DIIS#PR#PYL METHYLPH#SPH#NATE (DIMP) PROFILE OF DRINKING WATER CONTAMINANTS FOR EMERGENCY RESPONSE GENERAL INFORMATION Diisopropyl methylphosphonate (DIMP) is a stable by-product or contaminant in the effluent from the manufacture of the military nerve gas isopropyl methylphosphonofluoridate (GB). DIMP constitutes about 2-3% of crude GB. In the United States, active production of GB- containing DIMP occurred between 1953 and 1957 at the Rocky Mountain Arsenal in Colorado where it was subsequently stored. Remaining stockpiles of GB are mandated for destruction by 1994. DIMP that was disposed of in surface ponds at the Arsenal has contaminated ground water and is known to accumulate in plants. In water, DIMP is stable for over 2 years and is not af- fected by photolysis, biodegradation, or volatil- ization. In soil, it readily migrates with water. Biotransformation in soil is slow. DIMP is not likely to enter the atmosphere due to its low volatility. PHARMACOKINETICS DIMP is readily absorbed following oral ad- ministration to mice, rats, and dogs and is widely distributed throughout the body. Greater than 90% of the radiolabeled compound is excreted in urine. One major metabolite, isopropyl methyl phosphonic acid, accounts for 95% of the excreted compound. HEALTH EFFECTS Humans No data are available on the potential systemic human health effects of exposure to DIMP. A skin sensitization test performed on 215 volunteers showed no allergic dermatitis. HEALTH EFFECTS Experimental Animals Acute toxicity studies in a variety of species indicate that DIMP acts on the central nervous system to produce ataxia, copious salivation, lethargy, and coma. Cattle showed additional signs of cerebral edema and encephalitis. DIMP is a significant eye irritant in rabbits, but upon dermal application, it produces only minimal skin irritation. In guinea pigs, DIMP was not found to be a skin sensitizer following dermal application. Studies in mink and dogs fed DIMP for 21 days or less showed no DIMP toxicity. Blood, intestinal, and ophthalmologic?! changes seen in rats, mice, or dogs fed DIMP for 90 days were not clearly related to DIMP toxi- city. In a three-generation drinking water study with rats, decreases in the viability ratio and lac- tation viability of pups were observed. No other reproductive or developmental effects were found. Lifetime toxicity and carcinogenicity data are not available. \ No mutagenic effects were seen in in vitro bacterial assays. OTHER CRITERIA, ANALYSES, AND TREAT- MENT TECHNOLOGIES In 1984, the U.S. Army Medical Bioengineer- ing Research and Development Laboratory recom- mended an interim limit for DIMP of 26.3 mg/L in drinking water. Methods for the analysis of DIMP include gas chromatography with a flame photometric phos- phorus detector, infrared and Raman spectros- copy, thin layer and paper chromatography, nuclear magnetic resonance spectroscopy, and field ionization mass spectrometry. Gas chroma- tography using a flame photometric phosphorus detector is considered the method of choice. No data on treatment technologies were found although adsorption by activated carbon and several synthetic sorbents appear feasible. ------- Physical and Chemical Properties Empirical Formula Synonyms CAS Number Physical State Molecular Weight Boiling Point Liquid Density Vapor Pressure Solubility (at 25°C) WV DIMP, Diisopropyl methylphosphonate, Diisopropyl methanephosphonate, Phosphonic acid, Methyl-, bis-( 1 -methyl-ethyl) ester, Phosphonic acid, Methyl diisopropyl ester 1445-75-6 CH3 O CH3 Colorless liquid \ II / 180.18 CH-O-P-O-CH 174°C CH3 ch3 ch3 0.976 g/cm3 at 25°C 77 mm Hg at 10°C; 122 mm Hg at 100°C In water 1-2 g/L at 25°C and >11 g/L at >80°C. Health Effects Data and Advisory Values Genotoxicity Reproductive and Developmental Effects Cancer Classification DIMP did not induce genetic effects in Salmonella and Saccharomyces cerevisiae assays with or without activation. A significant decrease in the viability ratio of F3a rat pups and in the lactation viability of F3b pups were observed in a three-generation drinking water study with Sprague-Dawley rats. No other reproductive or developmental effects were found. The results of a mink study were considered inconclusive. EPA Group D, not classifiable as to human carcinogenicity. Reference Dose (RfD) 0.08 mg/kg/day Drinking Water 3 mg/L Equivalent Level (DWEL) Health Advisory Values One-Day 8 mg/L Ten-Day 8 mg/L Longer-Term (child) 8 mg/L Longer-Term (adult) 30 mg/L Lifetime 0.6 mg/L This summary was developed using information from the Drinking Water Health Advisory. For further information contact EPA's Office of Science and Technology at (202) 260-7571. Office of Science and Technology Office of Water U.S. Environmental Protection Agency 401 M Street, SW Washington, DC 20460 June 17,1991 ------- |