1973)
C-vp f bp
Calc
CC-Kow


•
F-TTR

M-OX R02. SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  86

-------
                                                                             60

                                                          Br
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
Compound Name:   pentabromobenzene
CAS Registry Number;    608-90-2
.Molecular Weight(g):
472.6
Parameters!

Water Solubility (ppm)

Melting Point (°C)
Boiling Point (°C)    .


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation      .
Rate Constant (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M-1hr~ )
                  Reference
0.25
160-161
sublimes

14.77
6.46
NHFG
NHFG
NHFG
3 x 10-12

INERT
C-Sw f Kow
Weast (1973)
Weast (1973)

Calc
CC-Kow



E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  87

-------
                                                                            61
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO.  15
                        Br

                    8rtbtBr
                      ^^•^ff^*» —
                     BrYBr
                         Br
Compound Name!
CAS Registry Number: 87-82-1
.Molecular Weight(g):
551.52
Parameters:

Water Solubility (ppm)
Melting Point  (°C).
Boiling Point  (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M  hr  )
                  Reference
9 x in"6
327


17.2
7.32
NHFG
NHFG
NHFG
3 x m-12

INERT
C-Sw f Kow
Weast (1973)


Hair-
CC-TCnw



E-KB

M-OX R02. SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used  in more detailed assessments,
                                  88

-------
                                                                            62
                       EPA CONTRACT  68-03-2981
                       WORK ASSIGNMENT NO.  15
                                                   OH
                                                -tbr"
Compound Name:    2,6-dibromophenol
CAS Registry Number;  608-33-3
                            .Molecular Weight(g):
                                                251.9
Parameters;

Water Solubility (ppm)

Melting Point (°C)
Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
                                             Reference
Alkaline
Constant
Hydrolysi
(M-ihr'1)
is Rate
Acid Hydrolysis Rate
Constant (M^hr"1)
Neutral Hydrolysis Rate
Constant (hr~  )
Microbial Degradation
Rate Constant (ml cell  hr  )
Photolysis Rate Constant (hr"1)
Oxidation Rate Constant (M^hr"1)      1 x 10
210
56-7
162/21 torr. (sub-
limes
2.5 x 10~3
7.87
"?.2n (parr-ia!}
NHFG
NHFG
NHFG
1 x lO'10

1 x 107
C-Sw f Row
Weast (1973)
Weast (1973}
I.
C-vp f bp
Calc
CC-Kow


•
E-KB

M-OX R02
 These data were estimated  for use  in a preliminary assessment to be
 conducted by the EPA,  and  should not be used in more detailed assessments.
                                 89

-------
                                                              »H
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                      Q
                                                             Br
                                                                            63
Compound Name:   3,4—dibromophenol
CAS Registry Number; 615-56-5
.Molecular Weight(g):
251.9
Parameters;

Water Solubility (ppm)


Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant
Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M-1hr~ )
                  Reference
440


7.87
3.20 (partial)
NTTFa
NHFfJ
NHFG
3 x 10~9

i -x in7
C-Sw f Row


Calc
CC-Kow


•
E-KB

M-OX R02
 These data were estimated for use in a preliminary assessment  to be
 conducted by the EPA, and should not be used in more detailed  assessments.
                                  90

-------
                                                                             64
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                           OH
                                        o
                                                           Br
                                                              ,Br
Compound Name:   2,4-dibromophenol
CAS Registry Number; 615-58-7
                    .Molecular Weight(g):
                                                                 251.9
Parameters;

Water Solubility (ppm)

Melting Point (°CX
Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
                                      Reference
         Hydrolysi
         (M-ihr'1)
is Rate
Alkaline
Constant
Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr  )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M-1hr~  )
310
40
238-9
1.9 x 10~3
7.87
3.20 (partial)
NHFG
NHFG
NHFG
3 x 10~9

1 x 107
C-Sw f Kow
Weast (1973")
Weast (1973)
C-vp f bp
Calc
CC-Kow



E-KB

M-OX R02
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  91

-------
                                                                            65
                                                           OH
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                  Br ^  Br
Compound Name:    3,5—dibromophenol
CAS Registry Number;  626-41-5
                                .Molecular Weight(g):
                                                251.9
Parameters;

Water Solubility (ppm)


Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
                                                  Reference
Acid
Constant
Hydrolysis Ra
,ant  (M'-'-hr-1)
Rate
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~  )
Photolysis Rate Constant  (hr-1)
Oxidation Rate Constant  (M   hr~  )
440

.
7.87
3.20 (partial)
NHFG
NHFG
NHFG
3 x 10~9

1 x 107
C-Sw f Kow


Calc
CC-Kow



F-KB

M-OX R02
 These data were estimated for use in a preliminary assessment to  be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  92

-------
                                                                             66
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                             OH
                                                          Br
Compound Name:    2,5-dibromophenol
CAS Registry Number; 28165-52-8
.Molecular WeightCg):
251.9
Parameters!

Water Solubility (ppm)


Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (OctanoI/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant       "
Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M  hr~  )
                  Reference
440


7.87
3.20 (partial)
NHFG
NHFG
NHFG
3 x 10~9

1 x 107
C-Sw f Row


Calc
CC-Kow



E-KR

M-OX R02
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  93

-------
                                                                            67
                                                        OH
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                              Br

                                                              Br
Compound Name:    dibromophgnol
CAS Registry Number;  28514-45-6	Molecular Weight(g):
                                                                  251.9
Parameters:
Water Solubility (ppm)
Boiling Point  (°C)
Vapor Pressure  (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
                                                       Reference
Alkaline
Constant
         Hydrolysi
         (M-ihr'1)
                 is Rate
Acid
Constant
     Hydrolysis Ra
     .ant  (M'-hir-1)
                Rate
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation       -
Rate Constant  (ml cell  hr~  )
Photolysis Rate Constant
Oxidation Rate Constant  (M  hr~  )
440


7.87
3.20 (partial)
NHFG
NHFG
NHFG
3 x 10~9

1 x 107
C-Sw f Row


Calc
CC-Kow


•
E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  94

-------
                                                                             68
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                            >H
Compound Name:    2,3-dibromophenol
CAS Registry Number: 57383-80-9
                                .Molecular Weight(g):
                                                  251.9
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant
                                                  Reference
Acid
Constant
Hydrolysis Ra
ant (M'Tir"1)
Rate
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation      ..
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant

440


7.87
V?n ("partial")
NHFG
NHFG
NHFG
3 x 10~9

1 x 107
C-Sw f Kow


Calc
CC-Kow


•
E-KB

M-OX R02
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  95

-------
                                                                            69
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                      Br
Compound Name:    decabromobiphenvl ether
CAS Registry Number;  1163-19-5
                                .Molecular Weight(g):
                                                 959.22
Parameters;

Water Solubility  (ppm)

Melting Point (°C)
Boiling Point (°C)


Vapor Pressure  (torr)


Molecular Weight/Oxygen
Log  (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
                                                 Reference
Acid
Constant
Hydrolysis Ra
ant (M'-hir-1)
Rate
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation     .
Rate Constant  (ml  cell  hr~  )
Photolysis Rate Constant  (hr-1)
Oxidation Rate Constant  (M-1hr~  )
1.3 x 1013"
294 - 296


30.00
12.87 foartial)
NHFG
NHFG
NHFG
3 x 10-12

INERT
C-Sw f Kow
Fluka (19821


Calf
CC-Kow



E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment  to  be
 conducted by the EPA, and should not be used in more detailed  assessments.
                                  96

-------
                                                                             70
                       EPA CONTRACT 68-03-^2981
                       WORK ASSIGNMENT NO. 15
Compound Name:   octabromobiphenyl ether
Parameters;
Boiling Point (°C)
Coefficient)
Constant
Constant  (M  hr")
Constant (hr~ )
umber: 32536-52-0 Molecular WeiehtCe): 442
ty (ppm)
(°C)
(torr)
ht/Oxygen 13.81
ater Partition
lysis Rate
r'1) NHFG
S-R*te NHFG
L )
.ysis Rate
) NHFG
adation _12
(ml cell "Mir ^ 3 x 10 ""
n Pnn^ t* in ^ ^V»T*™"^-^
t Constant (M-1hr~ ) INERT
Reference



Calc



•
E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  97

-------
                                                                             71
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                 H2N-C-N(CHJ2
Compound Name:    N.N-dimethylurea
CAS Registry Number;  598-94-7
.Molecular  Weight(g):
88.11
Parameters:

Water Solubility  (ppm)
Melting Point  (°C)
Boiling Point  (°C)


Vapor Pressure  (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M^hr""1)
                  Reference
Acid Hydrolysis Rate
Constant  (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml  cell"  hr~  )
Photolysis Rate Constant  (hr-1)
Oxidation Rate Constant  (M  hr~  )
7100
106
270
5.9 x 10~4
7.75
1 . fifi CparfiaT)
WNT?S
HNES
HNES
1 •«• in"9
PNER
INERT
C-Sw f Row
Hawley (1977)
Hawley (1977)
C-vp f bp
Calc
CC-Kow



E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments,
                                  98

-------
                                                                             72
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO.  15
              H2N-C-NH- CH-CH2CH3
                  O     CH,
Compound Name:    sec-butylurea
CAS Registry Number; 689-11-2
.Molecular Weight(g):
116.16
Parameters;

Water Solubility (ppm)
Melting Point (°C)
Boiling Point (°C)


Vapor Pressure (torr)


Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant
Acid Hydrolysis Rate
Constant (M  hr"1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant (ml cell  hr  )
Photolysis Rate Constant  (hr~l)
Oxidation Rate Constant  (M-1hr~ )
                  Reference
4.4 x 105
169-170


3.63
0.11
HNES
HNES
HNES
3 * in~9
PNER
INERT
C-Sw f Kow
Weast (1973)


Calc
CC-Kow



E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  99

-------
                                                                            73
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                         H
Compound Name:   dl—sec—butvlurea
CAS Registry Number; 869-79-4
.Molecular Weight(g):
172
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant
Acid Hydrolysis Rate
Constant  (M  hr-1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr~ )
Photolysis Rate Constant  (hr"1)
Oxidation Rate Constant  (M  hr  )
                  Reference
13


5.38
4.46 (partial)
HNES
HNES
HNES
1 v in"9
PNER
INERT
C-Sw f Kow


Calc
CC-Kow


•
•R-tTR

M-OX RO2. SO
 These data were estimated for use in a preliminary assessment  to be
 conducted by the EPA, and should not be used in more detailed  assessments,
                                 100

-------
                                                                 H
                       EPA CONTRACT 68-03-2981
                       WORK ASSIGNMENT NO. 15
                                                                 H
                                                                             74
Compound Name:    di-isopropylurea
CAS Registry Number;  4128-34-7
.Molecular Weight(g)
142
Parameters:
Water Solubility (ppm)
Boiling Point (°C)
Vapor Pressure (torr)
Molecular Weight/Oxygen
Log (Octanol/Water Partition
Coefficient)
Alkaline Hydrolysis Rate
Constant (M~1hr~1)
Acid Hydrolysis Rate
Constant  (M  hr""1)
Neutral Hydrolysis Rate
Constant (hr~ )
Microbial Degradation
Rate Constant  (ml cell  hr  )
Photolysis Rate Constant  (hr'1)
Oxidation Rate Constant  (M  hr~ )
                  Reference
160


4.43
3.38 (partial)
HNES
HNES
HNES
3 x 10~9
PNER
INERT
C-Sw f Row

•
Calc
CC-Kow


•
E-KB

M-OX R02, SO
 These data were estimated for use in a preliminary assessment to be
 conducted by the EPA, and should not be used in more detailed assessments.
                                  101

-------
                               REFERENCES

Aldrich Chemical Company.  1982-1983.  Aldrich Catalog/Handbook of Fine
     Chemicals.  Milwaukee, Wisconsin.

Aly, 0. A. 1976.  Water Res. .10, No. 12, 1047-1050.

Boublik, T., V. Fried, and E. Hala.  1973.  The Vapour Pressures of Pure
     Substances.  Elsevier Scientific Publishing Co., Amsterdam.

Dean, J. A., Ed. 1979.  Lange's Handbook of Chemistry,  Twelfth Edition.
     McGraw-Hill Book Co., New York.

Dreisbach, R. R. 1955.  Physical Properties of Chemical Compounds.
     Advances in Chemistry Series No. 15.  American Chemical Society,
     Washington, DC.

Dreisbach, R. R. 1959.  Physical Properties of Chemical Compdunds-II.
     Advances in Chemistry Series No. 22.  American Chemical Society,
     Washington, DC.

Dreisbach, R. R. 1961.  Physical Properties of Chemical Compounds-Ill.
     Advances in Chemistry Series No. 29.  American Chemical Society,
     Washington, DC.

Fluka Chemical Corporation.  1983/1983 Catalog.  Hauppauge, NY.

Grain, C. 1982.  Vapor Pressure.  In: Handbook of Chemical-Property
     Estimation Methods.  W. J. Lyman, W. F. Reehl, and D. K. Rosenblatt,
     Eds.  McGraw-Hill Book Company, New York.

Grover, R., W. F. Spencer, W. J. Farmer, and T. D. Shoup.  1978.  Weed
     Sci. 26, No. 5, 505-508.

Hawley, G. G. 1977.  The Condensed Chemical Dictionary.  Ninth Edition.
     Van Nostrand Reinhold Co., New York.

Jaber, H. M. , K. C. Irwin, and E. C. Gunderson.  1983.  Data Acquisition
     for Environmental Transport and Fate Screening for Compounds of
     Interest to the Office of Solid Waste.  Part II.  Vapor Pressure
     Measurements.  Final Report for U. S. EPA, Washington, DC.  Work
     Assignment No. 15 in partial fulfillment of EPA Contract No.
     68-03-2981.

Jordan, T. E. 1954.  Vapor Pressure of Organic Compounds.  Interscience
     Publishers, Inc., New York.

Karyakin, N. V., I. B. Rabinovich, and L. G. Pakhomov.  1968.  Zh. Fiz.
     . Khim. 42. No.  7, 1814-1816.

                                  102

-------
Mabey, W. R., and T. Mill. 1978.  J. Phys. Chem. Ref. Data.  7, No. 2,
     383-415.

The Merck Index.  1976.  9th Edition.  Merck and Co., Rahway, New Jersey.

Ouellette, R. P., and J. A. King.  1977.  Chemical Week Pesticide Register
     McGraw-Hill, Co., New York.  345 pp.               ""	 	

Osborn, A. G., and D. R. Douslin.  1966.  J. Chem. Eng. Data. 11, No. 4,
     502-509.

Sopach, E. D., and L. P. Boltromeyuk. 1974.  Gigiena i sanitariya. ]_,
     10-13.

Spencer, E. Y. 1973.  Guide to the Chemicals Used in Crop Protection.
     Agriculture Canada.  Publication 1093, Sixth Edition.  Ottawa,
     Ontario, Canada.

Van De Rostyne, C., and J. M. Prausnitz.  1980.  J. Chem. Eng. Data.  25,
     No. 1, 1-3.

Verschueren, K.  1977.  Handbook of Environmental Data on Organic Chemicals,
     Van Nostrand Reinhold Co., New York.

Vogel, T. 1983.  Unpublished work.  Stanford University, Stanford, CA.

Weast, R. C. Ed. 1973.  Handbook of Chemistry and Physics.  54th Edition.
     CRC Press, Cleveland, OH.

Weber, R. C., P. A. Parker, and M. Bowser.  1981.  Vapor Pressure Distrib-
     ution of Selected Organic Chemicals.  EPA Report No. 600/2-81-021.

Wiedemann, H. G.  1972.  Thermochim. Acta.  .3, No. 5, 355-366.

Yalkowsky, S. H., and S. C. Valvani.  1980.  J. Pharm. Sci. 69. No. 8,
     912-922.
                                   103

-------
                               SECTION 4

               CALCULATION OF PARTITION COEFFICIENTS OF
              ORGANIC CHEMICALS IN AQUATIC ENVIRONMENTS

     This section was taken in whole from W. R. Mabey^ J. H. Smith,
R. T. Podoll, et al.-, "Aquatic Fate Process Data for Organic Priority
Pollutants," EPA Report No. 440/4-81-014, December 1982.
                                     104

-------
                               Section 4
                CALCULATION OF PARTITION COEFFICIENT OF
               ORGANIC CHEMICALS IN AQUATIC ENVIRONMENTS

4.1  BACKGROUND
     The partitioning of a chemical between water and sediment and between
water and biota will affect the concentration of the chemical in water and
the rate of loss of the chemical from aquatic systems.  Solubility data,
on the other hand, are required for calculation of Henry's constants,
which are needed to calculate volatilization rates of chemicals in aquatic
systems.
     This section discusses the relationships between water solubility,
the partition coefficients for a chemical between sediment and biota, \and
the partition coefficient for a chemical between octanol and water.
Moreover, the theoretical basis for such relationships is explained, and
some of the published correlations for these data are discussed.  This
section also briefly discusses the calculation of the octanol-water
partition coefficient data used to calculate many of the other partitioning
constants.
     As discussed in Section 2, the partitioning of a chemical is given
by the equation
                               K  = C /C                           (4.1)
                                p    p  w
where C  and C  are the concentrations on a particulate material  (sediment
       p      w
or biota) and in water, respectively, and K  is the partitioning constant
                                           P
(or coefficient) whose units are determined by those of C  and C   (see
                                                         p      w
section 2).  In practice, C  is usually defined as the amount of chemical
per dry weight of sediment (or organisms) to correct for the variability
of the particulate water content.  The partition coefficient between
*
 This section was taken in whole from W. R. Mabey, J. H. Smith, R. Ti Podoll,
 et al., "Aquatic Fate Process Data for Organic Priority Pollutants," EPA
 Report No. 440/4-81-014, December 1982.
                                       105

-------
microorganism and water, ICg, given  for  individual organic chemicals in
Section 3, is in units  of micrograms  of  chemical per gram of microorganism
divided by grams of  chemical per  liter  of water.  Because the amount of
organic chemical sorbed to  sediments  has been found to depend on the
amount of organic carbon in the sediment, it is useful to normalize a
measured sediment partition coefficient  (K  ) for organic carbon content:

                              Koc - Vfoc                         (4'2)

where f   is the fraction of organic  carbon and K „ is the normalized
       oc                                        oc
(for organic carbon  content) partition  coefficient.  Karickhoff et al.
(1979) have also shown  that, because  f   varies with sediment particle
size, the distribution  of sediment  particle size will markedly affect
measured K   values.
          oc
     The octanol-water  partion coefficient  K   has commonly been used
as a measure of the  hydrophobicity  of a  chemical in medical and toxico-
logical applications as well as in  environmental chemistry  (Hansch and
Leo, 1979; Kenaga and Goring, 1978).  A large number of K   values is
therefore available  as  a result of  the  number of uses of such data.  Most
significantly, K   values can be  calculated from molecular structure  (.see
Section 4.4).  The K   data in Section  3 are given to allow calculations
of other properties  (partitioning coefficients for biota as well as toxi-
cological data) for  use in  environmental assessments of the organic
priority pollutants.

4.2  CALCULATION METHODS
     Several correlation equations  have  been proposed to calculate the
water solubility (S  ) ,  K , and iL,  from K   values and to calculate K
                   w' '   oc        B       ow                         oc
values from water solubility.  The  more  widely used of these equations
are discussed and analyzed  in Section 4.3.  Although we recognize that
better equations are evolving as  more experimental data are obtained,
the following equations are recommended  for use in environmental fate
assessments.
                                    106

-------
4.2.1  Correlation Equations

     In the following equations, all partition coefficients  (K   , K   and
    Vare unitless, and water solubility (S ) is in units of parts per million
      *
Cppm).   As discussed in Section 4.2.2, however, the solubility units of

molarity (moles per liter) or mole fraction are preferred.

     K   and K   are correlated by the following equation (Karickhoff, 1979):
      oc      ow


                      log Koc = 1.00 log KQW- 0.21                (4.3)


     Correlation of S  and K   was reported by Yalkowsky and Valvani  (1980).

For organic pollutants that are liquid in their pure state at 25°C:


                 log S  = -1.08 log K   + 3.70 + log MW            (4.4)


where MW is the molecular weight of the pollutant  (g mole  ).  For organic
pollutants that are solid in their pure state at 25°C:

                                                  /AS
          log Sw = -1.08 log KQW + 3.70 + log ^-(7^;  (mp-25)  (4.5)
where mp is the melting point of the pollutant  (°C) and ASf is the entropy
                                   -1    -1
of fusion of the pollutant  (cal mol   deg  ).   If AS- is not known, it
may be approximated by (Yalkowsky and Valvani,  1980):


                         ASf - 13.6 + 2.5  (n -  5)                  (4-6)


where n is the number flexible atoms (i.e., atoms not involved in double
bonds, triple bonds, or part of a ring structure) in the pollutant molecule,
other than hydrogen.  If n  is less than 5, (n - 5) is set equal to zero.
it
 The original equations in the literature are different if they were
 reported in different solubility units.  Refer to Section 4.2.2 for
 the appropriate solubility units conversion factors.
                                   107

-------
     Correlation of K   and S  is provided by  (Kenaga and Goring, 1978):
                     oc      w


                      log KQC = -0.55 log Sw 4- 3.64                 (4.7)
     K_ can be correlated with K   by
      B                         ow  3
                                   0.16 K                           (4.8)
                                         ow
4.2..2  Units and Conversion Factors
     Three commonly used units of  aqueous  solubility are defined below:

     (.1)  Mole fraction, x,  the unitless ratio of the number of moles of
          solute to the total number  of moles of solute plus water.  In
          symbols, for a binary solution of n moles of solute in n  moles
          of water

                             x = n/(n + nw)

                               — n/n  for  n  » n                   (4.9)
                                    w     w


     (.2)  Molarity, S, expressed in moles  of solute per liter of solution
          CM):
                      S(M) = n(mol)/liter  of  solution               (4.10)
     (3)  Weight fraction, expressed  in  milligrams of  solute per liter of
          water, or parts per million, ppm


              S  (ppm) = "  («ol) MM (8 mol"1)  1000  
-------
or

                                * 55.5 x  for  x  <  10
                                                    "2
                      (4.13)
     To convert from molarity to ppm is  straightforward  by substituting

Equation (4.10) into equation (4.11)  •
                     ppm - S(MW)  (1000)  for  S  <  1 M
                      (4.14)
     Thus to convert from mole fractions  to  ppm follows  from equations

(4.11) and (4.13)
                       ppm =  ,?5:5..*x  (MW)  (1000)
                              (1 - x  )
                            ^55.5(x)  (MW)  (1000)  for x < 10
These conversion factors are  summarized in Table 4.1.
                                                            -2
                      (.4-15)
                                 Table 4.1

                CONVERSION  FACTORS FOR COMPOSITION UNITS
FROM
ppm
(mole fraction)
    M
(Molarity)
                      TO
                               ppm
                                                                   M
(mole fraction)    (Molarity)
	
5.55 x 104(MW)
(UK) (103)
1.80 x 10~5
MW
	
1
55.5
ID'3
MW
55.5
	
                                    109

-------
     Concentration in aqueous solution is prereraoiy given in moie rraction
or molarity units since  these units are measures of the amount of solute
per amount of solution.  The weight fraction or ppm, on the other hand,
expresses the weight of  solute per weight of solution and is thus a
function of the molecular weight of the molecule, which is not relevant
to environmental or toxicological effects.

4.3  CALCULATION OF K    and S  FROM K
                     oc      w       ow
     The sediment partition coefficient, normalized for organic carbon
content (K  ), and aqueous solubility  (S ) of an organic pollutant are
critical to its environmental fate.  Because K   and S  values may ;be
                                              oc      w          J
unmeasured or unreliable, it is important to be able to correlate these
environmental parameters with other experimental quantitites, namely, to
predict unmeasured values and appraise the reliability of measured values.
     It is useful to correlate these parameters with octanol/water
partition coefficients  (K  ) for practical as well as theoretical reasons.
Practically, K   values  are easier to measure and, where K   measurements
          '   ow                                          ow
have not been made, calculated values may be used with confidence.  The
theoretical basis for expecting correlations of K   and S  with K   is
                                                 oc      w       ow
described below.  The correlation of 1C, with other partitioning constants
                                      o
is not discussed in this section since a recent review of the subject is
available.
4.3.1  Partitioning Thermodynamics
     This discussion first considers the partitioning of a chemical
between octanol and water, with octanol being a representative organic
phase.  If a small amount of a chemical is added to a closed vessel
containing n-octanol and water, the vessel is shaken, and the octanol
and water are allowed  to separate, the chemical will partition between
the two phases  (see Figure 4.1).  By convention, the small amount of
chemical in each phase is called  the solute.  The partitioning of the
solute molecules between the two  phases can be understood in terms of a
simple lattice model.   If we assume that every molecule (water, octanol,

                                  110

-------
                           0
     o      s       o      o      o

     w    w    w    w   w   w   w
     w    w    w    w    s   w   w
     w    w    w    w   w   w   w
     w    w    w    w   w   w   w
                                 SA -6729-8

FIGURE 4.1  LATTICE MODEL OF A SOLUTE (S)
           PARTITIONING BETWEEN OCTANOL
           (0) AND WATER (W) PHASES

           K   ' C/C  = 2
s
0
0
w
w
w
w
0 0
0 0
S 0
WWW
w s w
WWW
WWW
s o
0 0
0 S
WWW
WWW
WWW
w s . w
                                   SA-6729-9

FIGURE 4.2  LATTICE MODEL OF A HIGHER MOLE
           FRACTION OF SOLUTE (S) PARTITIONING
           BETWEEN OCTANOL (0> AND WATER
           (W) PHASES
           Because the environment of each solute mole-
           cule is the same. KQW = CQ/Cw =2 as in
           Figure 4.1.

-------
and solute) in both phases occupies a  particular site on a three-dimensional
lattice, with uniform  spacing between  sites, then the fraction of sites
in each phase occupied by the chemical is  the mole fraction x.  A two-
dimensional cross section of this lattice  is shown in Figures 4.1 and
4.2.
     The tendency for  a  solute molecule to leave either phase is propor-
tional to the solute mole fraction in  that phase and to the forces acting
on the solute in that  phase.  The forces acting on a solute molecule will
depend on which molecules occupy neighboring sites on the lattice.
Figures 4.1 and 4.2 show that, over the mole fraction range of x  = 1/28
to x  = 1/14, solute molecules in the  water phase are surrounded by water
molecules.  Thus, the  forces acting on the solute in the water phase are
independent of the solute mole fraction.   Consequently, the tendency (f)
of a solute molecule to  leave the water phase is directly proportional
to its mole fraction:
                                  f =  Hx                          (4.16)
where H is a constant  representing the forces exerted on the solute by
the solvent.  At higher  solute mole fractions, where solute-solute inter-
actions become important (that is, where the solute is concentrated
enough that solute molecules occupy neighboring lattice sites), H becomes
a function [H(x)] of the solute mole fraction, and thus f is no longer
directly proportional  to x:

                               f = H(x) x                         (4.17)

     The partitioning  of the chemical  between the octanol and water phases
depends on this relative tendency of the chemical to leave each phase (f),
which is conveniently  viewed as a force per unit area.  In thermodynamics,
                         *
f is called the fugacity and, as explained above, is proportional to the
relative amount of the solute in the phase, x, and the forces acting on
the solute within each phase; explicitly,
*
 See, for example, G.  L. Lewis  and M. Randall, Thermodynamics, revised
 by K. S. Pitzer and L.  Brewer  (McGraw-Hill, NY, 1961).

                                   112

-------
                             fw= (fV xw
                             fo =  CfV *0                        (4.19)





where subscripts w and o refer, respectively, to the water and octanol

             j^

phases, and f  and Y. are, respectively, the reference fugacity and


activity coefficient, which together represent the forces acting on the


solute in the i   phase.  At equilibrium
                                 fw- fo                           (4.20)
so that
                                   fR
                                   n

In general, at constant pressure, f  depends only on the temperature and


y. depends on the composition as well as the temperature of the i   phase.


In sufficiently dilute solutions , however , the forces acting on a solute


molecule will be independent of x. because, as explained above, the


environment of a solute molecule t


be a function only of temperature
                                                               o

environment of a solute molecule will remain constant.  Thus (f y.) will
                                (fRYi) = H±                         (4.22)





where H. is the Henry's constant for a very dilute solution of the solute


in phase i.  Thus





                              x /x  = H /H                         (4.23)
                               o  w    w  o




is a function only of temperature.  However, if x  or x  is large enough
                                                 o     w

that y  or y  is not constant, then K   will also no longer be constant.
      o     w                        ow                 °
                                  113

-------
     Because composition  is  commonly measured  in moles liter   (M), it


is convenient to define:
                   K   =  C  /C  = r   (x  /x  ) = r   (H /H )           (4.25)
                    ow    o  w    wo  o w    wo  w  o
where r   is a constant  equal  to. the ratio of the molar volume of water





                          r    - v /v    (= 0.115)                   (4.26)
                           wo     w  o
to that of octanol.   (In  terms of  the  lattice mode, r   is equal to the
                                                     wo     n

ratio of the number of  sites  per unit  volume of octanol to that of water.)



     Numerous workers have  correlated  the partitioning of chemicals be-


tween sediment and water  and  between biota  and water with octanol/water


partition coefficients.   Before discussing  these specific correlations


in detail, it is useful to  understand  the conditions that must be met


for these correlations  to be  successful.



     Partitioning of  a  solute between  water and any other water immiscible


phase p (i.e., biota, sediment) may be described by





                            K   = r   (H /H )                        (4.27)
                            pw    wp   w  p                             '





From equation (.4.25)  for  partitioning  between octanol and water
                            H  = K   H /r                          (4.28)
                             w    ow  o  wo
thus
               K   =  (r   /r   )(H  /H  )K   =  r   (H /H  )K             (.4.29)
                pw     wp wo   o  p  ow    op  o  p  ow
where r   is the ratio of  the molar volume  of octanol to that of phase
       op

p.  Thus, taking the  logarithm of both  sides of equation (.4.29)
                                   114

-------
                  log Kpw = log KQW 4- log CropHo/Hp)              (4.30)

Thus, for the second term on the right-hand side of equation (4.30) to
remain constant for a set of chemicals partitioning between water-octanol
and water-phase p, phase p must be chemically similar to octanol and both
K   and K   must be measured at low enough solute concentrations that
 ow      pw
solute-solute interactions are absent.
     The success of K.  -K   correlations (.to be discussed in detail below),
                     ow  oc
for example, may thus be understood.  First, by normalizing adsorption
for organic carbon content, we ensure the chemical similarity of phase p
(.that is, the organic content) and octanol.  Second, the partitioning of
the chemical between the water and sediment phases is usually measured
at very low surface coverage (in the linear region of the adsorption
isotherm) where adsorbate-adsorbate interactions are minimal.
     Octanol/water partition coefficients have been used not only to
correlate other partitioning data, but also to predict aqueous solubili-
ties.  The assumptions implicit in these predictions become apparent
on close examination of the octanol/water partition experiment.
     If it is assumed that the ratio of the number of solute molecules
in each phase remains constant up to the limit of solubility, then

                Kow = (Co/Cw) dilute = (-Co/(Vsaturated            C.4.31}

From equation (4.21), this means that the ratio of activity coefficients
Y /Y  remains constant up to saturation.  As explained above, however,
 wo
the ratio Y /Y  will depend on solute concentration, particularly if
           X  O
C  (saturated) is large enough that solute-solute interactions become
 w
 *Because of the chemical similarity of a neutral organic solute with
  n-octanol, it  is  expected that Y  will not vary significantly with C .
                                   115

-------
important.  Furthermore,  if we assume  that  the solubility of the chemical
in pure water equals its  solubility in the  octanol-saturated water phase
of the partition measurement, then
                              Kow = VSw
where S  and  S   are solubilities  in moles  liter   (M)  in  pure  octanol  and
       o      w
pure water, respectively.
     To correlate  aqueous  solubility with  K  , many authors have  proposed
                                            ow
an equation of  the form:

                       log  S   =  -(I/a) log  K  +  c                 (4.33)
                           w               ow
where a and  c  are  constants.   Equation (4.33) may  be  derived  by  modifying
equation  (4.32)  to account  for deviations  of real  systems  from model  be-
havior:
                              Kow
This  equation is  clearly identical to equation (4.32)  for a = 1.   Taking
the logarithm of  both sides of equation (4.34) and rearranging terms:

                 log S  = - (I/a) log K   + (I/a)  log S            (4.35)
                      w                ow              o
 If  S   is  assumed constant for a set of solutes in octanol, equation
    o
 (4.35)becomes
                 log S  = - (I/a) log K   + c                      (4.36)
                      w                ow
 and the correlation coefficients a and c may be calculated from a plot
 of  known values of log S  versus known values of log K   for the given
                                    116

-------
set of solutes.  Clearly, if the assumptions implicit in equation  (.4.32)
are reasonable, the calculated value of a_ should be close  to one.
     The variability of SQ for a set of solutes is difficult to  quantify
except by comparing liquid and solid solutes.  If two solutes are  identi-
cal except that one is a liquid and the other is a solid in its  pure  state
at temperature T, the solid will be less soluble than the  liquid because
of the additional energy required to remove solute molecules from  the
solid phase.  Thus, if we assume that all liquid solutes have the  same
solubilities in n-octanol, and we use this pure liquid solute as the  ref-
erence state, calculated solid solubilities must be corrected for  the
energy necessary to transform the solid to the liquid state.  This energy
is called the enthalpy of fusion, and from simple thermodynamic  argu-
ments, we can modify equation (.4.35) for solid solutes:

                                                *Hf     Tf- T
      log Sw = - d/a) log Kow 4-  c  -  (I/a)            -          (.4.37)
where AH^ is the enthalpy of fusion, R is the gas constant, and  T-  is
the melting temperature of the solute.  At  the melting point,
                             AHf = Tf ASf                          (.4.38)
Therefore at 25°C, equation  (.4.38) becomes
            log Sw - -  (I/a) log KQW + c - TrRT-Tvr ^P'25)         <-4-39>
where mp is the melting point  (.in  C) and  AS.  is  the entropy  of  fusion
           -1     -1
(in cal deg   mole  ).  This correction is  zero for solutes that are
liquid at 25 C, but substantial for solutes with  high melting points.
Assuming that the theory is approximately  correct and the  correlation
coefficient _a is approximately equal  to one, Table 4^2  and Figure 4.3
illustrate the magnitude of this correction as a  'function  of  melting
point for a hypothetical solute with  an uncorrected solubility of 100  ppm
and a typical entropy of fusion of 13.6 entropy units  (cal deg   mol  ).

                                   117

-------
                               Table 4.2

                  EFFECT OP MELTING POINT CORRECTION
                      ON WATER SOLUBILITY VALUES
 Solubility
(uncorrected)                    e
   (ppm)                        (°C)	              (ppm)

    100                         25                    100

    100                         50                     56

    100                         100                     18

    100                         200                      2

    100                         300                     0.2
*                                                              o
 log S  (.corrected) = log S   Cuncorrected) - 0.01  (mp-25) at 25 C,

 where AS  = 13.6 and a = 1 are assumed in equation  (4-39) and S

 is the water solubility in ppm.
                                  118

-------
 f  0.6  -
                                f = Sw(corrected)/Sw(uncorrected)
f = 10-(O.OD(mp-25)
     -50
50     100     150     200    250
   MELTING TEMPERATURE (°C)
                            300    350
                                                               SA-6729-10
FIGURE 4.3   ENTHALPY OF FUSION CORRECTION FACTOR FOR AQUEOUS SOLUBILITY
            AT 25°C AS A FUNCTION OF MELTING TEMPERATURE
                                 119

-------
4.3.2  Comparison of Reported Correlations
     Table 4.3 lists a representative sample of recently published
correlations among K   , K   , S  .  This section examines these correla-
                    ow   oc   w
tions in detail.
     K  -K  .  As discussed earlier, the sorption constant K   is the
      oc  ow                                r               oc
amount of chemical adsorbed per unit weight of organic carbon in the
sediment divided by the equilibrium concentration of the chemical in
the water phase.  This constant is useful because, once K   has been
determined for a chemical,  the  sorption partition coefficient may be
calculated if the fraction  organic content  Cf  ) is known:
                                             oc

                         K  = K  Cf  N = C  /C                     C4.40)
                          p     oc  oc)    s  w
where
     K   = Sorption partition coefficient
     K   = Sorption partition coefficient normalized for organic carbon
      oc      !.  _
           content
     f   = Fraction of  organic  content  in the sediment  CO < OC <1)
     C   = Concentration  of  the adsorbed chemical
      s
     C   = Equilibrium  solution concentration.

     Furthermore, it  is useful  to be able to predict K   values from
                                                      oc
the more easily measured  K   values.  The theoretical basis for expect-
ing good K  -K   correlations has been  discussed above.  Two recent
  & s     oc  ow
K  -K   correlations  that have  appeared in  the literature are listed in
 oc  ow
Table 4.3.  The significantly different correlation equations of Kenaga
and Goring  (1978) and Karickhoff et al.  (1979) probably reflect the
different data bases  used to correlate  K    with K
                                        oc       ow
                                  120

-------
                                                                     Table  4.3
                                                     REPORTED CORRELATIONS OF  K   .  K   AND  S
                                                                               ou   oc      v
Corrr l;ic Inn
 K   - K
  oc    ow
                                  Equ.it ion
                                                                                           Data  Base
                                                                                                                                    Authors
 K    -  K
 oc    ow
S  - K
 w    ow
log K   = 0.544 log K   + 1.377
     oc              ow
log
          1.00  log Kou - 0.21
               log  S  =  -  0.922  log K   + 4.184
                    w                ow
                 S   In ppm
               log  x   =  -  1.08  log  K    -  1.04
                   s             6  ow
                           AS,
              x   is  the mole  fraction solubility at  25°C
               8
              ASf Is the entropy of fusion in cal deg   mol

              mp Is the melting point In °C  (If mp i 25
              then the term in brackets Is zero)
(4.41)   Pollutants

         I  Aromatic hydrocarbons  (8)
           Carboxyllc acids and esters  (5)
           Phosphorus containing  lnsectlcic.es  (5)
           Ureas and uraclls  (7)
           Symmetrical trlazines  (6)
           Miscellaneous  (14)

         Adsorbents

           Variety of soils

(4.3)    Pollutants
           Polycycllc aromatics (8)
           Chlorinated hydrocarbons (2)

(4.42)   Substituted benzenes and halobenzenes (12)
         llalogenated blphenyls and diphenyl oxides (11)
         Aromatic hydrocarbons (9)
         Phosphorus containing insecticides (16)
         Carboxyllc acids and esters (9)
         Ureas and uraclls (7)
         Miscellaneous (24)

(4.43)   Simple aliphatics and arnmatics
         in the following groups (n <• 114)

           Alcohols
           Halogens
           Amines
           Carboxyllc  acids and esters
           Aldehydes and  ketones             •
           Ethers
           Nitro compounds
              *
               Number In parentheses refer to Che number of pollutants in the data base.
                                                                                                             Kenaga  and  Goring (1978)
Karlckhoff et al. (1979)
                                                                                                            Kenaga and Goring (1978)
                                                                                                            Yalkowsky (1980)

-------
                  x  In the mole fraction solubility
                                                                        Table 4.3 (continued)
                                                              REPORTED  CORRELATIONS OF K  ,  K   AND S
                                                                                        ow   oc      w
   C..r re l.it ion
                   Equation
K   - S       log K   " - 0.55 log S  + 3.64
 oc    w        B  oc               w
                                                                                              Data  Base
                                                                                                                                      Authors
                                                                    (4.7)    Similar to data base  for equation  (4.41)
                                                                                                             Kenaga  and  Coring (1978)
                       in ppn



    K   - S       log K   - - 0.56 log S + 0.70
     oc    u           OB               w
                  log KQC - - 0.56 log Su + 0.93
NJ
                                                 (4.44)   Pollutants




                                                 (4.45)
                                                                          Polychlorlnated blphenyls (3)

                                                                          Pesticides (4)

                                                                          Halogenated ethanes and propones (6)

                                                                          Tetrachloroethene

                                                                          1,2-Dlchlorobenzene


                                                                        Adsorbents


                                                                          Willamette silt loam

                                                                          Miscellaneous other soils
                                                                                                                          Chlou et al. (1979)
    K   - S
     oc    w
log K   » -  0.54  log x   +0.44
     oc          -a
                                                               (4.46)    Similar  to data base for equation (4.3)
Karlckhoff (1979)
                   K    is  the  sorptlon  partition  coefficient  normalized  for  organic matter reported by


                   Chlou et  al.  (1979).  Assuming K  -  1.7  K  ., equation (4.45)  Is  derived.

-------
     The theoretical equation of Table 4.4,
                   log K   =1.00 log K   + constant              (.4.47)
follows from assuming that the second term on the right-hand side of
equation (4.30) is constant; the data base required for a good fit with
equation C4.47) follows from the assumptions used in the derivation of
equation (4.30).  It is clear from Table 4.4 that the data base and
correlation equation of Karickhoff et al. (1979) closely conform with
the theoretical model; however, the data base and correlation equation
of Kenaga and Goring (1978) do not.
     The advantages and disadvantages of using these alternative equa-
tions are not as well defined, however.  Although the equation of
Karickhoff et al. (.1979) conforms to a simple model and accurately pre-
dicts sorption coefficients from K   data for a limited class of organic
chemicals, it has not been widely tested and may be highly inaccurate
for a more universal set of pollutants and soil/sediments.  The equation
of Kenaga and Goring (.1978), however, is strictly empirical and only
roughly predicts K   values from K   data, but it is applicable to a
more universal set of pollutant/adsorbent systems because of the data
base used.  When more precise K   and K   data are available, it will
                      r        oc      ow
be of interest to assess the predictive value of both of these correla-
tions for both the universal set and individual classes of pollutant/
adsorbent systems.  It may become apparent that several correlation
equations may be required to adequately predict K   values from K
values for the variety of systems of interest.
     S  - K     Several comparisons of the equations of Kenaga and Goring
(1978) and Yalkowsky (1980) can be made.  For reasons discussed earlier,
the mole fraction units of solubility used by Yalkowsky are to be pre-
ferred to the ppm units used by Kenaga and Goring.  In fact, to compare
equation (4.42) of Kenaga and Goring with equation (4.43) of Yalkowsky,
we must assume an average molecular weight for the chemicals in the data
                                 123

-------
                                               Table 4.4
                                  DATA BASES FOR K  -K   CORRELATIONS
                                                  oc  ow
log K   =
  "  oc

K
 ow
Kenaga and Goring (1978)

0.54 log K   + 1.38
       "  ow

Measured and calculated
values compiled from
literature
Karickhoff et al. (1979)

1.00 log K   - 0.21
          ow

Measured by Karickhoff
et al.
                                                                                      Theoretical
                                                               1.00 log K   + constant
                                                                      "  oW

                                                               Measured for very
                                                               dilute solution
 OC
Chemicals
Calculated average values
for each chemical from
adsorption coefficients
for widely differing soils

Very wide range of
organic classes
                                Measured values for the
                                silt (high organic content)
                                fractions of two natural
                                sediments

                                Nonpolar or slightly
                                polar organics
                               Uniform organic content
                               of soil/sediment.  Mea-
                               sured for adsorption
                               from very dilute solutions

                               Nonpolar organics

-------
base of Kenaga and Goring.  Converting equation  (4.42) from ppm to mole
fractions units
               log x  = - 0.922 log K   - 0.56 - log MW            (4.48)
where x  is the mole fraction solubility and MW is the average molecular
       s
weight.
     The variation of equation (4.48) with MW is shown in Figure 4.4
and compared with Yalkowsky's equation for liquid solutes.  Two observa-
tions can be made about Figure 4.4.  First, the molecular weight depen-
dence of equation (4.48) is not very great for chemicals in the molecular
weight range of 100-400.  Second, because the average molecular weight
of chemicals in the data base used to determine equation (4.48) is in
the range of 100-400, it is clear that solubilities predicted by equation
(4.48) will be approximately an order of magnitude lower than those
predicted by equation (4.43).
     A comparison of measured solubilities (in molarity units, M) with
those predicted by the equations of Kenaga and Goring and of Yalkowsky
is shown in Table 4.5 for a series of chlorinated methanes and ethanes.
Note that all the chemicals listed in Table 4.5 (except hexachloroethane,
which sublimes) are liquid at 25 C.  Furthermore, is is clear from
Table 4.5 that equation (4.43) of Yalkowsky predicts the aqueous solu-
bility of chlorinated methanes and ethanes very accurately, whereas the
corresponding prediction of equation (4.42) is  an order of magnitude
lower.  Table 4.6, which compares calculated and measured solubilities
for some low melting point aromatics, further supports these conclusions.
     The cause of this discrepancy becomes clear when we examine the con-
trasting methods and data bases used by Kenaga and Goring and by Yalkowsky
to develop their correlations.  Kenaga and Goring empirically correlated
K   with the solubility of a set of chemicals, most of which are solid
 ow
at 25°C.  In other words, Kenaga and Goring implicitly used a solid
solute reference state; consequently, their correlation equation cannot
accurately predict the solubility of a chemical that is liquid at 25 C.
                                   125

-------
-2
-3
-5
-7
       Kenaga and Goring
       (log xs = -0.922 log Kow -0.56 - log MW)
       Yalkowsky	
       (log xs - -1.08 log K^ -1.04)
       xs = Mole Fraction Solubility
       MW = Molecular Weight
      	I	   I	I	I
                                                            MW = 1
                                                           MW = 10
                                                           MW = 100
                                                           MW = 200
                                                           MW = 400
             1
                                                                6
                                   log K
                                        ow
                                                                 SA-6729-11
FIGURE  4.4  COMPARISON OF SOLUBILITY -
                                          EQUATIONS FOR LIQUID SOLUTES
                                   126

-------
                                           Table 4.5
          CALCULATED VERSUS MEASURED SOLUBILITIES FOR CHLORINATED METHANES AND ETHANES
Chloromethane
Dichloromethane
Chloroethane
1,1-Dichloroethane
Trichloromethane
1,1.2-Trichloroethane
1,1,1-Trichloroethane
1,1,2,2-Tetrachloroethane
Tetrachloromethane
Hexachloroethane
log K
ow
0.95
1.26
1.49
1.80
1.96
2.07
2.50
2.66
2.96
4.62
ui|j
-98
-95
-136
-97
-64
-37
-30
-36
-23
Sublimes

Kenaga and Goring
-1.4
-1.87
-2.03
-2.45
-2.67
-2.84
-3.25
-3.48
-3.70
-5.45
(M)
Yalkowsky
-0.32
-0.66
-0.91
-1.24
-1.41
-1.53
-2.00
-2.17
-2.49
-4.29

Measured
-0.89
-0.80
-1.05
-1.25
-1.16
-1.47
-2.27
-1.76
-2.29
-3.68

-------
Yalkowsky, on the other hand,  explicitly used a liquid solute reference
state.  To calculate  the  solubilities  of chemicals that are solid at
25 C, Yalkowsky included  an  entropy  of melting correction term.  Thus
the equation of Yalkowsky, assuming  accurate known values of the entropy
of fusion  CAS,) and melting  point  (.T-.), is equally valid for liquid
and solid solutes.
     As discussed earlier,  if  two  solutes  are  identical except that one
is a liquid and the other is a solid  in its pure state at 25°C, then the
solid will be less soluble  than the liquid by  a factor of
                     exp  [-2.303CASf/1360)(jnp-25)]                 (4.49)
where AS- is the entropy of  fusion and mp  is  the melting point  ( C).
If AS  is constant,  then it  is  clear  from  equation  (4.46) that  solu-
bility decreases as  the melting point increases.  Assuming AS,  = 13.6
entropy units and converting mole fraction solubilities to molarity
units, Figure 4.5 illustrates that equation  (4.43)  of Yalkowsky, in
contrast with equation  (.4.42) of Kenaga and Goring, successfully predicts
the decrease in solubility with increase in melting point for a-, S~>
$-, and y-
     Figure 4.5 also  indicates  that  implicit  in equation  (4.42) of
Kenaga and Goring  is  an  empirical  average  of  the solid solute correction
term.  Because the solubilities of liquid  solutes predicted by equation
C4.42) are approximately an  order  of magnitude lower than measured values,
we can assume that this  average correction term is  approximately equal
to 0.10, which is  the dashed line  in Figure 4.3.  Thus, the predicted
solubilities of equation (.4.42) should  approximate  those  of Yalkowsky
and measured values for  solutes with melting  points in the 100  to 200 C
temperature range.  Figure 4.6  illustrates, in fact, that for solutes
with an approximate molecular weight of 150,  an entropy of fusion of
13.6 and a melting point of  125 C, the  correlation  equations of Yalkowsky
and of Kenaga and  Goring are similar.   Moreover, Table 4.7 illustrates
                                   128

-------
                                                   Table 4.6
                     CALCULATED VERSUS MEASURED SOLUBILITIES FOR LOW MELTING POINT AROMATICS
K)
Nitrobenzene
Benzene
Toluene
Chlorobenzene
Ethylbenzene
1,2-Dichlorobenzene
log K

 1.87
 2.13
 2.79
 2.84
 3.34
 3.56
                                         ow
log S
Kenaga and Goring
-2.63
-2.63
-3.35
-3.48
-3.92
. -4.26
w (M)
Yalkowsky
-1.32
-1.60
-2.31
-2.37
-2.90
-3.14

Measured
-1.82
-1.64
-2.24
-2.37
-2.85
-3.00

-------
    -2.0



    -3.0



—  -4.0

C/J

~  -5.0



    -6.0



    -7.0
                                               Yalkowsky
                                               Kenaga and Goring
                                               Measured
                         5 - BHC
                    7 - BHC
                            a - BHC
                                                         /3-BHC  _
                      I
           50       100      150       200      250
                      MELTING TEMPERATURE (°C)
                                                               300
350
                                                              SA-6729-12
FIGURE 4.5   SOLUBILITIES OF HEXACHLOROCYCLOHEXANES (a-, 0-, 5-, 7-BHC)
            AS A FUNCTION OF MELTING TEMPERATURE
                               130

-------
      -3
      -5
  CT
  O
      -7
Kenaga and Goring 	
log xs - -0.922 log Kow -0.56 - log MW
       MW - 150
Yalkowsky	                            ^s
log xs = -1.08 log K^ -1.04 -[(mp - 25)ASf/1360]
       ASf - 13.6     mp = 125°C
       I	I	I	I	I
                  1
                          3
                       logK™
                                                            SA-6729-13
FIGURE 4.6   COMPARISON OF SOLUBILITY - KQW EQUATIONS FOR SOLID SOLUTES
                                   131

-------
                                                    Table 4.7


                         CALCULATED VERSUS MEASURED SOLUBILITIES FOR SELECTED PESTICIDES
10
ho

Llndane
Aid r in
Chlordane
ODD
DDT
log K
ow
3.89
5.30
5.48
6.20
6.91
MP
113
104
108
112
109
log
Kenaga and Goring
-4.85
-6.24
-6.46
-7.04
-7.74
S (M)
w
Yalkowsky
-4.38
-5.80
-6.04
-6.85
-7.59

Measured
-4.40 to -5.15
-6.30 to -7.35
-5.30 to -6.85
-6.5 to -7.2
-6.6 to -8.5

-------
that for selected pesticides with melting points around 110 C the cor-
relations of Yalkowsky and of Kenaga and Goring compare equally well
with measured values.
     Figure 4.5 also suggests that solubilities predicted from equation
(.4.42) of Kenaga and Goring will become progressively higher relative
to measured values as the melting temperature increases above 200 C.
Table 4.8 indicates that, indeed, measured solubilities of chemicals
with melting points above 200 C systematically fall below those pre-
dicted by Kenaga and Goring.
     In summary, equation C4.42) of Kenaga and Goring should be re-
stricted to chemicals with melting points in the 100  to 200 C range,
but equation (.4.43) of Yalkowsky, because it includes a melting point
correction factor is not limited by melting point restrictions.
     K   - S .   To compare equation (4.7) with equations  (.4.45) and
(4.46), it is again necessary to assume an average molecular weight
for the correlation equation of Kenaga and Goring.  If an average
molecular weight of 200 is assumed, converting equations  (4.7) and
(.4.45) to mole fraction solubility units gives

     log K   = - 0.55 log x  - 0.23    (Kenaga and Goring, 1978)  (4.50)
          o c               s

     log K   = - 0.56 log x  - 0.04    (.Chiou et al., 1979)       (4.51)
          oc               s

     log K   = - 0.54 log x  + 0.44    (Karickhoff et al., 1979)   (4.46)
          oc               s

     Several observations can be made about these equations.  First,
the similarity of equations  (4.50) and (4.51) is remarkable, consider-
ing the contrasting data bases used by Kenaga and Goring and by Chiou
et al. to determine their correlation coefficients.  In fact, equations
C4.50), (4.51), and  C4.46) may all be written in the form
                     K   =  (constant) ,-0-55(10.01)               (4.52)
                      oc               s
                                 133

-------
                               Table 4.8

        AQUEOUS  SOLUBILITIES OF HIGH MELTING POINT CHEMICALS
    Chemical Name
Benzo[k]fluoranthene

Anthracene

Benzo[g,h,i]perylene

Chrysene

Dibenz[a,h]anthracene

TCDD

B-BHC
Melting Point


    217

    219

    222

    258

    270

    303

    309
                                                   Solubilities
                                                       (ppm)
             Predicted by
Measured     Equation (4.42)'
5.6 x 10

0.045

2.6 x 10"

1.8 x 10"

5 x 10~4

2 x 10~4

0.24
0.04

1.2

0.015

0.1

9 x 10~3

7.5 x 10"

4.0
  Kenaga and Goring  (1978)
                                  134

-------
 It  is  not  clear why  the solubility coefficient of -0.55(±0.01) should
 appear in  each  of  these correlations.   If as expected from the above
 discussions  [see equations  (4.3),  (4.42), and (4.43)],
                     log K   =  a log K   + constant                (4.53)
                          oc          ow
 and
                     log K   = - a log x  + constant               (4.54)

where  a ** 1,  then by substituting equation (.4.54) into equation  (4.53)

                                 2
                    log  K   =..- a  log x  + constant               (4.55)
                           •*• - 1.0 log x  + constant
                                         s

      It  is  also  apparent  that none of these three equations accounts for
 the  variation  in solubility  and hence variation in K   value with the
 melting  point  of the adsorbed chemical.  The difference in adsorption
 behavior between solid and liquid solutes, in general, has been well
.documented  in  the literature (see, for example, Kipling, 1965).  In fact,
 Roe  (1975)  has accounted  for this difference in terms of the solid solute
 correction  factor discussed  earlier in this report.  Karickhoff et al.
 C1979),  in  discussing their  relatively poor correlation of K   with x
                                                             OC       S
 (.compared with their excellent correlation of K   with K  ) , mention
 that a correction term is probably needed in equation (4.40) to account
 for  the  enthalpy of fusion of the chemicals they studied.
      K_  - K  .   The partitioning of organic chemicals has recently been
       p     ow
 reviewed by Baughman and  Paris (1981), who noted the paucity of reliable
 data available for correlating K,, with other partitioning parameters.
 For  the  chemicals in Section 3, the following equation was used to cal-
 culate Kg

                              K_ = 0.16 K                       '   (.4.8)
                               B         ow
                                   135

-------
which is the simplified version of  the equation given by Baughman and
Paris (1981),
                      log Kg  =  0.907  log KQW - 0.21                (4.56)
The reader is referred  to the above review for an excellent exposition
on the problems of reliably measuring K_ and the use of correlation
                                       B
equations to calculate  K_ from  S or from K   or K   data.
                        B       w         oc     ow

4.4  CALCULATION OF K   FROM STRUCTURAL PARAMETERS
                     ow
     The thermodynamics of partitioning of a chemical solution between
octanol and water phases was discussed in 4.3.1, and the use of the
octanol/water partition coefficient, K  , for calculating S , K   and
              ^                     '  ow                °  w'  oc
K_ was described in Section 4.3.2.  Although K   is the symbol used by
 fi                                            ow
many scientists for this partition coefficient, earlier literature and
some current medical toxicology literature has commonly referred to the
logarithm value of K    as "log  P"  (Hansch and Leo, 1979).  For discussion
                    ow
in this section only, the log P nomenclature will be used instead of
log K  , although the K  term  will be used.
  °  ow'       e        ow
     The K   data on the data sheets in Section 3 were calculated using
a computer program developed at SRI; it uses the FRAGMENT method for
calculating log P values  (Bansch and Leo, 1979).  The theory and pro-
cedures for these calculations  are discussed in detail in that reference.
Briefly, the method assumes that select groups of atoms in a molecule
can be considered fragments, each  of which contributes to the total log
P value in an additive  manner

                                    n
                            log P  = X a f                         (4.57)
                                    1  n n
where a is  the number  of occurrences of  fragment  f of structural type n.
Values of f have  been  empirically  derived  from the vast body of log P
data available in the  literature.   Since the  calculation  of log P values

                                    136

-------
for complex molecules can be time-consuming and subject to numerous cal-
culation errors, the FRAGMENT calculation method and the data base for
fragment values have been incorporated into a computer program using the
                         *
PROPHET computer network.   The log P data are generated by first enter-
ing the structure on a graphic tablet.  The log P program then uses an
ordered substructure search routine to obtain fragment values for frag-
ments of the molecular structure.  Fragments are used, rather than atoms,
because atomic contributions to log P vary with certain structural en-
vironments.  The program then adds the fragment values to obtain log P
values.  It also identifies where the log P calculation may be incomplete
because of the absence of values for -particular fragments or because
polar interactions must be accommodated by manual calculations.  The log
P program is under continuing development and evaluation at SRI and
other laboratories .

     The manual calculation of log P values using the FRAGMENT method
is already established as a valid method for obtaining these data (Hansch
and Leo, 1979).  The calculations are, of course, subject to errors
arising from subtle structural differences that are not recognized or
cannot be accounted for when obtaining empirical values for the molecular
fragments.  In fact, the primary source of error is the original data
on which the fragment values are based.  The lack of reliable data is
also a dilemma for verification of calculated log P values.
     As an indicator of the accuracy of the log P calculation program
Table 4.9 compares the K   values recently published by Hasse-tt et al.
                        ow
(1980) with the K   values calculated by the log P program.  Although
                 ow
the chemicals are not  among  the organic priority pollutants, they do
represent some of the best K   data currently available.  The calculated
                            ow
and measured K   values agree within the factor of two for 8 of the 14
              ow
*PROPHET  is a NIH resource  available  to biological  and chemical
  scientists  on  a time-share  basis.   Information on the  log  P/PROPHET
  system can be obtained  from  Dr. Howard L.  Johnson  at SRI.
                                  137

-------
                                                    Table 4.9
                              CORRELATION OP MEASURED AND CALCULATED VALUES OF K
                                                                                ow

                                                                                Computer-Calculated
                      _       .                    Measured K   ± S.D.a              K            b
           	Compound	         	ow	           	ow         r
           Pyrene                                  124,000 ± 11,000                79,400      1.6
           7,12-Dimethylbenz[a]anthracene          953,000 ± 59,000               871,000      1.1
           Dibenz[a,h)anthracene                 3,170,000 ± 883,000            5,890,000      0.54
           3-Methylcholanthrene                  2,632,000 ± 701,000            9,330,000      0.28
           Dibenzothiophene                         24,000 ± 2,200                 33,900      0.71
w          Acridine                                  4,200 ± 940                    2,570      1.6
           13H-Dibenzo[a,i]carbazole             2,514,000 ± 761,000              692,000      3.6
           Acetophenone                               38.6 ± 1.2                     38.9      0.99
           1-Napthol                                   700 ±62                       417      1.7
           Benzidine                                  46.0 ± 2.2                     35.5      1.3
           2-Aminoanthracene                        13,400 ± 930                    1,660      8.1
           6-Aminochrysene                          96,600 ±4,200                 24,000      4.0
           Anthracene-9-carboxyllc acid              1,300 ± 130                   15,500      0.08
           3 Hassett et al. (1980).
           b Ratio of measured K   to calculated K  .
                                ow                ow

-------
compounds listed and agree within a factor of five for 12 of the 14
compounds.  It is also significant to note that the last three compounds
in Table 4.9 show the most disagreement between calculated and measured
K   values, and these compounds are large molecules containing groups
that may participate in H-bonding interactions.

     In general, the accuracy of log P calculations by this method
closely approaches the accuracy of experimental determinations performed
over the last ten or twenty years because the fragment values were
derived largely from those experimental data (by regression analysis)
and incorporate the same experimental errors.  It is not uncommon for
measured log P values for a given compound in the literature to vary
by 1 to 2 units; this corresponds to a factor of 10 to 100 in measured
K   variation.
 ow
                                  139

-------
1 TECHNICAL REPORT DATA
1 (Please read Instructions on the reverse before completing)
1. REPORT NO. 2.
OHEA-E-119
». TITLE AND SUBTITLE
Data Acquisition for Environmental Transport ancHFate
Screening for Compounds of Interest to the Office of
Solid Waste
?. AUTHOR(S)
H.M. Jaber, W. R. Mabey, A.T. Liu, T.W. Chou, H.L.
Johnson, T. Mill, R.T. Podoll, and J.S. Winterle
). PERFORMING ORGANIZATION NAME AND ADDRESS
SRI International
333 Ravenswood Avenue
Menlo Park, CA 94025
12. SPONSORING AGENCY NAME AND ADDRESS-
US Environmental Protection Agency, OHEA, ORD, .".-i
Exposure Assessment Group
Washington, DC 20460
3. RECIPIENT'S ACCESSION NO.
5. REPORT DATE
February 1984
6. PERFORMING ORGANIZATION CODE
8. PERFORMING ORGANIZATION REPORT NO.
10. PROGRAM ELEMENT NO.
11. CONTRACT/GRANT NO.
EPA Contract No. 68-03-2981
Work Assignment 15
13. TYPE OF REPORT AND PERIOD COVERED
Project Report 5/83-9/83
14. SPONSORING AGENCY CODE
15. SUPPLEMENTARY NOTES
16. ABSTRACT
      Physical properties, equilibrium,  and kinetic  constants  for  evaluating  the  trans-
 formation and transport  in aquatic systems for organic  chemicals  of  interest to  the
 US Environmental Protection Agency's Office of Solid Waste  during FY  1983  have been
 obtained from the  literature and calculated from  theoretical  or empirical  relations.
 Values for selected physical properties such  as melting point, boiling  point,  vapor
 pressure, water solubility, and octanol/water partitioning, and for  rate constants
 such as hydrolysis, microbial degradation, photolysis,  and  oxidation  are
 each chemical along with the source of  the data.  Values are  reported in
 suitable for use in a current aquatic fate model.   A discussion of the  empirical
 relationships between water solubility, octanol/water partition coefficients,  and
 partition coefficients for sediment and biota is  presented.
                                                     listed
                                                     units
for

17. KEY WORDS AND DOCUMENT ANALYSIS
a. DESCRIPTORS
-
18. DISTRIBUTION STATEMENT
Release Unlimited; Available through NTIS
b.lDENTIFIERS/OPEN ENDED TERMS

19. SECURITY CLASS (This Report)
Unclassified
20. SECURITY CLASS (This page/
Unclassified
c. COSATI Field/Group
•
21. NO. OF PAGES
146
22. PRICE
EPA Form 2220-1 (Rev. 4-77)
PREVIOUS EDITION IS OBSOLETE

-------
                                                          INSTRUCTIONS

   1.    REPORT NUMBER
        Insert the EPA report number as it appears on the cover of the publication.

   2.    LEAVE BLANK

   3.    RECIPIENTS ACCESSION NUMBER
        Reserved for use by each report recipient.

   4.    TITLE AND SUBTITLE
        Title  should indicate  clearly and briefly the subject coverage of the report, and be displayed prominently. Set subtitle, if used, in smaller
        type or otherwise subordinate it to main title. When a report  is prepared in more than one volume, repeat the primary title, add volume
        number and include subtitle for the specific title.

   5.    REPORT DATE
        Each  report shall carry a date indicating at least  month and year.  Indicate the basis on which it was selected (e.g.. dale of issue, date of
        approval, date of preparation, etc.).

   6.    PERFORMING ORGANIZATION CODE
        Leave blank.

   7.    AUTHOR(S)
        Give name(s) in conventional order (John R. Doe, J. Robert Doe, etc.).  List author's affiliation if it differs from the performing organi-
        zation.

   8.    PERFORMING ORGANIZATION REPORT NUMBER                                                           '.
        Insert if performing organization wishes to assign this number.

   9.    PERFORMING ORGANIZATION NAME AND ADDRESS
        Give name, street, city, state, and ZIP code.  List no more  than two levels of an organizational hirearchy.

   10.   PROGRAM ELEMENT NUMBER
        Use the program element number under which the report was prepared. Subordinate numbers may be included in parentheses.

   11.   CONTRACT/GRANT NUMBER
        Insert contract or grant number under which report was prepared.

   12.   SPONSORING AGENCY NAME AND ADDRESS
        Include ZIP code.

   13.   TYPE OF REPORT AND PERIOD COVERED
        Indicate interim final, etc., and if applicable, dates covered.

   14.   SPONSORING AGENCY CODE
        Insert appropriate code.

   15.   SUPPLEMENTARY  NOTES
        Enter information not included elsewhere but useful, such as:  Prepared in cooperation with. Translation  of, ('resented at conference of,
        To be published in, Supersedes, Supplements, etc.

   16.   ABSTRACT
        Include a brief (200 words or less) factual summary of the most significant information contained  in the report. If tlie report  contains a
        significant bibliography or literature survey, mention it here.

  . 17.   KEY  WORDS AND DOCUMENT ANALYSIS
        (a) DESCRIPTORS - Select from the Thesaurus  of Engineering and Scientific Terms the proper authori/.ed terms that  identify the major
        concept of the research and are sufficiently specific and precise to be used as index entries for cataloging.

        (b) IDENTIFIERS AND OPEN-ENDED TERMS - Use identifiers  for project names, code  names, equipment designators, etc. Use open-
        ended terms written in descriptor form for those subjects for which no descriptor exists.

        (c) COSATI HELD GROUP - Field and group assignments are to be taken from the 1965 C'OSATl Subject Category List.  Since the ma-
        jority of documents are multidisciplinary in nature, the Primary Field/Group assignment(s) will be specific discipline, area of human
        endeavor, or type of  physical object. The application(s) will be cross-referenced with secondary I ield/Croup assignments that will follow
        the primary posting(s).

   18.   DISTRIBUTION STATEMENT
        Denote releasability to the public or limitation for reasons other than security for example "Release Unlimited."  C'ite any availability to
        the public, with address and price.

   19. &20.  SECURITY CLASSIFICATION
        DO NOT submit classified reports to the National Technical Information service.

   21.   NUMBER OF PAGES
        Insert the total number of pages, including this one and unnumbered pages, but exclude distribution list,  if any.

   22.   PRICE
        Insert the price set by the National Technical Information Service or the Government Printing Office, if known.
EPA Form 2220-1  (Rev. 4-77) (Reverse)

-------