EPA/600/A-97/042
                                              Proceedings of healthy buildings '95
Mixtures of Volatile Organic Compounds: Detection of Odor, Nasal
Pungency, and Eye Irritation
      J, Enrique Cometto-Muniz and William S. Cain

      Chemosensory Perception Laboratory, Department of Surgery (Otolaryngology),
      University of California, San Diego, La Jolla, CA 92093-0957, USA.
INTRODUCTION

      Human beings can typically sense, in sufficient concentration, almost any organic
vapor via smell, though some substances have lower thresholds than others by as many as
nine orders of magnitude (see Cain, 1988; Devos, Patte, et al., 1990). The reasons for this
spread in potency remain surprisingly obscure. In part, it seems due to physicochemica!
properties, such as solubility. In aliphatic series, for example, more lipid- soluble members
generally have greater potency  (Cometto-Muniz and Cain, 1994). This holds only up to a
certain point  in the series, where potency shows either no further increase or an actual
decrease. Such an outcome suggests  that,  in  addition to solubility  or  some correlated
property, molecular size may also determine odor potency. That is, even with sufficient
vapor pressure to become airborne in quantity,  molecules can Be too  big to stimulate
effectively.
      At some concentration, typically above the odor threshold, organic vapors may also
trigger chemesthesis, i.e., may  be felt  rather than smelled. The  chemesthetic modality or
common chemical sense (CCS) is mediated in the mucosac of the face by the trigeminal
nerve. The difference in concentration between  when a substance can be smelled and when
that same substance can be felt depends in part upon its reactivity Towards mucosal tissue.
Aggressive vapors, such as formaldehyde, acrolein, ozone, and others, may damage tissue
and thereby be felt. In these cases, the vapors often  have chemesthetic thresholds in the
rough vicinity of their  odor thresholds. For formaldehyde, for example, nasal irritation
occurs at a concentration only  a few times higher than the odor threshold (Berglund and
Shams Esfandabad, 1992).
      Most organic vapors in  the environment do not react readily with mucosal tissue,
yet these too may have some ability to stimulate the chemesthetic sense. In such cases, the
concentration required for detection via feel lies at least an order of magnitude, and in some
instances many orders of magnitude, above that required for detection via odor. In recent
investigations, we  have  charted the difference between  olfactory and chemesthetic
thresholds  for various  aliphatic series of chemicals (Cometto-Muniz and Cain,  1990;
Cometto-Muniz  and Cain,  1991; Cometto-Muniz and Cain, 1993; Cometto-Muniz and
Cain, 1994). In general, the chemesthetic outcome of interest  was nasal pungency,  though
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 in some cases it was ocular pungency (eye irritation) (Comctto-Mun^ and Cain, 1995). As
 with odor potency, chcmesthetic potency increased with chain length, though not in exactly
 (he same way. Chemesthetic potency increased somewhat more predictably. For example, it
 increased with  chain  length in much the same way from one series to another. In this
 behavior, chemesthesis mimicked phenomena such as narcosis and anesthesia that these
 same organic vapors can induce under appropriate conditions.
       Our results have also implied that, to a  first approximation: a) chemesthctic
 detection via the eye occurs at about the same concentration as chemcsthetic detection via
 the nose, and b) the threshold of detection via  feel occurs at the same level of saturated
 vapor concentration irrespective of the substance or the series it comes from.  Decades ago,
 Ferguson (Ferguson, 1939; Ferguson, 1951) articulated a principle that various phenomena,
 e.g., anesthesia, occurred at fixed percentages of saturated vapor, or, as he expressed it, at
 criterion  levels of thermodynamic activity. This in turn suggested an equilibrium between
 concentration in the  vapor phase and concentration in  the biophasc where biological
 activation occurred. Insofar as a biological effect takes place at a criterion percentage of
 saturated vapor only for members within a particular scries, it is not  sufficient to imply the
 veracity of the Ferguson principle. Insofar as  the effect takes place at a criterion level
 across all series, it  does. For chemesthesis, it seems to hold roughly  (Abraham, Andonian-
 Haftvan, Comctto-Muniz, and Cain, 1995).
       Nielsen  and associates (Nielsen and Alarie, 1982;  Nielsen, 1991) argued  for a
 protein receptor as the site of transduction for chcmesthetic responses  to nonrcactive
 irritants,  though they  admitted that  such compounds might exert  their  action through
 nonspecific physical adsorption. It is tempting to speculate that the  rules of chemesthesis
 indicated  in  our various studies  imply stimulation  without need  to invoke  a receptor.
 Certainly, high quantities of organic chemicals can have direct effects on membranes. For
 example, high quantities can change fluidity and can allow ion  flux across a  membrane.
 Such phenomena can generally account  for narcosis and anesthesia, two  of the  very
 biological properties seen as analogous to sensory  irritation.  Regarding olfaction, recent
 studies point towards  the existence of many protein receptors (Buck and  Axel,  1991).
 Olfaction distinguishes itself from chemesthesis in remarkable variation in  sensory quality
 such as skunky, fishy, floral, minty, ethereal, and so on. The many receptors of olfaction
 presumably permit the discriminations upon which such qualitative variation is based.
 Chemesthesis exhibits only trivial qualitative variation in comparison.
       A quantitative  structure-activity relationship (QSAR) based upon a linear solvation
energy relationship (LSER) has described the  relative potency of organic  vapors for a
 number of biological  effects (e.g., anesthesia,  respiratory depression) in  animal  models
 (Abraham, 1993).  Abraham and colleagues have  demonstrated that a  five-parameter
equation that  describes the biophasc as a solvent for impinging vapors can account for 97%
or more of variance in potency (Abraham, Whiting, ct a!.. 1990; Abraham, 1993; Abraham.
 Nielsen, ct al., 1994).  A roughly analogous four-parameter solution  of an LSER for nasal
 irritation  in humans has accounted for 96% of the variance (Abraham, Andonian-Haftvan.
etal., 1995).
       Our cxpcrimcnial strategy has entailed testing subjects diagnosed (Cain, I9S9) as
 anosmic (i.e., lacking olfaction) to chart thresholds for nasal pungency independently from
smell. We also test normosmic subjects (i e., persons with normal olfaction) matched' to the
 anosmics in age, gender, and smoking-status to map corresponding odor thresholds. In the
 present extension of our series of studies, we explored thresholds for odor, nasal pungency,
and eye irritation for mixtures of the relatively nonrcactive compounds studied previously
 individually.
       Most  studies of mixtures of odoriferous vapors  have examined  suprathrcshold
perception  via ratings of intensity (e.g., Olsson, 1994). Such studies have found that the
perceived  intensity of mixtures falls short  of the sum of the intensities of their (unmixed)
components (e.g.,  Bcrglund and  Olsson,  1993). Perceived intensity  of  suprathreshold
mixtures also falls somewhat below predictions made from "addition" of concentration but
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much closer to it than addition of sensory  magnitude (Cain, Schict, et al.  1995).
Suprathreshold experiments with pungent odorants at concentrations that clearly appealed
also to the nasal CCS yielded a concentration-dependent degree of addition of perceived
intensity (Comctto-Muniz, Garcfa-Medina, ct al., 1989). Whereas suprathreshold odor in
such mixtures displayed hypoadditivity of sensation, nasal pungency displayed additivity or
even hyperadditivity (Cometto-Mufiiz and Hemdndez, 1990).
       Exploration  of differences in "additivity"  between  odor  and pungency  at
suprathreshold levels has had no counterpart at the threshold level.  Few investigations
have explored potency of odor in mixtures, and none has apparently explored potency of
nasal  pungency  in mixtures. The outcomes for odor have uncovered  simple stimulus
agonism (Guadagni, Buttery, et al.,  1963; Patterson,  Stevens, et al., 1993) and some
evidence of synergistic stimulus  agonism, particularly for  mixtures of three or more
components (Rosen, Peter, et al.,  1962; Baker, 1963; Laska and Hudson,  1991). Simple
agonism in, for example, a balanced three-component mixture  implies that when the
substances  are presented mixed, each needs to be at only  1/3 its  individual threshold
concentration for the mixture to be perceived. Synergistic agonism implies  — following
the same example of a three-component mixture — that  individual substances need to be at
a concentration even lower than 1/3 of their respective thresholds for the mixture to  be
perceived; whereas partial agonism implies that they need to be at a concentration higher
than  1/3 of their respective thresholds but less than the threshold value itself. Independence
implies that at least one of the components in the mixture needs to be at its individual
threshold for the mixture to be perceived. Finally, antagonism implies that the componenls
need to be at concentrations  higher than their individual thresholds for the mixture to  be
perceived.
      In view of earlier research  in olfaction and in view of the  success of an LSER to
predict nasal pungency, we  expected both olfaction  and chemesthesis to show  simple
agonism with some possibility of an increase in agonism toward synergy as the mixtures
increased in number of components.

METHODS

Stimuli

      The  stimuli  included  members of homologous  series of alcohols (1-propanol,  1-
butanol, 1-hexanol), esters (ethyl acetate,  hexyl acetate, heptyl acetate), ketones (2-
pentanone, 2-heptanone), and alkylbenzenes (toluene, ethyl benzene, and propyl benzene).
All were analytical-grade reagents. Single chemicals tested for the three relevant sensory
responses of odor, nasal pungency, and eye irritation were: 1-propanol, 1-hexanol, ethyl
acetate, heptyl acetate, 2-pcntanone, 2-heptanone, toluene,  ethyl benzene, and  propyl
benzene. Mineral oil served as solvent to prepare three-fold dilution steps of the pure (100
%v/v) substance (i.e.,  33, 11, 3.7, 1.1, etc., %v/v). Due to the limited solubility of 1-
propanol in  mineral oil,  the first two members of its series, 33 and 11 %v/v, were prepared
in deionizcd water.
      Five  mixtures were  prepared using mineral  oil as solvent:  two 3-component
mixtures (labeled A and B, below), two 6-component mixtures (labeled C and D), and one
9-component mixture (labeled E). Mixture A comprised: l-propanol, ethyl acetate, and 2-
pcntanone.  Mixture B comprised:  1-hexanol. heptyl acetate, and 2-heptanone. Mixture C
comprised:  1-propanol,  1-butanol,  ethyl acetate, 2-pentanone,  toluene, and ethyl benzene.
Mixture D comprised-  1-hexanol,  I-heptanol, hexyl acetate, heptyl acetate, 2-heptanone,
and propyl  benzene. Mixture E comprised:  1-propanol,  1-hexanol, ethyl acetate, heptyl
acetate, 2-pentanone, 2-heptanone, toluene, ethyl benzene, and propyl benzene. These
particular mixtures were chosen to give one 3-component (i.e., A) and one 6-component
('•e., C) mixture of relatively  low molecular weight, high vapor pressure chemicals; one 3-
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component (i.e., B) and one 6-component (i.e., D) mixture of higher molecular weight,
lower vapor pressure chemicals; and one 9-component mixture (i.e., E) having both kinds
of chemicals.
       Substances in each liquid mixture were present in proportions thai reflected their
odor thresholds measured  in  our  previous  studies (Cometto-Muniz and  Cain,  1990;
Cometto-Muniz and Cain,  1991; Cometto-Muniz and Cain, 1993; Cometto-Muniz and
Cain, 1994). This was done  by using a "reference" that contained, for each liquid mixture,
components at their individual odor thresholds as found previously. For example, the odor
thresholds for  1-propanol, ethyl acetate, and 2-pentanone equaled 0.0051, 0.0017, and
0.0017%v/v, respectively, and the reference for this three-component mixture therefore had
these concentrations. Based on such a  reference, threefold steps in concentration  were
prepared for each mixture both above and below the reference. Accordingly, the first step
for mixture A above the reference was: 0.015  (0.0051  X 3), 0.0051 (0.0017  X 3), and
0.0051 (0.0017 X 3)%v/v, respectively, for 1-propanol, ethyl acetate, and 2-pentanone. The
first step below the reference was:  0.0017 (0.0051 -K 3), 0.00056 (0.0017 H- 3), 0.00056
(0.0017 •*• 3)%v/v, respectively, for the same chemicals in the same order. Steps above the
reference  continued until they reached the maximum value that could  be presented in a
mixture of the specified proportions (e.g., for mixture A: 33, II, and 11 %v/v cf 1 -propanol,
ethyl acetate, and  2-pcntanone,  respectively). Steps below the threshold continued until
they fell definitively below the odor threshold for even the most sensitive subject.
       We prepared duplicate series for  each of the nine single chemicals and each of the
five mixtures. Stimuli were delivered from cylindrical, squeezable polyethylene bottles
(270 ml capacity) (Cain, 1989) containing 30 ml of solution. For measurements of odor and
nasal pungency, the bottle closure had a  pop-up spout that fit into the nostril  being tested.
Each nostril was tested separately. For measurements of eye irritation, the bottle caps held a
tube that  led  to a 25-ml  measuring chamber (of the  type used  in  variable  volume
dispensers), the rim of which was placed around the eye. Each eye was tested separately.
The tube that fed the chamber was connected to the headspace of the bottle. A squeeze of
the bottle delivered a puff of vapor into the measuring chamber where the eye was exposed.
A polyethylene dust cover closed the open end of the measuring chamber when the bottle
was not in use.
       The concentration of  each compound in the headspace of every bottle was measured
by a gas chromatograph (photoionization detector) equipped with  a gas sampling valve,
allowing direct sampling of the  headspace. For every single or mixed stimulus, repeated
chromatographic readings were taken at each dilution step. Readings were also taken from
bottles containing pure chemicals (100 %v/v). The  headspace of a bottle with  a pure
chemical contains  vapor saturated with  the chemical at room temperature (23 °C). The
concentration of the saturated vapor from each substance was retrieved from the literature.
Knowledge of saturated  vapor concentration (at 23°C) and  its  associated average
chromatographic reading allowed conversion of the readings from  the other bottles into
concentration units (ppm by volume), and derivation of a calibration curve.

Subjects

       Eight subjects, four  males and four females, provided values  for odor and eve
irritation thresholds. The subjects covered a wide range of age (21  to 60 years) in order to
match the group of anosmics available for testing nasal pungency thresholds. Participants
included a male and a female in each of the following categories: early twenties,  early
thirties, early forties, and late fifties/sixty. A  21 year-old male became unavailable after
being tested for odor thresholds. In order to complete the group, he was replaced by a 22
year-old male tested only for eye irritation thresholds.
       Four anosmic  subjects, two males and two females,  provided values for  nasal
pungency  thresholds. One participant was a head-trauma anosmic (male, 66 years old), the
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 other three were congenital anosmics (a male, 43 years old, and two females, 20 and 62
 years old, respectively),

 Procedure

       On odor and nasal pungency trials, participants delivered the stimulus by inserting
 the pop-out probe inside the specified nostril and squeezing the bottle as they sniffed. On
 eye irritation trials, they squeezed the bottle while the eye was exposed in the measuring
 chamber. Subjects quickly learned to squeeze and sniff with equal vigor on every trial.
       We used a forced-choice ascending method of limits to  measure threshold. The
 subject had to choose the stronger smelling or stronger feeling of two stimuli. One was a
 blank of mineral oil and, at the start, the other was a high dilution-step, low concentration
 of the  stimulus, either single chemical  or mixture. If the choice was correct, testing
 continued with the same step from the duplicate set, also paired with a blank. If the choice
 was incorrect, testing continued with the next step — a liquid-phase concentration three
 times higher — paired with a blank. In this way, correct choices entailed the presentation of
 the same concentration, whereas errors triggered  step-wise increments in concentration.
 The procedure continued until five correct choices were made in a row, in which case that
 step was  taken as threshold. Once the threshold was measured for one nostril or eye, the
 other nostril or eye was tested. After this, testing began again with another stimulus. Both
 (he ascending-concentration approach to the  threshold and the separate testing of each
 nostril  helped  to minimize effects of adaptation, frequently encountered in olfactory
 investigations (see Cometto-Muniz and Cain, 1995).
       Sessions typically lasted between one and two hours and were repeated until eight
 thresholds per subject, four for each nostril or eye, were obtained for each single compound
 and each  mixture. This equaled a total of 64 odor or eye irritation thresholds per stimulus
 and 32  nasal pungency thresholds per stimulus.

 Data analysis

       Geometric means served to summarize threshold concentrations within and among
subjects. The geometric mean acknowledges that threshold data for chemosensory stimuli
conform to log normal distributions (Brown, Mac  Lean, et al.,  1968; Amoore, 1986; Gain
and Gent, 1991).
       For analysis of agonism in mixtures, consider the case of a three-component
mixture with a formulation that reflects perfectly a subject's relative sensitivity to its three
components unmixed.  Such a mixture would be  perfectly balanced.  If the components
were simply to add their individual effects,  detection would occur when each component
fell at one-third the concentration of its unmixed threshold.  Hence, if component A had a
threshold of 3 ppm, component  B of 9 ppm, and component C of 27 ppm, and if the
mixture were made up in the proportions 1:3:9, respectively, for balance, then we would
expect detection  for the mixture to occur with component A at 1  ppm, component B at 3
ppm, and component C at 9 ppm.
       The relative contribution of components  in a just-detectable, three-component
mixture can be reflected in the formula: WS - a(RA) + b(Ru) + c(Rc), where WS stands
for weighted sum; RA = concentration of A in mixture •*• threshold A; RB = concentration
of B in  mixture -s- threshold B; RC — concentration of C in mixture * threshold C; and  with
a, b, and c as weighting coefficients to reflect the degree of balance in the mixture. These
weighting coefficients in our three-component mixture are defined as follows: a = [RA/(RA
+ RB + RC)] *  3; b = [RB/(RA + RB + Rc)l * 3; c = [RC/(RA + RB + RC)] * 3.  The
second  factor (3 in our case) of each coefficient represents the number of components in the
mixture.
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       In our example, WS = 1(1/3)  + 1(1/3) +1(1/3)  = 1, which implies complete
agonism of stimulating power. In an unbalanced mixture, which  occurs more commonly
than not because no single subject has exactly the same sensitivity as the reference group
used to formulate the mixture, a, b, and c will take on different values, but will always add
up to 3 for a three-component mixture, to 6 for a six-component mixture, and to 9 for a
nine-component mixture. Irrespective of the relative weights of the components, whenever
WS lies  at  1.0 simple  agonism will have held. Whenever WS lies significantly above or
below 1.0, then departure from simple agonism will have held, as follows: 1) WS above 1.0
implies that the components do not add their sensory potency completely when mixed
(partial agonism or even antagonism) and 2) WS beiow 1.0 implies that the components
have gained sensory potency when mixed (synergistic agonism).
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Figure 1. Thresholds (ppm ± SD) for nasal pungency (filled squares), eye irritation (triangles), and odor
(empty squares). The SD is indicated by the dots. The nine sections of the graph correspond lo nine
substances. Each section lists, first, the threshold  for  the substance by itself (e.g., 1-propanol), then,
consecutively, the level at which that substance was present when the threshold was achieved for mixtures
of increasing complexity, e.g., l-propanol in mixture & (3 components) when A achieved threshold, I-
propanol in C (6 components) when  C achieved threshold, 1-propane! in E (9 components) when E
achieved threshold.
RESULTS

       Figure 1 presents thresholds (ppm by  volume) for all three sensory responses
plotted  for each of the nine substances. The graph is divided in nine sections one per
substance. Within a section, the first value corresponds to the threshold (odor, eye irritation,
and  nasal pungency) of the substance  when  presented alone. Subsequent thresholds
correspond to the concentration at which the substance was present when that particular
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mixture reached threshold (e.g., l-propanol in A corresponds to the level of 1-propanol
found in mixture A when the mixture achieved threshold). A common trend in the three
sensory responses and all chemicals is for thresholds to decline with increasing number of
components in the mixture. This indicates that some degree of stimulus agonism is taking
place in the mixtures to help precipitate odor, eye irritation, and nasal pungency when each
component is below its individual sensory threshold. It should be pointed out that pungency
thresholds for hcptyl acetate and propyl benzene presented alone could only be measured in
two to four of eight repetitions per subject (depending on the anosmic). Probably as a result
of this, the pungency threshold for mixture D could only be measured in two  to five of the
eight repetitions. Hence, values given for the pungency of these two chemicals and of
mixture D do  not represent the average of all anosmics on  all repetitions, but do represent
the average of those cases where a threshold was obtained.
 Table I.
Weighted sum (WS) of ratios of mixed thresholds/unmixed thresholds.
Odor
Subject 1
2
3
4
5
6
7
8
Geo. Mean
Eye Irritation
Subject I
2
3
4
5
6
7
8
Gco, Mean
Nasal Pungency
Subject 1
2
3
4
Geo. Mean

1.0
4.9
6.4
3.7
2.6
5.9
5.0
2.8
3.6

2.2
1.6
1.9
1.9
1.0
2.1
3.3
2.0
1.9

2.1
2.2
1.3
2.4
1.9
                       Three Components
                Mixture A      Mixture B
                                6.6
                                2.8
                                1.9
                                3.0
                                6.3
                                1.4
                                0.3
                                4.7
                                2.5

                                6.0
                                0.9
                                1.4
                                1.6
                                0.6
                                1.1
                                2.2
                                4.6
                                1.7

                                0.7
                                2.3
                                2.0
                                0.9
                                1.3
                              Six Components        Nine Components
                             Mixture C   Mixture D     Mixture E
                                0.9
                                6.3
                                3.7
                                2.3
                                6.5
                                2.0
                                7.2
                                4.2
                                3.4
                                5.8
                                7.0
                                6.6
                                6.7
                                6.S
1.8
1.6
0.4
3.2
1.4
0.6
2.3
1.1
1,3
3.1
2.0
3.0
2.6
2.9
1.4
2.6
i.l
2.2
0.6
0.4
0.2
0.6
0.4
0.03
0.2
0.1
0.2
0.8
0.5
1.0
1.1
0.8
IA
1.3
1.2
2.0
1.8
1.0
2.0
3.0
1.6

O.S
0.5
0.6
0.6
0.7
0.3
0.9
0.3
0.6

1.7
1.5
1.5
1.8
1.6
       Table 1 shows, subject-by-subject, values of WS from the formula given in the
section on data analysis. For averages across subjects, 12 out of 15 cases yielded WS's
above  1.0 which implies a general tendency for components to act, at most, as partial
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agonists in mixtures. This varied, however, both with sense modality and with complexity
of a mixture.
       To  compare  odor with eye irritation, an analysis of variance (ANOVA) was
performed  on the logarithm of the values in Table I with the two variables modality (two
levels: odor vs eye irritation)  and  mixtures (five levels) in a repeated-measures design
(recall that seven subjects were common to all measures, with the eighth subject in each
group matched to a counterpart in the other). The results revealed a significant difference
between modalities (F[l,7]=25.86, p=0.001), with eye irritation showing higher stimulus
agonism; a significant difference among mixtures (F[4,28]=14.01, p<0.00005), with the
more complex mixtures tending to  show greater agonism; and a significant interaction of
modality by mixture (F[4,28]=4.37, p=0.007) which reflected the tendency  for complexity
to have more leverage for eye irritation.
       ANOVA on the same values, but excluding mixture E, which contained substances
of both low and high lipophilicity  gave a view of the variables  modality, complexity of
mixture, and lipophilicity. The results again revealed  significant  differences for modality
(F[l,7]=18.98, p=0.003), as well as  for three vs six components (F[l,7]=9.38, p=0.02), with
six showing greater agonism, and for lipophilicity (F[l,7)=l  1.18, p=0.01), with the
mixtures (B and D) of the more lipophilic substances  snowing greater agonism. The two-
way interaction of number of  components by lipophilicity and the three-way interaction
were also significant (F[I,7]=23.97, p=0.002 and F[ 1,7]=8.71, p=0.02,  respectively).

Table 2. Results of 95% confidence intervals on log WS. Expected value for agonism = 0, i.e., log of 1.0.
Modality	Mixture	n	Mean	S.D	Result


Odor



Eye
Irritation



Nasal
Pungency


A
B
C
D
E
A
B
C
D
E
A
B
C
D
E
8
8
8
8
8
8
8
8
8
8
4
4
4
.4
4
0.551
0.390
0.532
0.115
0.207
0.281
0.238
0.344
-0.645
-0.261
0.285
0.113
0.813
-0.093
0.203
0.263
0.436
0.317
0.296
• 0.151
0.145
0.343
0.167
0.444
0.180
0.124
0.246
0.035
0.157
0.046
Partial agonism
Partial agonism
Partial agonism
Agonism
Partial aponism
Partial agonism
Agonism
Partial agonism
Syncrgistic agonism
Svncrgistic agonism
Partial agonism
Agonism
Partial agonism
Agonism
Partial agonism
       Two ANOVAs were analogously performed on log WS for nasal pungency. The
first was a one-way  ANOVA  that  showed  significant differences among  mixtures
(F[4,12]=18.40, p<0.00005). The second was a two-way ANOVA that again  excluded
mixture E and showed significant differences  for lipophilicity (F[l,3]=50.26, p=0.006),
with the more lipophilic substances  showing greater agonism, and  for the interaction
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number-of-components by lipophilicity (F[1,3]=I2.10, p=0.04), but not for number of
components.
       Ninety-five  percent confidence intervals around  the log WSs allowed us to
determine if the values for each mixture and modality differed significantly from 0 (simple
agonism), i.e., if WS differed significantly from 1.0.  The results, shown in Table 2,
reinforce the picture that mixtures increase their degree of stimulus agonism with
increasing number of components and increasing lipophilicity of components. Eye irritation
even reached syncrgistic agonism for the most lipophilic (D) and the most complex (E)
mixtures.

DISCUSSION

       Studies of odor mixtures at threshold levels have been very few and have generally
entailed no vapor-phase calibration of the stimuli, typically liquid  solutions of odorant
presented in open containers.  Without such calibration, the data could in any instance
reflect departures from Raoult's law (proportionality between the vapor-pressure of a solute
and its mole fraction in solution) as readily as they do the biological rules of how humans
detect mixtures.
       A study of odor thresholds for three chemicals (1-butanol, p-cresol, and pyridine)
relevant to off-flavors in drinking water yielded simple agonism most commonly in binary
mixtures and synergistic agonism in  the ternary mixture (Rosen, Peter, et al., 1962). A
study of food-related chemicals by Guadagni et al. (Guadagni, Buttery, et al.,  1963) also
yielded simple agonism among components in all but one of 20 mixtures composed of two
to 10 components. The components  included various saturated and  unsaturated aliphatic
aldehydes, an alcohol, a carboxylic acid, a sulfide, and an aminc. Another study motivated
by the flavor of drinking water yielded synergistic agonism for many binary mixtures of
eight starting materials (m-cresol, pyridine,  1-butanol, acrylonitrile, n-amyl acetate, 2,4-
dichlorophenol, acetophenone, n-butyl  mcrcaptan) and for the eight-component mixture
(Baker,  1963).  The investigation yielded antagonism for the pair m-cresol—acetophenone.
       More recently,  Laska  and Hudson  (Laska and  Hudson, 1991) measured odor
thresholds for  various single chemicals (isoamyl acetate,  alpha-pinene, cyclohexanone,
cineole, linalool, (-)-carvone, t-butylcyclohexyl acetate, mcthylpropylkctone, and dccyl
acetate) and for three-component mixtures.  The general outcome suggested simple-to-
synergistic agonism.
       The trend of the data therefore lay  towards  simple-to-synergistic agonism, with
greater synergism for more complex mixtures.  When, in a recent investigation, we studied
a psychophysically balanced,  rigorously-calibrated ternary  mixture of 1-butanol, 2-
pentanone, and n-butyl acetate, we also obtained simple agonism (Patterson, Stevens, Cain,
and Cometto-Muniz, 1993).  Hence,  when the mixture  achieved odor threshold, the
headspacc concentration  of each component  was approximately  one third that of the
individual odor threshold of the component.  This outcome lent credence to earlier results
with non-calibrated stimuli insofar as it indicated that the olfactory  system could display
simple agonism.
       The present data argue for partial as opposed to simple agonism, though degree of
agonism tended toward simpte as the number of components increased.  Differences among
stimuli  and among people (see Table 1) both need further attention in the quest for
generalities. For at least  the present stimuli,  it  seems reasonably certain that irritation
exhibits more agonism than odor and that eye irritation exhibits the most. Lipophilicity
seems important in mixtures for both modalities.
       We have yet to  develop any theory to explain why agonism would increase with
complexity.  Theory might need to await definitive dismissal of the possibility that the
tendency for agonism to increase with complexity results  from  a complexity-dependent
vulnerability towards imbalance in mixtures, whether for odor or irritation.  For simple
mixtures (e.g., two or three components), small errors of measurement could  mimic just
                                        179

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about any outcome, from synergistic agonism to antagonism. Scrutiny of our data revealed
no significant correlation between degree of imbalance, measured as root-mean-squared
deviation from perfect balance, and degree of agonism.  Nevertheless, the matter merits
continued attention in the choice of conditions in future investigations. Despite the penalty
of additional work, complex mixtures will reveal more about agonism than will  simple
mixtures.
       As if to add insult to injury, the proper study of agonism  should  also include
variation in  the proportions of components in mixtures.  Measurements should therefore
include psychometric (stimulus-response) functions  for each component unmixed and
against the many backgrounds of various proportions of the components.  A ten-component
mixture, studied in  a few subjects, could consequently entail millions of sensory and
analytical measurements.  Would it be worth Ihe effort of a few person-years of work to
make such measurements in a strategically-chosen mixture. In our view, it would, both for
theoretical and practical understanding.  We see our present work and our work on single
chemicals chosen -from homologous chemical  series as relevant to the choice of. that
strategic mixture.
       What are the practical implications of what we  know now for human detection of
VOCs in indoor air, where scores may be present simultaneously?  In any such mixture,
the more lipophilic substances  will have much more weight as sensory stimuli.  The
LSER developed by  Abraham, Andonian-Haftvan, Comctto-Muniz, and Cain (1995)
gives quantitative predictions of exactly how much.  In mixtures, lipophilicity takes on
even more importance, for it may increase the "gain" in detection, but agonism would in
any case reduce the  amount by which any single substance needed to be present to
contribute to detection of irritation or odor. Conservatively predicted, the "gain"  from
complexity  would be just proportional to the level of complexity. In that case, a 100-
component mixture, balanced for the effect of its components, would require 1/100th of
the threshold of each component to cause a  sensory  effect.  The possibility thai
complexity-dependent agonism may actually lead to synergistic agonism, no matter what
the sensory channel, would make the prediction of a 100-fold gain conservative possibly
by orders of magnitude.  In reality, though, mixtures may be dominated by just a few
components  and until we know just how agonism operates in such unbalanced cases via
the study of varying proportions we will be left with an uncomfortable degree of
uncertainty.

Summary

       Thresholds for detection of odor, nasal pungency (irritation), and eye irritation were
measured for single volatile organic compounds (VOCs) (I-propanol, 1-hexanol, ethyl
acetate, heplyl acetate, 2-pentanone, 2-heptanone, toluene, ethyl benzene, and  propyl
benzene) and certain mixtures of them (two three-component mixtures, two six-component
mixtures and one nine-component mixture). Nasal pungency was measured in persons
lacking a functional sense of smell to avoid interference from olfaction. The results showed
the existence of various degrees of stimulus agonism (additive effects) in the three sensory
channels. Such agonism  increased with  the complexity of the mixtures and with the
lipophilicity  of their components. Eye irritation even showed synergistic stimulus agonism
for the  most lipophilic (one of the  six-component)  and the most  complex  (the nine-
component)  mixtures.  The results indicate that complex chemical environments  may
enable chemosensory, and particularly irritative, detection when single VOCs lie far below
their individual thresholds.  Even the present rather rudimentary state of knowledge  of how
lipophiticity influences detection of single VOCs and how it and complexity (number of
components) influence detection of mixtures would  presumably allow refinement of a
measure such as total mass (or concentration) of volatile organic compounds (TVOC) into a
much more meaningful index that we  might call the perceptually weighted level of VOCs,
                                        180

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or PWVOC.  Such an index, like the index dB(A) for sound, could make an otherwise
strictly physical measurement at least somewhat predictive of human responses.

 Acknowledgments

       The research described  in this article was supported by NIH Grant DC00284 and
by the United States Environmental Protection Agency through Cooperative Agreement N°
CR-816362-02 awarded to the  John  B. Pierce Laboratory. It has been reviewed by the
Agency  and cleared for publication, but does not necessarily reflect the views of the
Agency  and no official endorsement should be  inferred. Mention of  trade names or
commercial products does not constitute endorsement or recommendation for use. Thanks
are due  to Mrs. Robin.Babbitt and Mr. Todd  O'Hearn  for their excellent  technical
assistance.   Research performed while J.E.C.-M. was a member of  the Carrera de!
Investigador Cientifico, Consejo Nacional de Investigaciones CientiTicas  y  Tecnicas
(CONICET), Republica Argentina,  -
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NRMRL-RTP-P-202
           TECHNICAL RiPORT DATA
     (Please read Instructions on she reverse before comple\
1. REPORT NO.
:PA/600/A-97/042
                           2.
4. TITLE AND SUBTITLE
                                                      5. REPORT DATE
Mixtures of Volatile Organic Compounds: Detection of
 Odor, Nasal Pungency, and Eye Irritation
                                 6. PERFORMING ORGANIZATION CODE
7. AUTHOR(S)
J. Enrique Cometto-Muniz and William S. Cain
                                                      8. PERFORMING ORGANIZATION REPORT NO.
9. PERFORMING ORGANIZATION NAME AND ADDRESS
Chemosensory Perception Laboratory
Department of Surgery (Otolarygology)
University of California, San Diego
La Jolla,  California  92093-0957
                                                      10. PROGRAM ELEMENT NO.
                                 11. CONTRACT/GRANT NO.
                                  EPA  CR 816362-02
                                  NIH Grant DC00284
12, SPONSORING AGENCY NAME AND ADDRESS
 EPA, Office of Research and Development
 Air Pollution Prevention and Control Division
 Research Triangle Park, NC  27711
                                  13. TYPE OF REPORT AND PERIOD COVERED
                                  Published paper; 9/95	
                                  14. SPONSORING AGENCY CODE
                                   EPA/600/13
15. SUPPLEMENTARY NOTES A PPCD project officer is Mark A. Mason, Mail Drop 54,  919/541-
4835. Presented at Healthy Buildings '95, Milan, Italy,  9/10-14/95.
16. ABSTRACT
          The paper gives results of the measurement of threshold responses of
odor, nasal pungency (irritation), and eye irritation for single chemicals (l-propa-
nol,  1-hexanol, ethyl acetate, heptyl acetate,  2-pentanone, toluene,  ethyl benzene,
and propyl benzene),  and their mixtures (two  three-component mixtures,  two six-
component mixtures, and one nine-component mixture). Nasal pungency was mea-
sured in subjects lacking a functional sense of smell  (i. e., anosmics) to avoid inter-
ference from olfaction. Various degrees of stimulus  agonism (additive effects) were
observed for each of the three sensory channels when testing mixtures. As the num-
ber of components and the lipophilicity of such components in the mixtures increa-
sed, so did the degree of agonism. Synergistic stimulus agonism characterized the
eye irritation response for the most complex  (the nine-component) and the most lipo-
      (one of the six-component) mixtures. Physicochemical properties play a large
role in the determination of sensitivity to airborne chemicals, particularly to their
ability to evoke irritation. Whereas this has revealed itself previously with respect
to single chemicals, it seems to have relevance to mixtures as well.
17.
                             KEY WORDS AND DOCUMENT ANALYSIS
                DESCRIPTORS
                      b.IDENTIFIERS/OPEN ENDED TERMS C. COSATI Field/Group
Pollution
Measurement
Organic Compounds
Volatility
Smell
Odors
Olfactory Nerve
Senses
Pollution Control
Stationary Sources
Nasal Pungency
Nasal Irritation
Eye Irritation
Trigeniinal Nerve
13 B
14G
07C
20 M
360,05J
36P
18. DISTRIBUTION STATEMENT

 Release to Public
                      19. SECURITY CLASS (This Report)
                      Unclassified
                                                                   21. NO. OF PAGES
                      20. SECURITY CLASS (Thispage)
                      Unclassified
                                               22. PRICE
EPA Form 2220-1 (9-73J

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